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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-1-[2-(dimethylamino)ethyl]-5-[4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl]piperidin-2-one —— C18H30N6O3
(5R)-1-[2-(dimethylamino)ethyl]-5-[4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl]piperidin-2-one
—— 5-[[(5R)-6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl]sulfonyl]-1H-pyrimidine-2,4-dione —— C15H22N4O5S
5-[[(5R)-6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl]sulfonyl]-1H-pyrimidine-2,4-dione
—— (5S)-5-[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]-1-[[3-(trifluoromethyl)phenyl]methyl]piperidin-2-one —— C17H18F3N3O2S
(5S)-5-[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]-1-[[3-(trifluoromethyl)phenyl]methyl]piperidin-2-one
—— (5S)-2-methylsulfonyl-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C14H24N2O4S
(5S)-2-methylsulfonyl-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[2-(4-oxo-3H-quinazolin-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H21N3O3
(5S)-9-[2-(4-oxo-3H-quinazolin-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S,10bS)-5-(2-ethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H20N2O2S
(5S,10bS)-5-(2-ethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R)-7-ethyl-2-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O2
(5R)-7-ethyl-2-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(4-methylthiadiazol-5-yl)methyl]piperidin-2-one —— C18H21N3O3S
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(4-methylthiadiazol-5-yl)methyl]piperidin-2-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(4-methylthiadiazol-5-yl)methyl]piperidin-2-one —— C18H21N3O3S
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(4-methylthiadiazol-5-yl)methyl]piperidin-2-one
—— (5R)-1-cyclopentyl-5-[3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C21H34N4O2
(5R)-1-cyclopentyl-5-[3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5S)-7-methyl-2-(4-phenylmethoxybutyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H30N2O2
(5S)-7-methyl-2-(4-phenylmethoxybutyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(oxan-4-yl)-2-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O2
(5S)-7-(oxan-4-yl)-2-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-Methyl-1-(2-methyl-1-phenylbenzimidazol-5-yl)triazole-4-carboxylate —— C18H14N5O2-
5-Methyl-1-(2-methyl-1-phenylbenzimidazol-5-yl)triazole-4-carboxylate
—— (5R)-5-benzyl-1-(3-chlorophenyl)-4-(3-hydroxypropanoyl)piperazin-2-one —— C20H21ClN2O3
(5R)-5-benzyl-1-(3-chlorophenyl)-4-(3-hydroxypropanoyl)piperazin-2-one
—— 5-[[(3S)-1-[2-(1,1-dioxothian-4-yl)acetyl]pyrrolidin-3-yl]methyl]-1H-pyridin-2-one —— C17H24N2O4S
5-[[(3S)-1-[2-(1,1-dioxothian-4-yl)acetyl]pyrrolidin-3-yl]methyl]-1H-pyridin-2-one
—— 5-ethyl-N-[(3S,4S)-4-methoxypyrrolidin-3-yl]furan-2-carboxamide —— C12H18N2O3
5-ethyl-N-[(3S,4S)-4-methoxypyrrolidin-3-yl]furan-2-carboxamide
—— (5R)-7-(2-methoxyethyl)-2-thieno[3,2-d]pyrimidin-4-yl-2,7-diazaspiro[4.5]decan-6-one —— C17H22N4O2S
(5R)-7-(2-methoxyethyl)-2-thieno[3,2-d]pyrimidin-4-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[4-[5-[(2R)-oxan-2-yl]furan-2-yl]triazol-1-yl]methyl]-3-pyridin-3-yl-1,2-oxazole —— C20H19N5O3
5-[[4-[5-[(2R)-oxan-2-yl]furan-2-yl]triazol-1-yl]methyl]-3-pyridin-3-yl-1,2-oxazole
—— (5R)-5-(4-methoxyphenyl)-1,8,8-trimethyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione —— C21H23N3O4
(5R)-5-(4-methoxyphenyl)-1,8,8-trimethyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione
—— (5S)-1-ethyl-5-(4-methoxyphenyl)-8,8-dimethyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione —— C22H25N3O4
(5S)-1-ethyl-5-(4-methoxyphenyl)-8,8-dimethyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione
—— (5R)-5-(3,4-dimethoxyphenyl)-1,8,8-trimethyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione —— C22H25N3O5
(5R)-5-(3,4-dimethoxyphenyl)-1,8,8-trimethyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione
—— (5S,10bS)-5-(4-fluorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H15FN2OS
(5S,10bS)-5-(4-fluorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[(3,4-Dimethoxyphenyl)methylidene]-3-[3-(4-methylpiperazin-4-ium-1-yl)-3-oxopropyl]-1,3-thiazolidine-2,4-dione —— C20H26N3O5S+
5-[(3,4-Dimethoxyphenyl)methylidene]-3-[3-(4-methylpiperazin-4-ium-1-yl)-3-oxopropyl]-1,3-thiazolidine-2,4-dione
—— (5S)-7-cyclopentyl-2-(1,3-dimethylpyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5S)-7-cyclopentyl-2-(1,3-dimethylpyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-chloropyridin-2-yl)-[(2S,4R)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidin-1-yl]methanone —— C16H13ClF2N2O2
