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—— 5-[[2-[(1S)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-7-methyl-3,4-dihydro-2H-1,5-benzoxazepine —— C17H22N2O2S
5-[[2-[(1S)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-7-methyl-3,4-dihydro-2H-1,5-benzoxazepine
—— 5-[[(3aR,6aR)-3-(2-fluorophenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoic acid —— C16H17FN2O5S2
5-[[(3aR,6aR)-3-(2-fluorophenyl)-5,5-dioxo-3a,4,6,6a-tetrahydrothieno[3,4-d][1,3]thiazol-2-ylidene]amino]-5-oxopentanoic acid
—— 5-bromo-N-[2-[(3R,4S)-3-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C14H19BrN2O3S
5-bromo-N-[2-[(3R,4S)-3-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— (5-methyl-1,3,4-thiadiazol-2-yl)methyl (2R)-2-thiophen-3-ylpropanoate —— C11H12N2O2S2
(5-methyl-1,3,4-thiadiazol-2-yl)methyl (2R)-2-thiophen-3-ylpropanoate
—— (5aR)-3-methyl-6,11-dihydro-5aH-chromeno[2,3-b][1,5]benzodiazepin-13-one —— C17H14N2O2
(5aR)-3-methyl-6,11-dihydro-5aH-chromeno[2,3-b][1,5]benzodiazepin-13-one
—— 5-bromo-N-[2-[(3S,4R)-3-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C14H19BrN2O3S
5-bromo-N-[2-[(3S,4R)-3-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— 5-bromo-N-[2-[(3S,4S)-3-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C14H19BrN2O3S
5-bromo-N-[2-[(3S,4S)-3-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— 5-fluoro-2-hydroxy-N-[(1R,2R)-1-methoxy-1-(4-methoxyphenyl)propan-2-yl]benzamide —— C18H20FNO4
5-fluoro-2-hydroxy-N-[(1R,2R)-1-methoxy-1-(4-methoxyphenyl)propan-2-yl]benzamide
—— 5-[[[(3R)-1,4-dioxaspiro[4.4]nonan-3-yl]methylamino]methyl]-2-methoxybenzonitrile —— C17H22N2O3
5-[[[(3R)-1,4-dioxaspiro[4.4]nonan-3-yl]methylamino]methyl]-2-methoxybenzonitrile
—— (5aR)-2,3-dimethyl-6,11-dihydro-5aH-chromeno[2,3-b][1,5]benzodiazepin-13-one —— C18H16N2O2
(5aR)-2,3-dimethyl-6,11-dihydro-5aH-chromeno[2,3-b][1,5]benzodiazepin-13-one
—— 5-(2,3-dihydroindol-1-ylsulfonyl)-2-methoxy-N-(2-methylbutan-2-yl)benzamide —— C21H26N2O4S
5-(2,3-dihydroindol-1-ylsulfonyl)-2-methoxy-N-(2-methylbutan-2-yl)benzamide
—— (5-propan-2-yl-1H-pyrazol-3-yl)-[(3R)-3-(1,3,5-trimethylpyrazol-4-yl)morpholin-4-yl]methanone —— C17H25N5O2
(5-propan-2-yl-1H-pyrazol-3-yl)-[(3R)-3-(1,3,5-trimethylpyrazol-4-yl)morpholin-4-yl]methanone
—— 5-(difluoromethyl)-1-methyl-N-[(1S,2S)-2-[2-(trifluoromethyl)phenyl]cycloheptyl]pyrazole-4-carboxamide —— C20H22F5N3O
5-(difluoromethyl)-1-methyl-N-[(1S,2S)-2-[2-(trifluoromethyl)phenyl]cycloheptyl]pyrazole-4-carboxamide
—— 5-methyl-2-[(1S)-1-[4-(2-methyl-1H-indol-3-yl)piperidin-1-yl]ethyl]-1,3-oxazole —— C20H25N3O
5-methyl-2-[(1S)-1-[4-(2-methyl-1H-indol-3-yl)piperidin-1-yl]ethyl]-1,3-oxazole
—— 5-bromo-2-[(2R,5R)-2-ethyl-5-methylpyrrolidin-1-yl]pyridine —— C12H17BrN2
5-bromo-2-[(2R,5R)-2-ethyl-5-methylpyrrolidin-1-yl]pyridine
—— (5-methyl-1,2-oxazol-3-yl)methyl (E)-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enoate —— C15H12N2O7
(5-methyl-1,2-oxazol-3-yl)methyl (E)-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enoate
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 2,3-dimethylquinoxaline-6-carboxylate —— C20H15N5O5
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 2,3-dimethylquinoxaline-6-carboxylate
—— 5-[(4-Bromo-2-chloro-6-methylphenoxy)methyl]-1,3-benzodioxole —— C15H12BrClO3
5-[(4-Bromo-2-chloro-6-methylphenoxy)methyl]-1,3-benzodioxole
—— 5-bromo-2-[(2R,5S)-2-ethyl-5-methylpyrrolidin-1-yl]pyridine —— C12H17BrN2
5-bromo-2-[(2R,5S)-2-ethyl-5-methylpyrrolidin-1-yl]pyridine
—— 5-(9H-carbazol-2-yloxymethyl)-3-(2-methylphenyl)-1,2,4-oxadiazole —— C22H17N3O2
5-(9H-carbazol-2-yloxymethyl)-3-(2-methylphenyl)-1,2,4-oxadiazole
—— 5-bromo-2-[(2S,5S)-2-ethyl-5-methylpyrrolidin-1-yl]pyridine —— C12H17BrN2
5-bromo-2-[(2S,5S)-2-ethyl-5-methylpyrrolidin-1-yl]pyridine
—— (5R)-5-[(1R)-2-benzyl-3-oxo-1H-isoindol-1-yl]-1-butyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C23H23N3O3S
(5R)-5-[(1R)-2-benzyl-3-oxo-1H-isoindol-1-yl]-1-butyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-bromo-2-[(2S,5R)-2-ethyl-5-methylpyrrolidin-1-yl]pyridine —— C12H17BrN2
5-bromo-2-[(2S,5R)-2-ethyl-5-methylpyrrolidin-1-yl]pyridine
—— 5-[(3S)-4-(2-ethoxyethyl)-3-ethylpiperazin-1-yl]imidazo[1,2-a]pyrazine —— C16H25N5O
5-[(3S)-4-(2-ethoxyethyl)-3-ethylpiperazin-1-yl]imidazo[1,2-a]pyrazine
—— 5-methyl-2-[(1R)-1-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]ethyl]-1,3-oxazole —— C14H20N4O
5-methyl-2-[(1R)-1-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]ethyl]-1,3-oxazole
—— 5-methyl-2-[(1R)-1-[4-(2-methyl-1H-indol-3-yl)piperidin-1-yl]ethyl]-1,3-oxazole —— C20H25N3O
5-methyl-2-[(1R)-1-[4-(2-methyl-1H-indol-3-yl)piperidin-1-yl]ethyl]-1,3-oxazole
—— [5-(methoxymethyl)-1,2-oxazol-3-yl]-[(2S,3R)-2,3,4-trimethylpiperazin-1-yl]methanone —— C13H21N3O3
[5-(methoxymethyl)-1,2-oxazol-3-yl]-[(2S,3R)-2,3,4-trimethylpiperazin-1-yl]methanone
—— (5aS,9aS)-1-(5-bromopyrimidin-4-yl)-2,3,4,5,5a,6,7,8,9,9a-decahydrobenzo[b]azepine —— C14H20BrN3
(5aS,9aS)-1-(5-bromopyrimidin-4-yl)-2,3,4,5,5a,6,7,8,9,9a-decahydrobenzo[b]azepine
—— [5-(methoxymethyl)-1,2-oxazol-3-yl]-[(2S,3S)-2,3,4-trimethylpiperazin-1-yl]methanone —— C13H21N3O3
[5-(methoxymethyl)-1,2-oxazol-3-yl]-[(2S,3S)-2,3,4-trimethylpiperazin-1-yl]methanone
—— [5-(furan-2-yl)-1,3-oxazol-4-yl]-[(9R)-9-methyl-6-azaspiro[3.5]nonan-6-yl]methanone —— C17H20N2O3
[5-(furan-2-yl)-1,3-oxazol-4-yl]-[(9R)-9-methyl-6-azaspiro[3.5]nonan-6-yl]methanone
—— 5-methyl-2-[(1S)-1-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]ethyl]-1,3-oxazole —— C14H20N4O
5-methyl-2-[(1S)-1-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]ethyl]-1,3-oxazole
—— [5-(furan-2-yl)-1,3-oxazol-4-yl]-[(9S)-9-methyl-6-azaspiro[3.5]nonan-6-yl]methanone —— C17H20N2O3
[5-(furan-2-yl)-1,3-oxazol-4-yl]-[(9S)-9-methyl-6-azaspiro[3.5]nonan-6-yl]methanone
—— 5-methyl-2-[(1S)-1-[4-(1-methylpyrazol-4-yl)piperidin-1-yl]ethyl]-1,3-oxazole —— C15H22N4O
5-methyl-2-[(1S)-1-[4-(1-methylpyrazol-4-yl)piperidin-1-yl]ethyl]-1,3-oxazole
—— (5R,9S)-N-[4-(difluoromethylsulfonyl)phenyl]-2,6-dioxaspiro[4.5]decan-9-amine —— C15H19F2NO4S
