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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-methyl-N-[[(2S)-8-propan-2-yl-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl]-1,3,4-oxadiazol-2-amine —— C15H26N4O2
5-methyl-N-[[(2S)-8-propan-2-yl-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl]-1,3,4-oxadiazol-2-amine
—— (5S)-9-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-2-oxa-9-azaspiro[4.5]decane —— C16H21N3O2
(5S)-9-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-2-oxa-9-azaspiro[4.5]decane
—— (5R)-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-2-oxa-9-azaspiro[4.5]decane —— C16H19N3O2
(5R)-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-2-oxa-9-azaspiro[4.5]decane
—— 5,7-dimethyl-N-[[(2R)-1-methylpiperidin-2-yl]methyl]pyrido[2,3-d]pyrimidin-4-amine —— C16H23N5
5,7-dimethyl-N-[[(2R)-1-methylpiperidin-2-yl]methyl]pyrido[2,3-d]pyrimidin-4-amine
—— 5-methyl-N-[[(4S)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]pyrazine-2-carboxamide —— C17H19N3O2
5-methyl-N-[[(4S)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]pyrazine-2-carboxamide
—— (5R)-7-(cyclobutylmethyl)-2-pyridin-4-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O
(5R)-7-(cyclobutylmethyl)-2-pyridin-4-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R,10bR)-1',5'-dimethyl-2-(4-methylphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one —— C26H23N3O2
(5R,10bR)-1',5'-dimethyl-2-(4-methylphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one
—— 5-ethyl-4-N-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]pyrimidine-2,4-diamine —— C15H21N7
5-ethyl-4-N-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]pyrimidine-2,4-diamine
—— 5-[(3S)-1-(2-ethylbutanoyl)piperidin-3-yl]-3-[(4-fluorophenyl)methyl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C22H27FN6O2
5-[(3S)-1-(2-ethylbutanoyl)piperidin-3-yl]-3-[(4-fluorophenyl)methyl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-methyl-N-[[(4R)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]pyrazine-2-carboxamide —— C17H19N3O2
5-methyl-N-[[(4R)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]pyrazine-2-carboxamide
—— (5Z)-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-5-(thiophen-2-ylmethylidene)-1,3-thiazol-4-one —— C14H16N2O2S2
(5Z)-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-5-(thiophen-2-ylmethylidene)-1,3-thiazol-4-one
—— (5S)-2-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4O3S
(5S)-2-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(4-Methylpyrazol-1-yl)methyl]furan-2-carboxylate —— C10H9N2O3-
5-[(4-Methylpyrazol-1-yl)methyl]furan-2-carboxylate
—— 5-[(3S)-3-(2-chlorophenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-5-oxopentanoate —— C21H20ClN2O3-
5-[(3S)-3-(2-chlorophenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-5-oxopentanoate
—— (5S,10bR)-5-(4-chlorophenyl)-9-methoxy-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H19ClN2O2
(5S,10bR)-5-(4-chlorophenyl)-9-methoxy-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R)-7-cyclopentyl-2-[2-[methyl(pyridin-2-ylmethyl)amino]acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H32N4O2
(5R)-7-cyclopentyl-2-[2-[methyl(pyridin-2-ylmethyl)amino]acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— [5-(3-Amino-2-carbamoyl-3-oxopropyl)-2-ethoxyphenyl]methyl-dimethylazanium —— C15H24N3O3+
[5-(3-Amino-2-carbamoyl-3-oxopropyl)-2-ethoxyphenyl]methyl-dimethylazanium
—— 5-ethyl-4-N-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]pyrimidine-2,4-diamine —— C15H21N7
5-ethyl-4-N-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]pyrimidine-2,4-diamine
—— (5E)-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-[(3-methoxy-4-pentoxyphenyl)methylidene]-1,3-thiazol-4-one —— C22H30N2O4S
(5E)-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-[(3-methoxy-4-pentoxyphenyl)methylidene]-1,3-thiazol-4-one
—— 5-(morpholin-4-ylmethyl)-N-[(1S)-1-phenyl-2-pyrazol-1-ylethyl]furan-3-carboxamide —— C21H24N4O3
5-(morpholin-4-ylmethyl)-N-[(1S)-1-phenyl-2-pyrazol-1-ylethyl]furan-3-carboxamide
—— 5-Hydrazinyl-11-methyl-4-(4-methylphenyl)-8-thia-4,6-diaza-11-azoniatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one —— C17H20N5OS+
5-Hydrazinyl-11-methyl-4-(4-methylphenyl)-8-thia-4,6-diaza-11-azoniatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
—— 5-(2-methoxyphenyl)-7-(trifluoromethyl)-2,3-dihydro-1H-1,4-diazepin-1-ium —— C13H14F3N2O+
5-(2-methoxyphenyl)-7-(trifluoromethyl)-2,3-dihydro-1H-1,4-diazepin-1-ium
—— (5S,10bS)-9-methoxy-2-phenyl-5-(4-propan-2-ylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C26H26N2O2
(5S,10bS)-9-methoxy-2-phenyl-5-(4-propan-2-ylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R)-7-(2-methoxyethyl)-2-(6-methylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O2
(5R)-7-(2-methoxyethyl)-2-(6-methylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-(6-methyl-2-phenylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C20H25N3O2
(5S)-9-(6-methyl-2-phenylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-[(3R)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one —— C20H29N5O2
5-[(3R)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one
—— (5S)-7-(cyclobutylmethyl)-2-pyridin-4-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O
(5S)-7-(cyclobutylmethyl)-2-pyridin-4-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5,7-dimethyl-N-[[(2S)-1-methylpiperidin-2-yl]methyl]pyrido[2,3-d]pyrimidin-4-amine —— C16H23N5
5,7-dimethyl-N-[[(2S)-1-methylpiperidin-2-yl]methyl]pyrido[2,3-d]pyrimidin-4-amine
—— (5S)-7-(2-methoxyethyl)-2-(6-methylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O2
(5S)-7-(2-methoxyethyl)-2-(6-methylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(morpholin-4-ylmethyl)-N-[(1R)-1-phenyl-2-pyrazol-1-ylethyl]furan-3-carboxamide —— C21H24N4O3
5-(morpholin-4-ylmethyl)-N-[(1R)-1-phenyl-2-pyrazol-1-ylethyl]furan-3-carboxamide
—— (5R)-9-[(8-methoxyquinolin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C20H26N2O3
(5R)-9-[(8-methoxyquinolin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-[(3S)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one —— C20H29N5O2
5-[(3S)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one
—— (5R)-2-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4O3S
(5R)-2-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[(8-methoxyquinolin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C20H26N2O3
(5S)-9-[(8-methoxyquinolin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-9-(6-methyl-2-phenylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C20H25N3O2
(5R)-9-(6-methyl-2-phenylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5S)-7-cyclopentyl-2-[2-[methyl(pyridin-2-ylmethyl)amino]acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H32N4O2
(5S)-7-cyclopentyl-2-[2-[methyl(pyridin-2-ylmethyl)amino]acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(3-morpholin-4-ium-4-ylpropylamino)-2-[(E)-2-thiophen-2-ylethenyl]-1,3-oxazole-4-carbonitrile —— C17H21N4O2S+
5-(3-morpholin-4-ium-4-ylpropylamino)-2-[(E)-2-thiophen-2-ylethenyl]-1,3-oxazole-4-carbonitrile
—— 5,6-dimethyl-2-[2-[4-[(1R)-1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl]-2-oxoethyl]pyridazin-3-one —— C20H33N5O2
5,6-dimethyl-2-[2-[4-[(1R)-1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl]-2-oxoethyl]pyridazin-3-one
—— 5-[1-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]triazol-4-yl]pyrimidine —— C16H14N8
5-[1-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]triazol-4-yl]pyrimidine
—— (5S)-9-[(3-methylsulfonylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-2-oxa-9-azaspiro[4.5]decane —— C16H22N4O3S
(5S)-9-[(3-methylsulfonylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-2-oxa-9-azaspiro[4.5]decane
—— (5E)-3-[4-[(2R)-2-ethylpiperidin-1-yl]-4-oxobutyl]-2-sulfanylidene-5-(thiophen-2-ylmethylidene)-1,3-thiazolidin-4-one —— C19H24N2O2S3
(5E)-3-[4-[(2R)-2-ethylpiperidin-1-yl]-4-oxobutyl]-2-sulfanylidene-5-(thiophen-2-ylmethylidene)-1,3-thiazolidin-4-one
—— 5-ethyl-4-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-2-methylpyrimidine —— C19H26N8
5-ethyl-4-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-2-methylpyrimidine
—— 5-[1-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]triazol-4-yl]pyrimidine —— C16H14N8
5-[1-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]triazol-4-yl]pyrimidine
—— (5R)-9-[(3-methylsulfonylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-2-oxa-9-azaspiro[4.5]decane —— C16H22N4O3S
(5R)-9-[(3-methylsulfonylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-2-oxa-9-azaspiro[4.5]decane
—— 5-[1-[(2S)-2-methyl-3-[3-methyl-5-(trifluoromethyl)pyrazol-1-yl]propyl]triazol-4-yl]pyrimidine —— C15H16F3N7
5-[1-[(2S)-2-methyl-3-[3-methyl-5-(trifluoromethyl)pyrazol-1-yl]propyl]triazol-4-yl]pyrimidine
—— 5,6-dimethyl-2-[2-[4-[(1S)-1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl]-2-oxoethyl]pyridazin-3-one —— C20H33N5O2
5,6-dimethyl-2-[2-[4-[(1S)-1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl]-2-oxoethyl]pyridazin-3-one
—— 5-ethyl-4-[(3S)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-2-methylpyrimidine —— C19H26N8
5-ethyl-4-[(3S)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-2-methylpyrimidine
—— 5-[1-[(2R)-2-methyl-3-[3-methyl-5-(trifluoromethyl)pyrazol-1-yl]propyl]triazol-4-yl]pyrimidine —— C15H16F3N7
5-[1-[(2R)-2-methyl-3-[3-methyl-5-(trifluoromethyl)pyrazol-1-yl]propyl]triazol-4-yl]pyrimidine
—— (5S)-5-(1,3-benzodioxol-5-yl)-1-hexyl-4-[hydroxy(phenyl)methylidene]pyrrolidine-2,3-dione —— C24H25NO5
(5S)-5-(1,3-benzodioxol-5-yl)-1-hexyl-4-[hydroxy(phenyl)methylidene]pyrrolidine-2,3-dione
—— (5S)-1-hexyl-4-[hydroxy-(4-methylphenyl)methylidene]-5-(4-methylphenyl)pyrrolidine-2,3-dione —— C25H29NO3
(5S)-1-hexyl-4-[hydroxy-(4-methylphenyl)methylidene]-5-(4-methylphenyl)pyrrolidine-2,3-dione