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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4,5-dimethyl-2-[(3R)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]-1,3-thiazole —— C17H25N5S
4,5-dimethyl-2-[(3R)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]-1,3-thiazole
—— N-[(R)-(4-chlorophenyl)-thiophen-2-ylmethyl]-4-methyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide —— C20H15ClN4OS2
N-[(R)-(4-chlorophenyl)-thiophen-2-ylmethyl]-4-methyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide
—— [(1S)-1-[2-(4-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]ethyl] (1R,2S)-2-methylcyclopropane-1-carboxylate —— C17H18FNO2S
[(1S)-1-[2-(4-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]ethyl] (1R,2S)-2-methylcyclopropane-1-carboxylate
—— 2-[[5-(4-tert-butylphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N'-[(1Z)-1-(6-oxocyclohexa-2,4-dien-1-ylidene)ethyl]acetohydrazide —— C29H31N5O3S
2-[[5-(4-tert-butylphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N'-[(1Z)-1-(6-oxocyclohexa-2,4-dien-1-ylidene)ethyl]acetohydrazide
—— (1R,2R)-2-(3-chlorophenyl)-N-[[5-(4-methyl-1,3-thiazol-5-yl)-1,2,4-oxadiazol-3-yl]methyl]cyclopropane-1-carboxamide —— C17H15ClN4O2S
(1R,2R)-2-(3-chlorophenyl)-N-[[5-(4-methyl-1,3-thiazol-5-yl)-1,2,4-oxadiazol-3-yl]methyl]cyclopropane-1-carboxamide
—— (3S)-N-methyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-3-amine —— C17H27N5OS
(3S)-N-methyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-3-amine
—— N-[(1S)-1-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]ethyl]-4-methyl-1,3-thiazole-5-carboxamide —— C15H13ClN4O2S
N-[(1S)-1-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]ethyl]-4-methyl-1,3-thiazole-5-carboxamide
—— (1R)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)ethanamine —— C17H20N4OS
(1R)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)ethanamine
—— 4-methyl-N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]-2-pyridin-2-yl-1,3-thiazole-5-carboxamide —— C19H25N3O2S
4-methyl-N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]-2-pyridin-2-yl-1,3-thiazole-5-carboxamide
—— 1-(4,5-dimethyl-1,3-thiazol-2-yl)-3-[1-[(3R)-oxolan-3-yl]piperidin-4-yl]urea —— C15H24N4O2S
1-(4,5-dimethyl-1,3-thiazol-2-yl)-3-[1-[(3R)-oxolan-3-yl]piperidin-4-yl]urea
—— 3-(4-chlorophenyl)-6-[(E)-2-(2-chlorophenyl)ethenyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C17H10Cl2N4S
3-(4-chlorophenyl)-6-[(E)-2-(2-chlorophenyl)ethenyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3S)-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrrolidin-3-yl]acetamide —— C16H23N5O2S
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3S)-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrrolidin-3-yl]acetamide
—— [(2R)-2-(5-methyl-1,3,4-oxadiazol-2-yl)pyrrolidin-1-yl]-(4-methyl-2-phenyl-1,3-thiazol-5-yl)methanone —— C18H18N4O2S
[(2R)-2-(5-methyl-1,3,4-oxadiazol-2-yl)pyrrolidin-1-yl]-(4-methyl-2-phenyl-1,3-thiazol-5-yl)methanone
—— N-[[(2R)-4-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]morpholin-2-yl]methyl]-N-methylpyridazin-3-amine —— C16H23N5OS
N-[[(2R)-4-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]morpholin-2-yl]methyl]-N-methylpyridazin-3-amine
—— N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-4,5-dimethyl-1,3-thiazole-2-sulfonamide —— C16H23N3O3S2
N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-4,5-dimethyl-1,3-thiazole-2-sulfonamide
—— N-[(S)-(4-chlorophenyl)-thiophen-2-ylmethyl]-4-methyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide —— C20H15ClN4OS2
N-[(S)-(4-chlorophenyl)-thiophen-2-ylmethyl]-4-methyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide
—— 1-cyclopentyl-3-[(Z)-1-(4-methyl-1,3-thiazol-5-yl)ethylideneamino]urea —— C12H18N4OS
1-cyclopentyl-3-[(Z)-1-(4-methyl-1,3-thiazol-5-yl)ethylideneamino]urea
—— 2-[(S)-(2,4-dimethyl-1,3-thiazol-5-yl)methylsulfinyl]-N-methyl-N-(thiophen-2-ylmethyl)acetamide —— C14H18N2O2S3
2-[(S)-(2,4-dimethyl-1,3-thiazol-5-yl)methylsulfinyl]-N-methyl-N-(thiophen-2-ylmethyl)acetamide
—— (1R,2S)-2-(3-chlorophenyl)-N-[[5-(4-methyl-1,3-thiazol-5-yl)-1,2,4-oxadiazol-3-yl]methyl]cyclopropane-1-carboxamide —— C17H15ClN4O2S
(1R,2S)-2-(3-chlorophenyl)-N-[[5-(4-methyl-1,3-thiazol-5-yl)-1,2,4-oxadiazol-3-yl]methyl]cyclopropane-1-carboxamide
—— N'-[(5S)-5-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl]-4-methyl-1,3-thiazole-5-carbohydrazide —— C18H23N3O2S2
N'-[(5S)-5-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl]-4-methyl-1,3-thiazole-5-carbohydrazide
—— [(1S,6R,7S)-8,8-dimethyl-2-oxabicyclo[4.2.0]octan-7-yl] 4-methyl-1,3-thiazole-5-carboxylate —— C14H19NO3S
[(1S,6R,7S)-8,8-dimethyl-2-oxabicyclo[4.2.0]octan-7-yl] 4-methyl-1,3-thiazole-5-carboxylate
—— N-[(1S)-1-cyclopropylethyl]-N,4-dimethyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide —— C15H18N4OS
N-[(1S)-1-cyclopropylethyl]-N,4-dimethyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide
—— N-[(E)-1-(4-fluorophenyl)ethylideneamino]-3-(4-methylphenyl)-1H-pyrazole-5-carboxamide —— C19H17FN4O
N-[(E)-1-(4-fluorophenyl)ethylideneamino]-3-(4-methylphenyl)-1H-pyrazole-5-carboxamide
—— 4-methyl-5-[2-[[(2S)-oxolan-2-yl]methylsulfonyl]ethyl]-1,3-thiazole —— C11H17NO3S2
4-methyl-5-[2-[[(2S)-oxolan-2-yl]methylsulfonyl]ethyl]-1,3-thiazole
—— N-[(2R)-2-cyano-4-phenylbutan-2-yl]-4-methyl-1,3-thiazole-5-carboxamide —— C16H17N3OS
N-[(2R)-2-cyano-4-phenylbutan-2-yl]-4-methyl-1,3-thiazole-5-carboxamide
—— 2-[(1R)-cyclohex-2-en-1-yl]sulfanyl-5-(2,4-dimethyl-1,3-thiazol-5-yl)-1,3,4-oxadiazole —— C13H15N3OS2
2-[(1R)-cyclohex-2-en-1-yl]sulfanyl-5-(2,4-dimethyl-1,3-thiazol-5-yl)-1,3,4-oxadiazole
—— N,4-dimethyl-N-[(1S)-2,2,2-trifluoro-1-phenylethyl]-1,3-thiazole-5-carboxamide —— C14H13F3N2OS
N,4-dimethyl-N-[(1S)-2,2,2-trifluoro-1-phenylethyl]-1,3-thiazole-5-carboxamide
—— N-methyl-2-(4-methyl-2-sulfanylidene-3H-1,3-thiazol-5-yl)-N-[(1R)-1-thiophen-2-ylethyl]acetamide —— C13H16N2OS3
N-methyl-2-(4-methyl-2-sulfanylidene-3H-1,3-thiazol-5-yl)-N-[(1R)-1-thiophen-2-ylethyl]acetamide
—— N-[(1R,2S)-2-(2,4-difluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide —— C16H13F2N5OS
N-[(1R,2S)-2-(2,4-difluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide
—— [(1R)-1-[2-(4-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]ethyl] (1R,2S)-2-methylcyclopropane-1-carboxylate —— C17H18FNO2S
[(1R)-1-[2-(4-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]ethyl] (1R,2S)-2-methylcyclopropane-1-carboxylate
—— (3S)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]-3-methyl-3-(2-methylpropyl)pyrrolidine-2,5-dione —— C15H22N2O2S
(3S)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]-3-methyl-3-(2-methylpropyl)pyrrolidine-2,5-dione
—— 2-(4-fluorophenyl)-N-[(1S)-4-hydroxy-1-phenylbutyl]-4-methyl-1,3-thiazole-5-carboxamide —— C21H21FN2O2S
2-(4-fluorophenyl)-N-[(1S)-4-hydroxy-1-phenylbutyl]-4-methyl-1,3-thiazole-5-carboxamide
—— N-[(1S,2S)-2-(2-chlorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide —— C16H14ClN5OS
