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—— (5S)-2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C15H22ClN5O3
(5S)-2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H21N3O3
(5S)-9-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-(4-oxocyclohexa-2,5-dien-1-ylidene)-N-[(1S)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,2-dihydropyrazole-3-carboxamide —— C19H20N4O2S
5-(4-oxocyclohexa-2,5-dien-1-ylidene)-N-[(1S)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,2-dihydropyrazole-3-carboxamide
—— 5,6-dimethyl-N-[(2S)-2-pyridin-3-yloxypropyl]pyrimidin-4-amine —— C14H18N4O
5,6-dimethyl-N-[(2S)-2-pyridin-3-yloxypropyl]pyrimidin-4-amine
—— 5-(5-methylfuran-2-yl)-N-[(3R)-2-oxoazepan-3-yl]-1H-pyrazole-3-carboxamide —— C15H18N4O3
5-(5-methylfuran-2-yl)-N-[(3R)-2-oxoazepan-3-yl]-1H-pyrazole-3-carboxamide
—— (5S)-7-(cyclobutylmethyl)-2-(1,1-dioxothiane-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H30N2O4S
(5S)-7-(cyclobutylmethyl)-2-(1,1-dioxothiane-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H27N5O2
(5S)-7-(cyclobutylmethyl)-2-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one —— C18H24N4O
(5S)-1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
—— (5R)-1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one —— C18H24N4O
(5R)-1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
—— (5S)-9-[2-[(3-chlorophenyl)methylsulfanyl]ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H22ClNO2S
(5S)-9-[2-[(3-chlorophenyl)methylsulfanyl]ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-5-methyl-1-[(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)methyl]-5-phenylpiperidin-2-one —— C15H18N4O2
(5S)-5-methyl-1-[(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)methyl]-5-phenylpiperidin-2-one
—— 5-(3-fluorophenyl)-N-[(3S)-3-hydroxy-3-phenylpropyl]-N-methyl-1H-pyrazole-4-carboxamide —— C20H20FN3O2
5-(3-fluorophenyl)-N-[(3S)-3-hydroxy-3-phenylpropyl]-N-methyl-1H-pyrazole-4-carboxamide
—— [5-(imidazol-1-ylmethyl)furan-2-yl]-[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C18H21N5O3
[5-(imidazol-1-ylmethyl)furan-2-yl]-[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— (5R)-2-(3-hydroxypyridine-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H25N3O4
(5R)-2-(3-hydroxypyridine-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-[2-(2,3-difluorophenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H24F2N2O2
(5S)-7-(cyclopropylmethyl)-2-[2-(2,3-difluorophenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(2-chlorophenyl)-N-[(S)-cyclopropyl-(3-methylpyridin-2-yl)methyl]furan-2-carboxamide —— C21H19ClN2O2
5-(2-chlorophenyl)-N-[(S)-cyclopropyl-(3-methylpyridin-2-yl)methyl]furan-2-carboxamide
—— (5R)-7-propan-2-yl-2-(1-propan-2-ylpyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H29N3O2
(5R)-7-propan-2-yl-2-(1-propan-2-ylpyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclopropylmethyl)-2-[2-(2,3-difluorophenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H24F2N2O2
(5R)-7-(cyclopropylmethyl)-2-[2-(2,3-difluorophenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-methyl-5-phenyl-1-[3-(pyridin-3-ylamino)propyl]piperidin-2-one —— C20H25N3O
(5R)-5-methyl-5-phenyl-1-[3-(pyridin-3-ylamino)propyl]piperidin-2-one
—— 5-(4-oxocyclohexa-2,5-dien-1-ylidene)-N-[(2S)-2-pyridin-3-yloxypropyl]-1,2-dihydropyrazole-3-carboxamide —— C18H18N4O3
5-(4-oxocyclohexa-2,5-dien-1-ylidene)-N-[(2S)-2-pyridin-3-yloxypropyl]-1,2-dihydropyrazole-3-carboxamide
—— 5-(4-oxocyclohexa-2,5-dien-1-ylidene)-N-[(2R)-2-pyridin-3-yloxypropyl]-1,2-dihydropyrazole-3-carboxamide —— C18H18N4O3
5-(4-oxocyclohexa-2,5-dien-1-ylidene)-N-[(2R)-2-pyridin-3-yloxypropyl]-1,2-dihydropyrazole-3-carboxamide
—— 5-(2-chlorophenyl)-N-[(R)-cyclopropyl-(3-methylpyridin-2-yl)methyl]furan-2-carboxamide —— C21H19ClN2O2
5-(2-chlorophenyl)-N-[(R)-cyclopropyl-(3-methylpyridin-2-yl)methyl]furan-2-carboxamide
—— 5-(3-fluorophenyl)-N-[(3R)-3-hydroxy-3-phenylpropyl]-N-methyl-1H-pyrazole-4-carboxamide —— C20H20FN3O2
5-(3-fluorophenyl)-N-[(3R)-3-hydroxy-3-phenylpropyl]-N-methyl-1H-pyrazole-4-carboxamide
—— [5-(imidazol-1-ylmethyl)furan-2-yl]-[(2S)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C18H21N5O3
[5-(imidazol-1-ylmethyl)furan-2-yl]-[(2S)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— (5R)-2-(7-chloro-4-methylquinolin-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H24ClN3O2
(5R)-2-(7-chloro-4-methylquinolin-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(3-hydroxypyridine-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H25N3O4
(5S)-2-(3-hydroxypyridine-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-methyl-1-[(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)methyl]-5-phenylpiperidin-2-one —— C15H18N4O2
(5R)-5-methyl-1-[(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)methyl]-5-phenylpiperidin-2-one
—— (5R)-2-(1-methylpyrazole-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O3
(5R)-2-(1-methylpyrazole-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(7-chloro-4-methylquinolin-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H24ClN3O2
(5S)-2-(7-chloro-4-methylquinolin-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(3-fluorophenyl)-N-[(R)-(4-methylphenyl)-pyridin-4-ylmethyl]-1H-pyrazole-4-carboxamide —— C23H19FN4O
5-(3-fluorophenyl)-N-[(R)-(4-methylphenyl)-pyridin-4-ylmethyl]-1H-pyrazole-4-carboxamide
—— (5S)-2-[(3-benzylimidazol-4-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H28N4O2
(5S)-2-[(3-benzylimidazol-4-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— [(5S)-2-oxa-9-azaspiro[4.5]decan-9-yl]-(1-phenyltriazol-4-yl)methanone —— C17H20N4O2
[(5S)-2-oxa-9-azaspiro[4.5]decan-9-yl]-(1-phenyltriazol-4-yl)methanone
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(1-propylpyrazol-4-yl)methyl]piperidin-2-one —— C21H27N3O3
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(1-propylpyrazol-4-yl)methyl]piperidin-2-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(1-propylpyrazol-4-yl)methyl]piperidin-2-one —— C21H27N3O3
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(1-propylpyrazol-4-yl)methyl]piperidin-2-one
—— (5S)-7-propan-2-yl-2-(1-propan-2-ylpyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H29N3O2
(5S)-7-propan-2-yl-2-(1-propan-2-ylpyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-1-ethyl-6-oxopiperidine-3-carbonyl]-N-methyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C17H23N3O3S
5-[(3R)-1-ethyl-6-oxopiperidine-3-carbonyl]-N-methyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— (5R)-7-(2-hydroxyethyl)-2-[2-(methylamino)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H23N5O3
(5R)-7-(2-hydroxyethyl)-2-[2-(methylamino)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-hydroxyethyl)-2-[2-(methylamino)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H23N5O3
(5S)-7-(2-hydroxyethyl)-2-[2-(methylamino)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-cyclohexyl-N-[(2S)-2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1H-pyrazole-4-carboxamide —— C19H28N4O2
5-cyclohexyl-N-[(2S)-2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1H-pyrazole-4-carboxamide
—— (5S)-2-(1-methylpyrazole-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O3
(5S)-2-(1-methylpyrazole-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(3-methoxypropyl)-2-pyridin-3-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one —— C17H25N3O4S
(5R)-7-(3-methoxypropyl)-2-pyridin-3-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-(3-fluorophenyl)-N-[(S)-(4-methylphenyl)-pyridin-4-ylmethyl]-1H-pyrazole-4-carboxamide —— C23H19FN4O
5-(3-fluorophenyl)-N-[(S)-(4-methylphenyl)-pyridin-4-ylmethyl]-1H-pyrazole-4-carboxamide
—— 5-cyclohexyl-N-[(2R)-2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1H-pyrazole-4-carboxamide —— C19H28N4O2
5-cyclohexyl-N-[(2R)-2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1H-pyrazole-4-carboxamide
—— (5R)-2-(5-fluoro-1,3-dimethylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C20H24FN3O2
(5R)-2-(5-fluoro-1,3-dimethylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-(4-Methylphenyl)-2-[(2-methylphenyl)methylsulfanyl]-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one —— C24H22N2OS2
5-(4-Methylphenyl)-2-[(2-methylphenyl)methylsulfanyl]-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one
—— (5S)-5-methyl-5-phenyl-1-[3-(pyridin-3-ylamino)propyl]piperidin-2-one —— C20H25N3O
(5S)-5-methyl-5-phenyl-1-[3-(pyridin-3-ylamino)propyl]piperidin-2-one
—— (5S)-7-(cyclopropylmethyl)-2-(2-hydroxynaphthalene-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C23H26N2O3
(5S)-7-(cyclopropylmethyl)-2-(2-hydroxynaphthalene-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R,10bS)-5-(4-ethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H20N2O2S
(5R,10bS)-5-(4-ethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-(2-methylpropyl)-1'-pyridazin-3-ylspiro[6,7-dihydro-1H-imidazo[4,5-c]pyridine-4,4'-piperidine] —— C18H26N6
5-(2-methylpropyl)-1'-pyridazin-3-ylspiro[6,7-dihydro-1H-imidazo[4,5-c]pyridine-4,4'-piperidine]
—— (5S,10bS)-5-(2,4-dichlorophenyl)-2-(furan-2-yl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H14Cl2N2O2
(5S,10bS)-5-(2,4-dichlorophenyl)-2-(furan-2-yl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine