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—— 5-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-3-one —— C20H23N9O
5-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[4-(trifluoromethoxy)phenyl]-1H-pyrazol-3-one —— C22H24F3N5O2
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[4-(trifluoromethoxy)phenyl]-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4-fluorophenyl)-1H-pyrazol-3-one —— C21H24FN5O
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4-fluorophenyl)-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-fluorophenyl)-1H-pyrazol-3-one —— C21H24FN5O
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-fluorophenyl)-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[4-(trifluoromethyl)phenyl]-1H-pyrazol-3-one —— C22H24F3N5O
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[4-(trifluoromethyl)phenyl]-1H-pyrazol-3-one
—— 5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-3-one —— C21H27N7O
5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-phenyl-1H-pyrazol-3-one —— C21H25N5O
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-phenyl-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4-methoxyphenyl)-1H-pyrazol-3-one —— C22H27N5O2
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4-methoxyphenyl)-1H-pyrazol-3-one
—— 5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-pyridin-2-yl-1H-pyrazol-3-one —— C20H24N6O
5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-pyridin-2-yl-1H-pyrazol-3-one
—— 5-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-1,2-dihydropyrazol-3-one —— C15H21N5O
5-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-1,2-dihydropyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-methylphenyl)-1H-pyrazol-3-one —— C22H27N5O
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-methylphenyl)-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-3-one —— C20H23N9O
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-methylphenyl)-1H-pyrazol-3-one —— C22H27N5O
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-methylphenyl)-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-3-one —— C21H27N7O
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(6-methoxy-1,3-benzothiazol-2-yl)-1H-pyrazol-3-one —— C23H26N6O2S
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(6-methoxy-1,3-benzothiazol-2-yl)-1H-pyrazol-3-one
—— 5-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(6-methoxy-1,3-benzothiazol-2-yl)-1H-pyrazol-3-one —— C23H26N6O2S
5-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(6-methoxy-1,3-benzothiazol-2-yl)-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-3-one —— C21H25N9O
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[(3R)-1,1-dioxothiolan-3-yl]-1H-pyrazol-3-one —— C19H27N5O3S
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[(3R)-1,1-dioxothiolan-3-yl]-1H-pyrazol-3-one
—— 5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4-methoxyphenyl)-1H-pyrazol-3-one —— C22H27N5O2
5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4-methoxyphenyl)-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-1,2-dihydropyrazol-3-one —— C15H21N5O
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-1,2-dihydropyrazol-3-one
—— 5-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[(3R)-1,1-dioxothiolan-3-yl]-1H-pyrazol-3-one —— C19H27N5O3S
5-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[(3R)-1,1-dioxothiolan-3-yl]-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-methylphenyl)-1H-pyrazol-3-one —— C22H27N5O
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-methylphenyl)-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-methoxyphenyl)-1H-pyrazol-3-one —— C22H27N5O2
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-methoxyphenyl)-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4-methoxyphenyl)-1H-pyrazol-3-one —— C22H27N5O2
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4-methoxyphenyl)-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-pyridin-2-yl-1H-pyrazol-3-one —— C20H24N6O
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-pyridin-2-yl-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-fluorophenyl)-1H-pyrazol-3-one —— C21H24FN5O
