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—— (5S)-7-(cyclobutylmethyl)-2-[2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O3S
(5S)-7-(cyclobutylmethyl)-2-[2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[4-(Dimethylamino)phenyl]methylidene]-3-(2,4-dimethylphenyl)-2-(2-fluorophenyl)imidazol-4-one —— C26H24FN3O
5-[[4-(Dimethylamino)phenyl]methylidene]-3-(2,4-dimethylphenyl)-2-(2-fluorophenyl)imidazol-4-one
—— 5-[(1R)-1-(2-methylimidazol-1-yl)ethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole —— C12H12N6O
5-[(1R)-1-(2-methylimidazol-1-yl)ethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole
—— (5R)-7-(cyclopropylmethyl)-2-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H29FN2O3
(5R)-7-(cyclopropylmethyl)-2-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(oxan-4-yl)-2-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O2
(5R)-7-(oxan-4-yl)-2-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O3
(5R)-2-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-ethyl-N-[(3R,4S)-4-methoxypyrrolidin-3-yl]furan-2-carboxamide —— C12H18N2O3
5-ethyl-N-[(3R,4S)-4-methoxypyrrolidin-3-yl]furan-2-carboxamide
—— (5S)-2-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H25N3O2
(5S)-2-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-methyl-2-(4-phenylmethoxybutyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H30N2O2
(5R)-7-methyl-2-(4-phenylmethoxybutyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(4-fluorophenyl)-1,8,8-trimethyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione —— C20H20FN3O3
(5S)-5-(4-fluorophenyl)-1,8,8-trimethyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione
—— (5R)-9-[2-(4-oxo-3H-quinazolin-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H21N3O3
(5R)-9-[2-(4-oxo-3H-quinazolin-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-2-[2-(4-ethylpiperazin-1-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H32N4O3
(5S)-2-[2-(4-ethylpiperazin-1-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propyl-2-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O2
(5S)-7-propyl-2-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5,6-dimethyl-N-[(2R)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]-2-oxo-1H-pyridine-3-carboxamide —— C15H20N4O2
5,6-dimethyl-N-[(2R)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]-2-oxo-1H-pyridine-3-carboxamide
—— 5-[(2S)-oxolan-2-yl]-N-[2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)ethyl]thiophene-2-carboxamide —— C18H18N4O3S
5-[(2S)-oxolan-2-yl]-N-[2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)ethyl]thiophene-2-carboxamide
—— (5S)-7-(cyclopropylmethyl)-2-(4-methylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O2
(5S)-7-(cyclopropylmethyl)-2-(4-methylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-chloropyridin-2-yl)-[(2R,4S)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidin-1-yl]methanone —— C16H13ClF2N2O2
(5-chloropyridin-2-yl)-[(2R,4S)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidin-1-yl]methanone
—— 5-methyl-1-[2-oxo-2-[(5S)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decan-2-yl]ethyl]pyrimidine-2,4-dione —— C18H26N4O4
5-methyl-1-[2-oxo-2-[(5S)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decan-2-yl]ethyl]pyrimidine-2,4-dione
—— (5S)-2-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O3
(5S)-2-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[2-(dimethylamino)ethyl]-5-[4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl]piperidin-2-one —— C18H30N6O3
(5S)-1-[2-(dimethylamino)ethyl]-5-[4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl]piperidin-2-one
—— (5R)-5-[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]-1-[[3-(trifluoromethyl)phenyl]methyl]piperidin-2-one —— C17H18F3N3O2S
(5R)-5-[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]-1-[[3-(trifluoromethyl)phenyl]methyl]piperidin-2-one
—— (5R)-7-propyl-2-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O2
(5R)-7-propyl-2-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[2-(4-methylsulfonylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H22N2O4S
(5R)-2-[2-(4-methylsulfonylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H24N2O2S
(5R)-9-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5-chloropyridin-2-yl)-[(2R,4R)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidin-1-yl]methanone —— C16H13ClF2N2O2
(5-chloropyridin-2-yl)-[(2R,4R)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidin-1-yl]methanone
