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—— [5-(methylsulfanylmethyl)furan-2-yl]-[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methanone —— C16H18N2O2S
[5-(methylsulfanylmethyl)furan-2-yl]-[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methanone
—— 5-[5-methylsulfonyl-4-[(3S)-piperidin-3-yl]pyrimidin-2-yl]-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-2-amine —— C16H22N6O2S2
5-[5-methylsulfonyl-4-[(3S)-piperidin-3-yl]pyrimidin-2-yl]-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-2-amine
—— 5-[(E)-but-2-enyl]-2-[[(3S)-3-(imidazol-1-ylmethyl)piperidin-1-yl]methyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine —— C21H32N6
5-[(E)-but-2-enyl]-2-[[(3S)-3-(imidazol-1-ylmethyl)piperidin-1-yl]methyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine
—— (5R)-9-[(2-fluorophenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane —— C19H23FN4
(5R)-9-[(2-fluorophenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane
—— 5-[5-methylsulfonyl-4-[(3R)-piperidin-3-yl]pyrimidin-2-yl]-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-2-amine —— C16H22N6O2S2
5-[5-methylsulfonyl-4-[(3R)-piperidin-3-yl]pyrimidin-2-yl]-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-2-amine
—— 5-chloro-N-[2-(4-methylpiperazin-4-ium-1-yl)phenyl]thiophene-2-sulfonamide —— C15H19ClN3O2S2+
5-chloro-N-[2-(4-methylpiperazin-4-ium-1-yl)phenyl]thiophene-2-sulfonamide
—— [5-(methylsulfanylmethyl)furan-2-yl]-[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methanone —— C16H18N2O2S
[5-(methylsulfanylmethyl)furan-2-yl]-[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methanone
—— 5-chloro-N-[(3S)-2-oxopiperidin-3-yl]-3-phenyl-1H-indole-2-carboxamide —— C20H18ClN3O2
5-chloro-N-[(3S)-2-oxopiperidin-3-yl]-3-phenyl-1H-indole-2-carboxamide
—— 5-chloro-N-[(3R)-2-oxopiperidin-3-yl]-3-phenyl-1H-indole-2-carboxamide —— C20H18ClN3O2
5-chloro-N-[(3R)-2-oxopiperidin-3-yl]-3-phenyl-1H-indole-2-carboxamide
—— 5-bromo-N-(4-ethoxy-3-methoxyphenyl)thiophene-2-sulfonamide —— C13H14BrNO4S2
5-bromo-N-(4-ethoxy-3-methoxyphenyl)thiophene-2-sulfonamide
—— (5S)-9-furo[3,2-c]pyridin-4-yl-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H17N3O3
(5S)-9-furo[3,2-c]pyridin-4-yl-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-chloro-N-[4-(4-ethylpiperazin-1-yl)phenyl]thiophene-2-sulfonamide —— C16H20ClN3O2S2
5-chloro-N-[4-(4-ethylpiperazin-1-yl)phenyl]thiophene-2-sulfonamide
—— (5R)-9-[[3-(4-chlorophenoxy)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C21H23ClN2O3
(5R)-9-[[3-(4-chlorophenoxy)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-chloro-N-[4-(4-ethylpiperazin-4-ium-1-yl)phenyl]thiophene-2-sulfonamide —— C16H21ClN3O2S2+
5-chloro-N-[4-(4-ethylpiperazin-4-ium-1-yl)phenyl]thiophene-2-sulfonamide
—— (5R)-1-methyl-5-[[(5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]methyl]pyrrolidin-2-one —— C15H21N5O
(5R)-1-methyl-5-[[(5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]methyl]pyrrolidin-2-one
—— 5-chloro-N-(3-(2-methylthiazol-4-yl)phenyl)thiophene-2-sulfonamide —— C14H11ClN2O2S3
5-chloro-N-(3-(2-methylthiazol-4-yl)phenyl)thiophene-2-sulfonamide
—— (5R)-3-methyl-7-(2-phenylquinolin-4-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C22H21N3O2
(5R)-3-methyl-7-(2-phenylquinolin-4-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-ethyl-7-[3-[(2S)-2-methylpiperidin-1-yl]azetidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C17H25N5
5-ethyl-7-[3-[(2S)-2-methylpiperidin-1-yl]azetidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— (5-methyl-3-phenyl-1,2-oxazol-4-yl)-[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methanone —— C20H19N3O2
(5-methyl-3-phenyl-1,2-oxazol-4-yl)-[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methanone
—— 5-bromo-N-(4-ethoxy-3-methoxyphenyl)-2-methoxybenzenesulfonamide —— C16H18BrNO5S
5-bromo-N-(4-ethoxy-3-methoxyphenyl)-2-methoxybenzenesulfonamide
—— (5S)-1-methyl-5-[[(5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]methyl]pyrrolidin-2-one —— C15H21N5O
(5S)-1-methyl-5-[[(5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]methyl]pyrrolidin-2-one
—— 5-bromo-N-[4-(4-methylpiperazin-1-yl)phenyl]thiophene-2-sulfonamide —— C15H18BrN3O2S2
5-bromo-N-[4-(4-methylpiperazin-1-yl)phenyl]thiophene-2-sulfonamide
—— 5-[(1R)-1-[(2-methyl-5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]ethyl]-1,2-dihydro-1,2,4-triazol-3-one —— C14H19N7O
5-[(1R)-1-[(2-methyl-5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]ethyl]-1,2-dihydro-1,2,4-triazol-3-one
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-(diethylamino)benzoate —— C20H20N4O5
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-(diethylamino)benzoate
—— 5-ethyl-2,3-dimethyl-N-[(1R)-1-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H21N7O
5-ethyl-2,3-dimethyl-N-[(1R)-1-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-phenyl-N-[(1R)-1-thiophen-3-ylethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H16N4S
5-phenyl-N-[(1R)-1-thiophen-3-ylethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-(diethylamino)benzoate —— C18H19N3O4
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-(diethylamino)benzoate
—— (5R)-9-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H25N5O3
(5R)-9-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-2-[1-(2,3-dimethylphenyl)piperidin-4-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C22H33N3O
(5S)-2-[1-(2,3-dimethylphenyl)piperidin-4-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(2S)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one —— C18H20FN5O
5-[[(2S)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
—— 5-ethyl-2,3-dimethyl-N-[(1S)-1-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H21N7O
5-ethyl-2,3-dimethyl-N-[(1S)-1-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-ethyl-7-[3-[(2R)-2-methylpiperidin-1-yl]azetidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C17H25N5
5-ethyl-7-[3-[(2R)-2-methylpiperidin-1-yl]azetidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— (5-methyl-3-phenyl-1,2-oxazol-4-yl)-[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methanone —— C20H19N3O2
(5-methyl-3-phenyl-1,2-oxazol-4-yl)-[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methanone
—— 5-methyl-6-[(2R)-2-pyridin-2-ylpyrrolidine-1-carbonyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C17H16N4O2S
5-methyl-6-[(2R)-2-pyridin-2-ylpyrrolidine-1-carbonyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-[(1R)-1-(3-methylpyridin-2-yl)ethyl]pyridin-2-amine —— C18H21N5O2
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-[(1R)-1-(3-methylpyridin-2-yl)ethyl]pyridin-2-amine
—— (5R)-2-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C21H22FN5O
(5R)-2-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 3,5-dichlorobenzoate —— C14H8Cl2N2O4
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 3,5-dichlorobenzoate
—— 5-[[(2R)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one —— C18H20FN5O
5-[[(2R)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
—— (5S)-9-[[3-(4-chlorophenoxy)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C21H23ClN2O3
(5S)-9-[[3-(4-chlorophenoxy)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(1S)-1-[(2-methyl-5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]ethyl]-1,2-dihydro-1,2,4-triazol-3-one —— C14H19N7O
5-[(1S)-1-[(2-methyl-5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]ethyl]-1,2-dihydro-1,2,4-triazol-3-one
—— 5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]pyridin-2-amine —— C18H21N5O2
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]pyridin-2-amine
—— 5-ethyl-N-[(1S)-1-[1-(3-methoxyphenyl)pyrazol-4-yl]ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H22N6O
5-ethyl-N-[(1S)-1-[1-(3-methoxyphenyl)pyrazol-4-yl]ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-(diethylamino)benzoate —— C20H20ClN3O3
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-(diethylamino)benzoate
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 2,6-dichlorobenzoate —— C17H11Cl2NO3
(5-Phenyl-1,3-oxazol-2-yl)methyl 2,6-dichlorobenzoate
—— (5S)-2-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C21H22FN5O
(5S)-2-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[1-(2,3-dimethylphenyl)piperidin-4-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C22H33N3O
(5R)-2-[1-(2,3-dimethylphenyl)piperidin-4-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R,8S)-5-(4-methoxyphenyl)-8-(3-methylphenyl)-1,3,5,7,8,9-hexahydro-[1,2,5]oxadiazolo[3,4-b][1,4]benzodiazepin-6-one —— C23H22N4O3
(5R,8S)-5-(4-methoxyphenyl)-8-(3-methylphenyl)-1,3,5,7,8,9-hexahydro-[1,2,5]oxadiazolo[3,4-b][1,4]benzodiazepin-6-one
—— (5R,8R)-5-(3-methylphenyl)-8-phenyl-1,3,5,7,8,9-hexahydro-[1,2,5]oxadiazolo[3,4-b][1,4]benzodiazepin-6-one —— C22H20N4O2
(5R,8R)-5-(3-methylphenyl)-8-phenyl-1,3,5,7,8,9-hexahydro-[1,2,5]oxadiazolo[3,4-b][1,4]benzodiazepin-6-one
—— (5R,8R)-5-(4-methoxyphenyl)-8-(4-methylphenyl)-1,3,5,7,8,9-hexahydro-[1,2,5]oxadiazolo[3,4-b][1,4]benzodiazepin-6-one —— C23H22N4O3
(5R,8R)-5-(4-methoxyphenyl)-8-(4-methylphenyl)-1,3,5,7,8,9-hexahydro-[1,2,5]oxadiazolo[3,4-b][1,4]benzodiazepin-6-one
—— (5R,8S)-5-(4-hydroxyphenyl)-8-methyl-1,3,5,7,8,9-hexahydro-[1,2,5]oxadiazolo[3,4-b][1,4]benzodiazepin-6-one —— C16H16N4O3
(5R,8S)-5-(4-hydroxyphenyl)-8-methyl-1,3,5,7,8,9-hexahydro-[1,2,5]oxadiazolo[3,4-b][1,4]benzodiazepin-6-one