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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-7-cyclohexyl-2-[5-(methylsulfanylmethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O3S
(5R)-7-cyclohexyl-2-[5-(methylsulfanylmethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R)-2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one —— C17H16N6O3
5-[(2R)-2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one
—— (5S)-7-cyclohexyl-2-[5-(methylsulfanylmethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O3S
(5S)-7-cyclohexyl-2-[5-(methylsulfanylmethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-morpholin-4-ylsulfonyl-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C13H24N2O5S
(5R)-9-morpholin-4-ylsulfonyl-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-[(2S)-2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one —— C17H16N6O3
5-[(2S)-2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one
—— (5S)-9-morpholin-4-ylsulfonyl-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C13H24N2O5S
(5S)-9-morpholin-4-ylsulfonyl-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5S)-9-[2-(2H-triazol-4-ylsulfanyl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C12H18N4O2S
(5S)-9-[2-(2H-triazol-4-ylsulfanyl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-propyl-N-(pyridin-3-ylmethyl)-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1H-pyrazole-3-carboxamide —— C23H26N4O
5-propyl-N-(pyridin-3-ylmethyl)-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1H-pyrazole-3-carboxamide
—— 5-propyl-N-(pyridin-3-ylmethyl)-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-1H-pyrazole-3-carboxamide —— C23H26N4O
5-propyl-N-(pyridin-3-ylmethyl)-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-1H-pyrazole-3-carboxamide
—— (5S)-5-methyl-1-(2-morpholin-4-ylethyl)-5-phenylpiperidin-2-one —— C18H26N2O2
(5S)-5-methyl-1-(2-morpholin-4-ylethyl)-5-phenylpiperidin-2-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(3-ethylimidazol-4-yl)methyl]-5-methylpiperidin-2-one —— C20H25N3O3
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(3-ethylimidazol-4-yl)methyl]-5-methylpiperidin-2-one
—— (5R)-N'-[(2-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide —— C17H18N2O3S
(5R)-N'-[(2-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide
—— [(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]methanone —— C15H20F3N3O3
[(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]methanone
—— 5-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C19H20N6O2
5-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— (5S)-7-cyclohexyl-2-(4-hydroxy-3-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C22H30N2O3
(5S)-7-cyclohexyl-2-(4-hydroxy-3-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5S)-7-(cyclopropylmethyl)-2-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— [5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(2S)-2-phenylpyrrolidin-1-yl]methanone —— C20H18FN3O
[5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(2S)-2-phenylpyrrolidin-1-yl]methanone
—— (5R)-7-cyclohexyl-2-(2-pyridin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O2
(5R)-7-cyclohexyl-2-(2-pyridin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-N-benzyl-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H19NOS
(5S)-N-benzyl-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[2-[(3R)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C20H23N3O5
5-[2-[(3R)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— (5R)-7-(cyclopropylmethyl)-2-(2-methylsulfanylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H26N2O2S
(5R)-7-(cyclopropylmethyl)-2-(2-methylsulfanylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-tert-butyl-4-[[(5R)-7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl]furan-2-carboxamide —— C20H31N3O4
5-tert-butyl-4-[[(5R)-7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl]furan-2-carboxamide
—— (5R)-9-[2-(2-ethylimidazol-1-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C15H23N3O2
(5R)-9-[2-(2-ethylimidazol-1-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— [(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]methanone —— C15H20F3N3O3
[(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]methanone
—— (5R)-7-(2-methoxyethyl)-2-[(E)-3-(2-methoxyphenyl)prop-2-enyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O3
(5R)-7-(2-methoxyethyl)-2-[(E)-3-(2-methoxyphenyl)prop-2-enyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(5R)-7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione —— C18H24N4O4
5-[(5R)-7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione
—— (5Z)-5-[[2-(3-imidazol-1-ylpropylamino)-8-methyl-4-oxo-1H-quinolin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H19N5O2S2
(5Z)-5-[[2-(3-imidazol-1-ylpropylamino)-8-methyl-4-oxo-1H-quinolin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-7-(2-methoxyethyl)-2-[(E)-3-(2-methoxyphenyl)prop-2-enyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O3
(5S)-7-(2-methoxyethyl)-2-[(E)-3-(2-methoxyphenyl)prop-2-enyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[2-(2-ethylimidazol-1-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C15H23N3O2
(5S)-9-[2-(2-ethylimidazol-1-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— [(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(4-methylsulfonylphenyl)methanone —— C17H23NO5S
[(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(4-methylsulfonylphenyl)methanone
—— (5R)-9-[2-(2H-triazol-4-ylsulfanyl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C12H18N4O2S
(5R)-9-[2-(2H-triazol-4-ylsulfanyl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-5-ethyl-N'-[(7-ethylindol-3-ylidene)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide —— C22H25N3OS
(5R)-5-ethyl-N'-[(7-ethylindol-3-ylidene)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide
—— (5R)-5-methyl-1-(2-morpholin-4-ylethyl)-5-phenylpiperidin-2-one —— C18H26N2O2
(5R)-5-methyl-1-(2-morpholin-4-ylethyl)-5-phenylpiperidin-2-one
—— (5S)-7-cyclohexyl-2-(2-pyridin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O2
(5S)-7-cyclohexyl-2-(2-pyridin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-hydroxyethyl)-2-[[3-(trifluoromethyl)phenyl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H23F3N2O2
(5R)-7-(2-hydroxyethyl)-2-[[3-(trifluoromethyl)phenyl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— [(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(4-methylsulfonylphenyl)methanone —— C17H23NO5S
[(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(4-methylsulfonylphenyl)methanone
—— 5-tert-butyl-4-[[(5S)-7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl]furan-2-carboxamide —— C20H31N3O4
5-tert-butyl-4-[[(5S)-7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl]furan-2-carboxamide
—— (5R)-5-methyl-N-[(Z)-(2-oxoacenaphthylen-1-ylidene)amino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C22H18N2O2S
(5R)-5-methyl-N-[(Z)-(2-oxoacenaphthylen-1-ylidene)amino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,5-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C16H21N3O2S
(5R)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,5-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[(5S)-7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione —— C18H24N4O4
5-[(5S)-7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione
—— (5R)-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C14H18F3N3O2
(5R)-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-[[(3S)-3-[[4-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methyl]-2-methoxybenzoic acid —— C21H25NO4
5-[[(3S)-3-[[4-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methyl]-2-methoxybenzoic acid
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(3-ethylimidazol-4-yl)methyl]-5-methylpiperidin-2-one —— C20H25N3O3
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(3-ethylimidazol-4-yl)methyl]-5-methylpiperidin-2-one
—— (5S)-7-(cyclopropylmethyl)-2-(2-methylsulfanylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H26N2O2S
(5S)-7-(cyclopropylmethyl)-2-(2-methylsulfanylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(oxan-4-yl)-2-(2H-triazol-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H25N5O2
(5R)-7-(oxan-4-yl)-2-(2H-triazol-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4OS
(5S)-7-(cyclopropylmethyl)-2-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(2R)-2-phenylpyrrolidin-1-yl]methanone —— C20H18FN3O
[5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(2R)-2-phenylpyrrolidin-1-yl]methanone
—— (5R)-7-cyclohexyl-2-(4-hydroxy-3-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C22H30N2O3
(5R)-7-cyclohexyl-2-(4-hydroxy-3-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclopropylmethyl)-2-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4OS
(5R)-7-(cyclopropylmethyl)-2-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C14H18F3N3O2
(5S)-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol