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—— [5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C19H23N5O3
[5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— (5S)-9-[(4-pyrazol-1-ylphenyl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H21N3O2
(5S)-9-[(4-pyrazol-1-ylphenyl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-2-[2-(2-ethylimidazol-1-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O3
(5S)-2-[2-(2-ethylimidazol-1-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-methoxy-1-methyl-N-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]indole-2-carboxamide —— C20H23N5O2
5-methoxy-1-methyl-N-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]indole-2-carboxamide
—— (5S)-1-cyclopentyl-5-[4-(4-methyl-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidin-2-one —— C19H29N5O2
(5S)-1-cyclopentyl-5-[4-(4-methyl-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidin-2-one
—— [5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C19H23N5O3
[5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— (5S)-5-methyl-1-[(2-methylpyridin-4-yl)methyl]-5-phenylpiperidin-2-one —— C19H22N2O
(5S)-5-methyl-1-[(2-methylpyridin-4-yl)methyl]-5-phenylpiperidin-2-one
—— 5-[(3R)-1-tert-butyl-5-oxopyrrolidine-3-carbonyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C17H23N3O3S
5-[(3R)-1-tert-butyl-5-oxopyrrolidine-3-carbonyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— 5-fluoro-4-N,4-N-dimethyl-2-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]pyrimidine-2,4-diamine —— C11H17FN4O2S
5-fluoro-4-N,4-N-dimethyl-2-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]pyrimidine-2,4-diamine
—— (5R)-1-cyclopentyl-5-[4-(4-methyl-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidin-2-one —— C19H29N5O2
(5R)-1-cyclopentyl-5-[4-(4-methyl-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidin-2-one
—— (5R)-7-(cyclopropylmethyl)-2-(3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H25FN4O2
(5R)-7-(cyclopropylmethyl)-2-(3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5,6-dimethyl-3-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one —— C16H19N3O3
5,6-dimethyl-3-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one
—— 5-(3-fluorophenyl)-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide —— C13H12FN7O
5-(3-fluorophenyl)-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
—— 5-[[(1S)-2,3-dihydro-1H-inden-1-yl]methyl]-3-pyridazin-3-yl-1,2,4-oxadiazole —— C16H14N4O
5-[[(1S)-2,3-dihydro-1H-inden-1-yl]methyl]-3-pyridazin-3-yl-1,2,4-oxadiazole
—— 5-methoxy-1-methyl-N-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]indole-2-carboxamide —— C20H23N5O2
5-methoxy-1-methyl-N-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]indole-2-carboxamide
—— (5S)-2-[4-(morpholine-4-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O3
(5S)-2-[4-(morpholine-4-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-propyl-2-pyridin-3-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one —— C16H23N3O3S
(5R)-7-propyl-2-pyridin-3-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-methoxyethyl)-2-[3-(1,2,4-triazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H25N5O3
(5R)-7-(2-methoxyethyl)-2-[3-(1,2,4-triazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-methyl-2-[2-(5-oxo-2-phenylcyclopenten-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H26N2O3
(5R)-7-methyl-2-[2-(5-oxo-2-phenylcyclopenten-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propyl-2-pyridin-3-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one —— C16H23N3O3S
(5S)-7-propyl-2-pyridin-3-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-cyclopentyl-2-[6-(methoxymethyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5S)-7-cyclopentyl-2-[6-(methoxymethyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(3-fluorophenyl)-N-[(1R)-1-(2H-tetrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide —— C13H12FN7O
5-(3-fluorophenyl)-N-[(1R)-1-(2H-tetrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
—— (5R)-1-cyclopentyl-5-(3-phenylmethoxyazetidine-1-carbonyl)piperidin-2-one —— C21H28N2O3
(5R)-1-cyclopentyl-5-(3-phenylmethoxyazetidine-1-carbonyl)piperidin-2-one
—— [5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(2R)-2-(pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methanone —— C18H21N5O2S
[5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(2R)-2-(pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methanone
—— (5R)-7-methyl-2-[4-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O3
(5R)-7-methyl-2-[4-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[2-(4-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H25N3O2
(5S)-9-[2-(4-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-7-ethyl-2-[2-(2-oxopyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H23N3O3
(5R)-7-ethyl-2-[2-(2-oxopyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— [5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-(pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methanone —— C18H21N5O2S
[5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-(pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methanone
—— (5R)-2-[2-(2-ethylimidazol-1-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O3
(5R)-2-[2-(2-ethylimidazol-1-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-[2-(2-oxopyrimidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O3
(5S)-7-(cyclopropylmethyl)-2-[2-(2-oxopyrimidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[(4-pyrazol-1-ylphenyl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H21N3O2
(5R)-9-[(4-pyrazol-1-ylphenyl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-(4-methylpiperazin-1-yl)-2-nitro-N-[(1S)-1-phenylethyl]aniline —— C19H24N4O2
5-(4-methylpiperazin-1-yl)-2-nitro-N-[(1S)-1-phenylethyl]aniline
—— (5S)-4-[(4-butoxy-3-methylphenyl)-hydroxymethylidene]-1-(2-methoxyethyl)-5-pyridin-4-ylpyrrolidine-2,3-dione —— C24H28N2O5
(5S)-4-[(4-butoxy-3-methylphenyl)-hydroxymethylidene]-1-(2-methoxyethyl)-5-pyridin-4-ylpyrrolidine-2,3-dione
—— (5R)-7-methyl-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H22N4O2
(5R)-7-methyl-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-methoxy-1-methyl-N-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]indole-2-carboxamide —— C20H23N3O2
5-methoxy-1-methyl-N-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]indole-2-carboxamide
—— (5R)-7-(cyclopropylmethyl)-2-[2-(2-oxopyrimidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O3
(5R)-7-(cyclopropylmethyl)-2-[2-(2-oxopyrimidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-methoxy-1-methyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]indole-2-carboxamide —— C20H23N3O2
5-methoxy-1-methyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]indole-2-carboxamide
—— (5S)-2-(5-methoxyfuran-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C15H20N2O4
(5S)-2-(5-methoxyfuran-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(4-methoxypyrimidin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O2
(5R)-2-(4-methoxypyrimidin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(4-methoxypyrimidin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O2
(5S)-2-(4-methoxypyrimidin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-1-carbamoylpiperidine-3-carbonyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C15H20N4O3S
5-[(3R)-1-carbamoylpiperidine-3-carbonyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— (5R,10bS)-2-(4-chlorophenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-1H-indole]-2'-one —— C23H16ClN3O2
(5R,10bS)-2-(4-chlorophenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-1H-indole]-2'-one
—— (5R)-5-(diethylsulfamoylamino)-2-phenyl-5,6,7,8-tetrahydroquinazoline —— C18H24N4O2S
(5R)-5-(diethylsulfamoylamino)-2-phenyl-5,6,7,8-tetrahydroquinazoline
—— (5S)-7-cyclopentyl-2-morpholin-4-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one —— C17H29N3O4S
(5S)-7-cyclopentyl-2-morpholin-4-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(5-methoxyfuran-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C15H20N2O4
(5R)-2-(5-methoxyfuran-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24N4O3
(5S)-7-(cyclobutylmethyl)-2-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[3-(3,5-dimethylpyrazol-1-yl)propyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H30N4O2
(5S)-2-[3-(3,5-dimethylpyrazol-1-yl)propyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(6-fluoro-2-oxo-1H-quinoline-4-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C21H24FN3O3
(5S)-2-(6-fluoro-2-oxo-1H-quinoline-4-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(R)-[(2R,6S)-2,6-dimethylmorpholin-4-ium-4-yl]-(4-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O2S+
5-[(R)-[(2R,6S)-2,6-dimethylmorpholin-4-ium-4-yl]-(4-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(1S)-1-[4-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine —— C16H15N7OS2
5-[(1S)-1-[4-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine