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—— (5S,6S)-1-methyl-5-[(5S)-2-oxa-7-azaspiro[4.4]nonane-7-carbonyl]-6-thiophen-2-ylpiperidin-2-one —— C18H24N2O3S
(5S,6S)-1-methyl-5-[(5S)-2-oxa-7-azaspiro[4.4]nonane-7-carbonyl]-6-thiophen-2-ylpiperidin-2-one
—— (5S)-N-[(2R)-1-cyclopropylbutan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C15H26N2O2
(5S)-N-[(2R)-1-cyclopropylbutan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(S)-cyclobutyl(phenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H26N2O2
(5S)-N-[(S)-cyclobutyl(phenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5R)-7-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane —— C18H19N5O
(5R)-7-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane
—— (5S)-7-(3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-2-oxa-7-azaspiro[4.4]nonane —— C18H19N5O
(5S)-7-(3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-2-oxa-7-azaspiro[4.4]nonane
—— (5R)-N-[(1-phenylsulfanylcyclopropyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C18H24N2O2S
(5R)-N-[(1-phenylsulfanylcyclopropyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-7-(2-tert-butylpyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane —— C15H23N3O
(5S)-7-(2-tert-butylpyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane
—— (5S)-N-[(1S,2R)-2-(2,4-difluorophenyl)cyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C17H20F2N2O2
(5S)-N-[(1S,2R)-2-(2,4-difluorophenyl)cyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(1R,3R)-3-cyclopropylcyclohexyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C17H28N2O2
(5S)-N-[(1R,3R)-3-cyclopropylcyclohexyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-7-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2-oxa-7-azaspiro[4.4]nonane —— C15H18N4O2
(5S)-7-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2-oxa-7-azaspiro[4.4]nonane
—— (5R)-7-(3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-2-oxa-7-azaspiro[4.4]nonane —— C18H19N5O
(5R)-7-(3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-2-oxa-7-azaspiro[4.4]nonane
—— 5-chloro-N-[[(2R)-thiolan-2-yl]methyl]pyridine-2-carboxamide —— C11H13ClN2OS
5-chloro-N-[[(2R)-thiolan-2-yl]methyl]pyridine-2-carboxamide
—— (5S)-N-[(1-phenylsulfanylcyclopropyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C18H24N2O2S
(5S)-N-[(1-phenylsulfanylcyclopropyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5R)-2-methylsulfanyl-5-(4-nitrophenyl)-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C14H12N4O4S
(5R)-2-methylsulfanyl-5-(4-nitrophenyl)-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— 5-[(3R)-1-(2-methyl-4-nitrophenyl)sulfonylpiperidin-3-yl]-1H-pyrazole-3-carboxamide —— C16H19N5O5S
5-[(3R)-1-(2-methyl-4-nitrophenyl)sulfonylpiperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-(2-fluorophenyl)-N-[(2S)-2-pyridin-4-ylpropyl]-1H-pyrazole-4-carboxamide —— C18H17FN4O
5-(2-fluorophenyl)-N-[(2S)-2-pyridin-4-ylpropyl]-1H-pyrazole-4-carboxamide
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-(2-methylphenyl)sulfanylacetate —— C16H14N2O3S2
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-(2-methylphenyl)sulfanylacetate
—— 5-[(3R)-1-[4-(diethylcarbamoyl)phenyl]sulfonylpiperidin-3-yl]-1H-pyrazole-3-carboxamide —— C20H27N5O4S
5-[(3R)-1-[4-(diethylcarbamoyl)phenyl]sulfonylpiperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5S)-N-[(S)-1-benzofuran-2-yl(cyclopropyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C20H24N2O3
(5S)-N-[(S)-1-benzofuran-2-yl(cyclopropyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-[2-[(1S,3S)-3-methylcyclohexyl]ethylsulfanylmethyl]-3-(methylsulfonylmethyl)-1,2,4-oxadiazole —— C14H24N2O3S2
5-[2-[(1S,3S)-3-methylcyclohexyl]ethylsulfanylmethyl]-3-(methylsulfonylmethyl)-1,2,4-oxadiazole
—— (5R,6S)-1-methyl-5-[(5S)-2-oxa-7-azaspiro[4.4]nonane-7-carbonyl]-6-thiophen-2-ylpiperidin-2-one —— C18H24N2O3S
(5R,6S)-1-methyl-5-[(5S)-2-oxa-7-azaspiro[4.4]nonane-7-carbonyl]-6-thiophen-2-ylpiperidin-2-one
—— (5S)-N-[(1R,2S)-2-cyclohexylcyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C17H28N2O2
(5S)-N-[(1R,2S)-2-cyclohexylcyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5R)-N-[(2R)-1-cyclopropylbutan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C15H26N2O2
(5R)-N-[(2R)-1-cyclopropylbutan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-[(3R)-1-(4-pyrazol-1-ylpyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C16H18N8O
5-[(3R)-1-(4-pyrazol-1-ylpyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5S)-N-[(1S,2S)-2-cyclohexylcyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C17H28N2O2
(5S)-N-[(1S,2S)-2-cyclohexylcyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C17H27N5O2
(5S)-N-[2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5R)-N-[(S)-cyclobutyl(phenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H26N2O2
(5R)-N-[(S)-cyclobutyl(phenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-7-(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)-2-oxa-7-azaspiro[4.4]nonane —— C18H19N5O
(5S)-7-(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)-2-oxa-7-azaspiro[4.4]nonane
—— (5S)-N-[(1S,3S)-3-methoxy-2,2,3-trimethylcyclobutyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H28N2O3
(5S)-N-[(1S,3S)-3-methoxy-2,2,3-trimethylcyclobutyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(1S,5R,6S)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H26N2O3
(5S)-N-[(1S,5R,6S)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5R)-N-[(2R)-1-cyclopropylpropan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C14H24N2O2
(5R)-N-[(2R)-1-cyclopropylpropan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5R)-N-[(2S)-1-cyclopropylpropan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C14H24N2O2
(5R)-N-[(2S)-1-cyclopropylpropan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(1R,3S)-3-methoxy-2,2,3-trimethylcyclobutyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H28N2O3
(5S)-N-[(1R,3S)-3-methoxy-2,2,3-trimethylcyclobutyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(R)-cyclobutyl(phenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H26N2O2
(5S)-N-[(R)-cyclobutyl(phenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(1R)-1-[(1S,2S)-2-(3-methylphenyl)cyclopropyl]ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C20H28N2O2
(5S)-N-[(1R)-1-[(1S,2S)-2-(3-methylphenyl)cyclopropyl]ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(1R,2S)-2-(2,4-difluorophenyl)cyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C17H20F2N2O2
(5S)-N-[(1R,2S)-2-(2,4-difluorophenyl)cyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[[(1S,2S)-2-phenylcyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C18H24N2O2
(5S)-N-[[(1S,2S)-2-phenylcyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(1S,5S,6R)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H26N2O3
(5S)-N-[(1S,5S,6R)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(2R)-1-cyclopropylpropan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C14H24N2O2
(5S)-N-[(2R)-1-cyclopropylpropan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-(4-cycloheptyloxybutyl)-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H34N2O3
(5S)-N-(4-cycloheptyloxybutyl)-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(S)-cyclobutyl-(4-fluorophenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H25FN2O2
(5S)-N-[(S)-cyclobutyl-(4-fluorophenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-7-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane —— C18H19N5O
(5S)-7-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane
—— (5R)-N-[(R)-cyclobutyl(phenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H26N2O2
(5R)-N-[(R)-cyclobutyl(phenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5R)-N-[2-[cyclopropyl(cyclopropylmethyl)amino]ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C17H29N3O2
(5R)-N-[2-[cyclopropyl(cyclopropylmethyl)amino]ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(2S)-1-cyclopropylbutan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C15H26N2O2
(5S)-N-[(2S)-1-cyclopropylbutan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(1R,2R)-2-cyclohexylcyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C17H28N2O2
(5S)-N-[(1R,2R)-2-cyclohexylcyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(1S,5S,6S)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H26N2O3
(5S)-N-[(1S,5S,6S)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-[(3R)-1-(4-cyano-5,6-dimethylpyridazin-3-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C16H19N7O
5-[(3R)-1-(4-cyano-5,6-dimethylpyridazin-3-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5R)-N-[[1-(2-methoxyphenyl)cyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H26N2O3
(5R)-N-[[1-(2-methoxyphenyl)cyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-methyl-2-[(2R)-thiolan-2-yl]-3H-thieno[2,3-d]pyrimidin-4-one —— C11H12N2OS2
5-methyl-2-[(2R)-thiolan-2-yl]-3H-thieno[2,3-d]pyrimidin-4-one