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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-N-(4-cycloheptyloxybutyl)-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H34N2O3
(5R)-N-(4-cycloheptyloxybutyl)-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5R)-N-[(2-cyclobutyloxyphenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H26N2O3
(5R)-N-[(2-cyclobutyloxyphenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[[(1S,2R)-2-phenylcyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C18H24N2O2
(5S)-N-[[(1S,2R)-2-phenylcyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(1S,3R)-3-methoxy-2,2,3-trimethylcyclobutyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H28N2O3
(5S)-N-[(1S,3R)-3-methoxy-2,2,3-trimethylcyclobutyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-[(3S)-1-[4-(diethylcarbamoyl)phenyl]sulfonylpiperidin-3-yl]-1H-pyrazole-3-carboxamide —— C20H27N5O4S
5-[(3S)-1-[4-(diethylcarbamoyl)phenyl]sulfonylpiperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3R)-1-[4-fluoro-2-(trifluoromethylsulfonyl)phenyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C16H16F4N4O3S
5-[(3R)-1-[4-fluoro-2-(trifluoromethylsulfonyl)phenyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5R)-N-[(S)-cyclobutyl-(4-fluorophenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H25FN2O2
(5R)-N-[(S)-cyclobutyl-(4-fluorophenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(1S,2R)-2-cyclohexylcyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C17H28N2O2
(5S)-N-[(1S,2R)-2-cyclohexylcyclopropyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5R)-N-[[(4R)-6,7-dihydro-4H-thieno[3,2-c]pyran-4-yl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H22N2O3S
(5R)-N-[[(4R)-6,7-dihydro-4H-thieno[3,2-c]pyran-4-yl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-[(3S)-1-(4-cyano-5,6-dimethylpyridazin-3-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C16H19N7O
5-[(3S)-1-(4-cyano-5,6-dimethylpyridazin-3-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3S)-1-[4-fluoro-2-(trifluoromethylsulfonyl)phenyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C16H16F4N4O3S
5-[(3S)-1-[4-fluoro-2-(trifluoromethylsulfonyl)phenyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5R)-7-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2-oxa-7-azaspiro[4.4]nonane —— C15H18N4O2
(5R)-7-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2-oxa-7-azaspiro[4.4]nonane
—— (5S,6R)-1-methyl-5-[(5S)-2-oxa-7-azaspiro[4.4]nonane-7-carbonyl]-6-thiophen-2-ylpiperidin-2-one —— C18H24N2O3S
(5S,6R)-1-methyl-5-[(5S)-2-oxa-7-azaspiro[4.4]nonane-7-carbonyl]-6-thiophen-2-ylpiperidin-2-one
—— (5S)-N-[[(1R,2S,4S)-2-bicyclo[2.2.1]heptanyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H26N2O2
(5S)-N-[[(1R,2S,4S)-2-bicyclo[2.2.1]heptanyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5R)-7-[2-(methoxymethyl)-6-methylpyrimidin-4-yl]-2-oxa-7-azaspiro[4.4]nonane —— C14H21N3O2
(5R)-7-[2-(methoxymethyl)-6-methylpyrimidin-4-yl]-2-oxa-7-azaspiro[4.4]nonane
—— 5-[[[(3R)-1-(2,6-difluorophenyl)pyrrolidin-3-yl]amino]methyl]furan-2-carbonitrile —— C16H15F2N3O
5-[[[(3R)-1-(2,6-difluorophenyl)pyrrolidin-3-yl]amino]methyl]furan-2-carbonitrile
—— (5S)-N-[[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H26N2O2
(5S)-N-[[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-[(3R)-1-(6-chloro-2-methylpyrimidin-4-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C14H17ClN6O
5-[(3R)-1-(6-chloro-2-methylpyrimidin-4-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5R)-N-[(R)-cyclobutyl-(4-fluorophenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H25FN2O2
(5R)-N-[(R)-cyclobutyl-(4-fluorophenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-[(3R)-1-(6-ethylthieno[2,3-d]pyrimidin-4-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C17H20N6OS
5-[(3R)-1-(6-ethylthieno[2,3-d]pyrimidin-4-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5S)-N-[[1-(2-methoxyphenyl)cyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H26N2O3
(5S)-N-[[1-(2-methoxyphenyl)cyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(2S)-1-cyclopropylpropan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C14H24N2O2
(5S)-N-[(2S)-1-cyclopropylpropan-2-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[[(1R,2R)-2-phenylcyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C18H24N2O2
(5S)-N-[[(1R,2R)-2-phenylcyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[(1R)-1-[(1R,2R)-2-(3-methylphenyl)cyclopropyl]ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C20H28N2O2
(5S)-N-[(1R)-1-[(1R,2R)-2-(3-methylphenyl)cyclopropyl]ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-[[[(3S)-1-(2,6-difluorophenyl)pyrrolidin-3-yl]amino]methyl]furan-2-carbonitrile —— C16H15F2N3O
