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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-2-(4-bromophenoxy)-1-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]propan-1-one —— C21H21BrN4O2
(2S)-2-(4-bromophenoxy)-1-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]propan-1-one
—— 1-ethyl-3-[3-[(4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea —— C28H30N6O5S
1-ethyl-3-[3-[(4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea
—— (2S)-2-(4-bromophenoxy)-1-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]propan-1-one —— C21H21BrN4O2
(2S)-2-(4-bromophenoxy)-1-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]propan-1-one
—— (2R)-2-(4-bromophenoxy)-1-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]propan-1-one —— C21H21BrN4O2
(2R)-2-(4-bromophenoxy)-1-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]propan-1-one
—— N'-(2-aminophenyl)-N-[3-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]heptanediamide —— C46H46N4O6S
N'-(2-aminophenyl)-N-[3-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]heptanediamide
—— N'-(2-aminophenyl)-N-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]octanediamide —— C39H43N7O6S
N'-(2-aminophenyl)-N-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]octanediamide
—— 7-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methylamino]-7-oxoheptanoic acid —— C33H37N5O7S
7-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methylamino]-7-oxoheptanoic acid
—— 1-[(1S)-1-(furan-2-yl)-2-methoxyethyl]-3-[4-(1H-pyrazol-5-yl)phenyl]urea —— C17H18N4O3
1-[(1S)-1-(furan-2-yl)-2-methoxyethyl]-3-[4-(1H-pyrazol-5-yl)phenyl]urea
—— (3S)-5-N-(2-hydroxyethyl)-5-N-(2-methoxyethyl)-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide —— C16H22N4O4
(3S)-5-N-(2-hydroxyethyl)-5-N-(2-methoxyethyl)-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide
—— [5-(2-chlorophenyl)-1H-pyrazol-4-yl]-[(3R,4R)-3-hydroxy-4-methylpiperidin-1-yl]methanone —— C16H18ClN3O2
[5-(2-chlorophenyl)-1H-pyrazol-4-yl]-[(3R,4R)-3-hydroxy-4-methylpiperidin-1-yl]methanone
—— N'-hydroxy-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]heptanediamide —— C33H38N6O7S
N'-hydroxy-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]heptanediamide
—— N'-(2-aminophenyl)-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]heptanediamide —— C39H43N7O5S
N'-(2-aminophenyl)-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]heptanediamide
—— 1-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-(4-phenyltriazol-1-yl)ethanone —— C16H20N4O2
1-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-(4-phenyltriazol-1-yl)ethanone
—— (1R)-1-cyclopropyl-2-methoxy-N-[(1-phenylpyrazol-4-yl)methyl]ethanamine —— C16H21N3O
(1R)-1-cyclopropyl-2-methoxy-N-[(1-phenylpyrazol-4-yl)methyl]ethanamine
—— 1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-2-(4-phenyltriazol-1-yl)ethanone —— C16H20N4O2
1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-2-(4-phenyltriazol-1-yl)ethanone
—— methyl 3-[[(2S)-2-(1H-imidazol-2-yl)piperidin-1-yl]methyl]thiophene-2-carboxylate —— C15H19N3O2S
methyl 3-[[(2S)-2-(1H-imidazol-2-yl)piperidin-1-yl]methyl]thiophene-2-carboxylate
—— [5-(2-chlorophenyl)-1H-pyrazol-4-yl]-[(3S,4S)-3-hydroxy-4-methylpiperidin-1-yl]methanone —— C16H18ClN3O2
[5-(2-chlorophenyl)-1H-pyrazol-4-yl]-[(3S,4S)-3-hydroxy-4-methylpiperidin-1-yl]methanone
—— N'-hydroxy-N-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]hexanediamide —— C31H34N6O6S
N'-hydroxy-N-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]hexanediamide
—— 6-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid —— C32H35N5O7S
6-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid
—— 1-[(1R)-1-(furan-2-yl)-2-methoxyethyl]-3-[4-(1H-pyrazol-5-yl)phenyl]urea —— C17H18N4O3
1-[(1R)-1-(furan-2-yl)-2-methoxyethyl]-3-[4-(1H-pyrazol-5-yl)phenyl]urea
—— methyl (2R)-2-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-2-pyridin-3-ylacetate —— C23H18N2O3S
methyl (2R)-2-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-2-pyridin-3-ylacetate
—— 8-[[4-[(2S,4S,6R)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-8-oxooctanoic acid —— C30H35Cl2N3O6
8-[[4-[(2S,4S,6R)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-8-oxooctanoic acid
—— [5-(2-chlorophenyl)-1H-pyrazol-4-yl]-[(3S,4R)-3-hydroxy-4-methylpiperidin-1-yl]methanone —— C16H18ClN3O2
[5-(2-chlorophenyl)-1H-pyrazol-4-yl]-[(3S,4R)-3-hydroxy-4-methylpiperidin-1-yl]methanone
—— [5-(2-chlorophenyl)-1H-pyrazol-4-yl]-[(3R,4S)-3-hydroxy-4-methylpiperidin-1-yl]methanone —— C16H18ClN3O2
