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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-tert-butyl-2-[[(3S)-3-[(sulfamoylamino)methyl]piperidin-1-yl]methyl]-1,3-thiazole —— C14H26N4O2S2
4-tert-butyl-2-[[(3S)-3-[(sulfamoylamino)methyl]piperidin-1-yl]methyl]-1,3-thiazole
—— (5Z)-5-{[3-(3-chloro-4-propoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methylidene}-3-(3-ethoxypropyl)-2-thioxo-1,3-thiazolidin-4-one —— C27H28ClN3O3S2
(5Z)-5-{[3-(3-chloro-4-propoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methylidene}-3-(3-ethoxypropyl)-2-thioxo-1,3-thiazolidin-4-one
—— N-[(2R)-2-hydroxy-3-phenylpropyl]-2-(3-methyl-1,2,4-oxadiazol-5-yl)benzamide —— C19H19N3O3
N-[(2R)-2-hydroxy-3-phenylpropyl]-2-(3-methyl-1,2,4-oxadiazol-5-yl)benzamide
—— 2-(2-tert-butyl-1,3-thiazol-4-yl)-N-[(2R)-3-(dimethylamino)-2-hydroxy-2-methylpropyl]acetamide —— C15H27N3O2S
2-(2-tert-butyl-1,3-thiazol-4-yl)-N-[(2R)-3-(dimethylamino)-2-hydroxy-2-methylpropyl]acetamide
—— [2-(4-chlorophenyl)-5-(2-fluorophenyl)pyrazol-3-yl]-[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]methanone —— C29H26ClFN4O
[2-(4-chlorophenyl)-5-(2-fluorophenyl)pyrazol-3-yl]-[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]methanone
—— 4-tert-butyl-2-[[(3R)-3-[(sulfamoylamino)methyl]piperidin-1-yl]methyl]-1,3-thiazole —— C14H26N4O2S2
4-tert-butyl-2-[[(3R)-3-[(sulfamoylamino)methyl]piperidin-1-yl]methyl]-1,3-thiazole
—— (6R)-2-methyl-N-[4-(5-propan-2-yl-1,3-oxazol-2-yl)phenyl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide —— C23H23F3N4O2
(6R)-2-methyl-N-[4-(5-propan-2-yl-1,3-oxazol-2-yl)phenyl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide
—— 1-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-3-[1-[[(2R)-oxolan-2-yl]methyl]pyrazol-4-yl]urea —— C17H25N5O3
1-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-3-[1-[[(2R)-oxolan-2-yl]methyl]pyrazol-4-yl]urea
—— 2-(2-tert-butyl-1,3-thiazol-4-yl)-N-[(2S)-3-(dimethylamino)-2-hydroxy-2-methylpropyl]acetamide —— C15H27N3O2S
2-(2-tert-butyl-1,3-thiazol-4-yl)-N-[(2S)-3-(dimethylamino)-2-hydroxy-2-methylpropyl]acetamide
—— 3-[[5-[[(1R)-cyclopent-2-en-1-yl]methyl]-1,2,4-oxadiazol-3-yl]methyl]-5-methyl-1,2,4-oxadiazole —— C12H14N4O2
3-[[5-[[(1R)-cyclopent-2-en-1-yl]methyl]-1,2,4-oxadiazol-3-yl]methyl]-5-methyl-1,2,4-oxadiazole
—— 4-[[(3S)-1-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]pyrrolidin-3-yl]methyl]morpholine —— C17H29N3OS
4-[[(3S)-1-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]pyrrolidin-3-yl]methyl]morpholine
—— N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3R)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-3-yl]acetamide —— C15H21N5O2S
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3R)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-3-yl]acetamide
—— 1-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-3-[1-[[(2S)-oxolan-2-yl]methyl]pyrazol-4-yl]urea —— C17H25N5O3
1-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-3-[1-[[(2S)-oxolan-2-yl]methyl]pyrazol-4-yl]urea
—— N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3R)-1-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-yl]acetamide —— C17H25N5O3
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3R)-1-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-yl]acetamide
—— 1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-3-[(1R,2R)-2-(trifluoromethyl)cyclohexyl]urea —— C17H19F3N4O2
1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-3-[(1R,2R)-2-(trifluoromethyl)cyclohexyl]urea
—— (2R)-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-2,3-dihydro-1,4-benzoxathiine-2-carboxamide —— C18H15N3O3S
(2R)-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-2,3-dihydro-1,4-benzoxathiine-2-carboxamide
—— N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3S)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-3-yl]acetamide —— C15H21N5O2S
