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—— [5-[[[(2S)-butan-2-yl]-(2-methylbenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C21H27NO5S
[5-[[[(2S)-butan-2-yl]-(2-methylbenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— 5,6-dimethyl-3-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H25N5O2
5,6-dimethyl-3-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— (5S)-7-(2-methoxyethyl)-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H25N3O3
(5S)-7-(2-methoxyethyl)-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-cyclohexyl-2-[2-(2-oxopyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O3
(5S)-7-cyclohexyl-2-[2-(2-oxopyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-(1-ethylpyrazol-4-yl)sulfonyl-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4O3S
(5S)-7-(cyclobutylmethyl)-2-(1-ethylpyrazol-4-yl)sulfonyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-3-(1-ethylimidazol-2-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one —— C15H19N5O2
5-[(3S)-3-(1-ethylimidazol-2-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one
—— (5R)-9-[2-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H27N3O2
(5R)-9-[2-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-5-methyl-N-[[1-(pyrazol-1-ylmethyl)cyclopropyl]methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C18H23N3OS
(5S)-5-methyl-N-[[1-(pyrazol-1-ylmethyl)cyclopropyl]methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-7-(cyclobutylmethyl)-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C23H29N3O2
(5R)-7-(cyclobutylmethyl)-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)methyl]-N-[(2R)-3-methylbutan-2-yl]furan-2-carboxamide —— C21H24N2O5
5-[(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)methyl]-N-[(2R)-3-methylbutan-2-yl]furan-2-carboxamide
—— 5-[(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)methyl]-N-[(2S)-3-methylbutan-2-yl]furan-2-carboxamide —— C21H24N2O5
5-[(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)methyl]-N-[(2S)-3-methylbutan-2-yl]furan-2-carboxamide
—— 5-(3-fluorophenyl)-N-methyl-N-[(1R)-1-pyridin-3-ylpentyl]-1H-pyrazole-4-carboxamide —— C21H23FN4O
5-(3-fluorophenyl)-N-methyl-N-[(1R)-1-pyridin-3-ylpentyl]-1H-pyrazole-4-carboxamide
—— 5,6-dimethyl-3-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H25N5O2
5,6-dimethyl-3-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— (5S)-7-(cyclopropylmethyl)-N-(4-ethoxyphenyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide —— C21H29N3O3
(5S)-7-(cyclopropylmethyl)-N-(4-ethoxyphenyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
—— 5-methyl-1-propyl-N-[(1S)-1-(2-propyl-1,2,4-triazol-3-yl)ethyl]pyrazole-4-carboxamide —— C15H24N6O
5-methyl-1-propyl-N-[(1S)-1-(2-propyl-1,2,4-triazol-3-yl)ethyl]pyrazole-4-carboxamide
—— [5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone —— C19H23N5OS
[5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone
—— (5S)-1-(cyclohexylmethyl)-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C19H30N4O3
(5S)-1-(cyclohexylmethyl)-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5S)-7-(cyclobutylmethyl)-2-(2-methylsulfanylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4OS
(5S)-7-(cyclobutylmethyl)-2-(2-methylsulfanylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-methyl-1-propyl-N-[(1R)-1-(2-propyl-1,2,4-triazol-3-yl)ethyl]pyrazole-4-carboxamide —— C15H24N6O
5-methyl-1-propyl-N-[(1R)-1-(2-propyl-1,2,4-triazol-3-yl)ethyl]pyrazole-4-carboxamide
—— (5R)-7-(cyclobutylmethyl)-2-(1-ethylpyrazol-4-yl)sulfonyl-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4O3S
(5R)-7-(cyclobutylmethyl)-2-(1-ethylpyrazol-4-yl)sulfonyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-cyclohexyl-2-[2-(2-oxopyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O3
(5R)-7-cyclohexyl-2-[2-(2-oxopyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— [5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone —— C19H23N5OS
[5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone
—— 5-[(3R)-3-(1-ethylimidazol-2-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one —— C15H19N5O2
5-[(3R)-3-(1-ethylimidazol-2-yl)piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-(3-fluorophenyl)-N-methyl-N-[(1S)-1-pyridin-3-ylpentyl]-1H-pyrazole-4-carboxamide —— C21H23FN4O
5-(3-fluorophenyl)-N-methyl-N-[(1S)-1-pyridin-3-ylpentyl]-1H-pyrazole-4-carboxamide
—— [5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2R)-2-pyridin-3-ylpyrrolidin-1-yl]methanone —— C18H18N4O2
[5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2R)-2-pyridin-3-ylpyrrolidin-1-yl]methanone
