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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-2-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O4
(5R)-2-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclobutylmethyl)-2-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O3
(5R)-7-(cyclobutylmethyl)-2-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-1-(cyclohexylmethyl)-5-[3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C20H33N5O2
(5R)-1-(cyclohexylmethyl)-5-[3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5R)-9-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H20N2O4
(5R)-9-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-2-[2-(3-chloro-2,6-difluorophenyl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C17H19ClF2N2O2
(5S)-2-[2-(3-chloro-2,6-difluorophenyl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-1-(3-chlorophenyl)-5-methyl-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-2-one —— C18H20ClN3O2S
(5R)-1-(3-chlorophenyl)-5-methyl-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-2-one
—— (5S)-1-(3-chlorophenyl)-5-methyl-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-2-one —— C18H20ClN3O2S
(5S)-1-(3-chlorophenyl)-5-methyl-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-2-one
—— (5R)-7-cyclohexyl-2-[(3-hydroxy-4-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H32N2O3
(5R)-7-cyclohexyl-2-[(3-hydroxy-4-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H20N2O4
(5S)-9-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-7-(cyclopropylmethyl)-2-(4-methoxypyrimidin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24N4O2
(5S)-7-(cyclopropylmethyl)-2-(4-methoxypyrimidin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-N,N-dimethylpyridin-2-amine —— C17H20N2O
5-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-N,N-dimethylpyridin-2-amine
—— 5-methyl-4-[(3R)-3-(methylsulfonylmethyl)piperidin-1-yl]pyrimidin-2-amine —— C12H20N4O2S
5-methyl-4-[(3R)-3-(methylsulfonylmethyl)piperidin-1-yl]pyrimidin-2-amine
—— (5S)-2-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O4
(5S)-2-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-methoxyethyl)-2-[2-(6-oxo-1H-pyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H24N4O4
(5S)-7-(2-methoxyethyl)-2-[2-(6-oxo-1H-pyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-[2-(3-fluorophenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H27FN2O3
(5S)-7-(cyclobutylmethyl)-2-[2-(3-fluorophenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(1H-indol-3-yl)-5-phenyl-2,4-dihydro-1,2,4-triazin-3-one —— C17H14N4O
(5R)-5-(1H-indol-3-yl)-5-phenyl-2,4-dihydro-1,2,4-triazin-3-one
—— 5-[(2S)-oxolan-2-yl]-N-(2-pyridin-2-ylsulfanylethyl)thiophene-2-carboxamide —— C16H18N2O2S2
5-[(2S)-oxolan-2-yl]-N-(2-pyridin-2-ylsulfanylethyl)thiophene-2-carboxamide
—— (5R)-2-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H32N4O
(5R)-2-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-[2-(2,3-dimethylphenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H30N2O3
(5S)-7-(cyclopropylmethyl)-2-[2-(2,3-dimethylphenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-cyclopentyl-2-[(2,5-dimethyl-1,2,4-triazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H29N5O
(5R)-7-cyclopentyl-2-[(2,5-dimethyl-1,2,4-triazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-methyl-4-[(3S)-3-(methylsulfonylmethyl)piperidin-1-yl]pyrimidin-2-amine —— C12H20N4O2S
5-methyl-4-[(3S)-3-(methylsulfonylmethyl)piperidin-1-yl]pyrimidin-2-amine
—— (5R)-7-(cyclopropylmethyl)-2-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O
(5R)-7-(cyclopropylmethyl)-2-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R,7R)-N-(furan-2-ylmethyl)-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H19F3N4O2
(5R,7R)-N-(furan-2-ylmethyl)-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S)-2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C15H24N4O3
(5S)-2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[6-(dimethylamino)pyridine-3-carbonyl]-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O3
(5S)-2-[6-(dimethylamino)pyridine-3-carbonyl]-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
—— [(5S)-2-oxa-9-azaspiro[4.5]decan-9-yl]-(5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)methanone —— C18H25NO2S