(5-chloropyridin-2-yl)-[(2S,4R)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidin-1-yl]methanone
—— 5-methyl-1-[2-oxo-2-[(5R)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decan-2-yl]ethyl]pyrimidine-2,4-dione —— C18H26N4O4
5-methyl-1-[2-oxo-2-[(5R)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decan-2-yl]ethyl]pyrimidine-2,4-dione
—— (5S)-7-cyclohexyl-2-(5-methylpyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O
(5S)-7-cyclohexyl-2-(5-methylpyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5,6-dimethyl-N-[(2S)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]-2-oxo-1H-pyridine-3-carboxamide —— C15H20N4O2
5,6-dimethyl-N-[(2S)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]-2-oxo-1H-pyridine-3-carboxamide
—— (5R)-7-(cyclobutylmethyl)-2-[2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O3S
(5R)-7-(cyclobutylmethyl)-2-[2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O2
(5S)-7-(cyclobutylmethyl)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-propan-2-yl-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H21F3N4O2
(5R)-7-propan-2-yl-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(6S)-2-[2-(dimethylamino)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]pyridine-2-carbonitrile —— C20H27N5O2
5-[(6S)-2-[2-(dimethylamino)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]pyridine-2-carbonitrile
—— (5-methyl-4-phenylthiophen-3-yl)-[(5R)-2-oxa-9-azaspiro[4.5]decan-9-yl]methanone —— C20H23NO2S
(5-methyl-4-phenylthiophen-3-yl)-[(5R)-2-oxa-9-azaspiro[4.5]decan-9-yl]methanone
—— (5S)-5-benzyl-1-(3-chlorophenyl)-4-(3-hydroxypropanoyl)piperazin-2-one —— C20H21ClN2O3
(5S)-5-benzyl-1-(3-chlorophenyl)-4-(3-hydroxypropanoyl)piperazin-2-one
—— (5S)-2-[4-(methylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl]-2,7-diazaspiro[4.5]decan-6-one —— C16H23N5O
(5S)-2-[4-(methylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-amino-4-nitrobenzoate —— C14H10N4O5S
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-amino-4-nitrobenzoate
—— (5R)-7-propyl-2-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5R)-7-propyl-2-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-cyclohexyl-N-[[(3R)-1-(4-methylphenyl)pyrrolidin-3-yl]methyl]-1H-pyrazole-4-carboxamide —— C22H30N4O
5-cyclohexyl-N-[[(3R)-1-(4-methylphenyl)pyrrolidin-3-yl]methyl]-1H-pyrazole-4-carboxamide
—— (5R)-1-ethyl-8,8-dimethyl-5-phenyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione —— C21H23N3O3
(5R)-1-ethyl-8,8-dimethyl-5-phenyl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione
—— (5S)-2-[2-(4-methylsulfonylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H22N2O4S
(5S)-2-[2-(4-methylsulfonylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3R)-1-(4-methoxypiperidin-1-yl)sulfonylpyrrolidin-3-yl]methyl]-1H-pyridin-2-one —— C16H25N3O4S
5-[[(3R)-1-(4-methoxypiperidin-1-yl)sulfonylpyrrolidin-3-yl]methyl]-1H-pyridin-2-one
—— 5-[[(3R)-1-[2-(1,1-dioxothian-4-yl)acetyl]pyrrolidin-3-yl]methyl]-1H-pyridin-2-one —— C17H24N2O4S
5-[[(3R)-1-[2-(1,1-dioxothian-4-yl)acetyl]pyrrolidin-3-yl]methyl]-1H-pyridin-2-one
—— (5R)-2-[4-(methylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl]-2,7-diazaspiro[4.5]decan-6-one —— C16H23N5O
(5R)-2-[4-(methylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R,4S)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidine-1-carbonyl]-1-methylpyrrole-3-carboxamide —— C17H17F2N3O3
5-[(2R,4S)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidine-1-carbonyl]-1-methylpyrrole-3-carboxamide
—— (5R)-7-cyclohexyl-2-(5-methylpyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O
(5R)-7-cyclohexyl-2-(5-methylpyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S,10bS)-5-(2-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C21H18N2O2S
(5S,10bS)-5-(2-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R)-2-methylsulfonyl-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C14H24N2O4S
(5R)-2-methylsulfonyl-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-1,8,8-trimethyl-5-thiophen-2-yl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione —— C18H19N3O3S
(5R)-1,8,8-trimethyl-5-thiophen-2-yl-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione
—— (5R)-2-[2-(4-ethylpiperazin-1-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H32N4O3
(5R)-2-[2-(4-ethylpiperazin-1-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R)-oxolan-2-yl]-N-[2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)ethyl]thiophene-2-carboxamide —— C18H18N4O3S
5-[(2R)-oxolan-2-yl]-N-[2-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)ethyl]thiophene-2-carboxamide