5-[[[(3S)-1-(2,6-difluorophenyl)pyrrolidin-3-yl]amino]methyl]furan-2-carbonitrile
—— 5-[(3S)-1-(6-ethylthieno[2,3-d]pyrimidin-4-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C17H20N6OS
5-[(3S)-1-(6-ethylthieno[2,3-d]pyrimidin-4-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5S)-N-[[(4R)-6,7-dihydro-4H-thieno[3,2-c]pyran-4-yl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H22N2O3S
(5S)-N-[[(4R)-6,7-dihydro-4H-thieno[3,2-c]pyran-4-yl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-[(3S)-1-(2-methyl-4-nitrophenyl)sulfonylpiperidin-3-yl]-1H-pyrazole-3-carboxamide —— C16H19N5O5S
5-[(3S)-1-(2-methyl-4-nitrophenyl)sulfonylpiperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5S)-N-[(R)-cyclobutyl-(4-fluorophenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C19H25FN2O2
(5S)-N-[(R)-cyclobutyl-(4-fluorophenyl)methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[2-(cyclopropylmethoxy)ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C14H24N2O3
(5S)-N-[2-(cyclopropylmethoxy)ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-7-[2-(methoxymethyl)-6-methylpyrimidin-4-yl]-2-oxa-7-azaspiro[4.4]nonane —— C14H21N3O2
(5S)-7-[2-(methoxymethyl)-6-methylpyrimidin-4-yl]-2-oxa-7-azaspiro[4.4]nonane
—— (5S)-N-[(1R)-1-[(1S,2R)-2-(3-methylphenyl)cyclopropyl]ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C20H28N2O2
(5S)-N-[(1R)-1-[(1S,2R)-2-(3-methylphenyl)cyclopropyl]ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-Fluoro-4-methyl-2-(propan-2-ylamino)benzamide —— C11H15FN2O
5-Fluoro-4-methyl-2-(propan-2-ylamino)benzamide
—— (5R,6R)-1-methyl-5-[(5S)-2-oxa-7-azaspiro[4.4]nonane-7-carbonyl]-6-thiophen-2-ylpiperidin-2-one —— C18H24N2O3S
(5R,6R)-1-methyl-5-[(5S)-2-oxa-7-azaspiro[4.4]nonane-7-carbonyl]-6-thiophen-2-ylpiperidin-2-one
—— (5S)-N-[(1S,5R,6R)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C16H26N2O3
(5S)-N-[(1S,5R,6R)-7,7-dimethyl-2-oxabicyclo[3.2.0]heptan-6-yl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-[(3S)-1-(6-chloro-2-methylpyrimidin-4-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C14H17ClN6O
5-[(3S)-1-(6-chloro-2-methylpyrimidin-4-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5S)-7-(2-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane —— C14H18N4O
(5S)-7-(2-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane
—— 5-nitro-2-[[(3R)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methylamino]benzamide —— C14H17F3N4O3
5-nitro-2-[[(3R)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methylamino]benzamide
—— 5-nitro-2-[[(3S)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methylamino]benzamide —— C14H17F3N4O3
5-nitro-2-[[(3S)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methylamino]benzamide
—— (5R)-N-[2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C17H27N5O2
(5R)-N-[2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— (5S)-N-[[(1R,2S)-2-phenylcyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C18H24N2O2
(5S)-N-[[(1R,2S)-2-phenylcyclopropyl]methyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-[(3S)-1-(3-carbamoylphenyl)sulfonylpiperidin-3-yl]-1H-pyrazole-3-carboxamide —— C16H19N5O4S
5-[(3S)-1-(3-carbamoylphenyl)sulfonylpiperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5R)-7-(2-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane —— C14H18N4O
(5R)-7-(2-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane
—— 5-[(3S)-1-(4-pyrazol-1-ylpyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C16H18N8O
5-[(3S)-1-(4-pyrazol-1-ylpyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[[(R)-butylsulfinyl]methyl]-1-[4-(trifluoromethyl)phenyl]tetrazole —— C13H15F3N4OS
5-[[(R)-butylsulfinyl]methyl]-1-[4-(trifluoromethyl)phenyl]tetrazole
—— 5-(2-fluorophenyl)-3-[(2S)-2-methylbutyl]sulfanyl-1H-1,2,4-triazole —— C13H16FN3S
5-(2-fluorophenyl)-3-[(2S)-2-methylbutyl]sulfanyl-1H-1,2,4-triazole
—— (5R)-N-[2-(cyclopropylmethoxy)ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide —— C14H24N2O3
(5R)-N-[2-(cyclopropylmethoxy)ethyl]-2-oxa-7-azaspiro[4.4]nonane-7-carboxamide
—— 5-chloro-2-[[(3S)-1-methylsulfonylpiperidin-3-yl]methyl]-3,4-dihydro-1H-isoquinoline —— C16H23ClN2O2S
5-chloro-2-[[(3S)-1-methylsulfonylpiperidin-3-yl]methyl]-3,4-dihydro-1H-isoquinoline
—— 5-(2-fluorophenyl)-3-[(2R)-2-methylbutyl]sulfanyl-1H-1,2,4-triazole —— C13H16FN3S
5-(2-fluorophenyl)-3-[(2R)-2-methylbutyl]sulfanyl-1H-1,2,4-triazole
—— (5R)-5-[[[6-(2-methylpropoxy)pyrazin-2-yl]amino]methyl]pyrrolidin-2-one —— C13H20N4O2
(5R)-5-[[[6-(2-methylpropoxy)pyrazin-2-yl]amino]methyl]pyrrolidin-2-one