—— (5R)-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1-prop-2-enylpiperidin-2-one —— C15H17N5O2
(5R)-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1-prop-2-enylpiperidin-2-one
—— (5S)-7-(cyclopropylmethyl)-2-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H29FN2O3
(5S)-7-(cyclopropylmethyl)-2-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-methylthiophen-3-yl)-[(3S)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C20H22N4OS
(5-methylthiophen-3-yl)-[(3S)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (5S,10bS)-5-(4-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C21H18N2O2S
(5S,10bS)-5-(4-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[(2R,4R)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidine-1-carbonyl]-1-methylpyrrole-3-carboxamide —— C17H17F2N3O3
5-[(2R,4R)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidine-1-carbonyl]-1-methylpyrrole-3-carboxamide
—— (5S)-N-benzyl-5-hydroxy-N-methyl-1-oxa-9-azaspiro[5.5]undecane-9-sulfonamide —— C17H26N2O4S
(5S)-N-benzyl-5-hydroxy-N-methyl-1-oxa-9-azaspiro[5.5]undecane-9-sulfonamide
—— 5-[(1S)-1-[4-[2-(2-phenylethynyl)phenyl]triazol-1-yl]ethyl]-2H-tetrazole —— C19H15N7
5-[(1S)-1-[4-[2-(2-phenylethynyl)phenyl]triazol-1-yl]ethyl]-2H-tetrazole
—— (5S)-7-(2-methoxyethyl)-2-thieno[3,2-d]pyrimidin-4-yl-2,7-diazaspiro[4.5]decan-6-one —— C17H22N4O2S
(5S)-7-(2-methoxyethyl)-2-thieno[3,2-d]pyrimidin-4-yl-2,7-diazaspiro[4.5]decan-6-one
—— [(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(1,2,4-triazol-4-yl)piperidin-1-yl]methanone —— C17H22N4OS
[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(1,2,4-triazol-4-yl)piperidin-1-yl]methanone
—— (5S)-7-propan-2-yl-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H21F3N4O2
(5S)-7-propan-2-yl-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclobutylmethyl)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O2
(5R)-7-(cyclobutylmethyl)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclopropylmethyl)-2-(4-methylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O2
(5R)-7-(cyclopropylmethyl)-2-(4-methylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(4-hydroxyphenyl)-1,8,8-trimethyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione —— C20H21N3O4
(5R)-5-(4-hydroxyphenyl)-1,8,8-trimethyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione
—— (5S)-1-[[2-(dimethylamino)-1,3-thiazol-4-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one —— C18H29N3OS
(5S)-1-[[2-(dimethylamino)-1,3-thiazol-4-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one
—— 5-[(5S)-7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione —— C19H26N4O4
5-[(5S)-7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione
—— (5S)-9-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H24N2O2S
(5S)-9-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-cyclohexyl-N-[[(3S)-1-(4-methylphenyl)pyrrolidin-3-yl]methyl]-1H-pyrazole-4-carboxamide —— C22H30N4O
5-cyclohexyl-N-[[(3S)-1-(4-methylphenyl)pyrrolidin-3-yl]methyl]-1H-pyrazole-4-carboxamide
—— (5R)-1-[[2-(dimethylamino)-1,3-thiazol-4-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one —— C18H29N3OS
(5R)-1-[[2-(dimethylamino)-1,3-thiazol-4-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one
—— [(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(1,2,4-triazol-4-yl)piperidin-1-yl]methanone —— C17H22N4OS
[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-[4-(1,2,4-triazol-4-yl)piperidin-1-yl]methanone
—— 5-[[(3S)-1-(4-methoxypiperidin-1-yl)sulfonylpyrrolidin-3-yl]methyl]-1H-pyridin-2-one —— C16H25N3O4S
5-[[(3S)-1-(4-methoxypiperidin-1-yl)sulfonylpyrrolidin-3-yl]methyl]-1H-pyridin-2-one
—— 5-[(5R)-7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione —— C19H26N4O4
5-[(5R)-7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione
—— (5R)-7-cyclopentyl-2-(1,3-dimethylpyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5R)-7-cyclopentyl-2-(1,3-dimethylpyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-methylthiophen-3-yl)-[(3R)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C20H22N4OS
(5-methylthiophen-3-yl)-[(3R)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (5R)-1-(2-morpholin-4-ylethyl)-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C16H26N4O3
(5R)-1-(2-morpholin-4-ylethyl)-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5S)-2-(1-phenylcyclohexanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H28N2O2
(5S)-2-(1-phenylcyclohexanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one