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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-methyl-4-[(3S)-3-methyl-3-phenylpiperidin-1-yl]sulfonyl-1,2-oxazole —— C16H20N2O3S
5-methyl-4-[(3S)-3-methyl-3-phenylpiperidin-1-yl]sulfonyl-1,2-oxazole
—— (5-propylthiophen-3-yl)-[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone —— C18H25N3OS
(5-propylthiophen-3-yl)-[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone
—— (5-propylthiophen-3-yl)-[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone —— C18H25N3OS
(5-propylthiophen-3-yl)-[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone
—— (5S)-5-methyl-1-[2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethyl]-5-phenylpiperidin-2-one —— C17H22N4OS
(5S)-5-methyl-1-[2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethyl]-5-phenylpiperidin-2-one
—— (5S)-2-(1-benzoxepine-4-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C22H26N2O3
(5S)-2-(1-benzoxepine-4-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-O-tert-butyl 3-O-methyl (6S)-6-(benzylsulfanylmethyl)-6,7-dihydro-4H-triazolo[1,5-a]pyrazine-3,5-dicarboxylate —— C20H26N4O4S
5-O-tert-butyl 3-O-methyl (6S)-6-(benzylsulfanylmethyl)-6,7-dihydro-4H-triazolo[1,5-a]pyrazine-3,5-dicarboxylate
—— (5R)-7,7-dimethyl-2-morpholin-4-yl-N-quinolin-4-yl-6,8-dihydro-5H-quinazolin-5-amine —— C23H27N5O
(5R)-7,7-dimethyl-2-morpholin-4-yl-N-quinolin-4-yl-6,8-dihydro-5H-quinazolin-5-amine
—— (5R)-5-methyl-1-[2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethyl]-5-phenylpiperidin-2-one —— C17H22N4OS
(5R)-5-methyl-1-[2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethyl]-5-phenylpiperidin-2-one
—— (5S)-7,7-dimethyl-2-morpholin-4-yl-N-quinolin-4-yl-6,8-dihydro-5H-quinazolin-5-amine —— C23H27N5O
(5S)-7,7-dimethyl-2-morpholin-4-yl-N-quinolin-4-yl-6,8-dihydro-5H-quinazolin-5-amine
—— (5R)-2-(1-benzoxepine-4-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C22H26N2O3
(5R)-2-(1-benzoxepine-4-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-3-(2-aminoethyl)-5-propan-2-yl-2,5-dihydro-1H-1,2,4-triazin-6-one —— C8H16N4O
(5R)-3-(2-aminoethyl)-5-propan-2-yl-2,5-dihydro-1H-1,2,4-triazin-6-one
—— (5R)-7-(cyclopropylmethyl)-2-(4-propylthiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O2S
(5R)-7-(cyclopropylmethyl)-2-(4-propylthiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(4-chlorophenyl)-8,8-dimethyl-2-methylsulfanyl-5,7,9,10-tetrahydro-3H-pyrimido[4,5-b]quinoline-4,6-dione —— C20H20ClN3O2S
(5S)-5-(4-chlorophenyl)-8,8-dimethyl-2-methylsulfanyl-5,7,9,10-tetrahydro-3H-pyrimido[4,5-b]quinoline-4,6-dione
—— (5S)-7-cyclopentyl-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H26N2O4
(5S)-7-cyclopentyl-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-3-piperidin-4-yl-5-propan-2-yl-2,5-dihydro-1H-1,2,4-triazin-6-one —— C11H20N4O
(5S)-3-piperidin-4-yl-5-propan-2-yl-2,5-dihydro-1H-1,2,4-triazin-6-one
—— (5R)-5-(1,4-oxazepane-4-carbonyl)-1-(3-phenylpropyl)piperidin-2-one —— C20H28N2O3
(5R)-5-(1,4-oxazepane-4-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
—— (5R)-2-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H27N3O4
(5R)-2-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(1,3-benzothiazol-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H21N3O2S
(5R)-2-(1,3-benzothiazol-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5,6-dimethyl-4-N-[2-[5-[(2S)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]ethyl]pyrimidine-2,4-diamine —— C14H20N6O2
5,6-dimethyl-4-N-[2-[5-[(2S)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]ethyl]pyrimidine-2,4-diamine
—— 5-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-2-(phenoxymethyl)-1H-pyrimidin-6-one —— C20H20N4O4
5-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-2-(phenoxymethyl)-1H-pyrimidin-6-one
—— (5R)-3-piperidin-4-yl-5-propan-2-yl-2,5-dihydro-1H-1,2,4-triazin-6-one —— C11H20N4O
(5R)-3-piperidin-4-yl-5-propan-2-yl-2,5-dihydro-1H-1,2,4-triazin-6-one
—— (5S)-3-(2-aminoethyl)-5-propan-2-yl-2,5-dihydro-1H-1,2,4-triazin-6-one —— C8H16N4O
(5S)-3-(2-aminoethyl)-5-propan-2-yl-2,5-dihydro-1H-1,2,4-triazin-6-one
—— (5S)-7-(cyclopropylmethyl)-2-(5-methoxy-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H24N2O5
(5S)-7-(cyclopropylmethyl)-2-(5-methoxy-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H27N3O4
(5S)-2-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-O-tert-butyl 3-O-methyl (6R)-6-(benzylsulfanylmethyl)-6,7-dihydro-4H-triazolo[1,5-a]pyrazine-3,5-dicarboxylate —— C20H26N4O4S
5-O-tert-butyl 3-O-methyl (6R)-6-(benzylsulfanylmethyl)-6,7-dihydro-4H-triazolo[1,5-a]pyrazine-3,5-dicarboxylate
—— 5-(3-Methylphenyl)-2-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-ylmethyl)tetrazole —— C10H9N8-
