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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-2-[5-(piperidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O2
(5R)-2-[5-(piperidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-[2-(4,5-dimethylimidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5S)-7-(cyclopropylmethyl)-2-[2-(4,5-dimethylimidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C21H28N4O2
(5S)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]-1-(3-morpholin-4-ylpropyl)piperidin-2-one —— C16H26N4O3S
(5S)-5-[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]-1-(3-morpholin-4-ylpropyl)piperidin-2-one
—— (5S)-7-(cyclopropylmethyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O2S
(5S)-7-(cyclopropylmethyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propyl-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24N4O2S
(5S)-7-propyl-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-hydroxyethyl)-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C14H19F3N4O3
(5R)-7-(2-hydroxyethyl)-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-(pyridin-3-ylmethyl)-1,2-dihydropyrazole-3-carboxamide —— C16H14N4O2
5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-(pyridin-3-ylmethyl)-1,2-dihydropyrazole-3-carboxamide
—— (5R)-7-(2-methoxyethyl)-2-(1-methyl-2-oxopyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O4
(5R)-7-(2-methoxyethyl)-2-(1-methyl-2-oxopyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-fluoro-2-[(3R)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidin-1-yl]-3,8-dimethylquinoline —— C22H27FN4O
5-fluoro-2-[(3R)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidin-1-yl]-3,8-dimethylquinoline
—— (5S)-2-[3-(2-methyl-6-oxopyridin-1-yl)propanoyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O3
(5S)-2-[3-(2-methyl-6-oxopyridin-1-yl)propanoyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-(hydroxymethyl)-3-prop-2-enylpiperidine-1-carbonyl]-1-methylpyrimidine-2,4-dione —— C15H21N3O4
5-[(3R)-3-(hydroxymethyl)-3-prop-2-enylpiperidine-1-carbonyl]-1-methylpyrimidine-2,4-dione
—— [(5S)-3-methyl-4,5-dihydro-1,2-oxazol-5-yl]-[4-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C19H23N5O2
[(5S)-3-methyl-4,5-dihydro-1,2-oxazol-5-yl]-[4-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— 5-fluoro-2-[(3S)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidin-1-yl]-3,8-dimethylquinoline —— C22H27FN4O
5-fluoro-2-[(3S)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidin-1-yl]-3,8-dimethylquinoline
—— (5R)-7-(cyclopropylmethyl)-2-[2-(4,5-dimethylimidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5R)-7-(cyclopropylmethyl)-2-[2-(4,5-dimethylimidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C12H13N5O2
(5R)-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5S)-9-[(1-benzylpyrazol-4-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C19H23N3O2
(5S)-9-[(1-benzylpyrazol-4-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-[(2R)-oxolan-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]thiophene-2-carboxamide —— C20H21N3O2S
5-[(2R)-oxolan-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]thiophene-2-carboxamide
—— (5R)-7-(cyclopropylmethyl)-2-(2-methylimidazo[1,2-a]pyrimidine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5R)-7-(cyclopropylmethyl)-2-(2-methylimidazo[1,2-a]pyrimidine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2S)-oxolan-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]thiophene-2-carboxamide —— C20H21N3O2S
5-[(2S)-oxolan-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]thiophene-2-carboxamide
—— 5-ethyl-4-N-[(2R)-2-pyridin-3-yloxypropyl]pyrimidine-2,4-diamine —— C14H19N5O
5-ethyl-4-N-[(2R)-2-pyridin-3-yloxypropyl]pyrimidine-2,4-diamine
—— (5S)-7-(2-hydroxyethyl)-2-quinoxalin-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H22N4O2
(5S)-7-(2-hydroxyethyl)-2-quinoxalin-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-(3-indazol-1-ylpropyl)-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H23N3O2
(5R)-9-(3-indazol-1-ylpropyl)-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-2-(4-methylpyrimidine-5-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O3
(5R)-2-(4-methylpyrimidine-5-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[5-(piperidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O2
(5S)-2-[5-(piperidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-cyclopentyl-2-(5-fluoropyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24FN3O
