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—— (5S)-7-(2-methoxyethyl)-2-[(1-methyl-4-oxo-2H-pyrazolo[3,4-d]pyrimidin-6-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H26N6O3
(5S)-7-(2-methoxyethyl)-2-[(1-methyl-4-oxo-2H-pyrazolo[3,4-d]pyrimidin-6-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-1-ethyl-5-(4-pyrimidin-2-yl-1,4-diazepane-1-carbonyl)piperidin-2-one —— C17H25N5O2
(5R)-1-ethyl-5-(4-pyrimidin-2-yl-1,4-diazepane-1-carbonyl)piperidin-2-one
—— [(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(3-methoxy-5-methylthiophen-2-yl)methanone —— C16H23NO4S
[(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(3-methoxy-5-methylthiophen-2-yl)methanone
—— (5S)-2-(7-chloroquinolin-4-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H22ClN3O2
(5S)-2-(7-chloroquinolin-4-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-methyl-2-(3-pyridin-4-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H23N3O2
(5R)-7-methyl-2-(3-pyridin-4-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[(2-aminopyridin-3-yl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O
(5R)-2-[(2-aminopyridin-3-yl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(7-chloroquinolin-4-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H22ClN3O2
(5R)-2-(7-chloroquinolin-4-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-methyl-2-[2-methyl-2-(4-methylphenoxy)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H28N2O3
(5R)-7-methyl-2-[2-methyl-2-(4-methylphenoxy)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-[[2-(methylamino)-1,3-thiazol-4-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4OS
(5S)-7-(cyclobutylmethyl)-2-[[2-(methylamino)-1,3-thiazol-4-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-4-[[4-(2-aminoethyl)phenyl]methyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one —— C21H27N3O
(5S)-4-[[4-(2-aminoethyl)phenyl]methyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
—— (5S)-7-methyl-2-[2-methyl-2-(4-methylphenoxy)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H28N2O3
(5S)-7-methyl-2-[2-methyl-2-(4-methylphenoxy)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-(5,6-dimethylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O
(5S)-7-(cyclopropylmethyl)-2-(5,6-dimethylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[2-(methylamino)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H20N4O2
(5S)-2-[2-(methylamino)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-ethyl-5-(4-pyrimidin-2-yl-1,4-diazepane-1-carbonyl)piperidin-2-one —— C17H25N5O2
(5S)-1-ethyl-5-(4-pyrimidin-2-yl-1,4-diazepane-1-carbonyl)piperidin-2-one
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(5R)-2-oxa-9-azaspiro[4.5]decan-9-yl]methanone —— C17H22N4O2
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(5R)-2-oxa-9-azaspiro[4.5]decan-9-yl]methanone
—— 5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-[2-(1-oxophthalazin-2-yl)ethyl]-1,2-dihydropyrazole-3-carboxamide —— C20H17N5O3
5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-[2-(1-oxophthalazin-2-yl)ethyl]-1,2-dihydropyrazole-3-carboxamide
—— (5R)-9-(2-phenoxyethylsulfonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C17H25NO5S
(5R)-9-(2-phenoxyethylsulfonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-1-[2-(1H-imidazol-5-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one —— C17H21N3O
(5R)-1-[2-(1H-imidazol-5-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
—— 5-[2-oxo-2-[(3R)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]ethyl]-1H-pyrimidine-2,4-dione —— C20H22N6O3
5-[2-oxo-2-[(3R)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]ethyl]-1H-pyrimidine-2,4-dione
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl]-5-methylpiperidin-2-one —— C20H25N3O5
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl]-5-methylpiperidin-2-one
—— (5R)-2-[2-(azepan-1-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H31N3O3
(5R)-2-[2-(azepan-1-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[2-(1H-imidazol-5-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one —— C17H21N3O
(5S)-1-[2-(1H-imidazol-5-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
—— (5S)-7-(cyclobutylmethyl)-2-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H28N4OS
(5S)-7-(cyclobutylmethyl)-2-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[2-(azepan-1-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H31N3O3
(5S)-2-[2-(azepan-1-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclobutylmethyl)-2-[[2-(methylamino)-1,3-thiazol-4-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4OS
(5R)-7-(cyclobutylmethyl)-2-[[2-(methylamino)-1,3-thiazol-4-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C15H24ClN3O2S
(5S)-9-[[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— [5-[1-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]triazol-4-yl]furan-2-yl]methanol —— C16H18N6O2
[5-[1-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]triazol-4-yl]furan-2-yl]methanol
—— [5-[1-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]triazol-4-yl]furan-2-yl]methanol —— C16H18N6O2
[5-[1-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]triazol-4-yl]furan-2-yl]methanol
—— (5S)-2-[(2-aminopyridin-3-yl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O
(5S)-2-[(2-aminopyridin-3-yl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-3-[(4-methylpiperidin-1-yl)methyl]-5-(naphthalen-1-yloxymethyl)-1,3-oxazolidin-2-one —— C21H26N2O3
(5R)-3-[(4-methylpiperidin-1-yl)methyl]-5-(naphthalen-1-yloxymethyl)-1,3-oxazolidin-2-one
—— (5R)-1-(4-hydroxybutyl)-5-methyl-5-phenylpiperidin-2-one —— C16H23NO2
(5R)-1-(4-hydroxybutyl)-5-methyl-5-phenylpiperidin-2-one
—— (5S)-9-[5-(trifluoromethyl)pyridin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C15H19F3N2O2
(5S)-9-[5-(trifluoromethyl)pyridin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-2-[3-(2-fluorophenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C22H23FN2O2
(5R)-2-[3-(2-fluorophenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclobutylmethyl)-2-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H28N4OS
(5R)-7-(cyclobutylmethyl)-2-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-propyl-1H-pyrazol-3-yl)-[(2S)-2-(2-pyridin-2-ylethyl)piperidin-1-yl]methanone —— C19H26N4O
(5-propyl-1H-pyrazol-3-yl)-[(2S)-2-(2-pyridin-2-ylethyl)piperidin-1-yl]methanone
—— (5S)-2-[3-(2-fluorophenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C22H23FN2O2
(5S)-2-[3-(2-fluorophenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5-propyl-1H-pyrazol-3-yl)-[(2R)-2-(2-pyridin-2-ylethyl)piperidin-1-yl]methanone —— C19H26N4O
(5-propyl-1H-pyrazol-3-yl)-[(2R)-2-(2-pyridin-2-ylethyl)piperidin-1-yl]methanone
—— (5S)-7-(2-hydroxyethyl)-2-[1-(2-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one —— C22H33N3O2
(5S)-7-(2-hydroxyethyl)-2-[1-(2-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C15H24ClN3O2S
(5R)-9-[[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R,10bR)-2-phenylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-1H-indole]-2'-one —— C23H17N3O2
(5R,10bR)-2-phenylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-1H-indole]-2'-one
—— (5S)-2-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C16H26N4O2S
(5S)-2-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl]-5-methylpiperidin-2-one —— C20H25N3O5
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl]-5-methylpiperidin-2-one
—— (5S)-7-cyclohexyl-2-(3-pyridin-4-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C22H31N3O2
(5S)-7-cyclohexyl-2-(3-pyridin-4-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H26ClN3O3
(5R)-2-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[2-[(5S)-7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C19H26N4O4
5-[2-[(5S)-7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— (5R)-7-(2-hydroxyethyl)-2-[(3-methylquinoxalin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H26N4O2
(5R)-7-(2-hydroxyethyl)-2-[(3-methylquinoxalin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C15H24N2O3
(5S)-9-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-[(4aS,7aR)-3-benzyl-2,4-dioxo-4a,6,7,7a-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-5-yl]-5-oxopentanoic acid —— C18H21N3O5
5-[(4aS,7aR)-3-benzyl-2,4-dioxo-4a,6,7,7a-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-5-yl]-5-oxopentanoic acid
—— (5R)-2-[4-(2-methylimidazol-1-yl)butanoyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C19H30N4O2
(5R)-2-[4-(2-methylimidazol-1-yl)butanoyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(3-methoxypropyl)-2-[(4-methylthiadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H26N4O2S
(5R)-7-(3-methoxypropyl)-2-[(4-methylthiadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one