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中文名称 英文名称 CAS号 化学式 结构式图片
—— (1S)-1-(4-fluorophenyl)-2,2-dimethyl-N-[[2-(1,2,4-triazol-1-yl)phenyl]methyl]cyclopropane-1-carboxamide —— C21H21FN4O
(1S)-1-(4-fluorophenyl)-2,2-dimethyl-N-[[2-(1,2,4-triazol-1-yl)phenyl]methyl]cyclopropane-1-carboxamide
—— 2-[[3-(3-fluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C18H18FN5O2S
2-[[3-(3-fluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 4-(benzenesulfonyl)-5-[(2S)-butan-2-yl]sulfanyl-2-(4-methylphenyl)-1,3-oxazole —— C20H21NO3S2
4-(benzenesulfonyl)-5-[(2S)-butan-2-yl]sulfanyl-2-(4-methylphenyl)-1,3-oxazole
—— 1-[(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-2-(2-phenylimidazol-1-yl)ethanone —— C23H23N5O
1-[(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-2-(2-phenylimidazol-1-yl)ethanone
—— 1-N'-[(4S)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]cyclopropane-1,1-dicarboxamide —— C21H26N4O2
1-N'-[(4S)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]cyclopropane-1,1-dicarboxamide
—— 5-(3-fluorophenyl)-N-[(1R)-2,2,2-trifluoro-1-pyridin-2-ylethyl]-1H-pyrazole-4-carboxamide —— C17H12F4N4O
5-(3-fluorophenyl)-N-[(1R)-2,2,2-trifluoro-1-pyridin-2-ylethyl]-1H-pyrazole-4-carboxamide
—— (2-methylsulfanylpyrimidin-5-yl)-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C18H17N5O2S
(2-methylsulfanylpyrimidin-5-yl)-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— ethyl (2S)-2-[3-(4-fluorophenyl)triazolo[4,5-d]pyrimidin-7-yl]sulfanylpropanoate —— C15H14FN5O2S
ethyl (2S)-2-[3-(4-fluorophenyl)triazolo[4,5-d]pyrimidin-7-yl]sulfanylpropanoate
—— (5R)-7-(cyclopropylmethyl)-2-[(2-pyrazol-1-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H28N4O
(5R)-7-(cyclopropylmethyl)-2-[(2-pyrazol-1-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 3-(4-fluorophenyl)-N-[(1S)-1-phenyl-2-pyrazol-1-ylethyl]-1H-pyrazole-5-carboxamide —— C21H18FN5O
3-(4-fluorophenyl)-N-[(1S)-1-phenyl-2-pyrazol-1-ylethyl]-1H-pyrazole-5-carboxamide
—— (4S)-1-(4-tert-butylphenyl)-4-(dimethylsulfamoylamino)-4,5,6,7-tetrahydroindazole —— C19H28N4O2S
(4S)-1-(4-tert-butylphenyl)-4-(dimethylsulfamoylamino)-4,5,6,7-tetrahydroindazole
—— (5R)-9-[[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C19H23N3O5
(5R)-9-[[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-methyl-N-[(1S)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-1-propylpyrazole-4-carboxamide —— C21H27N5O
5-methyl-N-[(1S)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-1-propylpyrazole-4-carboxamide
—— (5S)-7-(cyclopropylmethyl)-2-[(2-pyrazol-1-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H28N4O
(5S)-7-(cyclopropylmethyl)-2-[(2-pyrazol-1-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (2-methylsulfanylpyrimidin-5-yl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C18H17N5O2S
(2-methylsulfanylpyrimidin-5-yl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— 1-tert-butyl-3-[(4S)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]urea —— C18H22F2N4O
1-tert-butyl-3-[(4S)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]urea
—— 5-methyl-N-[(1R)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-1-propylpyrazole-4-carboxamide —— C21H27N5O
5-methyl-N-[(1R)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-1-propylpyrazole-4-carboxamide
—— 3-(4-fluorophenyl)-N-[(1R)-1-phenyl-2-pyrazol-1-ylethyl]-1H-pyrazole-5-carboxamide —— C21H18FN5O
3-(4-fluorophenyl)-N-[(1R)-1-phenyl-2-pyrazol-1-ylethyl]-1H-pyrazole-5-carboxamide
—— 5-(3-fluorophenyl)-N-[(1S)-2,2,2-trifluoro-1-pyridin-2-ylethyl]-1H-pyrazole-4-carboxamide —— C17H12F4N4O
5-(3-fluorophenyl)-N-[(1S)-2,2,2-trifluoro-1-pyridin-2-ylethyl]-1H-pyrazole-4-carboxamide
—— (5R)-7-cyclohexyl-2-(1-phenyltetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one —— C21H28N6O
(5R)-7-cyclohexyl-2-(1-phenyltetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 1-N'-[(4R)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]cyclopropane-1,1-dicarboxamide —— C21H26N4O2
1-N'-[(4R)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]cyclopropane-1,1-dicarboxamide
—— (5S)-7-cyclohexyl-2-(1-phenyltetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one —— C21H28N6O
(5S)-7-cyclohexyl-2-(1-phenyltetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 1-[(3S)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-2-(2-phenylimidazol-1-yl)ethanone —— C23H23N5O
1-[(3S)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-2-(2-phenylimidazol-1-yl)ethanone
—— (7-methylpyrazolo[1,5-a]pyrimidin-6-yl)-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C20H18N6O2
(7-methylpyrazolo[1,5-a]pyrimidin-6-yl)-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— 1-(4-methoxyphenyl)-5-[(3S)-3-pyrrolidin-1-ylbutyl]-1,2,4-triazole —— C17H24N4O
1-(4-methoxyphenyl)-5-[(3S)-3-pyrrolidin-1-ylbutyl]-1,2,4-triazole
