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—— (5-ethyl-1H-pyrazol-4-yl)-[(2S)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methanone —— C18H21N5O
(5-ethyl-1H-pyrazol-4-yl)-[(2S)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methanone
—— 5-(4-fluorophenyl)-N-[(3R)-thiolan-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H15FN4S
5-(4-fluorophenyl)-N-[(3R)-thiolan-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-2-[(2,4-dimethyl-6-pyrazol-1-ylphenyl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C21H28N4O
(5S)-2-[(2,4-dimethyl-6-pyrazol-1-ylphenyl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]pyrimidin-2-amine —— C15H22N6O2S
5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]pyrimidin-2-amine
—— 5-ethyl-2,3-dimethyl-7-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C21H27N5O
5-ethyl-2,3-dimethyl-7-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— 5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-(2-propan-2-ylsulfanylethyl)pyridazin-3-one —— C15H26N4O2S
5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-(2-propan-2-ylsulfanylethyl)pyridazin-3-one
—— 5,6-Dimethyl-3-prop-2-enyl-2-(quinolin-2-ylmethylsulfanyl)thieno[2,3-d]pyrimidin-4-one —— C21H19N3OS2
5,6-Dimethyl-3-prop-2-enyl-2-(quinolin-2-ylmethylsulfanyl)thieno[2,3-d]pyrimidin-4-one
—— (5S)-7-[[2-(benzylamino)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C19H23N5O2
(5S)-7-[[2-(benzylamino)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-7-[(E)-3-(4-methoxyphenyl)prop-2-enyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H22N2O3
(5R)-7-[(E)-3-(4-methoxyphenyl)prop-2-enyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-7-[(E)-3-(4-methoxyphenyl)prop-2-enyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H22N2O3
(5S)-7-[(E)-3-(4-methoxyphenyl)prop-2-enyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[[4-(3-hydroxy-3-methylbutyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H30N2O3
(5S)-9-[[4-(3-hydroxy-3-methylbutyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5,6-dimethyl-2-[(1S)-1-(3-nitrophenyl)ethyl]sulfanyl-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one —— C19H19N3O3S2
5,6-dimethyl-2-[(1S)-1-(3-nitrophenyl)ethyl]sulfanyl-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one
—— 5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-(2-propan-2-ylsulfanylethyl)pyridazin-3-one —— C15H26N4O2S
5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-(2-propan-2-ylsulfanylethyl)pyridazin-3-one
—— 5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]pyrimidin-2-amine —— C15H22N6O2S
5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]pyrimidin-2-amine
—— (5R)-9-[5-(tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C12H14N8O3
(5R)-9-[5-(tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-propyl-N-[(5S)-4,5,6,7-tetrahydro-1H-indazol-5-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H20N6
5-propyl-N-[(5S)-4,5,6,7-tetrahydro-1H-indazol-5-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(4-fluorophenyl)-N-[(3S)-thiolan-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H15FN4S
5-(4-fluorophenyl)-N-[(3S)-thiolan-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-ethyl-2,3-dimethyl-7-[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C21H27N5O
5-ethyl-2,3-dimethyl-7-[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— (5R)-7-methyl-2-[[5-[2-(methylamino)acetyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H30N6O2
(5R)-7-methyl-2-[[5-[2-(methylamino)acetyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-methyl-2-[[5-[2-(methylamino)acetyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H30N6O2
(5S)-7-methyl-2-[[5-[2-(methylamino)acetyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— [(5S)-5-methyl-4,5,6,7-tetrahydro-1H-indazol-3-yl]-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methanone —— C19H26N4OS
[(5S)-5-methyl-4,5,6,7-tetrahydro-1H-indazol-3-yl]-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methanone
—— (5R)-9-[[4-(3-hydroxy-3-methylbutyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H30N2O3
(5R)-9-[[4-(3-hydroxy-3-methylbutyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-chloro-N-[(3R)-2-oxopyrrolidin-3-yl]-3-phenyl-1H-indole-2-carboxamide —— C19H16ClN3O2
5-chloro-N-[(3R)-2-oxopyrrolidin-3-yl]-3-phenyl-1H-indole-2-carboxamide
—— (5-Chloro-2-methoxyphenyl)methyl 2-[(3,4-dimethylbenzoyl)amino]acetate —— C19H20ClNO4
(5-Chloro-2-methoxyphenyl)methyl 2-[(3,4-dimethylbenzoyl)amino]acetate
—— (5-methyl-1,2-oxazol-3-yl)-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C18H26N6O2
(5-methyl-1,2-oxazol-3-yl)-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— (5S)-9-(6-chloro-8-methylquinolin-4-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20ClN3O2
(5S)-9-(6-chloro-8-methylquinolin-4-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[2-[(2S)-2-(aminomethyl)morpholin-4-yl]pyrimidin-4-yl]-2-ethoxybenzoic acid —— C18H22N4O4
5-[2-[(2S)-2-(aminomethyl)morpholin-4-yl]pyrimidin-4-yl]-2-ethoxybenzoic acid
—— (5R)-9-[[2-[3-(dimethylamino)propoxy]phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H31N3O3
(5R)-9-[[2-[3-(dimethylamino)propoxy]phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-(piperidin-1-ylmethyl)-2-[(2S)-1-pyrrolidin-1-ylhex-5-en-2-yl]oxypyridine —— C21H33N3O
5-(piperidin-1-ylmethyl)-2-[(2S)-1-pyrrolidin-1-ylhex-5-en-2-yl]oxypyridine
—— (5S)-3-methyl-9-[(3-phenoxyphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C21H24N2O3
(5S)-3-methyl-9-[(3-phenoxyphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[2-[(2R)-2-(aminomethyl)morpholin-4-yl]pyrimidin-4-yl]-2-ethoxybenzoic acid —— C18H22N4O4
5-[2-[(2R)-2-(aminomethyl)morpholin-4-yl]pyrimidin-4-yl]-2-ethoxybenzoic acid
—— 5-(piperidin-1-ylmethyl)-2-[(2R)-1-pyrrolidin-1-ylhex-5-en-2-yl]oxypyridine —— C21H33N3O
5-(piperidin-1-ylmethyl)-2-[(2R)-1-pyrrolidin-1-ylhex-5-en-2-yl]oxypyridine
—— (5-ethylthiophen-2-yl)-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone —— C18H28N2O2S
(5-ethylthiophen-2-yl)-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone
—— 5-chloro-N-[(3S)-2-oxopyrrolidin-3-yl]-3-phenyl-1H-indole-2-carboxamide —— C19H16ClN3O2
5-chloro-N-[(3S)-2-oxopyrrolidin-3-yl]-3-phenyl-1H-indole-2-carboxamide
—— (5-ethylthiophen-2-yl)-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone —— C18H28N2O2S
(5-ethylthiophen-2-yl)-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone
—— 5-(4-fluorophenyl)-N-[(1S)-1-(2-propyl-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H20FN7
5-(4-fluorophenyl)-N-[(1S)-1-(2-propyl-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-9-[2-amino-6-(4-methylphenyl)sulfanylpyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H23N5O2S
(5R)-9-[2-amino-6-(4-methylphenyl)sulfanylpyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[[2-[3-(dimethylamino)propoxy]phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H31N3O3
(5S)-9-[[2-[3-(dimethylamino)propoxy]phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-(4-fluorophenyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C22H18FN7
5-(4-fluorophenyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(4-fluorophenyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C22H18FN7
5-(4-fluorophenyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5-methyl-1,2-oxazol-3-yl)-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C18H26N6O2
(5-methyl-1,2-oxazol-3-yl)-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— [5-[[(4S)-4-(3-methyl-1-benzofuran-2-yl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methyl]furan-2-yl]methanol —— C21H21N3O3
[5-[[(4S)-4-(3-methyl-1-benzofuran-2-yl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methyl]furan-2-yl]methanol
—— 5-ethyl-N-[3-[(3R)-oxolan-3-yl]propyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C15H22N4O
5-ethyl-N-[3-[(3R)-oxolan-3-yl]propyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-ethyl-N-[3-[(3S)-oxolan-3-yl]propyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C15H22N4O
5-ethyl-N-[3-[(3S)-oxolan-3-yl]propyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-chloro-4-[(2Z)-2-[[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]methylidene]hydrazinyl]-1H-pyridazin-6-one —— C13H13ClN4O2
5-chloro-4-[(2Z)-2-[[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]methylidene]hydrazinyl]-1H-pyridazin-6-one
—— (5S)-9-[2-amino-6-(4-methylphenyl)sulfanylpyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H23N5O2S
(5S)-9-[2-amino-6-(4-methylphenyl)sulfanylpyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(4S)-5-(furan-2-ylmethyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-3-phenyl-1,2-oxazole —— C20H18N4O2
5-[(4S)-5-(furan-2-ylmethyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-3-phenyl-1,2-oxazole
—— 5-chloro-4-[(2Z)-2-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methylidene]hydrazinyl]-1H-pyridazin-6-one —— C13H13ClN4O2
5-chloro-4-[(2Z)-2-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methylidene]hydrazinyl]-1H-pyridazin-6-one
—— (5R)-3-methyl-9-[(3-phenoxyphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C21H24N2O3
(5R)-3-methyl-9-[(3-phenoxyphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-(4-fluorophenyl)-N-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H21FN6
5-(4-fluorophenyl)-N-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine