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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5,7-dimethyl-4-[(3S)-3-(propoxymethyl)pyrrolidin-1-yl]pyrido[2,3-d]pyrimidine —— C17H24N4O
5,7-dimethyl-4-[(3S)-3-(propoxymethyl)pyrrolidin-1-yl]pyrido[2,3-d]pyrimidine
—— 5-methyl-N-[(2R)-2-piperidin-1-yl-2-pyridin-3-ylethyl]pyrimidin-2-amine —— C17H23N5
5-methyl-N-[(2R)-2-piperidin-1-yl-2-pyridin-3-ylethyl]pyrimidin-2-amine
—— (5S)-1-butyl-5-(4-chlorophenyl)-4-[hydroxy(phenyl)methylidene]pyrrolidine-2,3-dione —— C21H20ClNO3
(5S)-1-butyl-5-(4-chlorophenyl)-4-[hydroxy(phenyl)methylidene]pyrrolidine-2,3-dione
—— (5S)-1-(2-hydroxyethyl)-4-[hydroxy-(4-methoxyphenyl)methylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione —— C21H21NO6
(5S)-1-(2-hydroxyethyl)-4-[hydroxy-(4-methoxyphenyl)methylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione
—— 5-bromo-N-[3-(6-ethoxypyridazin-3-yl)phenyl]furan-2-carboxamide —— C17H14BrN3O3
5-bromo-N-[3-(6-ethoxypyridazin-3-yl)phenyl]furan-2-carboxamide
—— (5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(4-fluorophenyl)-5-phenylpyrrolidine-2,3-dione —— C23H15ClFNO3
(5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(4-fluorophenyl)-5-phenylpyrrolidine-2,3-dione
—— 5-methyl-N-[(2S)-2-piperidin-1-yl-2-pyridin-3-ylethyl]pyrimidin-2-amine —— C17H23N5
5-methyl-N-[(2S)-2-piperidin-1-yl-2-pyridin-3-ylethyl]pyrimidin-2-amine
—— (5S)-4-[hydroxy-(4-methylphenyl)methylidene]-5-phenyl-1-pyridin-2-ylpyrrolidine-2,3-dione —— C23H18N2O3
(5S)-4-[hydroxy-(4-methylphenyl)methylidene]-5-phenyl-1-pyridin-2-ylpyrrolidine-2,3-dione
—— 5,6-dimethyl-2-[(1S)-1-(1,3,4-thiadiazol-2-ylsulfanyl)ethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C12H12N4OS3
5,6-dimethyl-2-[(1S)-1-(1,3,4-thiadiazol-2-ylsulfanyl)ethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 5,6-dimethyl-N-[(1R)-1-(1,3-thiazol-2-yl)propyl]pyrimidin-4-amine —— C12H16N4S
5,6-dimethyl-N-[(1R)-1-(1,3-thiazol-2-yl)propyl]pyrimidin-4-amine
—— (5S)-7-(3-bromophenyl)-1,2,7-triazaspiro[4.4]non-1-ene-6,8-dione —— C12H10BrN3O2
(5S)-7-(3-bromophenyl)-1,2,7-triazaspiro[4.4]non-1-ene-6,8-dione
—— 5,6-dimethyl-2-[(1R)-1-[(5-methyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C16H19N5OS2
5,6-dimethyl-2-[(1R)-1-[(5-methyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5S)-2-(5-chloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H22ClN3O2
(5S)-2-(5-chloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(4-chlorophenyl)-4-[hydroxy(phenyl)methylidene]-1-(3-methylphenyl)pyrrolidine-2,3-dione —— C24H18ClNO3
(5S)-5-(4-chlorophenyl)-4-[hydroxy(phenyl)methylidene]-1-(3-methylphenyl)pyrrolidine-2,3-dione
—— (5R)-5-(4-chlorophenyl)-4-[hydroxy-(4-methoxy-2-methylphenyl)methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione —— C22H22ClNO5
(5R)-5-(4-chlorophenyl)-4-[hydroxy-(4-methoxy-2-methylphenyl)methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione
—— [(5S)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(2-pyridin-3-ylpyrimidin-5-yl)methanone —— C20H24N4O3
[(5S)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(2-pyridin-3-ylpyrimidin-5-yl)methanone
—— 5,6-dimethyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C12H12N4OS3
5,6-dimethyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5S)-4-[hydroxy(phenyl)methylidene]-5-(2-methoxyphenyl)-1-(3-methylphenyl)pyrrolidine-2,3-dione —— C25H21NO4
(5S)-4-[hydroxy(phenyl)methylidene]-5-(2-methoxyphenyl)-1-(3-methylphenyl)pyrrolidine-2,3-dione
—— (5R)-7-(4-ethylphenyl)-1,2,7-triazaspiro[4.4]non-1-ene-6,8-dione —— C14H15N3O2
(5R)-7-(4-ethylphenyl)-1,2,7-triazaspiro[4.4]non-1-ene-6,8-dione
—— (5-fluoropyridin-3-yl)-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C18H20FN7O
(5-fluoropyridin-3-yl)-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— (5S)-9-[(4-chlorophenyl)methylsulfonyl]-2-oxa-9-azaspiro[4.5]decane —— C15H20ClNO3S
(5S)-9-[(4-chlorophenyl)methylsulfonyl]-2-oxa-9-azaspiro[4.5]decane
—— (5R)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(3-hydroxypropyl)-5-(4-methoxyphenyl)pyrrolidine-2,3-dione —— C22H23NO5
(5R)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(3-hydroxypropyl)-5-(4-methoxyphenyl)pyrrolidine-2,3-dione
—— 5-[[(3S)-3-(4-fluorophenyl)oxolan-3-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine —— C17H20FN3O
5-[[(3S)-3-(4-fluorophenyl)oxolan-3-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine
—— (5S)-1-butyl-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(4-nitrophenyl)pyrrolidine-2,3-dione —— C21H19ClN2O5
(5S)-1-butyl-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(4-nitrophenyl)pyrrolidine-2,3-dione
—— (5R)-4-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-1-(3-methoxypropyl)-5-thiophen-2-ylpyrrolidine-2,3-dione —— C21H23NO5S
(5R)-4-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-1-(3-methoxypropyl)-5-thiophen-2-ylpyrrolidine-2,3-dione
—— 5,7-dimethyl-N-[1-[[(2S)-oxolan-2-yl]methyl]piperidin-4-yl]pyrido[2,3-d]pyrimidin-4-amine —— C19H27N5O
5,7-dimethyl-N-[1-[[(2S)-oxolan-2-yl]methyl]piperidin-4-yl]pyrido[2,3-d]pyrimidin-4-amine
—— (5R)-2-(6-aminopyrimidin-4-yl)-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O
(5R)-2-(6-aminopyrimidin-4-yl)-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one
—— (5-fluoropyridin-3-yl)-[(3S)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C18H20FN7O
(5-fluoropyridin-3-yl)-[(3S)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— (5R)-4-[hydroxy-(4-methoxy-2-methylphenyl)methylidene]-1-(2-methoxyethyl)-5-(2-methoxyphenyl)pyrrolidine-2,3-dione —— C23H25NO6
(5R)-4-[hydroxy-(4-methoxy-2-methylphenyl)methylidene]-1-(2-methoxyethyl)-5-(2-methoxyphenyl)pyrrolidine-2,3-dione
—— (5R)-2-(5-chloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H22ClN3O2
(5R)-2-(5-chloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[(4-chlorophenyl)methylsulfonyl]-2-oxa-9-azaspiro[4.5]decane —— C15H20ClNO3S
(5R)-9-[(4-chlorophenyl)methylsulfonyl]-2-oxa-9-azaspiro[4.5]decane
—— (5R)-5-(4-ethylphenyl)-1-(furan-2-ylmethyl)-4-[hydroxy-(4-methoxyphenyl)methylidene]pyrrolidine-2,3-dione —— C25H23NO5
(5R)-5-(4-ethylphenyl)-1-(furan-2-ylmethyl)-4-[hydroxy-(4-methoxyphenyl)methylidene]pyrrolidine-2,3-dione
—— (5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-(3-methoxypropyl)pyrrolidine-2,3-dione —— C21H19ClFNO4
(5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-(3-methoxypropyl)pyrrolidine-2,3-dione
—— 5-[(3R)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrimidin-6-one —— C18H26N6O2
5-[(3R)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrimidin-6-one
—— (5S)-1-ethyl-5-[3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C15H25N5O2
(5S)-1-ethyl-5-[3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— 5-[1-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]triazol-4-yl]pyrimidine —— C15H16N6
5-[1-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]triazol-4-yl]pyrimidine
—— (5S,10bR)-5-(3-bromophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H15BrN2OS
(5S,10bR)-5-(3-bromophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[[(3R)-3-(4-fluorophenyl)oxolan-3-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine —— C17H20FN3O
5-[[(3R)-3-(4-fluorophenyl)oxolan-3-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine
—— 5,6-dimethyl-N-[1-(2-methylsulfanylethyl)piperidin-4-yl]pyrimidin-4-amine —— C14H24N4S
5,6-dimethyl-N-[1-(2-methylsulfanylethyl)piperidin-4-yl]pyrimidin-4-amine
—— 5,7-dimethyl-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrido[2,3-d]pyrimidin-4-amine —— C20H25N5O2
5,7-dimethyl-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrido[2,3-d]pyrimidin-4-amine
—— 5-[(3S)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrimidin-6-one —— C18H26N6O2
5-[(3S)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrimidin-6-one
—— (5R)-1-ethyl-5-[3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C15H25N5O2
(5R)-1-ethyl-5-[3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— 5-ethyl-N-[[(3R)-1-propylpiperidin-3-yl]methyl]pyrimidin-2-amine —— C15H26N4
5-ethyl-N-[[(3R)-1-propylpiperidin-3-yl]methyl]pyrimidin-2-amine
—— 5-ethyl-N-[[(3S)-1-propylpiperidin-3-yl]methyl]pyrimidin-2-amine —— C15H26N4
5-ethyl-N-[[(3S)-1-propylpiperidin-3-yl]methyl]pyrimidin-2-amine
—— 5,7-dimethyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrido[2,3-d]pyrimidin-4-amine —— C20H25N5O2
5,7-dimethyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrido[2,3-d]pyrimidin-4-amine
—— 5,7-dimethyl-N-[1-[[(2R)-oxolan-2-yl]methyl]piperidin-4-yl]pyrido[2,3-d]pyrimidin-4-amine —— C19H27N5O
5,7-dimethyl-N-[1-[[(2R)-oxolan-2-yl]methyl]piperidin-4-yl]pyrido[2,3-d]pyrimidin-4-amine
—— 5-cyclopropyl-N-[(1R)-1-(2-oxo-1,3-dihydroindol-5-yl)ethyl]-1,2-oxazole-3-carboxamide —— C17H17N3O3
5-cyclopropyl-N-[(1R)-1-(2-oxo-1,3-dihydroindol-5-yl)ethyl]-1,2-oxazole-3-carboxamide
—— 5-[1-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]triazol-4-yl]pyrimidine —— C15H16N6
5-[1-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]triazol-4-yl]pyrimidine
—— (5S)-2-(6-aminopyrimidin-4-yl)-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O
(5S)-2-(6-aminopyrimidin-4-yl)-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-(morpholin-4-ylmethyl)-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]furan-3-carboxamide —— C17H22N4O3
5-(morpholin-4-ylmethyl)-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]furan-3-carboxamide