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—— 5-[(R)-(2-fluorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H20FN4O2S+
5-[(R)-(2-fluorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[[(3R)-1-[2-[cyclopentyl(methyl)amino]acetyl]pyrrolidin-3-yl]methyl]-1H-pyridin-2-one —— C18H27N3O2
5-[[(3R)-1-[2-[cyclopentyl(methyl)amino]acetyl]pyrrolidin-3-yl]methyl]-1H-pyridin-2-one
—— 5-[(S)-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-(4-ethoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O3S
5-[(S)-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-(4-ethoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-methoxy-1-methyl-N-[2-[5-[(2S)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]ethyl]indole-2-carboxamide —— C19H22N4O4
5-methoxy-1-methyl-N-[2-[5-[(2S)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]ethyl]indole-2-carboxamide
—— 5-methoxy-1-methyl-N-[(4R)-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl]indole-2-carboxamide —— C19H21N3O2S
5-methoxy-1-methyl-N-[(4R)-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl]indole-2-carboxamide
—— 5-[3-[(3S)-3-(hydroxymethyl)-3-propylpiperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one —— C18H29N3O3
5-[3-[(3S)-3-(hydroxymethyl)-3-propylpiperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one
—— 5-[(S)-(3,4-dichlorophenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C16H17Cl2N4O2S+
5-[(S)-(3,4-dichlorophenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(4-ethylpiperazine-1,4-diium-1-yl)-(2-fluorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H24FN5OS+2
5-[(R)-(4-ethylpiperazine-1,4-diium-1-yl)-(2-fluorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5R)-5-methyl-5-(4-methylpent-3-enyl)-1-[2-(1,3-thiazol-4-yl)ethyl]piperidin-2-one —— C17H26N2OS
(5R)-5-methyl-5-(4-methylpent-3-enyl)-1-[2-(1,3-thiazol-4-yl)ethyl]piperidin-2-one
—— 5-[(S)-(2-chlorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H21ClN4OS
5-[(S)-(2-chlorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[3-[(3R)-3-(hydroxymethyl)-3-propylpiperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one —— C18H29N3O3
5-[3-[(3R)-3-(hydroxymethyl)-3-propylpiperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one
—— 5-[(S)-(2-chlorophenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C16H18ClN4O2S+
5-[(S)-(2-chlorophenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(4-ethoxy-3-methoxyphenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O4S+
5-[(R)-(4-ethoxy-3-methoxyphenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H24N4O3S
5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-Cyclopentylsulfanyl-7-(3-fluorophenyl)-1,3-dimethylpyrimido[4,5-d]pyrimidine-2,4-dione —— C19H19FN4O2S
5-Cyclopentylsulfanyl-7-(3-fluorophenyl)-1,3-dimethylpyrimido[4,5-d]pyrimidine-2,4-dione
—— 5-cyclopropyl-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methyl-1,3,4-oxadiazol-2-amine —— C15H17N3O3
5-cyclopropyl-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methyl-1,3,4-oxadiazol-2-amine
—— 5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H25N4O3S+
5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(4-ethoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O3S
5-[(R)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(4-ethoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4OS+
5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2-chlorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H21ClN4OS
5-[(R)-(2-chlorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— (5R)-7-(2-methoxyethyl)-2-[2-(methylamino)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O3
(5R)-7-(2-methoxyethyl)-2-[2-(methylamino)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(R)-(4-ethoxyphenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H25N5O2S
5-[(R)-(4-ethoxyphenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— (5S)-2-(2-amino-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one —— C20H29N5O
(5S)-2-(2-amino-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-Cyclopentylsulfanyl-7-(2-methoxyphenyl)-1,3-dimethylpyrimido[4,5-d]pyrimidine-2,4-dione —— C20H22N4O3S
5-Cyclopentylsulfanyl-7-(2-methoxyphenyl)-1,3-dimethylpyrimido[4,5-d]pyrimidine-2,4-dione
—— 5-[(R)-(4-ethoxy-3-methoxyphenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O4S+
5-[(R)-(4-ethoxy-3-methoxyphenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5S)-7-(cyclobutylmethyl)-2-(2,4-dimethyl-6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O3
(5S)-7-(cyclobutylmethyl)-2-(2,4-dimethyl-6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(R)-(3,4-difluorophenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C17H18F2N4OS
5-[(R)-(3,4-difluorophenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(2-fluorophenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C16H18FN4O2S+
5-[(R)-(2-fluorophenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(2-fluorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22FN4O2S+
5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(2-fluorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(3,4-difluorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H21F2N4OS+
5-[(R)-(3,4-difluorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5-chlorofuran-2-yl)-[(3S)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]methanone —— C15H22ClNO4
(5-chlorofuran-2-yl)-[(3S)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]methanone
—— 5-cyclopropyl-3-[[(3R)-3-methyl-3-phenylpiperidin-1-yl]methyl]-1,2,4-oxadiazole —— C18H23N3O
5-cyclopropyl-3-[[(3R)-3-methyl-3-phenylpiperidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-[(R)-(4-carbamoylpiperidin-1-ium-1-yl)-(3,4-difluorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H19F2N5O2S
5-[(R)-(4-carbamoylpiperidin-1-ium-1-yl)-(3,4-difluorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(2-chlorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H24ClN5O2S+2
5-[(S)-(2-chlorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(4-carbamoylpiperidin-1-ium-1-yl)-(2-chlorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H20ClN5O2S
5-[(R)-(4-carbamoylpiperidin-1-ium-1-yl)-(2-chlorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(4-ethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H26N4O2S
5-[(S)-(4-ethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(4-ethoxy-3-methoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4O3S+
5-[(R)-(4-ethoxy-3-methoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(3,4-difluorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C17H19F2N5OS
5-[(S)-(3,4-difluorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(3,4-difluorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H21F2N4OS+
5-[(S)-(3,4-difluorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2-fluorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H21FN4OS
5-[(S)-(2-fluorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(4-carbamoylpiperidin-1-ium-1-yl)-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H23N5O3S
5-[(S)-(4-carbamoylpiperidin-1-ium-1-yl)-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— (5R)-7-(cyclobutylmethyl)-2-(2,4-dimethyl-6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O3
(5R)-7-(cyclobutylmethyl)-2-(2,4-dimethyl-6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(S)-(4-ethoxy-3-methoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H24N4O4S
5-[(S)-(4-ethoxy-3-methoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2-chlorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22ClN4OS+
5-[(R)-(2-chlorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5S)-7-(oxan-4-yl)-2-[2-(2-oxopyrrolidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H29N3O4
(5S)-7-(oxan-4-yl)-2-[2-(2-oxopyrrolidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-methyl-1-[(1-methylpyrazol-4-yl)methyl]-5-phenylpiperidin-2-one —— C17H21N3O
(5S)-5-methyl-1-[(1-methylpyrazol-4-yl)methyl]-5-phenylpiperidin-2-one
—— 5-[(S)-(3,4-dichlorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C17H19Cl2N5OS
5-[(S)-(3,4-dichlorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— (5R)-N-[2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C16H21N3O3S
(5R)-N-[2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[(S)-(4-ethoxycarbonylpiperidin-1-ium-1-yl)-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C21H26N4O3S
5-[(S)-(4-ethoxycarbonylpiperidin-1-ium-1-yl)-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— (5R)-5-methyl-1-[(1-methylpyrazol-4-yl)methyl]-5-phenylpiperidin-2-one —— C17H21N3O
(5R)-5-methyl-1-[(1-methylpyrazol-4-yl)methyl]-5-phenylpiperidin-2-one