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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-5-tert-butyl-N-[(1S)-1-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C21H30N4OS
(5R)-5-tert-butyl-N-[(1S)-1-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-5-tert-butyl-N-[(1R)-1-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C21H30N4OS
(5R)-5-tert-butyl-N-[(1R)-1-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5-Chloro-2,3-dihydro-1,4-benzodioxin-7-yl)methyl 3-(trifluoromethyl)benzoate —— C17H12ClF3O4
(5-Chloro-2,3-dihydro-1,4-benzodioxin-7-yl)methyl 3-(trifluoromethyl)benzoate
—— (5S,10bS)-2-(1,3-benzodioxol-5-yl)-5-(4-chlorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17ClN2O3
(5S,10bS)-2-(1,3-benzodioxol-5-yl)-5-(4-chlorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S)-5-tert-butyl-N-[(1S)-1-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C21H30N4OS
(5S)-5-tert-butyl-N-[(1S)-1-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-5-tert-butyl-N-[(1R)-1-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C21H30N4OS
(5S)-5-tert-butyl-N-[(1R)-1-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-1,3-dihydrobenzimidazol-2-one —— C15H16N4O3S
5-[[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-1,3-dihydrobenzimidazol-2-one
—— 5-(4-Ethylpiperazin-1-yl)sulfonyl-1,3-dihydrobenzimidazol-2-one —— C13H18N4O3S
5-(4-Ethylpiperazin-1-yl)sulfonyl-1,3-dihydrobenzimidazol-2-one
—— (5R)-N-[(1-benzylimidazol-2-yl)methyl]-9-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C22H25N3O
(5R)-N-[(1-benzylimidazol-2-yl)methyl]-9-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— 5-[(1-butyltetrazol-5-yl)methylsulfanyl]-N-(3-methylphenyl)-1,3,4-thiadiazol-2-amine —— C15H19N7S2
5-[(1-butyltetrazol-5-yl)methylsulfanyl]-N-(3-methylphenyl)-1,3,4-thiadiazol-2-amine
—— (5S,7R)-3-chloro-N-[2-[2-(4-ethylbenzoyl)hydrazinyl]-2-oxoethyl]adamantane-1-carboxamide —— C22H28ClN3O3
(5S,7R)-3-chloro-N-[2-[2-(4-ethylbenzoyl)hydrazinyl]-2-oxoethyl]adamantane-1-carboxamide
—— 5-(3-Amino-5-methyl-4-nitrothiophen-2-yl)pentanoate —— C10H13N2O4S-
5-(3-Amino-5-methyl-4-nitrothiophen-2-yl)pentanoate
—— (5S)-N'-(3-chlorobenzoyl)-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide —— C18H19ClN2O2S
(5S)-N'-(3-chlorobenzoyl)-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide
—— 5-[(E)-2-(4-methoxyphenyl)ethenyl]-N,N-dimethyl-3-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-1,2,4-triazole-2-sulfonamide —— C19H20N4O4S
5-[(E)-2-(4-methoxyphenyl)ethenyl]-N,N-dimethyl-3-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-1,2,4-triazole-2-sulfonamide
—— 5-bromo-N-[2-oxo-2-(2,2,2-trifluoroethylamino)ethyl]furan-2-carboxamide —— C9H8BrF3N2O3
5-bromo-N-[2-oxo-2-(2,2,2-trifluoroethylamino)ethyl]furan-2-carboxamide
—— (5S)-5-[[4-[(4-methylphenyl)diazenyl]anilino]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C17H16N4OS2
(5S)-5-[[4-[(4-methylphenyl)diazenyl]anilino]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S,7R)-N-[2-(2-benzoylhydrazinyl)-2-oxoethyl]-3-chloroadamantane-1-carboxamide —— C20H24ClN3O3
(5S,7R)-N-[2-(2-benzoylhydrazinyl)-2-oxoethyl]-3-chloroadamantane-1-carboxamide