(5R,9S)-N-[4-(difluoromethylsulfonyl)phenyl]-2,6-dioxaspiro[4.5]decan-9-amine
—— 5-[(3R)-4-(2-ethoxyethyl)-3-ethylpiperazin-1-yl]imidazo[1,2-a]pyrazine —— C16H25N5O
5-[(3R)-4-(2-ethoxyethyl)-3-ethylpiperazin-1-yl]imidazo[1,2-a]pyrazine
—— [5-(methoxymethyl)-1,2-oxazol-3-yl]-[(2R,3R)-2,3,4-trimethylpiperazin-1-yl]methanone —— C13H21N3O3
[5-(methoxymethyl)-1,2-oxazol-3-yl]-[(2R,3R)-2,3,4-trimethylpiperazin-1-yl]methanone
—— (5R)-5-[[2-[(2,4-dichlorophenyl)methoxy]phenyl]methyl]-3-propyl-4,5-dihydro-1,2-oxazole —— C20H21Cl2NO2
(5R)-5-[[2-[(2,4-dichlorophenyl)methoxy]phenyl]methyl]-3-propyl-4,5-dihydro-1,2-oxazole
—— (5R)-3-[4-(difluoromethoxy)phenyl]-1',3',3'-trimethylspiro[4H-1,2-oxazole-5,2'-indole] —— C20H20F2N2O2
(5R)-3-[4-(difluoromethoxy)phenyl]-1',3',3'-trimethylspiro[4H-1,2-oxazole-5,2'-indole]
—— (5R,9R)-N-[4-(difluoromethylsulfonyl)phenyl]-2,6-dioxaspiro[4.5]decan-9-amine —— C15H19F2NO4S
(5R,9R)-N-[4-(difluoromethylsulfonyl)phenyl]-2,6-dioxaspiro[4.5]decan-9-amine
—— (5aR,9aS)-1-[5-(methoxymethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]-2,3,4,5,5a,6,7,8,9,9a-decahydrobenzo[b]azepine —— C17H25N5O
(5aR,9aS)-1-[5-(methoxymethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]-2,3,4,5,5a,6,7,8,9,9a-decahydrobenzo[b]azepine
—— 5-methyl-2-[(1R)-1-[4-(1-methylpyrazol-4-yl)piperidin-1-yl]ethyl]-1,3-oxazole —— C15H22N4O
5-methyl-2-[(1R)-1-[4-(1-methylpyrazol-4-yl)piperidin-1-yl]ethyl]-1,3-oxazole
—— (5S,9S)-N-[4-(difluoromethylsulfonyl)phenyl]-2,6-dioxaspiro[4.5]decan-9-amine —— C15H19F2NO4S
(5S,9S)-N-[4-(difluoromethylsulfonyl)phenyl]-2,6-dioxaspiro[4.5]decan-9-amine
—— (5S,9R)-N-[4-(difluoromethylsulfonyl)phenyl]-2,6-dioxaspiro[4.5]decan-9-amine —— C15H19F2NO4S
(5S,9R)-N-[4-(difluoromethylsulfonyl)phenyl]-2,6-dioxaspiro[4.5]decan-9-amine
—— [5-(methoxymethyl)-1,2-oxazol-3-yl]-[(2R,3S)-2,3,4-trimethylpiperazin-1-yl]methanone —— C13H21N3O3
[5-(methoxymethyl)-1,2-oxazol-3-yl]-[(2R,3S)-2,3,4-trimethylpiperazin-1-yl]methanone
—— (5R,9R)-N-[[2-(cyclopropylmethoxy)phenyl]methyl]-2,6-dioxaspiro[4.5]decan-9-amine —— C19H27NO3
(5R,9R)-N-[[2-(cyclopropylmethoxy)phenyl]methyl]-2,6-dioxaspiro[4.5]decan-9-amine
—— (5S,9S)-N-[(6-chloropyridin-3-yl)methyl]-2,6-dioxaspiro[4.5]decan-9-amine —— C14H19ClN2O2
(5S,9S)-N-[(6-chloropyridin-3-yl)methyl]-2,6-dioxaspiro[4.5]decan-9-amine
—— (5S,9S)-N-[(2,4,6-trimethylphenyl)methyl]-2,6-dioxaspiro[4.5]decan-9-amine —— C18H27NO2
(5S,9S)-N-[(2,4,6-trimethylphenyl)methyl]-2,6-dioxaspiro[4.5]decan-9-amine
—— (5R,9S)-N-[(3-bromo-4-methoxyphenyl)methyl]-2,6-dioxaspiro[4.5]decan-9-amine —— C16H22BrNO3
(5R,9S)-N-[(3-bromo-4-methoxyphenyl)methyl]-2,6-dioxaspiro[4.5]decan-9-amine
—— (5S,9R)-N-[[5-(4-methylphenyl)-1H-pyrazol-4-yl]methyl]-2,6-dioxaspiro[4.5]decan-9-amine —— C19H25N3O2
(5S,9R)-N-[[5-(4-methylphenyl)-1H-pyrazol-4-yl]methyl]-2,6-dioxaspiro[4.5]decan-9-amine
—— (5S,9R)-N-[[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-2,6-dioxaspiro[4.5]decan-9-amine —— C20H26ClN3O2
(5S,9R)-N-[[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-2,6-dioxaspiro[4.5]decan-9-amine