[5-(2-chlorophenyl)-1H-pyrazol-4-yl]-[(3R,4S)-3-hydroxy-4-methylpiperidin-1-yl]methanone
—— methyl 3-[[(2R)-2-(1H-imidazol-2-yl)piperidin-1-yl]methyl]thiophene-2-carboxylate —— C15H19N3O2S
methyl 3-[[(2R)-2-(1H-imidazol-2-yl)piperidin-1-yl]methyl]thiophene-2-carboxylate
—— (1S)-1-cyclopropyl-2-methoxy-N-[(1-phenylpyrazol-4-yl)methyl]ethanamine —— C16H21N3O
(1S)-1-cyclopropyl-2-methoxy-N-[(1-phenylpyrazol-4-yl)methyl]ethanamine
—— (3R)-5-N-(2-hydroxyethyl)-5-N-(2-methoxyethyl)-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide —— C16H22N4O4
(3R)-5-N-(2-hydroxyethyl)-5-N-(2-methoxyethyl)-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide
—— methyl 2-[(2S)-4-[[1-(4-fluorophenyl)pyrazol-3-yl]methyl]morpholin-2-yl]acetate —— C17H20FN3O3
methyl 2-[(2S)-4-[[1-(4-fluorophenyl)pyrazol-3-yl]methyl]morpholin-2-yl]acetate
—— methyl 2-[(2R)-4-[[1-(4-fluorophenyl)pyrazol-3-yl]methyl]morpholin-2-yl]acetate —— C17H20FN3O3
methyl 2-[(2R)-4-[[1-(4-fluorophenyl)pyrazol-3-yl]methyl]morpholin-2-yl]acetate
—— methyl (2S)-2-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-2-pyridin-3-ylacetate —— C23H18N2O3S
methyl (2S)-2-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-2-pyridin-3-ylacetate
—— methyl (4R)-1-[(5-thiophen-2-yl-1,2-oxazol-3-yl)methyl]-4,5,6,7-tetrahydroindazole-4-carboxylate —— C17H17N3O3S
methyl (4R)-1-[(5-thiophen-2-yl-1,2-oxazol-3-yl)methyl]-4,5,6,7-tetrahydroindazole-4-carboxylate
—— N'-(2-aminophenyl)-N-[3-[(2R,4R,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]pentanediamide —— C44H42N4O6S
N'-(2-aminophenyl)-N-[3-[(2R,4R,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]pentanediamide
—— N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]octanediamide —— C39H43N7O6S
N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]octanediamide
—— 6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid —— C32H35N5O7S
6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid
—— methyl 2-[(2R)-4-[(4-imidazol-1-ylphenyl)methyl]morpholin-2-yl]acetate —— C17H21N3O3
methyl 2-[(2R)-4-[(4-imidazol-1-ylphenyl)methyl]morpholin-2-yl]acetate
—— methyl (4S)-1-[(5-thiophen-2-yl-1,2-oxazol-3-yl)methyl]-4,5,6,7-tetrahydroindazole-4-carboxylate —— C17H17N3O3S
methyl (4S)-1-[(5-thiophen-2-yl-1,2-oxazol-3-yl)methyl]-4,5,6,7-tetrahydroindazole-4-carboxylate
—— methyl (6R)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-6-carboxylate —— C12H16N2O2
methyl (6R)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-6-carboxylate
—— methyl (6S)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-6-carboxylate —— C12H16N2O2
methyl (6S)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-6-carboxylate
—— methyl 2-[(2S)-4-[(4-imidazol-1-ylphenyl)methyl]morpholin-2-yl]acetate —— C17H21N3O3
methyl 2-[(2S)-4-[(4-imidazol-1-ylphenyl)methyl]morpholin-2-yl]acetate
—— (3S)-3-(3-chlorophenyl)-N-methyl-5-phenyl-3,4-dihydropyrazole-2-carbothioamide —— C17H16ClN3S
(3S)-3-(3-chlorophenyl)-N-methyl-5-phenyl-3,4-dihydropyrazole-2-carbothioamide
—— 5-[3-[(2R,4R,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C38H36N2O7S
5-[3-[(2R,4R,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]pentanediamide —— C36H37N7O6S
N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]pentanediamide
—— N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]heptanediamide —— C38H41N7O6S
N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]heptanediamide
—— 6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C31H33N5O7S
6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— 6-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C31H33N5O7S
6-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— (3R)-3-(3-bromophenyl)-N-methyl-5-phenyl-3,4-dihydropyrazole-2-carbothioamide —— C17H16BrN3S
(3R)-3-(3-bromophenyl)-N-methyl-5-phenyl-3,4-dihydropyrazole-2-carbothioamide
—— (3S)-3-(3-bromophenyl)-N-methyl-5-phenyl-3,4-dihydropyrazole-2-carbothioamide —— C17H16BrN3S
(3S)-3-(3-bromophenyl)-N-methyl-5-phenyl-3,4-dihydropyrazole-2-carbothioamide
—— N-[(1S)-7-fluoro-1,2,3,4-tetrahydronaphthalen-1-yl]-4-(1,2,4-triazol-4-yl)benzamide —— C19H17FN4O
N-[(1S)-7-fluoro-1,2,3,4-tetrahydronaphthalen-1-yl]-4-(1,2,4-triazol-4-yl)benzamide
—— N-[[4-[(2R,4R,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]-N'-hydroxyoctanediamide —— C42H45N3O7S
N-[[4-[(2R,4R,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]-N'-hydroxyoctanediamide
—— [2-(4-methoxyphenyl)-1,3-thiazol-4-yl]-[(3R)-3-(4-methylpiperazin-1-yl)azepan-1-yl]methanone —— C22H30N4O2S
[2-(4-methoxyphenyl)-1,3-thiazol-4-yl]-[(3R)-3-(4-methylpiperazin-1-yl)azepan-1-yl]methanone