—— 1-(4-methoxyphenyl)-5-[(3R)-3-pyrrolidin-1-ylbutyl]-1,2,4-triazole —— C17H24N4O
1-(4-methoxyphenyl)-5-[(3R)-3-pyrrolidin-1-ylbutyl]-1,2,4-triazole
—— (4R)-1-(4-tert-butylphenyl)-4-(dimethylsulfamoylamino)-4,5,6,7-tetrahydroindazole —— C19H28N4O2S
(4R)-1-(4-tert-butylphenyl)-4-(dimethylsulfamoylamino)-4,5,6,7-tetrahydroindazole
—— (2-fluoro-6-methoxyphenyl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C20H18FN3O3
(2-fluoro-6-methoxyphenyl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— 1-methyl-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1-[(2S)-3,3,3-trifluoro-2-hydroxypropyl]urea —— C12H16F3N3O2S
1-methyl-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1-[(2S)-3,3,3-trifluoro-2-hydroxypropyl]urea
—— (7-methylpyrazolo[1,5-a]pyrimidin-6-yl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C20H18N6O2
(7-methylpyrazolo[1,5-a]pyrimidin-6-yl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— (5S)-9-[[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C19H23N3O5
(5S)-9-[[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 1-tert-butyl-3-[(4R)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]urea —— C18H22F2N4O
1-tert-butyl-3-[(4R)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]urea
—— 5-methyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-3-ylethyl]-1-propylpyrazole-4-carboxamide —— C19H27N5O2
5-methyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-3-ylethyl]-1-propylpyrazole-4-carboxamide
—— 1-methyl-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1-[(2R)-3,3,3-trifluoro-2-hydroxypropyl]urea —— C12H16F3N3O2S
1-methyl-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1-[(2R)-3,3,3-trifluoro-2-hydroxypropyl]urea
—— methyl (2R)-2-[[3-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl]propanoate —— C15H13FN4O2S
methyl (2R)-2-[[3-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl]propanoate
—— N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-5-ethyl-1,3,4-oxadiazol-2-amine —— C11H16N4OS
N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-5-ethyl-1,3,4-oxadiazol-2-amine
—— (5S)-5-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid —— C9H12N2O2
(5S)-5-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
—— (3R)-8-methoxy-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3,4-dihydro-2H-chromene-3-carboxamide —— C20H19N3O4
(3R)-8-methoxy-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3,4-dihydro-2H-chromene-3-carboxamide
—— (3S)-8-methoxy-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3,4-dihydro-2H-chromene-3-carboxamide —— C20H19N3O4
(3S)-8-methoxy-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3,4-dihydro-2H-chromene-3-carboxamide
—— 5-methyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-3-ylethyl]-1-propylpyrazole-4-carboxamide —— C19H27N5O2
5-methyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-3-ylethyl]-1-propylpyrazole-4-carboxamide
—— [3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-[(2R)-2-(2-methoxyphenyl)pyrrolidin-1-yl]methanone —— C22H23N3O3
[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-[(2R)-2-(2-methoxyphenyl)pyrrolidin-1-yl]methanone
—— N-[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-5-ethyl-1,3,4-oxadiazol-2-amine —— C11H16N4OS
N-[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-5-ethyl-1,3,4-oxadiazol-2-amine
—— [3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-[(2S)-2-(2-methoxyphenyl)pyrrolidin-1-yl]methanone —— C22H23N3O3
[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-[(2S)-2-(2-methoxyphenyl)pyrrolidin-1-yl]methanone
—— N-[(4S)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]-5-ethyl-4-methyl-1H-pyrazole-3-carboxamide —— C23H29N5O
N-[(4S)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]-5-ethyl-4-methyl-1H-pyrazole-3-carboxamide
—— N-[(4R)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]-5-ethyl-4-methyl-1H-pyrazole-3-carboxamide —— C23H29N5O
N-[(4R)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]-5-ethyl-4-methyl-1H-pyrazole-3-carboxamide
—— [(2S)-oxolan-2-yl]-[4-[4-(1H-pyrazol-5-yl)benzoyl]piperazin-1-yl]methanone —— C19H22N4O3
[(2S)-oxolan-2-yl]-[4-[4-(1H-pyrazol-5-yl)benzoyl]piperazin-1-yl]methanone
—— 1-(2-methoxyphenyl)-N-[(2S)-1-thiophen-2-ylpropan-2-yl]pyrazole-4-carboxamide —— C18H19N3O2S
1-(2-methoxyphenyl)-N-[(2S)-1-thiophen-2-ylpropan-2-yl]pyrazole-4-carboxamide
—— 1-(2-methoxyphenyl)-N-[(2R)-1-thiophen-2-ylpropan-2-yl]pyrazole-4-carboxamide —— C18H19N3O2S
1-(2-methoxyphenyl)-N-[(2R)-1-thiophen-2-ylpropan-2-yl]pyrazole-4-carboxamide
—— (5-cyclohexyl-1H-pyrazol-4-yl)-[(2R)-2-(furan-2-yl)pyrrolidin-1-yl]methanone —— C18H23N3O2
(5-cyclohexyl-1H-pyrazol-4-yl)-[(2R)-2-(furan-2-yl)pyrrolidin-1-yl]methanone
—— 1-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-propan-2-ylurea —— C19H26N4O
1-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-propan-2-ylurea