N-[(1S,2S)-2-(2-chlorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide
—— N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-2-pyrrol-1-yl-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxamide —— C19H21N3OS3
N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-2-pyrrol-1-yl-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxamide
—— methyl (2R)-3-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoylamino]-2-phenylpropanoate —— C16H19N3O3S
methyl (2R)-3-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoylamino]-2-phenylpropanoate
—— (Z)-4-methyl-2-(2-(pyridin-2-ylmethylene)hydrazinyl)thiazole —— C10H10N4S
(Z)-4-methyl-2-(2-(pyridin-2-ylmethylene)hydrazinyl)thiazole
—— 1-(4,5-dimethyl-1,3-thiazol-2-yl)-3-[(1R)-2-methylsulfonyl-1-phenylethyl]urea —— C15H19N3O3S2
1-(4,5-dimethyl-1,3-thiazol-2-yl)-3-[(1R)-2-methylsulfonyl-1-phenylethyl]urea
—— 1-[[(3S,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-3-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]urea —— C15H24N4O2S
1-[[(3S,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-3-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]urea
—— (3R)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]-3-methyl-3-(2-methylpropyl)pyrrolidine-2,5-dione —— C15H22N2O2S
(3R)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]-3-methyl-3-(2-methylpropyl)pyrrolidine-2,5-dione
—— N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-1-[(2S,3S)-2-(1-methylpyrazol-4-yl)oxolan-3-yl]methanamine —— C15H22N4OS
N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-1-[(2S,3S)-2-(1-methylpyrazol-4-yl)oxolan-3-yl]methanamine
—— (2,4-dimethyl-1,3-thiazol-5-yl)methyl (2R)-2-(3-methylbutoxy)propanoate —— C14H23NO3S
(2,4-dimethyl-1,3-thiazol-5-yl)methyl (2R)-2-(3-methylbutoxy)propanoate
—— N-[(1S,2S)-2-(2,4-difluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide —— C16H13F2N5OS
N-[(1S,2S)-2-(2,4-difluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide
—— (5R)-N-[5-[(2-fluorophenyl)methyl]-4-methyl-1,3-thiazol-2-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C21H18FN3O2S
(5R)-N-[5-[(2-fluorophenyl)methyl]-4-methyl-1,3-thiazol-2-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— 1-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[3-(2-oxopyridin-1-yl)propyl]urea —— C16H22N4O2S
1-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[3-(2-oxopyridin-1-yl)propyl]urea
—— 2-[(3R)-1,1-dioxo-2,3-dihydrothiophen-3-yl]-N-[5-[(2-fluorophenyl)methyl]-4-methyl-1,3-thiazol-2-yl]acetamide —— C17H17FN2O3S2
2-[(3R)-1,1-dioxo-2,3-dihydrothiophen-3-yl]-N-[5-[(2-fluorophenyl)methyl]-4-methyl-1,3-thiazol-2-yl]acetamide
—— [(2S)-2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)methanone —— C17H22N4O2S
[(2S)-2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)methanone
—— N-[(E)-1-(2-tert-butyl-4-methyl-1,3-thiazol-5-yl)ethylideneamino]-5-(trifluoromethyl)pyridin-2-amine —— C16H19F3N4S
N-[(E)-1-(2-tert-butyl-4-methyl-1,3-thiazol-5-yl)ethylideneamino]-5-(trifluoromethyl)pyridin-2-amine
—— (2,4-dimethyl-1,3-thiazol-5-yl)methyl (2S)-2-(3-methylbutoxy)propanoate —— C14H23NO3S
(2,4-dimethyl-1,3-thiazol-5-yl)methyl (2S)-2-(3-methylbutoxy)propanoate
—— (5R)-3-(2,4-dichlorophenyl)-N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H17Cl2N3O2S
(5R)-3-(2,4-dichlorophenyl)-N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [(1R,2R)-2-methoxycyclohexyl] 2-benzyl-4-methyl-1,3-thiazole-5-carboxylate —— C19H23NO3S
[(1R,2R)-2-methoxycyclohexyl] 2-benzyl-4-methyl-1,3-thiazole-5-carboxylate