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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[4-[[(S)-cyclopentyl(thiophen-2-yl)methyl]carbamoylamino]pyrazol-1-yl]acetamide —— C16H21N5O2S
2-[4-[[(S)-cyclopentyl(thiophen-2-yl)methyl]carbamoylamino]pyrazol-1-yl]acetamide
—— [(4aS,8aR)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[2-(furan-2-yl)-1,3-thiazol-4-yl]methanone —— C15H16N2O3S2
[(4aS,8aR)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[2-(furan-2-yl)-1,3-thiazol-4-yl]methanone
—— N-(furan-2-ylmethyl)-2-imidazo[2,1-b][1,3]thiazol-6-yl-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C17H19N3O3S
N-(furan-2-ylmethyl)-2-imidazo[2,1-b][1,3]thiazol-6-yl-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[4-[[(R)-cyclopentyl(thiophen-2-yl)methyl]carbamoylamino]pyrazol-1-yl]acetamide —— C16H21N5O2S
2-[4-[[(R)-cyclopentyl(thiophen-2-yl)methyl]carbamoylamino]pyrazol-1-yl]acetamide
—— [(4aR,8aR)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[2-(furan-2-yl)-1,3-thiazol-4-yl]methanone —— C15H16N2O3S2
[(4aR,8aR)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[2-(furan-2-yl)-1,3-thiazol-4-yl]methanone
—— [4-(tetrazol-1-yl)phenyl] (1S,2S)-2-(furan-2-yl)cyclopropane-1-carboxylate —— C15H12N4O3
[4-(tetrazol-1-yl)phenyl] (1S,2S)-2-(furan-2-yl)cyclopropane-1-carboxylate
—— [4-(tetrazol-1-yl)phenyl] (1R,2R)-2-(furan-2-yl)cyclopropane-1-carboxylate —— C15H12N4O3
[4-(tetrazol-1-yl)phenyl] (1R,2R)-2-(furan-2-yl)cyclopropane-1-carboxylate
—— [4-(tetrazol-1-yl)phenyl] (1S,2R)-2-(furan-2-yl)cyclopropane-1-carboxylate —— C15H12N4O3
[4-(tetrazol-1-yl)phenyl] (1S,2R)-2-(furan-2-yl)cyclopropane-1-carboxylate
—— N-(furan-2-ylmethyl)-2-imidazo[2,1-b][1,3]thiazol-6-yl-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C17H19N3O3S
N-(furan-2-ylmethyl)-2-imidazo[2,1-b][1,3]thiazol-6-yl-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— [(4aS,8aS)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[2-(furan-2-yl)-1,3-thiazol-4-yl]methanone —— C15H16N2O3S2
[(4aS,8aS)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[2-(furan-2-yl)-1,3-thiazol-4-yl]methanone
—— 2-[(3S)-4-[[2-(furan-2-yl)-1,3-thiazol-4-yl]methyl]morpholin-3-yl]ethanol —— C14H18N2O3S
2-[(3S)-4-[[2-(furan-2-yl)-1,3-thiazol-4-yl]methyl]morpholin-3-yl]ethanol
—— [4-(tetrazol-1-yl)phenyl] (1R,2S)-2-(furan-2-yl)cyclopropane-1-carboxylate —— C15H12N4O3
[4-(tetrazol-1-yl)phenyl] (1R,2S)-2-(furan-2-yl)cyclopropane-1-carboxylate
—— 2-[(3R)-4-[[2-(furan-2-yl)-1,3-thiazol-4-yl]methyl]morpholin-3-yl]ethanol —— C14H18N2O3S
2-[(3R)-4-[[2-(furan-2-yl)-1,3-thiazol-4-yl]methyl]morpholin-3-yl]ethanol
—— 3-[(3S)-oxolan-3-yl]-5-(3-thiophen-2-ylpropyl)-1,2,4-oxadiazole —— C13H16N2O2S
3-[(3S)-oxolan-3-yl]-5-(3-thiophen-2-ylpropyl)-1,2,4-oxadiazole
—— [(4aR,8aR)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[1-(4-fluorophenyl)pyrazol-3-yl]methanone —— C17H18FN3O2S
[(4aR,8aR)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[1-(4-fluorophenyl)pyrazol-3-yl]methanone
—— 3-(4-bromophenyl)-N'-[(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-1-phenylpyrazole-4-carbohydrazide —— C24H19BrN4O3
3-(4-bromophenyl)-N'-[(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-1-phenylpyrazole-4-carbohydrazide
—— 4-[4-[(3-bromo-5-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-3-oxo-5-(trifluoromethyl)-1H-pyrazol-2-yl]benzoate —— C19H11BrF3N2O5-
4-[4-[(3-bromo-5-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-3-oxo-5-(trifluoromethyl)-1H-pyrazol-2-yl]benzoate
—— (3R)-N-[4-(1H-pyrazol-5-yl)phenyl]-3-pyridin-3-yloxypyrrolidine-1-carboxamide —— C19H19N5O2
(3R)-N-[4-(1H-pyrazol-5-yl)phenyl]-3-pyridin-3-yloxypyrrolidine-1-carboxamide
—— [(4aR,8aR)-2,3,4,4a,5,7,8,8a-octahydropyrano[3,2-c]pyridin-6-yl]-[2-(4-fluorophenyl)triazol-4-yl]methanone —— C17H19FN4O2
[(4aR,8aR)-2,3,4,4a,5,7,8,8a-octahydropyrano[3,2-c]pyridin-6-yl]-[2-(4-fluorophenyl)triazol-4-yl]methanone
—— N-[(5E)-5-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)hydrazinylidene]-1,3-thiazol-2-ylidene]-3-pyrrolidin-1-ylsulfonylbenzamide —— C25H25N7O4S2
N-[(5E)-5-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)hydrazinylidene]-1,3-thiazol-2-ylidene]-3-pyrrolidin-1-ylsulfonylbenzamide
—— 2-(4-fluorophenyl)-4-[[(3S)-3-pyrrolidin-1-ylpyrrolidin-1-yl]methyl]-1,3-oxazole —— C18H22FN3O
2-(4-fluorophenyl)-4-[[(3S)-3-pyrrolidin-1-ylpyrrolidin-1-yl]methyl]-1,3-oxazole
—— 2-[(3S)-1-[[1-(4-chlorophenyl)triazol-4-yl]methyl]piperidin-3-yl]ethanol —— C16H21ClN4O
2-[(3S)-1-[[1-(4-chlorophenyl)triazol-4-yl]methyl]piperidin-3-yl]ethanol
—— N-[(5E)-5-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)hydrazinylidene]-1,3-thiazol-2-ylidene]benzamide —— C21H18N6O2S
N-[(5E)-5-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)hydrazinylidene]-1,3-thiazol-2-ylidene]benzamide
—— (2S)-3-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]propane-1,2-diol —— C12H13ClN2O3S
(2S)-3-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]propane-1,2-diol
—— 2-[(7S)-5,7-dihydro-4H-thieno[2,3-c]pyran-7-yl]-N-[2-[2-(4-fluorophenyl)-1,3-oxazol-4-yl]ethyl]acetamide —— C20H19FN2O3S
2-[(7S)-5,7-dihydro-4H-thieno[2,3-c]pyran-7-yl]-N-[2-[2-(4-fluorophenyl)-1,3-oxazol-4-yl]ethyl]acetamide
—— [(4aS,8aR)-2,3,4,4a,5,7,8,8a-octahydropyrano[3,2-c]pyridin-6-yl]-[2-(4-fluorophenyl)triazol-4-yl]methanone —— C17H19FN4O2
[(4aS,8aR)-2,3,4,4a,5,7,8,8a-octahydropyrano[3,2-c]pyridin-6-yl]-[2-(4-fluorophenyl)triazol-4-yl]methanone
—— [(4aS,8aS)-2,3,4,4a,5,7,8,8a-octahydropyrano[3,2-c]pyridin-6-yl]-[2-(4-fluorophenyl)triazol-4-yl]methanone —— C17H19FN4O2
[(4aS,8aS)-2,3,4,4a,5,7,8,8a-octahydropyrano[3,2-c]pyridin-6-yl]-[2-(4-fluorophenyl)triazol-4-yl]methanone
—— (2R)-3-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]propane-1,2-diol —— C12H13ClN2O3S
(2R)-3-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]propane-1,2-diol
—— [(4aS,8aR)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[1-(4-fluorophenyl)pyrazol-3-yl]methanone —— C17H18FN3O2S
[(4aS,8aR)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[1-(4-fluorophenyl)pyrazol-3-yl]methanone
—— (5R)-2-[[2-(4-fluorophenyl)-1,3-oxazol-4-yl]methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione —— C17H15FN2O3S
(5R)-2-[[2-(4-fluorophenyl)-1,3-oxazol-4-yl]methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione
—— N-(cyclopropylmethyl)-2-[(2S)-oxolan-2-yl]-N-pyridin-3-yl-1,3-thiazole-4-carboxamide —— C17H19N3O2S
N-(cyclopropylmethyl)-2-[(2S)-oxolan-2-yl]-N-pyridin-3-yl-1,3-thiazole-4-carboxamide
—— [(4aR,8aS)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[1-(4-fluorophenyl)pyrazol-3-yl]methanone —— C17H18FN3O2S
[(4aR,8aS)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[1-(4-fluorophenyl)pyrazol-3-yl]methanone
—— 1-[(2S)-2-hydroxy-3-morpholin-4-ylpropyl]-3-[4-(triazol-2-yl)phenyl]urea —— C16H22N6O3
1-[(2S)-2-hydroxy-3-morpholin-4-ylpropyl]-3-[4-(triazol-2-yl)phenyl]urea
—— 1-[[(2R)-oxolan-2-yl]methyl]-1-(pyridin-3-ylmethyl)-3-[4-(1,2,4-triazol-1-yl)phenyl]urea —— C20H22N6O2
1-[[(2R)-oxolan-2-yl]methyl]-1-(pyridin-3-ylmethyl)-3-[4-(1,2,4-triazol-1-yl)phenyl]urea
—— [(4aS,8aS)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[1-(4-fluorophenyl)pyrazol-3-yl]methanone —— C17H18FN3O2S
[(4aS,8aS)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-[1-(4-fluorophenyl)pyrazol-3-yl]methanone
—— (3R)-N-(4-pyrazol-1-ylphenyl)-3-pyridin-3-yloxypyrrolidine-1-carboxamide —— C19H19N5O2
(3R)-N-(4-pyrazol-1-ylphenyl)-3-pyridin-3-yloxypyrrolidine-1-carboxamide
—— methyl (2R)-2-[[4-amino-5-(3-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-3-methylbutanoate —— C14H17BrN4O2S
methyl (2R)-2-[[4-amino-5-(3-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-3-methylbutanoate
—— [2-(4-fluorophenyl)triazol-4-yl]-[(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone —— C16H17FN4O2
[2-(4-fluorophenyl)triazol-4-yl]-[(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone
—— 1-[(2S)-2-(dimethylamino)-3-methylbutyl]-3-[(1R)-1-(4-methyl-1,2,4-triazol-3-yl)ethyl]urea —— C13H26N6O
1-[(2S)-2-(dimethylamino)-3-methylbutyl]-3-[(1R)-1-(4-methyl-1,2,4-triazol-3-yl)ethyl]urea
—— [(4aR,8aS)-2,3,4,4a,5,7,8,8a-octahydropyrano[3,2-c]pyridin-6-yl]-[2-(4-fluorophenyl)triazol-4-yl]methanone —— C17H19FN4O2
[(4aR,8aS)-2,3,4,4a,5,7,8,8a-octahydropyrano[3,2-c]pyridin-6-yl]-[2-(4-fluorophenyl)triazol-4-yl]methanone
—— 2-[(3R)-1-[[1-(4-chlorophenyl)triazol-4-yl]methyl]piperidin-3-yl]ethanol —— C16H21ClN4O
2-[(3R)-1-[[1-(4-chlorophenyl)triazol-4-yl]methyl]piperidin-3-yl]ethanol
—— 2-(4-fluorophenyl)-4-[[(3R)-3-pyrrolidin-1-ylpyrrolidin-1-yl]methyl]-1,3-oxazole —— C18H22FN3O
2-(4-fluorophenyl)-4-[[(3R)-3-pyrrolidin-1-ylpyrrolidin-1-yl]methyl]-1,3-oxazole
—— [2-(4-fluorophenyl)triazol-4-yl]-[(5R)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone —— C16H17FN4O2
[2-(4-fluorophenyl)triazol-4-yl]-[(5R)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone
—— (3S)-N-[4-(1H-pyrazol-5-yl)phenyl]-3-pyridin-3-yloxypyrrolidine-1-carboxamide —— C19H19N5O2
(3S)-N-[4-(1H-pyrazol-5-yl)phenyl]-3-pyridin-3-yloxypyrrolidine-1-carboxamide
—— 2-[[5-(4-fluorophenyl)-1H-imidazol-2-yl]sulfanyl]-1-[(3S)-3-(trifluoromethyl)piperidin-1-yl]ethanone —— C17H17F4N3OS
2-[[5-(4-fluorophenyl)-1H-imidazol-2-yl]sulfanyl]-1-[(3S)-3-(trifluoromethyl)piperidin-1-yl]ethanone
—— (5S)-2-[[2-(4-fluorophenyl)-1,3-oxazol-4-yl]methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione —— C17H15FN2O3S
(5S)-2-[[2-(4-fluorophenyl)-1,3-oxazol-4-yl]methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione
—— (3S)-N-(4-pyrazol-1-ylphenyl)-3-pyridin-3-yloxypyrrolidine-1-carboxamide —— C19H19N5O2
(3S)-N-(4-pyrazol-1-ylphenyl)-3-pyridin-3-yloxypyrrolidine-1-carboxamide
—— (3S)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-3-carboxamide —— C13H13ClN4O2
(3S)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-3-carboxamide
—— 3-hydroxy-4-[4-(4-phenyl-1,2,4-triazol-3-yl)-5-(trifluoromethyl)-1,2-dihydropyrazol-3-ylidene]cyclohexa-2,5-dien-1-one —— C18H12F3N5O2
3-hydroxy-4-[4-(4-phenyl-1,2,4-triazol-3-yl)-5-(trifluoromethyl)-1,2-dihydropyrazol-3-ylidene]cyclohexa-2,5-dien-1-one
—— (3R)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-3-carboxamide —— C13H13ClN4O2
(3R)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-3-carboxamide