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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-methoxy-2-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyran-4-one —— C19H17N3O5
5-methoxy-2-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyran-4-one
—— 5-methoxy-2-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyran-4-one —— C19H17N3O5
5-methoxy-2-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyran-4-one
—— 5-[(3R)-1-acetylpiperidine-3-carbonyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C18H25N3O3S
5-[(3R)-1-acetylpiperidine-3-carbonyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— 5-[(3S)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C19H27N5O2
5-[(3S)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— (5R)-9-[(5,7-dimethyl-2,1,3-benzoxadiazol-4-yl)sulfonyl]-2-oxa-9-azaspiro[4.5]decane —— C16H21N3O4S
(5R)-9-[(5,7-dimethyl-2,1,3-benzoxadiazol-4-yl)sulfonyl]-2-oxa-9-azaspiro[4.5]decane
—— {5-Oxo-5H-[1,3]thiazolo[3,2-A]pyrimidin-7-YL}methyl 3-(thiophene-2-amido)benzoate —— C19H13N3O4S2
{5-Oxo-5H-[1,3]thiazolo[3,2-A]pyrimidin-7-YL}methyl 3-(thiophene-2-amido)benzoate
—— 5-ethyl-N-[(2R)-2-pyridin-3-yloxypropyl]pyrimidin-2-amine —— C14H18N4O
5-ethyl-N-[(2R)-2-pyridin-3-yloxypropyl]pyrimidin-2-amine
—— 5-ethyl-N-[(2S)-2-pyridin-3-yloxypropyl]pyrimidin-2-amine —— C14H18N4O
5-ethyl-N-[(2S)-2-pyridin-3-yloxypropyl]pyrimidin-2-amine
—— (5S)-7-methyl-2-(2-methylquinolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H23N3O
(5S)-7-methyl-2-(2-methylquinolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R)-2-(furan-2-yl)azepane-1-carbonyl]-1H-pyrazin-2-one —— C15H17N3O3
5-[(2R)-2-(furan-2-yl)azepane-1-carbonyl]-1H-pyrazin-2-one
—— 5-ethyl-4-N-[(1S)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]pyrimidine-2,4-diamine —— C14H23N7
5-ethyl-4-N-[(1S)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]pyrimidine-2,4-diamine
—— 5-[(dimethylamino)methyl]-N-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]furan-2-carboxamide —— C19H24N2O4
5-[(dimethylamino)methyl]-N-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]furan-2-carboxamide
—— (5S)-7-(2-methoxyethyl)-2-[1-(4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one —— C23H35N3O2
(5S)-7-(2-methoxyethyl)-2-[1-(4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-(5,6,7,8-tetrahydroquinolin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C18H26N2O2
(5R)-9-(5,6,7,8-tetrahydroquinolin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5S)-1-(2-methoxyethyl)-5-(7-methoxy-1,2,4,5-tetrahydro-3-benzazepine-3-carbonyl)piperidin-2-one —— C20H28N2O4
(5S)-1-(2-methoxyethyl)-5-(7-methoxy-1,2,4,5-tetrahydro-3-benzazepine-3-carbonyl)piperidin-2-one
—— (5R)-7-methyl-2-(2-methylquinolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H23N3O
(5R)-7-methyl-2-(2-methylquinolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(dimethylamino)methyl]-N-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]furan-2-carboxamide —— C19H24N2O4
5-[(dimethylamino)methyl]-N-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]furan-2-carboxamide
—— (5R)-2-(3-methylpyridine-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H27N3O3
(5R)-2-(3-methylpyridine-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C19H27N5O2
5-[(3R)-3-[1-[3-(dimethylamino)propyl]imidazol-2-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— (5S)-9-[[2-(2-imidazol-1-ylethoxy)phenyl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C21H29N3O3
(5S)-9-[[2-(2-imidazol-1-ylethoxy)phenyl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-[(3R)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]-3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazole —— C19H26N4O
5-[(3R)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]-3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazole
—— (5R)-9-[[1-(3-fluorophenyl)pyrazol-4-yl]methyl]-2-oxa-9-azaspiro[4.5]decane —— C18H22FN3O
(5R)-9-[[1-(3-fluorophenyl)pyrazol-4-yl]methyl]-2-oxa-9-azaspiro[4.5]decane
—— 5,7-dimethyl-4-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrido[2,3-d]pyrimidine —— C20H23N5O
5,7-dimethyl-4-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrido[2,3-d]pyrimidine
—— 5,7-dimethyl-4-[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrido[2,3-d]pyrimidine —— C20H23N5O
5,7-dimethyl-4-[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrido[2,3-d]pyrimidine
—— 5,6-dimethyl-N-[(3R)-1-pyrazin-2-ylpiperidin-3-yl]pyrimidin-4-amine —— C15H20N6
5,6-dimethyl-N-[(3R)-1-pyrazin-2-ylpiperidin-3-yl]pyrimidin-4-amine
—— (5S)-9-[[1-(3-fluorophenyl)pyrazol-4-yl]methyl]-2-oxa-9-azaspiro[4.5]decane —— C18H22FN3O
(5S)-9-[[1-(3-fluorophenyl)pyrazol-4-yl]methyl]-2-oxa-9-azaspiro[4.5]decane
—— 5-chloro-6-oxo-N-[[(4S)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]-1H-pyridine-3-carboxamide —— C17H17ClN2O3
5-chloro-6-oxo-N-[[(4S)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]-1H-pyridine-3-carboxamide
—— (5S)-2-(3-methylpyridine-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H27N3O3
(5S)-2-(3-methylpyridine-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 1-benzothiophene-2-carboxylate —— C18H11N3O5S
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 1-benzothiophene-2-carboxylate
—— 5-(3-Fluorophenyl)-2-[(2-fluorophenyl)methyl]tetrazole —— C14H10F2N4
5-(3-Fluorophenyl)-2-[(2-fluorophenyl)methyl]tetrazole
—— 5-ethyl-N-methyl-N-[(2R)-2-morpholin-4-ylpropyl]pyrimidin-2-amine —— C14H24N4O
5-ethyl-N-methyl-N-[(2R)-2-morpholin-4-ylpropyl]pyrimidin-2-amine
—— [(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-[5-(3-methoxyphenyl)-1H-pyrazol-4-yl]methanone —— C20H25N3O4
[(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-[5-(3-methoxyphenyl)-1H-pyrazol-4-yl]methanone
—— 5-[(3S)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]-3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazole —— C19H26N4O
5-[(3S)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]-3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazole
—— 5-(3-Chlorophenyl)-2-[2-(2,4-dichlorophenoxy)ethyl]tetrazole —— C15H11Cl3N4O
5-(3-Chlorophenyl)-2-[2-(2,4-dichlorophenoxy)ethyl]tetrazole
—— 5-(4-Bromophenyl)-2-[(3-methylphenyl)methyl]tetrazole —— C15H13BrN4
5-(4-Bromophenyl)-2-[(3-methylphenyl)methyl]tetrazole
—— 5-(4-Bromophenyl)-2-[(4-chlorophenyl)methyl]tetrazole —— C14H10BrClN4
5-(4-Bromophenyl)-2-[(4-chlorophenyl)methyl]tetrazole
—— 5-(3-Chlorophenyl)-2-[(4-methylphenyl)methyl]tetrazole —— C15H13ClN4
5-(3-Chlorophenyl)-2-[(4-methylphenyl)methyl]tetrazole
—— 5-(4-Propan-2-ylphenyl)-2-[(4-propan-2-ylphenyl)methyl]tetrazole —— C20H24N4
5-(4-Propan-2-ylphenyl)-2-[(4-propan-2-ylphenyl)methyl]tetrazole
—— 5-(4-Bromophenyl)-2-[(4-propan-2-ylphenyl)methyl]tetrazole —— C17H17BrN4
5-(4-Bromophenyl)-2-[(4-propan-2-ylphenyl)methyl]tetrazole
—— 5-(3-Chlorophenyl)-2-[(3-methylphenyl)methyl]tetrazole —— C15H13ClN4
5-(3-Chlorophenyl)-2-[(3-methylphenyl)methyl]tetrazole
—— 5-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]pyridazin-3-one —— C20H26N4O
5-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]pyridazin-3-one
—— 5-ethyl-N-methyl-N-[(2S)-2-morpholin-4-ylpropyl]pyrimidin-2-amine —— C14H24N4O
5-ethyl-N-methyl-N-[(2S)-2-morpholin-4-ylpropyl]pyrimidin-2-amine
—— (5R)-2-(4-fluorophenyl)sulfonyl-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H23FN2O4S
(5R)-2-(4-fluorophenyl)sulfonyl-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— [(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-[5-(3-methoxyphenyl)-1H-pyrazol-4-yl]methanone —— C20H25N3O4
[(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-[5-(3-methoxyphenyl)-1H-pyrazol-4-yl]methanone
—— 5,6-dimethyl-N-[(3S)-1-pyrazin-2-ylpiperidin-3-yl]pyrimidin-4-amine —— C15H20N6
5,6-dimethyl-N-[(3S)-1-pyrazin-2-ylpiperidin-3-yl]pyrimidin-4-amine
—— (5R)-9-[[2-(2-imidazol-1-ylethoxy)phenyl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C21H29N3O3
(5R)-9-[[2-(2-imidazol-1-ylethoxy)phenyl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-chloro-6-oxo-N-[[(4R)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]-1H-pyridine-3-carboxamide —— C17H17ClN2O3
5-chloro-6-oxo-N-[[(4R)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]-1H-pyridine-3-carboxamide
—— 5-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]pyridazin-3-one —— C20H26N4O
5-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]pyridazin-3-one
—— (5S)-2-(4-fluorophenyl)sulfonyl-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H23FN2O4S
(5S)-2-(4-fluorophenyl)sulfonyl-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(4-Bromophenyl)-2-(naphthalen-1-ylmethyl)tetrazole —— C18H13BrN4
5-(4-Bromophenyl)-2-(naphthalen-1-ylmethyl)tetrazole