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3S)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-3-yl]acetamide
—— 1-(4-chlorophenyl)-N-[(2R)-2-cyano-1-(3,4-difluorophenoxy)propan-2-yl]-5-methyl-1,2,4-triazole-3-carboxamide —— C20H16ClF2N5O2
1-(4-chlorophenyl)-N-[(2R)-2-cyano-1-(3,4-difluorophenoxy)propan-2-yl]-5-methyl-1,2,4-triazole-3-carboxamide
—— (2S)-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-2,3-dihydro-1,4-benzoxathiine-2-carboxamide —— C18H15N3O3S
(2S)-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-2,3-dihydro-1,4-benzoxathiine-2-carboxamide
—— N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3S)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-3-yl]acetamide —— C15H21N5O2S
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3S)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-3-yl]acetamide
—— (4S)-4-methyl-N-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carboxamide —— C18H18N4O2S
(4S)-4-methyl-N-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carboxamide
—— (2R)-2-[(2-chlorophenyl)methyl]-N-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]pyrrolidine-1-carboxamide —— C21H21ClN4O2
(2R)-2-[(2-chlorophenyl)methyl]-N-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]pyrrolidine-1-carboxamide
—— 3-[[5-[[(1S)-cyclopent-2-en-1-yl]methyl]-1,2,4-oxadiazol-3-yl]methyl]-5-methyl-1,2,4-oxadiazole —— C12H14N4O2
3-[[5-[[(1S)-cyclopent-2-en-1-yl]methyl]-1,2,4-oxadiazol-3-yl]methyl]-5-methyl-1,2,4-oxadiazole
—— 1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-3-[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]urea —— C20H26N4O2
1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-3-[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]urea
—— N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3S)-1-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-yl]acetamide —— C17H25N5O3
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3S)-1-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-yl]acetamide
—— N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3R)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-3-yl]acetamide —— C15H21N5O2S
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[(3R)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-3-yl]acetamide
—— 1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-3-[(1S,2S)-2-(trifluoromethyl)cyclohexyl]urea —— C17H19F3N4O2
1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-3-[(1S,2S)-2-(trifluoromethyl)cyclohexyl]urea
—— 1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-3-[(1R,2S)-2-(trifluoromethyl)cyclohexyl]urea —— C17H19F3N4O2
1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-3-[(1R,2S)-2-(trifluoromethyl)cyclohexyl]urea
—— N-[(1S)-1-(furan-2-yl)ethyl]-N,5-dimethyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carboxamide —— C20H24N4O2
N-[(1S)-1-(furan-2-yl)ethyl]-N,5-dimethyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carboxamide
—— (3R,6R)-1-[5-methyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carbonyl]-6-(trifluoromethyl)piperidine-3-carboxamide —— C20H24F3N5O2
(3R,6R)-1-[5-methyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carbonyl]-6-(trifluoromethyl)piperidine-3-carboxamide
—— 1-(4-chlorophenyl)-N-[(2S)-2-cyano-1-(3,4-difluorophenoxy)propan-2-yl]-5-methyl-1,2,4-triazole-3-carboxamide —— C20H16ClF2N5O2
1-(4-chlorophenyl)-N-[(2S)-2-cyano-1-(3,4-difluorophenoxy)propan-2-yl]-5-methyl-1,2,4-triazole-3-carboxamide
—— (3S,6R)-1-[5-methyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carbonyl]-6-(trifluoromethyl)piperidine-3-carboxamide —— C20H24F3N5O2
(3S,6R)-1-[5-methyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carbonyl]-6-(trifluoromethyl)piperidine-3-carboxamide
—— (3S,6S)-1-[5-methyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carbonyl]-6-(trifluoromethyl)piperidine-3-carboxamide —— C20H24F3N5O2
(3S,6S)-1-[5-methyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carbonyl]-6-(trifluoromethyl)piperidine-3-carboxamide
—— 1-(4-chlorophenyl)-5-methyl-N-[2-[(1R)-1-pyridin-4-ylethyl]pyrazol-3-yl]-1,2,4-triazole-3-carboxamide —— C20H18ClN7O
1-(4-chlorophenyl)-5-methyl-N-[2-[(1R)-1-pyridin-4-ylethyl]pyrazol-3-yl]-1,2,4-triazole-3-carboxamide
—— (1R)-N-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)phenyl]-3,4-dihydro-1H-isothiochromene-1-carboxamide —— C20H20N4OS
(1R)-N-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)phenyl]-3,4-dihydro-1H-isothiochromene-1-carboxamide
—— 1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)phenyl]-3-[(2S)-2-hydroxy-2-thiophen-3-ylpropyl]urea —— C18H21N5O2S
1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)phenyl]-3-[(2S)-2-hydroxy-2-thiophen-3-ylpropyl]urea
—— (1S)-N-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)phenyl]-3,4-dihydro-1H-isothiochromene-1-carboxamide —— C20H20N4OS
(1S)-N-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)phenyl]-3,4-dihydro-1H-isothiochromene-1-carboxamide
—— 5-methyl-N-[(1S)-1-(1-phenyltriazol-4-yl)ethyl]-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carboxamide —— C23H25N7O
5-methyl-N-[(1S)-1-(1-phenyltriazol-4-yl)ethyl]-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carboxamide
—— 5-(4-methoxyphenyl)-3-[[(S)-(2-methyl-1,3-thiazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole —— C15H15N3O3S2
5-(4-methoxyphenyl)-3-[[(S)-(2-methyl-1,3-thiazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole
—— methyl (1R,2S)-2-[4-(2-methyl-1,3-thiazol-4-yl)butanoylamino]cycloheptane-1-carboxylate —— C17H26N2O3S
methyl (1R,2S)-2-[4-(2-methyl-1,3-thiazol-4-yl)butanoylamino]cycloheptane-1-carboxylate
—— N-[(2S)-2-hydroxy-3,3-dimethylbutyl]-5-methyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carboxamide —— C19H28N4O2
N-[(2S)-2-hydroxy-3,3-dimethylbutyl]-5-methyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carboxamide
—— N-[(1R)-1-(furan-2-yl)ethyl]-N,5-dimethyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carboxamide —— C20H24N4O2
N-[(1R)-1-(furan-2-yl)ethyl]-N,5-dimethyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carboxamide
—— 5-methyl-N-[(1R)-1-(1-phenyltriazol-4-yl)ethyl]-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carboxamide —— C23H25N7O
5-methyl-N-[(1R)-1-(1-phenyltriazol-4-yl)ethyl]-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carboxamide
—— 5-(4-methoxyphenyl)-3-[[(R)-(2-methyl-1,3-thiazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole —— C15H15N3O3S2
5-(4-methoxyphenyl)-3-[[(R)-(2-methyl-1,3-thiazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole
—— 1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)phenyl]-3-[(2R)-2-hydroxy-2-thiophen-3-ylpropyl]urea —— C18H21N5O2S
1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)phenyl]-3-[(2R)-2-hydroxy-2-thiophen-3-ylpropyl]urea
—— 1-(4-chlorophenyl)-5-methyl-N-[2-[(1S)-1-pyridin-4-ylethyl]pyrazol-3-yl]-1,2,4-triazole-3-carboxamide —— C20H18ClN7O
1-(4-chlorophenyl)-5-methyl-N-[2-[(1S)-1-pyridin-4-ylethyl]pyrazol-3-yl]-1,2,4-triazole-3-carboxamide
—— 3-[(3R)-1-tert-butyl-5-oxopyrrolidin-3-yl]-1-methyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]urea —— C15H24N4O2S
3-[(3R)-1-tert-butyl-5-oxopyrrolidin-3-yl]-1-methyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]urea
—— (3R,6S)-1-[5-methyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carbonyl]-6-(trifluoromethyl)piperidine-3-carboxamide —— C20H24F3N5O2
(3R,6S)-1-[5-methyl-1-(2-propan-2-ylphenyl)-1,2,4-triazole-3-carbonyl]-6-(trifluoromethyl)piperidine-3-carboxamide
—— N-[(3R)-1,1-dioxothiolan-3-yl]-1-(4-fluorophenyl)-N,5-dimethyl-1,2,4-triazole-3-carboxamide —— C15H17FN4O3S
N-[(3R)-1,1-dioxothiolan-3-yl]-1-(4-fluorophenyl)-N,5-dimethyl-1,2,4-triazole-3-carboxamide
—— N,5-dimethyl-1-(2-propan-2-ylphenyl)-N-[(1R)-1-pyridin-2-ylethyl]-1,2,4-triazole-3-carboxamide —— C21H25N5O
N,5-dimethyl-1-(2-propan-2-ylphenyl)-N-[(1R)-1-pyridin-2-ylethyl]-1,2,4-triazole-3-carboxamide