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-fluorophenyl)-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-pyridin-2-yl-1H-pyrazol-3-one —— C20H24N6O
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-pyridin-2-yl-1H-pyrazol-3-one
—— 5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-methylphenyl)-1H-pyrazol-3-one —— C22H27N5O
5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-methylphenyl)-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[4-(trifluoromethyl)phenyl]-1H-pyrazol-3-one —— C22H24F3N5O
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[4-(trifluoromethyl)phenyl]-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4-fluorophenyl)-1H-pyrazol-3-one —— C21H24FN5O
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(4-fluorophenyl)-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-methoxyphenyl)-1H-pyrazol-3-one —— C22H27N5O2
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(2-methoxyphenyl)-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-phenyl-1H-pyrazol-3-one —— C21H25N5O
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-phenyl-1H-pyrazol-3-one
—— 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[(3R)-1,1-dioxothiolan-3-yl]-1H-pyrazol-3-one —— C19H27N5O3S
5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[(3R)-1,1-dioxothiolan-3-yl]-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-3-one —— C21H25N9O
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-3-one
—— (5-methyl-1,2-oxazol-3-yl)methyl (2R)-1-(1,1-dioxo-1,2-benzothiazol-3-yl)piperidine-2-carboxylate —— C18H19N3O5S
(5-methyl-1,2-oxazol-3-yl)methyl (2R)-1-(1,1-dioxo-1,2-benzothiazol-3-yl)piperidine-2-carboxylate
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-fluorophenyl)-1H-pyrazol-3-one —— C21H24FN5O
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-fluorophenyl)-1H-pyrazol-3-one
—— 5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[4-(trifluoromethoxy)phenyl]-1H-pyrazol-3-one —— C22H24F3N5O2
5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-[4-(trifluoromethoxy)phenyl]-1H-pyrazol-3-one
—— 5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-fluorophenyl)-1H-pyrazol-3-one —— C21H24FN5O
5-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-fluorophenyl)-1H-pyrazol-3-one
—— 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-methylphenyl)-1H-pyrazol-3-one —— C22H27N5O
5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-methylphenyl)-1H-pyrazol-3-one
—— (5-Chloro-2-methoxyphenyl)methyl 2-(1,2-benzoxazol-3-yl)acetate —— C17H14ClNO4
(5-Chloro-2-methoxyphenyl)methyl 2-(1,2-benzoxazol-3-yl)acetate
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate —— C19H15N3O4S
(5-Phenyl-1,2-oxazol-3-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate —— C19H15N3O4S
(5-Phenyl-1,3-oxazol-2-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate
—— (5-Acetyl-2-methoxyphenyl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate —— C19H18N2O5S
(5-Acetyl-2-methoxyphenyl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate —— C16H12N4O4S2
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate —— C18H14N4O4S
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate
—— 5-ethoxy-1-[[(3R)-3-hydroxypiperidin-1-yl]methyl]-3-[[(3S)-3-hydroxypiperidin-1-yl]methyl]benzimidazole-2-thione —— C21H32N4O3S
5-ethoxy-1-[[(3R)-3-hydroxypiperidin-1-yl]methyl]-3-[[(3S)-3-hydroxypiperidin-1-yl]methyl]benzimidazole-2-thione
—— 5-bromo-N-[2-(4-methylpiperazin-4-ium-1-yl)phenyl]thiophene-2-sulfonamide —— C15H19BrN3O2S2+
5-bromo-N-[2-(4-methylpiperazin-4-ium-1-yl)phenyl]thiophene-2-sulfonamide
—— 5-ethoxy-1-[[(3R)-3-hydroxypiperidin-1-ium-1-yl]methyl]-3-[[(3S)-3-hydroxypiperidin-1-ium-1-yl]methyl]benzimidazole-2-thione —— C21H34N4O3S+2
5-ethoxy-1-[[(3R)-3-hydroxypiperidin-1-ium-1-yl]methyl]-3-[[(3S)-3-hydroxypiperidin-1-ium-1-yl]methyl]benzimidazole-2-thione
—— (5E)-5-[(4-tert-butylphenyl)methylidene]-3-(2,6-diethylphenyl)-1-methyl-2-sulfanylideneimidazolidin-4-one —— C25H30N2OS
(5E)-5-[(4-tert-butylphenyl)methylidene]-3-(2,6-diethylphenyl)-1-methyl-2-sulfanylideneimidazolidin-4-one
—— 5-chloro-N-(4-ethoxy-3-methoxyphenyl)thiophene-2-sulfonamide —— C13H14ClNO4S2
5-chloro-N-(4-ethoxy-3-methoxyphenyl)thiophene-2-sulfonamide