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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(2R)-2-[2-(dimethylamino)ethyl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one —— C15H24N4O2
5-[(2R)-2-[2-(dimethylamino)ethyl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one
—— (5S)-3-methyl-7-(quinolin-4-ylmethyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H19N3O2
(5S)-3-methyl-7-(quinolin-4-ylmethyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(3R)-3-(1H-benzimidazol-2-yl)piperidine-1-carbonyl]-3-methyl-1,3-benzoxazol-2-one —— C21H20N4O3
5-[(3R)-3-(1H-benzimidazol-2-yl)piperidine-1-carbonyl]-3-methyl-1,3-benzoxazol-2-one
—— 5-acetyl-N-[(1R)-1-(1,3-benzothiazol-2-yl)ethyl]-N-methylthiophene-2-carboxamide —— C17H16N2O2S2
5-acetyl-N-[(1R)-1-(1,3-benzothiazol-2-yl)ethyl]-N-methylthiophene-2-carboxamide
—— (5R)-7-[(2-aminopyridin-3-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C13H18N4O2
(5R)-7-[(2-aminopyridin-3-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(3S)-3-(1H-benzimidazol-2-yl)piperidine-1-carbonyl]-3-methyl-1,3-benzoxazol-2-one —— C21H20N4O3
5-[(3S)-3-(1H-benzimidazol-2-yl)piperidine-1-carbonyl]-3-methyl-1,3-benzoxazol-2-one
—— (5R)-3-methyl-7-(quinolin-4-ylmethyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H19N3O2
(5R)-3-methyl-7-(quinolin-4-ylmethyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[6-[(3R)-3-(methoxymethyl)pyrrolidin-1-yl]pyridin-3-yl]-3-(3-phenylpropyl)-1,2,4-oxadiazole —— C22H26N4O2
5-[6-[(3R)-3-(methoxymethyl)pyrrolidin-1-yl]pyridin-3-yl]-3-(3-phenylpropyl)-1,2,4-oxadiazole
—— 5-methyl-7-[(3R)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C20H22N6
5-methyl-7-[(3R)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— 5-methylsulfonyl-N-(oxan-4-ylmethyl)-4-[(3S)-piperidin-3-yl]pyrimidin-2-amine —— C16H26N4O3S
5-methylsulfonyl-N-(oxan-4-ylmethyl)-4-[(3S)-piperidin-3-yl]pyrimidin-2-amine
—— 5-methyl-7-[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C20H22N6
5-methyl-7-[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— (5S)-5-[[2-[3-(3,5-dimethylpyrazol-1-yl)phenyl]imidazol-1-yl]methyl]-1-methylpyrrolidin-2-one —— C20H23N5O
(5S)-5-[[2-[3-(3,5-dimethylpyrazol-1-yl)phenyl]imidazol-1-yl]methyl]-1-methylpyrrolidin-2-one
—— 5-methyl-N-[(2R)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C13H16N6
5-methyl-N-[(2R)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]-5-oxopentanamide —— C18H30N6O2
5-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]-5-oxopentanamide
—— 5-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]-5-oxopentanamide —— C18H30N6O2
5-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]-5-oxopentanamide
—— (5R)-5-[[2-[3-(3,5-dimethylpyrazol-1-yl)phenyl]imidazol-1-yl]methyl]-1-methylpyrrolidin-2-one —— C20H23N5O
(5R)-5-[[2-[3-(3,5-dimethylpyrazol-1-yl)phenyl]imidazol-1-yl]methyl]-1-methylpyrrolidin-2-one
—— 5-methylsulfonyl-N-(oxan-4-ylmethyl)-4-[(3R)-piperidin-3-yl]pyrimidin-2-amine —— C16H26N4O3S
5-methylsulfonyl-N-(oxan-4-ylmethyl)-4-[(3R)-piperidin-3-yl]pyrimidin-2-amine
—— 5-methyl-N-[(2S)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C13H16N6
5-methyl-N-[(2S)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-3-methyl-7-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C20H21N5O2
(5R)-3-methyl-7-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[6-[(3S)-3-(methoxymethyl)pyrrolidin-1-yl]pyridin-3-yl]-3-(3-phenylpropyl)-1,2,4-oxadiazole —— C22H26N4O2
5-[6-[(3S)-3-(methoxymethyl)pyrrolidin-1-yl]pyridin-3-yl]-3-(3-phenylpropyl)-1,2,4-oxadiazole
—— 5-(4-fluorophenyl)-N-[(2R)-1-pyridin-4-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H18FN5
5-(4-fluorophenyl)-N-[(2R)-1-pyridin-4-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(2,4-dichlorophenyl)-N-[(2S)-1-(ethylamino)-1-oxopropan-2-yl]furan-2-carboxamide —— C16H16Cl2N2O3
5-(2,4-dichlorophenyl)-N-[(2S)-1-(ethylamino)-1-oxopropan-2-yl]furan-2-carboxamide
—— 5-(2,4-dichlorophenyl)-N-[(2R)-1-(ethylamino)-1-oxopropan-2-yl]furan-2-carboxamide —— C16H16Cl2N2O3
5-(2,4-dichlorophenyl)-N-[(2R)-1-(ethylamino)-1-oxopropan-2-yl]furan-2-carboxamide
—— 5-(4-fluorophenyl)-N-[(2S)-1-pyridin-4-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H18FN5
5-(4-fluorophenyl)-N-[(2S)-1-pyridin-4-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(piperidin-4-ylmethyl)pyrimidin-2-amine —— C16H27N5O2S
