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—— 5-phenyl-7-[(3S)-3-phenylpiperazin-1-yl]pyrazolo[1,5-a]pyrimidine —— C22H21N5
5-phenyl-7-[(3S)-3-phenylpiperazin-1-yl]pyrazolo[1,5-a]pyrimidine
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-11-methyl-3-pyridin-4-yl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C18H15N5O4S
5-[(3S)-1,1-dioxothiolan-3-yl]-11-methyl-3-pyridin-4-yl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-11-methyl-3-pyridin-3-yl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C18H15N5O4S
5-[(3R)-1,1-dioxothiolan-3-yl]-11-methyl-3-pyridin-3-yl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-3-(4-methoxyphenyl)-11-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H18N4O5S
5-[(3R)-1,1-dioxothiolan-3-yl]-3-(4-methoxyphenyl)-11-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-(4-fluorophenyl)-N-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H16FN5S
5-(4-fluorophenyl)-N-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-7-(9H-fluoren-2-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C21H22N2O2
(5S)-7-(9H-fluoren-2-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-11-methyl-3-phenyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C19H16N4O4S
5-[(3R)-1,1-dioxothiolan-3-yl]-11-methyl-3-phenyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-11-methyl-3-phenyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C19H16N4O4S
5-[(3S)-1,1-dioxothiolan-3-yl]-11-methyl-3-phenyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-3-(4-methoxyphenyl)-11-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H18N4O5S
5-[(3S)-1,1-dioxothiolan-3-yl]-3-(4-methoxyphenyl)-11-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one —— C18H22N4O3
5-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one
—— (5S)-9-[[5-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H19N5O3S
(5S)-9-[[5-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[3-[(3S)-3-[5-[(dimethylamino)methyl]-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C17H26N6O3
5-[3-[(3S)-3-[5-[(dimethylamino)methyl]-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— [5-(hydroxymethyl)furan-2-yl]-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone —— C17H26N2O4
[5-(hydroxymethyl)furan-2-yl]-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(2-nitrophenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C19H15N5O6S
5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(2-nitrophenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[3-[(3R)-3-[5-[(dimethylamino)methyl]-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C17H26N6O3
5-[3-[(3R)-3-[5-[(dimethylamino)methyl]-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— 5-ethyl-N-[(1R)-1-[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine —— C17H25N7O
5-ethyl-N-[(1R)-1-[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-tert-butyl-4-[[(3R)-4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl]furan-2-carboxamide —— C21H35N3O3
5-tert-butyl-4-[[(3R)-4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl]furan-2-carboxamide
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-11-(4-methoxyphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H18N4O5S
5-[(3R)-1,1-dioxothiolan-3-yl]-11-(4-methoxyphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(4-methylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H18N4O4S
5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(4-methylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-11-(2-fluoro-4-methylphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H17FN4O4S
5-[(3S)-1,1-dioxothiolan-3-yl]-11-(2-fluoro-4-methylphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— (5S)-7-[(3,4-difluorophenyl)methyl]-2-(1,3-dihydroxypropan-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24F2N2O3
(5S)-7-[(3,4-difluorophenyl)methyl]-2-(1,3-dihydroxypropan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-11-(2-fluorophenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C19H15FN4O4S
5-[(3S)-1,1-dioxothiolan-3-yl]-11-(2-fluorophenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-[4-(trifluoromethoxy)phenyl]-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H15F3N4O5S
5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-[4-(trifluoromethoxy)phenyl]-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— (5R)-9-[[5-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H19N5O3S
(5R)-9-[[5-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(4-Benzyl-5-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-3-(3-chlorophenyl)-1,2,4-oxadiazole —— C19H16ClN5OS
5-[(4-Benzyl-5-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-3-(3-chlorophenyl)-1,2,4-oxadiazole
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(4-propan-2-ylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C22H22N4O4S
5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(4-propan-2-ylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(4-Benzyl-5-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-3-(4-ethylphenyl)-1,2,4-oxadiazole —— C21H21N5OS
5-[(4-Benzyl-5-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-3-(4-ethylphenyl)-1,2,4-oxadiazole
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(3,4,5-trimethoxyphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C22H22N4O7S
5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(3,4,5-trimethoxyphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— (5R)-3-methyl-N-[4-morpholin-4-yl-1-(2,2,2-trifluoroethyl)indazol-3-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H20F3N5O3
(5R)-3-methyl-N-[4-morpholin-4-yl-1-(2,2,2-trifluoroethyl)indazol-3-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(2-phenylethyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C21H20N4O4S
5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(2-phenylethyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(2-phenylethyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C21H20N4O4S
5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(2-phenylethyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-[3-(trifluoromethoxy)phenyl]-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H15F3N4O5S
5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-[3-(trifluoromethoxy)phenyl]-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— (5S)-3-methyl-N-[4-morpholin-4-yl-1-(2,2,2-trifluoroethyl)indazol-3-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H20F3N5O3
(5S)-3-methyl-N-[4-morpholin-4-yl-1-(2,2,2-trifluoroethyl)indazol-3-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-11-(2-fluoro-4-methylphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H17FN4O4S
5-[(3R)-1,1-dioxothiolan-3-yl]-11-(2-fluoro-4-methylphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-11-(2-methoxyphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H18N4O5S
5-[(3R)-1,1-dioxothiolan-3-yl]-11-(2-methoxyphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-[3-(trifluoromethyl)phenyl]-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H15F3N4O4S
5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-[3-(trifluoromethyl)phenyl]-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-11-(4-methoxyphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H18N4O5S
5-[(3S)-1,1-dioxothiolan-3-yl]-11-(4-methoxyphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[[(2R)-2-[4-[(dimethylamino)methyl]phenyl]piperidin-1-yl]methyl]-N,N-dimethyl-1,3-thiazol-2-amine —— C20H30N4S
5-[[(2R)-2-[4-[(dimethylamino)methyl]phenyl]piperidin-1-yl]methyl]-N,N-dimethyl-1,3-thiazol-2-amine
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(2-methylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H18N4O4S
5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(2-methylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-11-(2-methoxyphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H18N4O5S
5-[(3S)-1,1-dioxothiolan-3-yl]-11-(2-methoxyphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(3,4,5-trimethoxyphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C22H22N4O7S
5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(3,4,5-trimethoxyphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— (5S)-9-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H17N5O3
(5S)-9-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H17N5O3
(5R)-9-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-11-(3-methoxyphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H18N4O5S
5-[(3S)-1,1-dioxothiolan-3-yl]-11-(3-methoxyphenyl)-3-methyl-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-[4-(trifluoromethoxy)phenyl]-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H15F3N4O5S
5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-[4-(trifluoromethoxy)phenyl]-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(4-propan-2-ylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C22H22N4O4S
5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(4-propan-2-ylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(4-nitrophenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C19H15N5O6S
5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(4-nitrophenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(3-methylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H18N4O4S
5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(3-methylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(2-methylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C20H18N4O4S
5-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-11-(2-methylphenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione
—— 5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(3-nitrophenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione —— C19H15N5O6S
5-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-11-(3-nitrophenyl)-4,5,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8-tetraene-10,12-dione