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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-2-[[6-(dimethylamino)pyridin-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O
(5S)-2-[[6-(dimethylamino)pyridin-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[(3-morpholin-4-ylphenyl)methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C22H33N3O2
(5S)-2-[(3-morpholin-4-ylphenyl)methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[6-(dimethylamino)pyridine-3-carbonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5S)-2-[6-(dimethylamino)pyridine-3-carbonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S,7S)-5-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H23F3N4O2
(5S,7S)-5-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R)-2-[(3-morpholin-4-ylphenyl)methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C22H33N3O2
(5R)-2-[(3-morpholin-4-ylphenyl)methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-hydroxyethyl)-2-[4-(1,3-oxazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H23N3O4
(5S)-7-(2-hydroxyethyl)-2-[4-(1,3-oxazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-[(5-methylthiophen-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H26N2OS
(5S)-7-(cyclopropylmethyl)-2-[(5-methylthiophen-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O3S
(5R)-2-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[4-(4-chlorophenyl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H23ClN2O2
(5S)-2-[4-(4-chlorophenyl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O3S
(5S)-2-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-chloro-6-[(5S)-7-ethyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carboxylic acid —— C16H20ClN3O3
5-chloro-6-[(5S)-7-ethyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carboxylic acid
—— (5R)-2-(1-ethyl-2,5-dimethylpyrrole-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H31N3O3
(5R)-2-(1-ethyl-2,5-dimethylpyrrole-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(3-methoxyphenyl)-3-[[4-[(3R)-oxolan-3-yl]triazol-1-yl]methyl]-1,2-oxazole —— C17H18N4O3
5-(3-methoxyphenyl)-3-[[4-[(3R)-oxolan-3-yl]triazol-1-yl]methyl]-1,2-oxazole
—— (5R)-7-(cyclopropylmethyl)-2-[(2,4-dimethoxy-3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H32N2O3
(5R)-7-(cyclopropylmethyl)-2-[(2,4-dimethoxy-3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[[6-(dimethylamino)pyridin-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O
(5R)-2-[[6-(dimethylamino)pyridin-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-hydroxyethyl)-2-(2-methylsulfanylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C15H22N4O2S
(5R)-7-(2-hydroxyethyl)-2-(2-methylsulfanylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-hydroxyethyl)-2-([1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H22N6O2
(5R)-7-(2-hydroxyethyl)-2-([1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-hydroxyethyl)-2-([1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H22N6O2
(5S)-7-(2-hydroxyethyl)-2-([1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R,7S)-5-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H23F3N4O2
(5R,7S)-5-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(3-methoxyphenyl)-3-[[4-[(3S)-oxolan-3-yl]triazol-1-yl]methyl]-1,2-oxazole —— C17H18N4O3
5-(3-methoxyphenyl)-3-[[4-[(3S)-oxolan-3-yl]triazol-1-yl]methyl]-1,2-oxazole
—— (5S,8R,9R,10S,13R,14R)-10,13-dimethyl-1,2,4,5,6,7,8,9,11,12,14,15-dodecahydrocyclopenta[a]phenanthren-3-one —— C19H28O
(5S,8R,9R,10S,13R,14R)-10,13-dimethyl-1,2,4,5,6,7,8,9,11,12,14,15-dodecahydrocyclopenta[a]phenanthren-3-one
—— (5R)-2-[(2-aminopyridin-3-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O2
(5R)-2-[(2-aminopyridin-3-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-cyclohexyl-N-[(1S)-1-(5-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazole-4-carboxamide —— C17H25N5O
5-cyclohexyl-N-[(1S)-1-(5-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
—— 5-cyclohexyl-N-[(1R)-1-(5-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazole-4-carboxamide —— C17H25N5O
5-cyclohexyl-N-[(1R)-1-(5-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
—— (5S)-5-methyl-5-(4-methylpent-3-enyl)-1-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)piperidin-2-one —— C19H26N4O
(5S)-5-methyl-5-(4-methylpent-3-enyl)-1-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)piperidin-2-one
—— (5S)-7-(2-methoxyethyl)-2-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H32N4O3
