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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[1-(2-fluorophenyl)pyrazol-4-yl]-3-[(4R)-4-hydroxy-2,2-dimethylpentyl]urea —— C17H23FN4O2
1-[1-(2-fluorophenyl)pyrazol-4-yl]-3-[(4R)-4-hydroxy-2,2-dimethylpentyl]urea
—— (4-pyrazol-1-ylphenyl)methyl (3R)-3-pyridin-4-ylbutanoate —— C19H19N3O2
(4-pyrazol-1-ylphenyl)methyl (3R)-3-pyridin-4-ylbutanoate
—— N-[(2R,4R)-4-hydroxy-4-phenylbutan-2-yl]-1,3-thiazole-4-carboxamide —— C14H16N2O2S
N-[(2R,4R)-4-hydroxy-4-phenylbutan-2-yl]-1,3-thiazole-4-carboxamide
—— N-[(2S,4S)-4-hydroxy-4-phenylbutan-2-yl]-1,3-thiazole-4-carboxamide —— C14H16N2O2S
N-[(2S,4S)-4-hydroxy-4-phenylbutan-2-yl]-1,3-thiazole-4-carboxamide
—— 2-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-N-[(2R,4R)-4-hydroxy-4-phenylbutan-2-yl]acetamide —— C21H21ClN2O2S
2-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-N-[(2R,4R)-4-hydroxy-4-phenylbutan-2-yl]acetamide
—— methyl (2S)-4-(3-fluoro-4-imidazol-1-ylanilino)-2-methyl-4-oxobutanoate —— C15H16FN3O3
methyl (2S)-4-(3-fluoro-4-imidazol-1-ylanilino)-2-methyl-4-oxobutanoate
—— tert-butyl N-[(1S)-1-[(2R)-4-[(3S)-3-carbamoyl-2-phenyl-3,4-dihydropyrazole-5-carbonyl]morpholin-2-yl]ethyl]carbamate —— C22H31N5O5
tert-butyl N-[(1S)-1-[(2R)-4-[(3S)-3-carbamoyl-2-phenyl-3,4-dihydropyrazole-5-carbonyl]morpholin-2-yl]ethyl]carbamate
—— (5E)-5-[[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]methylidene]-3-[(4-methylphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H20FN3OS2
(5E)-5-[[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]methylidene]-3-[(4-methylphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— tert-butyl N-[(1R)-1-[(2S)-4-[(3S)-3-carbamoyl-2-phenyl-3,4-dihydropyrazole-5-carbonyl]morpholin-2-yl]ethyl]carbamate —— C22H31N5O5
tert-butyl N-[(1R)-1-[(2S)-4-[(3S)-3-carbamoyl-2-phenyl-3,4-dihydropyrazole-5-carbonyl]morpholin-2-yl]ethyl]carbamate
—— 2-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-N-[(2R,4S)-4-hydroxy-4-phenylbutan-2-yl]acetamide —— C21H21ClN2O2S
2-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-N-[(2R,4S)-4-hydroxy-4-phenylbutan-2-yl]acetamide
—— 2-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-N-[(2S,4S)-4-hydroxy-4-phenylbutan-2-yl]acetamide —— C21H21ClN2O2S
2-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-N-[(2S,4S)-4-hydroxy-4-phenylbutan-2-yl]acetamide
—— N-[(1S)-1-cyclopropylethyl]-3-(5-phenylpyrazol-1-yl)benzamide —— C21H21N3O
N-[(1S)-1-cyclopropylethyl]-3-(5-phenylpyrazol-1-yl)benzamide
—— methyl (2R)-4-(3-fluoro-4-imidazol-1-ylanilino)-2-methyl-4-oxobutanoate —— C15H16FN3O3
methyl (2R)-4-(3-fluoro-4-imidazol-1-ylanilino)-2-methyl-4-oxobutanoate
—— 1-[(5Z)-5-({3-[4-(ethylsulfanyl)phenyl]-1-phenyl-1H-pyrazol-4-yl}methylidene)-4-oxo-4,5-dihydro-1,3-thiazol-2-yl]piperidine-4-carboxamide —— C27H27N5O2S2
1-[(5Z)-5-({3-[4-(ethylsulfanyl)phenyl]-1-phenyl-1H-pyrazol-4-yl}methylidene)-4-oxo-4,5-dihydro-1,3-thiazol-2-yl]piperidine-4-carboxamide
—— 2-[[5-(4-tert-butylphenyl)-4-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-1-(furan-2-yl)ethylideneamino]acetamide —— C27H29N5O2S
2-[[5-(4-tert-butylphenyl)-4-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-1-(furan-2-yl)ethylideneamino]acetamide
—— N-[(Z)-(4-methylphenyl)methylideneamino]-1,5-diphenylpyrazole-3-carboxamide —— C24H20N4O
N-[(Z)-(4-methylphenyl)methylideneamino]-1,5-diphenylpyrazole-3-carboxamide
—— tert-butyl N-[(1S)-1-[(2S)-4-[(3S)-3-carbamoyl-2-phenyl-3,4-dihydropyrazole-5-carbonyl]morpholin-2-yl]ethyl]carbamate —— C22H31N5O5
tert-butyl N-[(1S)-1-[(2S)-4-[(3S)-3-carbamoyl-2-phenyl-3,4-dihydropyrazole-5-carbonyl]morpholin-2-yl]ethyl]carbamate
—— methyl 4-[(Z)-{6-oxo-2-[4-(pentyloxy)phenyl][1,3]thiazolo[3,2-b][1,2,4]triazol-5(6H)-ylidene}methyl]benzoate —— C24H23N3O4S
methyl 4-[(Z)-{6-oxo-2-[4-(pentyloxy)phenyl][1,3]thiazolo[3,2-b][1,2,4]triazol-5(6H)-ylidene}methyl]benzoate
—— 2-[[4-(4-ethoxyphenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-1-(4-fluorophenyl)ethylideneamino]acetamide —— C26H24FN5O2S
2-[[4-(4-ethoxyphenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-1-(4-fluorophenyl)ethylideneamino]acetamide
—— N-[(1R,2R)-2-(4-fluorophenyl)cyclopropyl]-2-(2-propan-2-yl-1,3-thiazol-4-yl)acetamide —— C17H19FN2OS
N-[(1R,2R)-2-(4-fluorophenyl)cyclopropyl]-2-(2-propan-2-yl-1,3-thiazol-4-yl)acetamide
—— 2-[[4,5-bis(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-[(E)-2-methyl-3-phenylprop-2-enylidene]amino]acetamide —— C28H27N5O3S
2-[[4,5-bis(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-[(E)-2-methyl-3-phenylprop-2-enylidene]amino]acetamide
—— N-[(1R)-1-cyclopropylethyl]-3-(5-phenylpyrazol-1-yl)benzamide —— C21H21N3O
N-[(1R)-1-cyclopropylethyl]-3-(5-phenylpyrazol-1-yl)benzamide
—— (4-pyrazol-1-ylphenyl)methyl (3S)-3-pyridin-4-ylbutanoate —— C19H19N3O2
(4-pyrazol-1-ylphenyl)methyl (3S)-3-pyridin-4-ylbutanoate
—— (4E)-4-[[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-2-phenyl-1,3-oxazol-5-one —— C26H19N3O3
(4E)-4-[[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-2-phenyl-1,3-oxazol-5-one
—— 1-[1-(2-fluorophenyl)pyrazol-4-yl]-3-[(4S)-4-hydroxy-2,2-dimethylpentyl]urea —— C17H23FN4O2
1-[1-(2-fluorophenyl)pyrazol-4-yl]-3-[(4S)-4-hydroxy-2,2-dimethylpentyl]urea
—— ethyl (3Z)-4,4,4-trifluoro-3-[2-(4-phenyl-1,3-thiazol-2-yl)hydrazinylidene]butanoate —— C15H14F3N3O2S
ethyl (3Z)-4,4,4-trifluoro-3-[2-(4-phenyl-1,3-thiazol-2-yl)hydrazinylidene]butanoate
—— (1R)-1-cyclopropyl-N-[[4-[3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]ethanamine —— C16H18F3N3
(1R)-1-cyclopropyl-N-[[4-[3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]ethanamine
—— tert-butyl N-[[(1R,2R)-2-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)amino]cyclopentyl]methyl]carbamate —— C16H28N4O3
tert-butyl N-[[(1R,2R)-2-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)amino]cyclopentyl]methyl]carbamate
—— N-[(2S)-1-cyanopropan-2-yl]-1-(4-fluorophenyl)-4,5,6,7-tetrahydroindazole-3-carboxamide —— C18H19FN4O
N-[(2S)-1-cyanopropan-2-yl]-1-(4-fluorophenyl)-4,5,6,7-tetrahydroindazole-3-carboxamide
—— 1-[(2R)-2,3-dihydroxypropyl]-3-(2-propan-2-ylpyrazol-3-yl)urea —— C10H18N4O3
1-[(2R)-2,3-dihydroxypropyl]-3-(2-propan-2-ylpyrazol-3-yl)urea
—— (2E,5E)-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-[(4-nitrophenyl)methylidene]-2-[(Z)-(4-nitrophenyl)methylidenehydrazinylidene]-1,3-thiazolidin-4-one —— C28H21N7O6S
(2E,5E)-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-[(4-nitrophenyl)methylidene]-2-[(Z)-(4-nitrophenyl)methylidenehydrazinylidene]-1,3-thiazolidin-4-one
—— 1-(2,6-dichlorophenyl)-N-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-5-propan-2-yl-1,2,4-triazole-3-carboxamide —— C17H19Cl2N5O2
1-(2,6-dichlorophenyl)-N-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-5-propan-2-yl-1,2,4-triazole-3-carboxamide
—— N-[(1S,2R)-2-(4-fluorophenyl)cyclopropyl]-2-(2-propan-2-yl-1,3-thiazol-4-yl)acetamide —— C17H19FN2OS
N-[(1S,2R)-2-(4-fluorophenyl)cyclopropyl]-2-(2-propan-2-yl-1,3-thiazol-4-yl)acetamide
—— [(9aR)-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[1-propan-2-yl-5-(trifluoromethyl)pyrazol-4-yl]methanone —— C16H23F3N4O
[(9aR)-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[1-propan-2-yl-5-(trifluoromethyl)pyrazol-4-yl]methanone
—— N-[(3R)-1-(cyclobutylmethyl)pyrrolidin-3-yl]-N-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]acetamide —— C18H29N3O2
N-[(3R)-1-(cyclobutylmethyl)pyrrolidin-3-yl]-N-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]acetamide
—— (6E)-6-{4-[(4-methylbenzyl)oxy]benzylidene}-3-phenyl[1,3]thiazolo[2,3-c][1,2,4]triazol-5(6H)-one —— C25H19N3O2S
(6E)-6-{4-[(4-methylbenzyl)oxy]benzylidene}-3-phenyl[1,3]thiazolo[2,3-c][1,2,4]triazol-5(6H)-one
—— tert-butyl N-[(1R)-1-[(2R)-4-[(3S)-3-carbamoyl-2-phenyl-3,4-dihydropyrazole-5-carbonyl]morpholin-2-yl]ethyl]carbamate —— C22H31N5O5
tert-butyl N-[(1R)-1-[(2R)-4-[(3S)-3-carbamoyl-2-phenyl-3,4-dihydropyrazole-5-carbonyl]morpholin-2-yl]ethyl]carbamate
—— 1-[(2S)-2-hydroxy-2-thiophen-3-ylpropyl]-3-(1-propan-2-ylpyrazol-4-yl)urea —— C14H20N4O2S
1-[(2S)-2-hydroxy-2-thiophen-3-ylpropyl]-3-(1-propan-2-ylpyrazol-4-yl)urea
—— [(9aS)-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[1-propan-2-yl-5-(trifluoromethyl)pyrazol-4-yl]methanone —— C16H23F3N4O
[(9aS)-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[1-propan-2-yl-5-(trifluoromethyl)pyrazol-4-yl]methanone
—— N-(2-acetyloxyethyl)-1-[1-(2-acetyloxyethyl)-5-nitroimidazol-2-yl]methanimine oxide —— C12H16N4O7
N-(2-acetyloxyethyl)-1-[1-(2-acetyloxyethyl)-5-nitroimidazol-2-yl]methanimine oxide
—— N-[(1S)-1-cyclopropylethyl]-2-(4-oxo-7-phenylpyrazolo[3,4-d]triazin-3-yl)acetamide —— C17H18N6O2
N-[(1S)-1-cyclopropylethyl]-2-(4-oxo-7-phenylpyrazolo[3,4-d]triazin-3-yl)acetamide
—— 2-propan-2-yl-5-[[(3R)-3-(4-propan-2-yl-1,3-thiazol-2-yl)piperidin-1-yl]methyl]-1,3,4-oxadiazole —— C17H26N4OS
2-propan-2-yl-5-[[(3R)-3-(4-propan-2-yl-1,3-thiazol-2-yl)piperidin-1-yl]methyl]-1,3,4-oxadiazole
—— N-[(2R)-2-(furan-2-yl)-2-hydroxypropyl]-3-(2-propan-2-ylimidazol-1-yl)propanamide —— C16H23N3O3
N-[(2R)-2-(furan-2-yl)-2-hydroxypropyl]-3-(2-propan-2-ylimidazol-1-yl)propanamide
—— methyl 2-[(3S)-4-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]thiomorpholin-3-yl]acetate —— C14H22N2O2S2
methyl 2-[(3S)-4-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]thiomorpholin-3-yl]acetate
—— N-[(3S)-1-(2-cyanoethyl)pyrrolidin-3-yl]-N-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]acetamide —— C16H24N4O2
N-[(3S)-1-(2-cyanoethyl)pyrrolidin-3-yl]-N-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]acetamide
—— 1-(2,6-dichlorophenyl)-N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-5-propan-2-yl-1,2,4-triazole-3-carboxamide —— C17H19Cl2N5O2
1-(2,6-dichlorophenyl)-N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-5-propan-2-yl-1,2,4-triazole-3-carboxamide
—— N-[(1S,2S)-2-(4-fluorophenyl)cyclopropyl]-2-(2-propan-2-yl-1,3-thiazol-4-yl)acetamide —— C17H19FN2OS
N-[(1S,2S)-2-(4-fluorophenyl)cyclopropyl]-2-(2-propan-2-yl-1,3-thiazol-4-yl)acetamide
—— N-[(1R)-1-cyclopropylethyl]-2-(4-oxo-7-phenylpyrazolo[3,4-d]triazin-3-yl)acetamide —— C17H18N6O2
N-[(1R)-1-cyclopropylethyl]-2-(4-oxo-7-phenylpyrazolo[3,4-d]triazin-3-yl)acetamide
—— (2Z)-3-[3-(4-chlorophenyl)-1-phenyl-1H-pyrazol-4-yl]-2-cyano-N-(furan-2-ylmethyl)prop-2-enamide —— C24H17ClN4O2
(2Z)-3-[3-(4-chlorophenyl)-1-phenyl-1H-pyrazol-4-yl]-2-cyano-N-(furan-2-ylmethyl)prop-2-enamide
—— (5E)-3-(3-methoxypropyl)-5-[(2-phenyl-5-thiophen-2-ylpyrazol-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C21H19N3O2S3
(5E)-3-(3-methoxypropyl)-5-[(2-phenyl-5-thiophen-2-ylpyrazol-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one