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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-2-[(2-methylpropan-2-yl)oxycarbonyl]-7-phenylmethoxycarbonyl-2,7-diazaspiro[3.5]nonane-5-carboxylic acid —— C21H28N2O6
(5R)-2-[(2-methylpropan-2-yl)oxycarbonyl]-7-phenylmethoxycarbonyl-2,7-diazaspiro[3.5]nonane-5-carboxylic acid
—— (5R)-7-bromo-4-(3-bromobenzoyl)-5-phenyl-3,5-dihydro-1H-1,4-benzodiazepin-2-one —— C22H16Br2N2O2
(5R)-7-bromo-4-(3-bromobenzoyl)-5-phenyl-3,5-dihydro-1H-1,4-benzodiazepin-2-one
—— 5-O-benzyl 1-O'-tert-butyl (3aR,6aS)-spiro[1,2,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-3,4'-piperidine]-1',5-dicarboxylate —— C23H33N3O4
5-O-benzyl 1-O'-tert-butyl (3aR,6aS)-spiro[1,2,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-3,4'-piperidine]-1',5-dicarboxylate
—— (5R)-7-methyl-4-(3-methylbenzoyl)-5-phenyl-3,5-dihydro-1H-1,4-benzodiazepin-2-one —— C24H22N2O2
(5R)-7-methyl-4-(3-methylbenzoyl)-5-phenyl-3,5-dihydro-1H-1,4-benzodiazepin-2-one
—— (5S)-2-[(2-methylpropan-2-yl)oxycarbonyl]-7-phenylmethoxycarbonyl-2,7-diazaspiro[3.5]nonane-5-carboxylic acid —— C21H28N2O6
(5S)-2-[(2-methylpropan-2-yl)oxycarbonyl]-7-phenylmethoxycarbonyl-2,7-diazaspiro[3.5]nonane-5-carboxylic acid
—— 5-(4-Methoxyphenyl)sulfanyl-1,2,3-triaza-4-azanidacyclopenta-2,5-diene —— C8H7N4OS-
5-(4-Methoxyphenyl)sulfanyl-1,2,3-triaza-4-azanidacyclopenta-2,5-diene
—— (5E)-5-[(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylidene]-1,3-thiazolidine-2,4-dione —— C14H10ClN3O2S
(5E)-5-[(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylidene]-1,3-thiazolidine-2,4-dione
—— (5R)-7-chloro-4-(2,2-dimethylpropanoyl)-5-phenyl-3,5-dihydro-1H-1,4-benzodiazepin-2-one —— C20H21ClN2O2
(5R)-7-chloro-4-(2,2-dimethylpropanoyl)-5-phenyl-3,5-dihydro-1H-1,4-benzodiazepin-2-one
—— 5-O-benzyl 1-O'-tert-butyl (3aS,6aS)-spiro[1,2,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-3,4'-piperidine]-1',5-dicarboxylate —— C23H33N3O4
5-O-benzyl 1-O'-tert-butyl (3aS,6aS)-spiro[1,2,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-3,4'-piperidine]-1',5-dicarboxylate
—— 5-bromo-3-[4-chloro-2-[(S)-hydroxy(phenyl)methyl]phenyl]imino-1H-indol-2-one —— C21H14BrClN2O2
5-bromo-3-[4-chloro-2-[(S)-hydroxy(phenyl)methyl]phenyl]imino-1H-indol-2-one
—— 5-Bromo-2-[(6-bromo-2-oxochromene-3-carbonyl)amino]benzoate —— C17H8Br2NO5-
5-Bromo-2-[(6-bromo-2-oxochromene-3-carbonyl)amino]benzoate
—— 5-fluoro-1-[(2R,3S,4R,5R)-3,4,5-trihydroxyoxan-2-yl]pyrimidine-2,4-dione —— C9H11FN2O6
5-fluoro-1-[(2R,3S,4R,5R)-3,4,5-trihydroxyoxan-2-yl]pyrimidine-2,4-dione
—— 5-O-benzyl 1-O-tert-butyl (3aR,6aR)-3a,4,6,6a-tetrahydro-3H-pyrrolo[3,4-c][1,2]oxazole-1,5-dicarboxylate —— C18H24N2O5
5-O-benzyl 1-O-tert-butyl (3aR,6aR)-3a,4,6,6a-tetrahydro-3H-pyrrolo[3,4-c][1,2]oxazole-1,5-dicarboxylate
—— 5-bromo-N-[(1R)-1-phenylethyl]pyridine-3-carboxamide —— C14H13BrN2O
5-bromo-N-[(1R)-1-phenylethyl]pyridine-3-carboxamide
—— 5-O-benzyl 1-O'-tert-butyl (3aS,6aR)-spiro[1,2,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-3,4'-piperidine]-1',5-dicarboxylate —— C23H33N3O4
5-O-benzyl 1-O'-tert-butyl (3aS,6aR)-spiro[1,2,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-3,4'-piperidine]-1',5-dicarboxylate
—— 5-[(1S)-1-[4-(phenylmethoxymethyl)triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine —— C14H16N6OS
5-[(1S)-1-[4-(phenylmethoxymethyl)triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine
—— [5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(5S)-2-oxa-9-azaspiro[4.5]decan-9-yl]methanone —— C17H22N4O3
[5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(5S)-2-oxa-9-azaspiro[4.5]decan-9-yl]methanone
—— (5S)-N-(3-fluoropyridin-2-yl)-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-amine —— C19H17FN4
(5S)-N-(3-fluoropyridin-2-yl)-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-amine
—— (5S)-2-(4-chloro-1-methylpyrrole-2-carbonyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H26ClN3O2
(5S)-2-(4-chloro-1-methylpyrrole-2-carbonyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[(2-methylpropan-2-yl)oxycarbonyl]-3-phenylmethoxycarbonyl-3,9-diazaspiro[5.5]undecane-5-carboxylic acid —— C23H32N2O6
(5R)-9-[(2-methylpropan-2-yl)oxycarbonyl]-3-phenylmethoxycarbonyl-3,9-diazaspiro[5.5]undecane-5-carboxylic acid
—— 5-cyclohexyl-N-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]-1H-pyrazole-4-carboxamide —— C16H26N4O4S
5-cyclohexyl-N-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]-1H-pyrazole-4-carboxamide
—— (5S)-5-methyl-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-5-phenylpiperidin-2-one —— C18H24N2O2
(5S)-5-methyl-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-5-phenylpiperidin-2-one
—— (5S)-9-[(2-methylpropan-2-yl)oxycarbonyl]-3-phenylmethoxycarbonyl-3,9-diazaspiro[5.5]undecane-5-carboxylic acid —— C23H32N2O6
(5S)-9-[(2-methylpropan-2-yl)oxycarbonyl]-3-phenylmethoxycarbonyl-3,9-diazaspiro[5.5]undecane-5-carboxylic acid
—— (5R)-4-[hydroxy(phenyl)methylidene]-1-(2-morpholin-4-ium-4-ylethyl)-5-pyridin-4-ylpyrrolidine-2,3-dione —— C22H24N3O4+
(5R)-4-[hydroxy(phenyl)methylidene]-1-(2-morpholin-4-ium-4-ylethyl)-5-pyridin-4-ylpyrrolidine-2,3-dione
—— (5S)-2-(4-methoxypiperidin-1-yl)sulfonyl-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C17H31N3O4S
(5S)-2-(4-methoxypiperidin-1-yl)sulfonyl-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(3-morpholin-4-ium-4-ylpropyl)-5-phenylpyrrolidine-2,3-dione —— C24H26ClN2O4+
(5R)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(3-morpholin-4-ium-4-ylpropyl)-5-phenylpyrrolidine-2,3-dione
—— (5R)-5-methyl-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-5-phenylpiperidin-2-one —— C18H24N2O2
(5R)-5-methyl-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-5-phenylpiperidin-2-one
—— (5S)-5-methyl-5-phenyl-1-(2-pyridin-2-ylethyl)piperidin-2-one —— C19H22N2O
(5S)-5-methyl-5-phenyl-1-(2-pyridin-2-ylethyl)piperidin-2-one
—— (5R)-7-(cyclopropylmethyl)-2-[(2,5-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H24F2N2O
(5R)-7-(cyclopropylmethyl)-2-[(2,5-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-methoxy-1-methyl-N-[(5R)-4,5,6,7-tetrahydro-1H-indazol-5-yl]indole-2-carboxamide —— C18H20N4O2
5-methoxy-1-methyl-N-[(5R)-4,5,6,7-tetrahydro-1H-indazol-5-yl]indole-2-carboxamide
—— (5R)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[(3-fluorophenyl)methyl]piperidin-2-one —— C16H18FN3O2
(5R)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[(3-fluorophenyl)methyl]piperidin-2-one
—— [5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(5R)-2-oxa-9-azaspiro[4.5]decan-9-yl]methanone —— C17H22N4O3
[5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(5R)-2-oxa-9-azaspiro[4.5]decan-9-yl]methanone
—— (5R)-1-[2-(dimethylamino)ethyl]-5-[2-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]ethyl]pyrrolidin-2-one —— C17H25N5OS
(5R)-1-[2-(dimethylamino)ethyl]-5-[2-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]ethyl]pyrrolidin-2-one
—— (5S)-7-(2-hydroxyethyl)-2-[2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H22N4O4S
(5S)-7-(2-hydroxyethyl)-2-[2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(3-morpholin-4-ium-4-ylpropyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dione —— C27H32ClN2O4+
(5R)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(3-morpholin-4-ium-4-ylpropyl)-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dione
—— (5E)-5-[(4-nitrophenyl)methylidene]-3-(piperidin-1-ium-1-ylmethyl)-2-sulfanylidene-1,3-thiazolidin-4-one —— C16H18N3O3S2+
(5E)-5-[(4-nitrophenyl)methylidene]-3-(piperidin-1-ium-1-ylmethyl)-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-2-[2-(benzimidazol-1-yl)ethyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O
(5S)-2-[2-(benzimidazol-1-yl)ethyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[(3-fluorophenyl)methyl]piperidin-2-one —— C16H18FN3O2
(5S)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[(3-fluorophenyl)methyl]piperidin-2-one
—— 5-[(1R)-1-[4-(phenylmethoxymethyl)triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine —— C14H16N6OS
5-[(1R)-1-[4-(phenylmethoxymethyl)triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine
—— (5S)-7-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide —— C20H29N3O3
(5S)-7-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5R)-1-[(3-fluorophenyl)methyl]-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C21H27FN4O2
(5R)-1-[(3-fluorophenyl)methyl]-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5S)-1-[(3-fluorophenyl)methyl]-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C21H27FN4O2
(5S)-1-[(3-fluorophenyl)methyl]-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— 5-cyclohexyl-N-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]-1H-pyrazole-4-carboxamide —— C16H26N4O4S
5-cyclohexyl-N-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]-1H-pyrazole-4-carboxamide
—— (5R)-7-(2-methoxyethyl)-2-(1,2-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C15H21N3O3S
(5R)-7-(2-methoxyethyl)-2-(1,2-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-[(2,5-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H24F2N2O
(5S)-7-(cyclopropylmethyl)-2-[(2,5-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-methoxy-1-methyl-N-[(5S)-4,5,6,7-tetrahydro-1H-indazol-5-yl]indole-2-carboxamide —— C18H20N4O2
5-methoxy-1-methyl-N-[(5S)-4,5,6,7-tetrahydro-1H-indazol-5-yl]indole-2-carboxamide
—— (5S)-1-[2-(dimethylamino)ethyl]-5-[2-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]ethyl]pyrrolidin-2-one —— C17H25N5OS
(5S)-1-[2-(dimethylamino)ethyl]-5-[2-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]ethyl]pyrrolidin-2-one
—— (5R)-7-(cyclopropylmethyl)-2-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H28N4O2
(5R)-7-(cyclopropylmethyl)-2-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R,7S)-3-(acetamidomethyl)adamantane-1-carboxylate —— C14H20NO3-
(5R,7S)-3-(acetamidomethyl)adamantane-1-carboxylate
—— (5R)-2-(4-methoxypiperidin-1-yl)sulfonyl-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C17H31N3O4S
(5R)-2-(4-methoxypiperidin-1-yl)sulfonyl-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one