5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(piperidin-4-ylmethyl)pyrimidin-2-amine
—— 5-chloro-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-2-fluorobenzamide —— C17H14Cl2FNO3
5-chloro-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-2-fluorobenzamide
—— 5-chloro-N-[3-(dimethylsulfamoyl)-4-ethoxyphenyl]-2-fluorobenzamide —— C17H18ClFN2O4S
5-chloro-N-[3-(dimethylsulfamoyl)-4-ethoxyphenyl]-2-fluorobenzamide
—— 5-ethyl-N-[(1R)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine —— C17H23N5O
5-ethyl-N-[(1R)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(2-fluorophenyl)-N-[(3R)-thiolan-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H15FN4S
5-(2-fluorophenyl)-N-[(3R)-thiolan-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-acetyl-N-[(2-methoxy-5-methylphenyl)methyl]-N-methylthiophene-2-carboxamide —— C17H19NO3S
5-acetyl-N-[(2-methoxy-5-methylphenyl)methyl]-N-methylthiophene-2-carboxamide
—— (5S)-3-methyl-7-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C20H21N5O2
(5S)-3-methyl-7-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-chloro-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-2-nitrobenzamide —— C17H14Cl2N2O5
5-chloro-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-2-nitrobenzamide
—— 5-(4-fluorophenyl)-N-[(2-methoxy-5-methylphenyl)methyl]-N-methylfuran-2-carboxamide —— C21H20FNO3
5-(4-fluorophenyl)-N-[(2-methoxy-5-methylphenyl)methyl]-N-methylfuran-2-carboxamide
—— 5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(piperidin-4-ylmethyl)pyrimidin-2-amine —— C16H27N5O2S
5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(piperidin-4-ylmethyl)pyrimidin-2-amine
—— 5-(2-chlorophenyl)-N-[2-(2-nitroanilino)ethyl]furan-2-carboxamide —— C19H16ClN3O4
5-(2-chlorophenyl)-N-[2-(2-nitroanilino)ethyl]furan-2-carboxamide
—— (5R)-2-(1,3-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C16H22N6O
(5R)-2-(1,3-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-(4-fluorophenyl)-N-[2-(2-nitroanilino)ethyl]furan-2-carboxamide —— C19H16FN3O4
5-(4-fluorophenyl)-N-[2-(2-nitroanilino)ethyl]furan-2-carboxamide
—— 5-[[(3S)-3-(3-methylphenyl)piperidin-1-yl]methyl]-2-pyrrolidin-1-yl-1,3-thiazole —— C20H27N3S
5-[[(3S)-3-(3-methylphenyl)piperidin-1-yl]methyl]-2-pyrrolidin-1-yl-1,3-thiazole
—— 5-(4-fluorophenyl)-N-methyl-N-[[(2R)-oxan-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H21FN4O
5-(4-fluorophenyl)-N-methyl-N-[[(2R)-oxan-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[3-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C17H27N3O4
5-[3-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— 5-chloro-2-nitro-N-[2-(2-nitroanilino)ethyl]benzamide —— C15H13ClN4O5
5-chloro-2-nitro-N-[2-(2-nitroanilino)ethyl]benzamide
—— 5-[2-[(2S)-2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl]-3-methyl-1H-pyrimidine-2,4-dione —— C17H18FN3O3
5-[2-[(2S)-2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl]-3-methyl-1H-pyrimidine-2,4-dione
—— 5-acetyl-N-[2-(2-nitroanilino)ethyl]thiophene-2-carboxamide —— C15H15N3O4S
5-acetyl-N-[2-(2-nitroanilino)ethyl]thiophene-2-carboxamide
—— 5-[6-[(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]pyridin-3-yl]-3-(methoxymethyl)-1,2,4-oxadiazole —— C21H22N6O2
5-[6-[(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]pyridin-3-yl]-3-(methoxymethyl)-1,2,4-oxadiazole
—— 5-(1,3-benzothiazol-2-yl)-N-[2-(2-nitroanilino)ethyl]furan-2-carboxamide —— C20H16N4O4S
5-(1,3-benzothiazol-2-yl)-N-[2-(2-nitroanilino)ethyl]furan-2-carboxamide
—— 5-fluoro-3-methyl-N-[2-(2-nitroanilino)ethyl]-1-benzofuran-2-carboxamide —— C18H16FN3O4
5-fluoro-3-methyl-N-[2-(2-nitroanilino)ethyl]-1-benzofuran-2-carboxamide
—— [5-(methylsulfanylmethyl)furan-2-yl]-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone —— C18H28N2O3S
[5-(methylsulfanylmethyl)furan-2-yl]-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone
—— 5-[2-[(2R)-2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl]-3-methyl-1H-pyrimidine-2,4-dione —— C17H18FN3O3
5-[2-[(2R)-2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl]-3-methyl-1H-pyrimidine-2,4-dione
—— 5-chloro-2-fluoro-N-[2-(2-nitroanilino)ethyl]benzamide —— C15H13ClFN3O3
5-chloro-2-fluoro-N-[2-(2-nitroanilino)ethyl]benzamide
—— 5-acetyl-N-[(1R)-1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]thiophene-2-carboxamide —— C19H21NO2S
5-acetyl-N-[(1R)-1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]thiophene-2-carboxamide