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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-9-[3-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H22N4O2
(5S)-9-[3-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,5-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C16H21N3O2S
(5S)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,5-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-7-(cyclopropylmethyl)-2-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5R)-7-(cyclopropylmethyl)-2-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5,6-dimethyl-N-[(1R)-1-(6-methyl-1H-benzimidazol-2-yl)ethyl]-2-oxo-1H-pyridine-3-carboxamide —— C18H20N4O2
5,6-dimethyl-N-[(1R)-1-(6-methyl-1H-benzimidazol-2-yl)ethyl]-2-oxo-1H-pyridine-3-carboxamide
—— 5-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C19H20N6O2
5-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— (5S)-7-(2-hydroxyethyl)-2-[[3-(trifluoromethyl)phenyl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H23F3N2O2
(5S)-7-(2-hydroxyethyl)-2-[[3-(trifluoromethyl)phenyl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-Imidazo[1,2-c]quinazolin-3-ylsulfanylpentanoate —— C15H14N3O2S-
5-Imidazo[1,2-c]quinazolin-3-ylsulfanylpentanoate
—— (5R)-N-benzyl-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H19NOS
(5R)-N-benzyl-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-5-methyl-5-(4-methylpent-3-enyl)-1-[3-(1-methylpyrazol-4-yl)propyl]piperidin-2-one —— C19H31N3O
(5R)-5-methyl-5-(4-methylpent-3-enyl)-1-[3-(1-methylpyrazol-4-yl)propyl]piperidin-2-one
—— [5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(1S)-1-pyridin-2-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone —— C21H19N5O2
[5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(1S)-1-pyridin-2-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone
—— (5R)-7-(2-methoxyethyl)-2-[(2-methyl-6-oxo-1H-pyrimidin-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O3
(5R)-7-(2-methoxyethyl)-2-[(2-methyl-6-oxo-1H-pyrimidin-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5E)-5-(5-methoxy-3-methyl-1,3-benzothiazol-2(3H)-ylidene)-3-phenyl-2-thioxo-1,3-thiazolidin-4-one —— C18H14N2O2S3
(5E)-5-(5-methoxy-3-methyl-1,3-benzothiazol-2(3H)-ylidene)-3-phenyl-2-thioxo-1,3-thiazolidin-4-one
—— (5R)-2-(5-methyl-1,2,4-oxadiazol-3-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O3
(5R)-2-(5-methyl-1,2,4-oxadiazol-3-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-N'-[(5-hydroxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide —— C17H18N2O3S
(5R)-N'-[(5-hydroxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide
—— 5-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]-2-(phenoxymethyl)-1H-pyrimidin-6-one —— C20H20N4O4
5-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]-2-(phenoxymethyl)-1H-pyrimidin-6-one
—— 5,6-dimethyl-N-[(1S)-1-(6-methyl-1H-benzimidazol-2-yl)ethyl]-2-oxo-1H-pyridine-3-carboxamide —— C18H20N4O2
5,6-dimethyl-N-[(1S)-1-(6-methyl-1H-benzimidazol-2-yl)ethyl]-2-oxo-1H-pyridine-3-carboxamide
—— (5S)-9-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C19H27NO5
(5S)-9-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-indol-3-ylidene-4-[[(2S)-oxolan-2-yl]methyl]-2-(pyrrolidin-1-ylmethyl)-1,2,4-triazolidine-3-thione —— C20H25N5OS
5-indol-3-ylidene-4-[[(2S)-oxolan-2-yl]methyl]-2-(pyrrolidin-1-ylmethyl)-1,2,4-triazolidine-3-thione
—— (5S)-7-(2-methoxyethyl)-2-[(2-methyl-6-oxo-1H-pyrimidin-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O3
(5S)-7-(2-methoxyethyl)-2-[(2-methyl-6-oxo-1H-pyrimidin-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C19H27NO5
(5R)-9-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-[(3S)-1-tert-butyl-5-oxopyrrolidine-3-carbonyl]-N-methyl-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide —— C17H24N4O4
5-[(3S)-1-tert-butyl-5-oxopyrrolidine-3-carbonyl]-N-methyl-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
—— 5-[(3R)-1-tert-butyl-5-oxopyrrolidine-3-carbonyl]-N-methyl-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide —— C17H24N4O4
5-[(3R)-1-tert-butyl-5-oxopyrrolidine-3-carbonyl]-N-methyl-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
—— (5R)-7-(2-methoxyethyl)-2-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O3S
(5R)-7-(2-methoxyethyl)-2-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-methyl-5-(4-methylpent-3-enyl)-1-[3-(1-methylpyrazol-4-yl)propyl]piperidin-2-one —— C19H31N3O
(5S)-5-methyl-5-(4-methylpent-3-enyl)-1-[3-(1-methylpyrazol-4-yl)propyl]piperidin-2-one
—— 5-[(5S)-7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione —— C19H26N4O4
5-[(5S)-7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione
—— 5-indol-3-ylidene-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazolidine-3-thione —— C15H16N4OS
5-indol-3-ylidene-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazolidine-3-thione
—— 5-[(5R)-7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione —— C19H26N4O4
5-[(5R)-7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrimidine-2,4-dione
—— (5S)-7-(2-methoxyethyl)-2-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O3S
(5S)-7-(2-methoxyethyl)-2-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-cyclohexyl-2-[2-(5-methyl-1H-1,2,4-triazol-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H29N5O2
(5S)-7-cyclohexyl-2-[2-(5-methyl-1H-1,2,4-triazol-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R)-oxolan-2-yl]-N-[3-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]thiophene-2-carboxamide —— C18H20N4O2S
5-[(2R)-oxolan-2-yl]-N-[3-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]thiophene-2-carboxamide
—— 5-[(3R)-3-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one —— C20H23N5O3
5-[(3R)-3-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one
—— 5-[(2S)-oxolan-2-yl]-N-[3-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]thiophene-2-carboxamide —— C18H20N4O2S
5-[(2S)-oxolan-2-yl]-N-[3-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]thiophene-2-carboxamide
—— (5S)-7-cyclopentyl-2-(6-propan-2-ylpyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C21H31N3O
(5S)-7-cyclopentyl-2-(6-propan-2-ylpyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[2-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H20N4O3
(5S)-9-[2-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-[3-[[4-[(2S)-pentan-2-yl]triazol-1-yl]methyl]phenyl]-2H-tetrazole —— C15H19N7
5-[3-[[4-[(2S)-pentan-2-yl]triazol-1-yl]methyl]phenyl]-2H-tetrazole
—— (5R)-7-(2-methoxyethyl)-2-(1-methylpyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H25N3O3
(5R)-7-(2-methoxyethyl)-2-(1-methylpyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclopropylmethyl)-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O2
(5R)-7-(cyclopropylmethyl)-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(5-methyl-1,2,4-oxadiazol-3-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O3
(5S)-2-(5-methyl-1,2,4-oxadiazol-3-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[3-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H22N4O2
(5R)-9-[3-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-9-[2-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H20N4O3
(5R)-9-[2-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-[3-oxo-3-[(5S)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]propyl]-1,2-oxazol-3-one —— C14H19N3O4
5-[3-oxo-3-[(5S)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]propyl]-1,2-oxazol-3-one
—— (5R)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-cyclopentylpiperidin-2-one —— C19H21N5O2
(5R)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-cyclopentylpiperidin-2-one
—— (5R)-7-cyclohexyl-2-[2-(5-methyl-1H-1,2,4-triazol-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H29N5O2
(5R)-7-cyclohexyl-2-[2-(5-methyl-1H-1,2,4-triazol-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— [5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(1R)-1-pyridin-2-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone —— C21H19N5O2
[5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(1R)-1-pyridin-2-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone
—— (5S)-2-(2-ethyl-6-oxo-1H-pyridine-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O3
(5S)-2-(2-ethyl-6-oxo-1H-pyridine-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[2-(4-fluorophenoxy)ethyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H27FN2O3
(5R)-2-[2-(4-fluorophenoxy)ethyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-hydroxyethyl)-2-(2-methyl-5-propan-2-ylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N2O4
(5R)-7-(2-hydroxyethyl)-2-(2-methyl-5-propan-2-ylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3S)-1-(3-methylbut-2-enoyl)pyrrolidin-3-yl]methyl]-1H-pyridin-2-one —— C15H20N2O2
5-[[(3S)-1-(3-methylbut-2-enoyl)pyrrolidin-3-yl]methyl]-1H-pyridin-2-one
—— (5S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]-5-methyl-5-phenylpiperidin-2-one —— C18H23N3O
(5S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]-5-methyl-5-phenylpiperidin-2-one
—— 5-[(3S)-3-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one —— C20H23N5O3
5-[(3S)-3-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one