(5S)-7-(2-methoxyethyl)-2-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(4-hydroxyphenyl)-4-[hydroxy(phenyl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C23H24N2O5
(5S)-5-(4-hydroxyphenyl)-4-[hydroxy(phenyl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— (5R)-7-(2-hydroxyethyl)-2-[4-(1,3-oxazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H23N3O4
(5R)-7-(2-hydroxyethyl)-2-[4-(1,3-oxazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-methyl-N-[1-[[(2S)-oxolan-2-yl]methyl]piperidin-4-yl]-1-propylpyrazole-4-carboxamide —— C18H30N4O2
5-methyl-N-[1-[[(2S)-oxolan-2-yl]methyl]piperidin-4-yl]-1-propylpyrazole-4-carboxamide
—— (5-Acetyl-2-methoxyphenyl)methyl 4-(2,5-dioxopyrrolidin-1-yl)benzoate —— C21H19NO6
(5-Acetyl-2-methoxyphenyl)methyl 4-(2,5-dioxopyrrolidin-1-yl)benzoate
—— (5S)-7-(cyclobutylmethyl)-2-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H25N5O
(5S)-7-(cyclobutylmethyl)-2-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(morpholine-4-carbonyl)-1-(3-phenylpropyl)piperidin-2-one —— C19H26N2O3
(5R)-5-(morpholine-4-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
—— (5R)-1-ethyl-5-[4-(1-methylbenzimidazol-2-yl)piperidine-1-carbonyl]piperidin-2-one —— C21H28N4O2
(5R)-1-ethyl-5-[4-(1-methylbenzimidazol-2-yl)piperidine-1-carbonyl]piperidin-2-one
—— (5S)-2-[(2-aminopyridin-3-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O2
(5S)-2-[(2-aminopyridin-3-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(methoxymethyl)thiophen-2-yl]-[(2R)-2-(2-pyrrolidin-1-ylethyl)piperidin-1-yl]methanone —— C18H28N2O2S
[5-(methoxymethyl)thiophen-2-yl]-[(2R)-2-(2-pyrrolidin-1-ylethyl)piperidin-1-yl]methanone
—— 5-[(3S)-3-aminopyrrolidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]-1H-pyrimidin-6-one —— C16H16Cl2N4O2
5-[(3S)-3-aminopyrrolidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]-1H-pyrimidin-6-one
—— 5-[(5S)-7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridine-2-carbonitrile —— C21H26N4O2
5-[(5S)-7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridine-2-carbonitrile
—— (5-chloro-2-methoxyphenyl)-[(3S)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]methanone —— C18H26ClNO4
(5-chloro-2-methoxyphenyl)-[(3S)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]methanone
—— 5-methyl-N-[1-[[(2R)-oxolan-2-yl]methyl]piperidin-4-yl]-1-propylpyrazole-4-carboxamide —— C18H30N4O2
5-methyl-N-[1-[[(2R)-oxolan-2-yl]methyl]piperidin-4-yl]-1-propylpyrazole-4-carboxamide
—— [5-[(2R)-oxolan-2-yl]thiophen-2-yl]-[4-(1,3-thiazol-2-yl)piperazin-1-yl]methanone —— C16H19N3O2S2
[5-[(2R)-oxolan-2-yl]thiophen-2-yl]-[4-(1,3-thiazol-2-yl)piperazin-1-yl]methanone
—— (5R)-N-(imidazo[1,2-a]pyrimidin-2-ylmethyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H18N4OS
(5R)-N-(imidazo[1,2-a]pyrimidin-2-ylmethyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-7-(3-methoxypropyl)-2-thieno[3,2-d]pyrimidin-4-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O2S
(5S)-7-(3-methoxypropyl)-2-thieno[3,2-d]pyrimidin-4-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5-chloro-2-methoxyphenyl)-[(3R)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]methanone —— C18H26ClNO4
(5-chloro-2-methoxyphenyl)-[(3R)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]methanone
—— 5-[(5R)-7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridine-2-carbonitrile —— C21H26N4O2
5-[(5R)-7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridine-2-carbonitrile
—— (5S)-1-ethyl-5-[4-(1-methylbenzimidazol-2-yl)piperidine-1-carbonyl]piperidin-2-one —— C21H28N4O2
(5S)-1-ethyl-5-[4-(1-methylbenzimidazol-2-yl)piperidine-1-carbonyl]piperidin-2-one
—— (5R)-7-(2-methoxyethyl)-2-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H32N4O3
(5R)-7-(2-methoxyethyl)-2-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one —— C17H27N7O
(5S)-2-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-5-methyl-5-phenylpiperidin-2-one —— C19H25N3O
(5S)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-5-methyl-5-phenylpiperidin-2-one
—— (5R)-5-methyl-5-(4-methylpent-3-enyl)-1-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)piperidin-2-one —— C19H26N4O
(5R)-5-methyl-5-(4-methylpent-3-enyl)-1-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)piperidin-2-one
—— (5R)-7-(cyclobutylmethyl)-2-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H25N5O
(5R)-7-(cyclobutylmethyl)-2-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one