—— (5S)-N-[(1-benzylimidazol-2-yl)methyl]-8-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C22H25N3O
(5S)-N-[(1-benzylimidazol-2-yl)methyl]-8-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— (5S)-N-[(1-benzylimidazol-2-yl)methyl]-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C22H25N3O
(5S)-N-[(1-benzylimidazol-2-yl)methyl]-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— (5S)-N-[(1-benzylimidazol-2-yl)methyl]-9-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C22H25N3O
(5S)-N-[(1-benzylimidazol-2-yl)methyl]-9-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— (5S)-N'-[2-(2-fluorophenoxy)acetyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide —— C18H19FN2O3S
(5S)-N'-[2-(2-fluorophenoxy)acetyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbohydrazide
—— (5S,7R)-3-chloro-N-[2-[2-(2,5-dimethylfuran-3-carbonyl)hydrazinyl]-2-oxoethyl]adamantane-1-carboxamide —— C20H26ClN3O4
(5S,7R)-3-chloro-N-[2-[2-(2,5-dimethylfuran-3-carbonyl)hydrazinyl]-2-oxoethyl]adamantane-1-carboxamide
—— (5S)-5-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C15H17NOS2
(5S)-5-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-N-[(1-benzylimidazol-2-yl)methyl]-8-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C22H25N3O
(5R)-N-[(1-benzylimidazol-2-yl)methyl]-8-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— 5-[2-(1,3-Dioxolan-2-yl)ethyl]-1-(2-hydroxyethyl)pyrazolo[3,4-d]pyrimidin-4-one —— C12H16N4O4
5-[2-(1,3-Dioxolan-2-yl)ethyl]-1-(2-hydroxyethyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 5-[2-(Diethylamino)ethyl]-1-(2-hydroxyethyl)pyrazolo[3,4-d]pyrimidin-4-one —— C13H21N5O2
5-[2-(Diethylamino)ethyl]-1-(2-hydroxyethyl)pyrazolo[3,4-d]pyrimidin-4-one
—— (5R)-N-[(1-benzylimidazol-2-yl)methyl]-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C22H25N3O
(5R)-N-[(1-benzylimidazol-2-yl)methyl]-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— 5-(2-(azepan-1-yl)-2-oxoethyl)-1-(2-hydroxyethyl)-1H-pyrazolo[3,4-d]pyrimidin-4(5H)-one —— C15H21N5O3
5-(2-(azepan-1-yl)-2-oxoethyl)-1-(2-hydroxyethyl)-1H-pyrazolo[3,4-d]pyrimidin-4(5H)-one
—— 5-Methyl-7-[4-(2-methylprop-2-enyl)piperazin-4-ium-1-yl]-3-phenyl-6-prop-2-enylpyrazolo[1,5-a]pyrimidine —— C24H30N5+
5-Methyl-7-[4-(2-methylprop-2-enyl)piperazin-4-ium-1-yl]-3-phenyl-6-prop-2-enylpyrazolo[1,5-a]pyrimidine
—— (5-methyl-1,2-oxazol-3-yl)methyl 1H-indazole-3-carboxylate —— C13H11N3O3
(5-methyl-1,2-oxazol-3-yl)methyl 1H-indazole-3-carboxylate
—— (5S)-N-[3-[[(3S)-oxolan-3-yl]methoxy]propyl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine —— C18H27NO2S
(5S)-N-[3-[[(3S)-oxolan-3-yl]methoxy]propyl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine
—— (5S)-N-[3-[[(3R)-oxolan-3-yl]methoxy]propyl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine —— C18H27NO2S
(5S)-N-[3-[[(3R)-oxolan-3-yl]methoxy]propyl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine
—— (5R)-N-[3-[[(3R)-oxolan-3-yl]methoxy]propyl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine —— C18H27NO2S
(5R)-N-[3-[[(3R)-oxolan-3-yl]methoxy]propyl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine
—— (5R)-5-[[(1R)-1-(2,3-dichlorophenyl)ethyl]amino]-1-methylpiperidin-2-one —— C14H18Cl2N2O
(5R)-5-[[(1R)-1-(2,3-dichlorophenyl)ethyl]amino]-1-methylpiperidin-2-one
—— (5R)-5-[[(1S)-1-(5-chloro-2-methoxyphenyl)ethyl]amino]-1-methylpiperidin-2-one —— C15H21ClN2O2
(5R)-5-[[(1S)-1-(5-chloro-2-methoxyphenyl)ethyl]amino]-1-methylpiperidin-2-one
—— (5S)-5-[[(7S)-2-ethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-yl]amino]-1-methylpiperidin-2-one —— C15H23N3OS
(5S)-5-[[(7S)-2-ethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-yl]amino]-1-methylpiperidin-2-one
—— (5S)-1-methyl-5-[[(5R)-1,2,4,5-tetrahydro-3-benzothiepin-5-yl]amino]piperidin-2-one —— C16H22N2OS
(5S)-1-methyl-5-[[(5R)-1,2,4,5-tetrahydro-3-benzothiepin-5-yl]amino]piperidin-2-one
—— (5R)-1-methyl-5-[[(7R)-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-yl]amino]piperidin-2-one —— C14H21N3OS
(5R)-1-methyl-5-[[(7R)-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-yl]amino]piperidin-2-one
—— (5S)-5-[[(1S)-1-[2-(difluoromethoxy)-4-fluorophenyl]ethyl]amino]-1-methylpiperidin-2-one —— C15H19F3N2O2
(5S)-5-[[(1S)-1-[2-(difluoromethoxy)-4-fluorophenyl]ethyl]amino]-1-methylpiperidin-2-one
—— (5S)-5-[[(1R)-1-[2-(difluoromethoxy)-4-fluorophenyl]ethyl]amino]-1-methylpiperidin-2-one —— C15H19F3N2O2
(5S)-5-[[(1R)-1-[2-(difluoromethoxy)-4-fluorophenyl]ethyl]amino]-1-methylpiperidin-2-one
—— (5R)-1-methyl-5-[[(2S,4R)-2-methyl-3,4-dihydro-2H-thiochromen-4-yl]amino]piperidin-2-one —— C16H22N2OS
(5R)-1-methyl-5-[[(2S,4R)-2-methyl-3,4-dihydro-2H-thiochromen-4-yl]amino]piperidin-2-one
—— (5R)-5-[[(3S,5R)-1,5-dimethylpyrrolidin-3-yl]amino]-1-methylpiperidin-2-one —— C12H23N3O
(5R)-5-[[(3S,5R)-1,5-dimethylpyrrolidin-3-yl]amino]-1-methylpiperidin-2-one
—— (5R)-5-[[(7R)-2-ethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-yl]amino]-1-methylpiperidin-2-one —— C15H23N3OS
(5R)-5-[[(7R)-2-ethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-yl]amino]-1-methylpiperidin-2-one
—— (5S)-5-[[(1R)-1-[4-methoxy-3-(pyrazol-1-ylmethyl)phenyl]ethyl]amino]-1-methylpiperidin-2-one —— C19H26N4O2
(5S)-5-[[(1R)-1-[4-methoxy-3-(pyrazol-1-ylmethyl)phenyl]ethyl]amino]-1-methylpiperidin-2-one
—— (5R)-5-[[(1R)-1-[4-methoxy-3-(pyrazol-1-ylmethyl)phenyl]ethyl]amino]-1-methylpiperidin-2-one —— C19H26N4O2
(5R)-5-[[(1R)-1-[4-methoxy-3-(pyrazol-1-ylmethyl)phenyl]ethyl]amino]-1-methylpiperidin-2-one
—— (5R)-1-methyl-5-[[(5R)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one —— C16H22N2O2
(5R)-1-methyl-5-[[(5R)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one
—— (5S)-1-methyl-5-[[(4S,6S)-6-methyl-5,6-dihydro-4H-thieno[2,3-b]thiopyran-4-yl]amino]piperidin-2-one —— C14H20N2OS2
(5S)-1-methyl-5-[[(4S,6S)-6-methyl-5,6-dihydro-4H-thieno[2,3-b]thiopyran-4-yl]amino]piperidin-2-one
—— (5R)-5-[[(1S)-1-[2-(difluoromethoxy)-4-fluorophenyl]ethyl]amino]-1-methylpiperidin-2-one —— C15H19F3N2O2
(5R)-5-[[(1S)-1-[2-(difluoromethoxy)-4-fluorophenyl]ethyl]amino]-1-methylpiperidin-2-one
—— (5S)-5-[[(1S)-1-[4-methoxy-3-(pyrazol-1-ylmethyl)phenyl]ethyl]amino]-1-methylpiperidin-2-one —— C19H26N4O2
(5S)-5-[[(1S)-1-[4-methoxy-3-(pyrazol-1-ylmethyl)phenyl]ethyl]amino]-1-methylpiperidin-2-one
—— (5R)-5-[[(3S,5S)-1,5-dimethylpyrrolidin-3-yl]amino]-1-methylpiperidin-2-one —— C12H23N3O
(5R)-5-[[(3S,5S)-1,5-dimethylpyrrolidin-3-yl]amino]-1-methylpiperidin-2-one