—— (5R)-7-propan-2-yl-2-[5-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one —— C17H22F3N3O
(5R)-7-propan-2-yl-2-[5-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
—— [5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-pyridin-3-ylpyrrolidin-1-yl]methanone —— C18H18N4O2
[5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-pyridin-3-ylpyrrolidin-1-yl]methanone
—— 5-(3-fluorophenyl)-N-[(3S)-1-oxaspiro[4.5]decan-3-yl]-1H-pyrazole-4-carboxamide —— C19H22FN3O2
5-(3-fluorophenyl)-N-[(3S)-1-oxaspiro[4.5]decan-3-yl]-1H-pyrazole-4-carboxamide
—— 5-(3-chlorophenyl)-N-(1,3-dihydro-2-benzofuran-5-yl)-1,2-oxazole-3-carboxamide —— C18H13ClN2O3
5-(3-chlorophenyl)-N-(1,3-dihydro-2-benzofuran-5-yl)-1,2-oxazole-3-carboxamide
—— (5R)-7-cyclohexyl-2-(2-methylsulfanylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O2S
(5R)-7-cyclohexyl-2-(2-methylsulfanylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-methyl-4-N-[(1S)-1-(2-propyl-1,2,4-triazol-3-yl)ethyl]pyrimidine-2,4-diamine —— C12H19N7
5-methyl-4-N-[(1S)-1-(2-propyl-1,2,4-triazol-3-yl)ethyl]pyrimidine-2,4-diamine
—— (5R)-7-(cyclobutylmethyl)-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H26N2O4
(5R)-7-(cyclobutylmethyl)-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-(1H-benzimidazol-2-ylmethyl)piperidine-1-carbonyl]-2-cyclopropyl-1H-pyrimidin-6-one —— C21H23N5O2
5-[(3R)-3-(1H-benzimidazol-2-ylmethyl)piperidine-1-carbonyl]-2-cyclopropyl-1H-pyrimidin-6-one
—— (5S)-2-(5-ethylsulfanylthiophene-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24N2O3S2
(5S)-2-(5-ethylsulfanylthiophene-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-methyl-2-[2-(4-pyrimidin-2-ylpiperazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H28N6O2
(5S)-7-methyl-2-[2-(4-pyrimidin-2-ylpiperazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(3-methoxyphenyl)-N-[(1S)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide —— C18H21N5O3
5-(3-methoxyphenyl)-N-[(1S)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
—— (5R)-7-methyl-2-[2-(4-pyrimidin-2-ylpiperazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H28N6O2
(5R)-7-methyl-2-[2-(4-pyrimidin-2-ylpiperazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-propyl-4-[(3R)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidine —— C21H26N6
5-propyl-4-[(3R)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidine
—— (5R)-2-[2-[methyl(pyridin-3-ylmethyl)amino]acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O2
(5R)-2-[2-[methyl(pyridin-3-ylmethyl)amino]acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-propyl-4-[(3S)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidine —— C21H26N6
5-propyl-4-[(3S)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidine
—— (5S)-7-(cyclobutylmethyl)-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H26N2O4
(5S)-7-(cyclobutylmethyl)-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propan-2-yl-2-[5-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one —— C17H22F3N3O
(5S)-7-propan-2-yl-2-[5-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(5-ethylsulfanylthiophene-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24N2O3S2
(5R)-2-(5-ethylsulfanylthiophene-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-methyl-4-N-[(1R)-1-(2-propyl-1,2,4-triazol-3-yl)ethyl]pyrimidine-2,4-diamine —— C12H19N7
5-methyl-4-N-[(1R)-1-(2-propyl-1,2,4-triazol-3-yl)ethyl]pyrimidine-2,4-diamine
—— 5-(3-fluorophenyl)-N-[(3R)-1-oxaspiro[4.5]decan-3-yl]-1H-pyrazole-4-carboxamide —— C19H22FN3O2
5-(3-fluorophenyl)-N-[(3R)-1-oxaspiro[4.5]decan-3-yl]-1H-pyrazole-4-carboxamide
—— (5R)-7-(cyclobutylmethyl)-2-[6-(dimethylamino)pyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H30N4O2
(5R)-7-(cyclobutylmethyl)-2-[6-(dimethylamino)pyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[2-[[cyclopropanecarbonyl(propyl)amino]methyl]pyrrol-1-yl]methyl]-N-(2-pyrrolidin-1-ium-1-ylethyl)furan-2-carboxamide —— C24H35N4O3+
5-[[2-[[cyclopropanecarbonyl(propyl)amino]methyl]pyrrol-1-yl]methyl]-N-(2-pyrrolidin-1-ium-1-ylethyl)furan-2-carboxamide
—— (5S)-7-cyclohexyl-2-(2-methylsulfanylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O2S
(5S)-7-cyclohexyl-2-(2-methylsulfanylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(3-methoxyphenyl)-N-[(1R)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide —— C18H21N5O3
5-(3-methoxyphenyl)-N-[(1R)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
—— 5-methylsulfonyl-1'-[[(3S)-oxolan-3-yl]methyl]spiro[6,7-dihydro-1H-imidazo[4,5-c]pyridine-4,4'-piperidine] —— C16H26N4O3S
5-methylsulfonyl-1'-[[(3S)-oxolan-3-yl]methyl]spiro[6,7-dihydro-1H-imidazo[4,5-c]pyridine-4,4'-piperidine]