(5R)-7-cyclopentyl-2-(5-fluoropyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[2-(4-chlorophenyl)ethyl]-5-(3-ethyl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C17H20ClN3O2
(5S)-1-[2-(4-chlorophenyl)ethyl]-5-(3-ethyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5S)-2-(4-methylpyrimidine-5-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O3
(5S)-2-(4-methylpyrimidine-5-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S,10bS)-9-chloro-5-(3-nitrophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H14ClN3O3S
(5S,10bS)-9-chloro-5-(3-nitrophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R)-1-[2-(4-chlorophenyl)ethyl]-5-(3-ethyl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C17H20ClN3O2
(5R)-1-[2-(4-chlorophenyl)ethyl]-5-(3-ethyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— 5,6-dimethyl-2-[2-[(3S)-3-methyl-3-phenylpiperidin-1-yl]-2-oxoethyl]pyridazin-3-one —— C20H25N3O2
5,6-dimethyl-2-[2-[(3S)-3-methyl-3-phenylpiperidin-1-yl]-2-oxoethyl]pyridazin-3-one
—— (5S)-7-methyl-2-(2-methylsulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C12H22N2O3S
(5S)-7-methyl-2-(2-methylsulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S,10bR)-5-(2-chlorophenyl)-2-(4-chlorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H16Cl2N2O
(5S,10bR)-5-(2-chlorophenyl)-2-(4-chlorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-tert-butyl-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3,4-oxadiazol-2-amine —— C11H18N6O
5-tert-butyl-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3,4-oxadiazol-2-amine
—— (5S)-7-(cyclopropylmethyl)-2-(2-methylimidazo[1,2-a]pyrimidine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5S)-7-(cyclopropylmethyl)-2-(2-methylimidazo[1,2-a]pyrimidine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S,10bR)-5-(3-chlorophenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H16ClFN2O
(5S,10bR)-5-(3-chlorophenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— [5-(2-chlorophenyl)furan-2-yl]-[(2S)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]methanone —— C16H14ClNO3
[5-(2-chlorophenyl)furan-2-yl]-[(2S)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]methanone
—— 5-[(3R)-1-carbamoylpiperidine-3-carbonyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C17H24N4O3S
5-[(3R)-1-carbamoylpiperidine-3-carbonyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— 5-[(3S)-1-carbamoylpiperidine-3-carbonyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C17H24N4O3S
5-[(3S)-1-carbamoylpiperidine-3-carbonyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— (5S,10bS)-9-chloro-5-(4-methoxyphenyl)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H21ClN2O2
(5S,10bS)-9-chloro-5-(4-methoxyphenyl)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— [(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone —— C16H24N2O3S
[(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
—— 5-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-6-methylpyridin-2-amine —— C16H18N2O
5-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-6-methylpyridin-2-amine
—— (5S,10bS)-9-bromo-5-phenyl-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H15BrN2OS
(5S,10bS)-9-bromo-5-phenyl-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S)-7-cyclopentyl-2-(5-fluoropyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24FN3O
(5S)-7-cyclopentyl-2-(5-fluoropyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one —— C18H23N3O2
(5S)-1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
—— (5R)-7-(2-hydroxyethyl)-2-quinoxalin-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H22N4O2
(5R)-7-(2-hydroxyethyl)-2-quinoxalin-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-methoxyethyl)-2-(3-pyrazin-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O3
(5S)-7-(2-methoxyethyl)-2-(3-pyrazin-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2S)-oxolan-2-yl]-N-[[3-(pyrrolidin-1-ylmethyl)phenyl]methyl]thiophene-2-carboxamide —— C21H26N2O2S
5-[(2S)-oxolan-2-yl]-N-[[3-(pyrrolidin-1-ylmethyl)phenyl]methyl]thiophene-2-carboxamide
—— (5R)-7-methyl-2-(2-methylsulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C12H22N2O3S
(5R)-7-methyl-2-(2-methylsulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[1-(2-fluorophenyl)cyclopropanecarbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C21H27FN2O2
(5S)-2-[1-(2-fluorophenyl)cyclopropanecarbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one