[(5S)-2-oxa-9-azaspiro[4.5]decan-9-yl]-(5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)methanone
—— (5R)-7-propyl-2-quinoxalin-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C19H24N4O
(5R)-7-propyl-2-quinoxalin-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-cyclohexyl-2-(1-methylpyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5R)-7-cyclohexyl-2-(1-methylpyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-(aminomethyl)pyrrolidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]-1H-pyrimidin-6-one —— C17H18Cl2N4O2
5-[(3R)-3-(aminomethyl)pyrrolidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]-1H-pyrimidin-6-one
—— (5S)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one —— C16H24N4O3
(5S)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
—— 5-[[(3S)-3,4-dihydro-2H-chromen-3-yl]methyl]pyridine-3-carboxamide —— C16H16N2O2
5-[[(3S)-3,4-dihydro-2H-chromen-3-yl]methyl]pyridine-3-carboxamide
—— 5-[(3S)-3-(aminomethyl)pyrrolidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]-1H-pyrimidin-6-one —— C17H18Cl2N4O2
5-[(3S)-3-(aminomethyl)pyrrolidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]-1H-pyrimidin-6-one
—— (5R)-7-(cyclopropylmethyl)-2-[2-(2,3-dimethylphenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H30N2O3
(5R)-7-(cyclopropylmethyl)-2-[2-(2,3-dimethylphenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-N-[[3-(methoxymethyl)-1H-pyrazol-5-yl]methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C16H21N3O2S
(5R)-N-[[3-(methoxymethyl)-1H-pyrazol-5-yl]methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— [(5R)-2-oxa-9-azaspiro[4.5]decan-9-yl]-(5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)methanone —— C18H25NO2S
[(5R)-2-oxa-9-azaspiro[4.5]decan-9-yl]-(5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)methanone
—— 5-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]pyridine-3-carboxamide —— C16H16N2O2
5-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]pyridine-3-carboxamide
—— (5R)-9-(3-indol-1-ylpropyl)-2-oxa-9-azaspiro[4.5]decan-8-one —— C19H24N2O2
(5R)-9-(3-indol-1-ylpropyl)-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-2-[2-(azepan-1-yl)-2-oxoethyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H31N3O3
(5R)-2-[2-(azepan-1-yl)-2-oxoethyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5,8-dimethyl-2-[[[(3R)-5-oxo-1-propylpyrrolidin-3-yl]amino]methyl]-1H-quinolin-4-one —— C19H25N3O2
5,8-dimethyl-2-[[[(3R)-5-oxo-1-propylpyrrolidin-3-yl]amino]methyl]-1H-quinolin-4-one
—— (5R)-N-(2-chloro-6-methylphenyl)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decane-2-carboxamide —— C19H26ClN3O2
(5R)-N-(2-chloro-6-methylphenyl)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5S)-2-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C14H20FN5O
(5S)-2-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(1-methylpyrrole-2-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C17H25N3O2
(5S)-2-(1-methylpyrrole-2-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C15H24N4O3
(5R)-2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(2-morpholin-4-ylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H25N3O3
(5S)-2-(2-morpholin-4-ylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5,8-dimethyl-2-[[[(3S)-5-oxo-1-propylpyrrolidin-3-yl]amino]methyl]-1H-quinolin-4-one —— C19H25N3O2
5,8-dimethyl-2-[[[(3S)-5-oxo-1-propylpyrrolidin-3-yl]amino]methyl]-1H-quinolin-4-one
—— (5R)-7-(2-methoxyethyl)-2-[3-(2-methylimidazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H30N4O2
(5R)-7-(2-methoxyethyl)-2-[3-(2-methylimidazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one —— C16H24N4O3
(5R)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
—— (5R)-2-[2-(N-methylanilino)acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O2
(5R)-2-[2-(N-methylanilino)acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-N-(2-chloro-6-methylphenyl)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decane-2-carboxamide —— C19H26ClN3O2
(5S)-N-(2-chloro-6-methylphenyl)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5S)-7-cyclohexyl-2-(1-methylpyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5S)-7-cyclohexyl-2-(1-methylpyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one