5-(3-Methylphenyl)-2-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-ylmethyl)tetrazole
—— 5-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-2-(phenoxymethyl)-1H-pyrimidin-6-one —— C20H20N4O4
5-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-2-(phenoxymethyl)-1H-pyrimidin-6-one
—— 5-ethyl-4-N-[(1R)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine —— C11H15N5S
5-ethyl-4-N-[(1R)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine
—— (5-propylthiophen-3-yl)-[(3S)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]methanone —— C19H24N2O2S
(5-propylthiophen-3-yl)-[(3S)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]methanone
—— (5S)-7-cyclohexyl-2-(5-propyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H32N4O2
(5S)-7-cyclohexyl-2-(5-propyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[2-(4-methoxyphenyl)ethyl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C17H21N3O3
(5S)-1-[2-(4-methoxyphenyl)ethyl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— 5-ethyl-4-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine —— C11H15N5S
5-ethyl-4-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine
—— (5R)-1-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-5-methyl-5-phenylpiperidin-2-one —— C17H21N3O3
(5R)-1-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-5-methyl-5-phenylpiperidin-2-one
—— 5-[(2R)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-2-(1,2,4-triazol-1-ylmethyl)-1H-pyrimidin-6-one —— C15H15N7O2S
5-[(2R)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-2-(1,2,4-triazol-1-ylmethyl)-1H-pyrimidin-6-one
—— 5-[(5S)-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridine-2-carbonitrile —— C18H22N4O3
5-[(5S)-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridine-2-carbonitrile
—— (5R)-7-cyclopentyl-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H26N2O4
(5R)-7-cyclopentyl-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(2-chlorophenyl)-N-[(R)-cyclopropyl-(2-ethyl-1,2,4-triazol-3-yl)methyl]furan-2-carboxamide —— C19H19ClN4O2
5-(2-chlorophenyl)-N-[(R)-cyclopropyl-(2-ethyl-1,2,4-triazol-3-yl)methyl]furan-2-carboxamide
—— (5S)-7-(cyclopropylmethyl)-2-(4-propylthiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O2S
(5S)-7-(cyclopropylmethyl)-2-(4-propylthiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-1-[2-(4-methoxyphenyl)ethyl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C17H21N3O3
(5R)-1-[2-(4-methoxyphenyl)ethyl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5S)-5-(1,4-oxazepane-4-carbonyl)-1-(3-phenylpropyl)piperidin-2-one —— C20H28N2O3
(5S)-5-(1,4-oxazepane-4-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidin-2-one —— C19H25N3O4
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidin-2-one
—— (5R)-7-cyclohexyl-2-(5-propyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H32N4O2
(5R)-7-cyclohexyl-2-(5-propyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5,6-dimethyl-3-(pyridin-4-ylmethyl)-3,4-dihydro-2H-thieno[2,3-d]pyrimidin-3-ium-1-yl]-(furan-2-yl)methanone —— C19H20N3O2S+
[5,6-dimethyl-3-(pyridin-4-ylmethyl)-3,4-dihydro-2H-thieno[2,3-d]pyrimidin-3-ium-1-yl]-(furan-2-yl)methanone
—— (5S,10bS)-2-phenyl-5-(4-prop-2-enoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C25H22N2O2
(5S,10bS)-2-phenyl-5-(4-prop-2-enoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— [(5E)-5-{3,5-dibromo-4-[2-nitro-4-(trifluoromethyl)phenoxy]benzylidene}-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetic acid —— C19H9Br2F3N2O6S2
[(5E)-5-{3,5-dibromo-4-[2-nitro-4-(trifluoromethyl)phenoxy]benzylidene}-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetic acid
—— (5S)-2,2-dimethyl-5-[4-(1-propan-2-ylimidazol-2-yl)piperidine-1-carbonyl]thiomorpholin-3-one —— C18H28N4O2S
(5S)-2,2-dimethyl-5-[4-(1-propan-2-ylimidazol-2-yl)piperidine-1-carbonyl]thiomorpholin-3-one
—— (5S)-7-(cyclopropylmethyl)-2-(1-phenyltriazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H25N5O2
(5S)-7-(cyclopropylmethyl)-2-(1-phenyltriazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(6S)-10-(cyclopropylmethyl)-1-methyl-9-oxo-1,4,10-triazaspiro[5.6]dodecan-4-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C18H28N6O3
5-[[(6S)-10-(cyclopropylmethyl)-1-methyl-9-oxo-1,4,10-triazaspiro[5.6]dodecan-4-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-fluoro-2-[[(3S)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-N-methylpyrimidin-4-amine —— C16H18FN3O2
5-fluoro-2-[[(3S)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-N-methylpyrimidin-4-amine
—— (5S)-1-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-5-methyl-5-phenylpiperidin-2-one —— C17H21N3O3
(5S)-1-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-5-methyl-5-phenylpiperidin-2-one