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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-(5-chloro-2-methoxyphenyl)-3-[[4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methylsulfanyl]-1H-1,2,4-triazole —— C21H22ClN3O3S
5-(5-chloro-2-methoxyphenyl)-3-[[4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methylsulfanyl]-1H-1,2,4-triazole
—— (3R)-7-methoxy-N-[2-(1H-1,2,4-triazol-5-yl)phenyl]-3,4-dihydro-2H-chromene-3-carboxamide —— C19H18N4O3
(3R)-7-methoxy-N-[2-(1H-1,2,4-triazol-5-yl)phenyl]-3,4-dihydro-2H-chromene-3-carboxamide
—— N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]-1-(4-methoxyphenyl)pyrazole-3-carboxamide —— C20H25N3O4
N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]-1-(4-methoxyphenyl)pyrazole-3-carboxamide
—— 2-[(7R)-5,7-dihydro-4H-thieno[2,3-c]pyran-7-yl]-N-[[1-(4-methoxyphenyl)triazol-4-yl]methyl]acetamide —— C19H20N4O3S
2-[(7R)-5,7-dihydro-4H-thieno[2,3-c]pyran-7-yl]-N-[[1-(4-methoxyphenyl)triazol-4-yl]methyl]acetamide
—— [1-(4-methoxyphenyl)pyrazol-3-yl]-[(2S)-2-(1H-pyrazol-4-yl)piperidin-1-yl]methanone —— C19H21N5O2
[1-(4-methoxyphenyl)pyrazol-3-yl]-[(2S)-2-(1H-pyrazol-4-yl)piperidin-1-yl]methanone
—— 5-(4-methoxyphenyl)-3-[[(2S)-oxolan-2-yl]methylsulfonylmethyl]-1,2,4-oxadiazole —— C15H18N2O5S
5-(4-methoxyphenyl)-3-[[(2S)-oxolan-2-yl]methylsulfonylmethyl]-1,2,4-oxadiazole
—— [1-(4-methoxyphenyl)pyrazol-3-yl]-[(2R)-2-(1H-pyrazol-4-yl)piperidin-1-yl]methanone —— C19H21N5O2
[1-(4-methoxyphenyl)pyrazol-3-yl]-[(2R)-2-(1H-pyrazol-4-yl)piperidin-1-yl]methanone
—— (2R)-1-benzyl-2-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]imidazolidin-4-one —— C20H20N4O2
(2R)-1-benzyl-2-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]imidazolidin-4-one
—— N-[(3R)-1-(5-chloro-2-methoxyphenyl)pyrrolidin-3-yl]-3-(2-methylsulfanylimidazol-1-yl)benzamide —— C22H23ClN4O2S
N-[(3R)-1-(5-chloro-2-methoxyphenyl)pyrrolidin-3-yl]-3-(2-methylsulfanylimidazol-1-yl)benzamide
—— (2S)-N-[(3R)-1-(cyclopentylmethyl)pyrrolidin-3-yl]-2-(2-phenylimidazol-1-yl)propanamide —— C22H30N4O
(2S)-N-[(3R)-1-(cyclopentylmethyl)pyrrolidin-3-yl]-2-(2-phenylimidazol-1-yl)propanamide
—— (2S)-1-benzyl-2-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]imidazolidin-4-one —— C20H20N4O2
(2S)-1-benzyl-2-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]imidazolidin-4-one
—— 2-[(7S)-5,7-dihydro-4H-thieno[2,3-c]pyran-7-yl]-N-[[1-(4-methoxyphenyl)triazol-4-yl]methyl]acetamide —— C19H20N4O3S
2-[(7S)-5,7-dihydro-4H-thieno[2,3-c]pyran-7-yl]-N-[[1-(4-methoxyphenyl)triazol-4-yl]methyl]acetamide
—— 5-(4-methoxyphenyl)-3-[[(2R)-oxolan-2-yl]methylsulfonylmethyl]-1,2,4-oxadiazole —— C15H18N2O5S
5-(4-methoxyphenyl)-3-[[(2R)-oxolan-2-yl]methylsulfonylmethyl]-1,2,4-oxadiazole
—— (4S)-N-[[1-(4-methoxyphenyl)pyrazol-3-yl]methyl]-2-oxoimidazolidine-4-carboxamide —— C15H17N5O3
(4S)-N-[[1-(4-methoxyphenyl)pyrazol-3-yl]methyl]-2-oxoimidazolidine-4-carboxamide
—— 5-[[4-[(2S,4S,5R,6R)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methylamino]-5-oxopentanoic acid —— C28H31Cl2N3O6
5-[[4-[(2S,4S,5R,6R)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methylamino]-5-oxopentanoic acid
—— 1-(5-ethyl-3-methyl-1,2-oxazol-4-yl)-3-[(1R)-1-(5-methyl-1,2,4-oxadiazol-3-yl)propyl]urea —— C13H19N5O3
1-(5-ethyl-3-methyl-1,2-oxazol-4-yl)-3-[(1R)-1-(5-methyl-1,2,4-oxadiazol-3-yl)propyl]urea
—— 1-(5-ethyl-3-methyl-1,2-oxazol-4-yl)-3-[(1S)-1-(5-methyl-1,2,4-oxadiazol-3-yl)propyl]urea —— C13H19N5O3
1-(5-ethyl-3-methyl-1,2-oxazol-4-yl)-3-[(1S)-1-(5-methyl-1,2,4-oxadiazol-3-yl)propyl]urea
—— (2S)-N-cyclopropyl-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]propanamide —— C16H19N3OS
(2S)-N-cyclopropyl-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]propanamide
—— (2R)-N-[(3R)-1-(cyclopentylmethyl)pyrrolidin-3-yl]-2-(2-phenylimidazol-1-yl)propanamide —— C22H30N4O
(2R)-N-[(3R)-1-(cyclopentylmethyl)pyrrolidin-3-yl]-2-(2-phenylimidazol-1-yl)propanamide
—— N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]-1-(4-methoxyphenyl)pyrazole-3-carboxamide —— C20H25N3O4
N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]-1-(4-methoxyphenyl)pyrazole-3-carboxamide
—— (2R)-N-[(3S)-1-(cyclopentylmethyl)pyrrolidin-3-yl]-2-(2-phenylimidazol-1-yl)propanamide —— C22H30N4O
(2R)-N-[(3S)-1-(cyclopentylmethyl)pyrrolidin-3-yl]-2-(2-phenylimidazol-1-yl)propanamide
—— (2S)-N-[(3S)-1-(cyclopentylmethyl)pyrrolidin-3-yl]-2-(2-phenylimidazol-1-yl)propanamide —— C22H30N4O
(2S)-N-[(3S)-1-(cyclopentylmethyl)pyrrolidin-3-yl]-2-(2-phenylimidazol-1-yl)propanamide
—— (2R)-N-cyclopropyl-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]propanamide —— C16H19N3OS
(2R)-N-cyclopropyl-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]propanamide
—— (4R)-N-[[1-(4-methoxyphenyl)pyrazol-3-yl]methyl]-2-oxoimidazolidine-4-carboxamide —— C15H17N5O3
(4R)-N-[[1-(4-methoxyphenyl)pyrazol-3-yl]methyl]-2-oxoimidazolidine-4-carboxamide
—— 3-(2-methoxyphenyl)-4-[(3R)-5-(4-methoxyphenyl)-2-methylsulfonyl-3,4-dihydropyrazol-3-yl]-1-phenylpyrazole —— C27H26N4O4S
3-(2-methoxyphenyl)-4-[(3R)-5-(4-methoxyphenyl)-2-methylsulfonyl-3,4-dihydropyrazol-3-yl]-1-phenylpyrazole
—— [(2R)-2-[(S)-hydroxy-(4-methoxyphenyl)methyl]pyrrolidin-1-yl]-(2-phenyltriazol-4-yl)methanone —— C21H22N4O3
[(2R)-2-[(S)-hydroxy-(4-methoxyphenyl)methyl]pyrrolidin-1-yl]-(2-phenyltriazol-4-yl)methanone
—— (3S)-3-(2,4-dimethoxyphenyl)-N,5-diphenyl-3,4-dihydropyrazole-2-carbothioamide —— C24H23N3O2S
(3S)-3-(2,4-dimethoxyphenyl)-N,5-diphenyl-3,4-dihydropyrazole-2-carbothioamide
—— (3R)-3-(2,4-dimethoxyphenyl)-N,5-diphenyl-3,4-dihydropyrazole-2-carbothioamide —— C24H23N3O2S
(3R)-3-(2,4-dimethoxyphenyl)-N,5-diphenyl-3,4-dihydropyrazole-2-carbothioamide
—— 3-(2-methoxyphenyl)-4-[(3S)-5-(4-methoxyphenyl)-2-methylsulfonyl-3,4-dihydropyrazol-3-yl]-1-phenylpyrazole —— C27H26N4O4S
3-(2-methoxyphenyl)-4-[(3S)-5-(4-methoxyphenyl)-2-methylsulfonyl-3,4-dihydropyrazol-3-yl]-1-phenylpyrazole
—— [(2S)-2-[(R)-hydroxy-(4-methoxyphenyl)methyl]pyrrolidin-1-yl]-(2-phenyltriazol-4-yl)methanone —— C21H22N4O3
[(2S)-2-[(R)-hydroxy-(4-methoxyphenyl)methyl]pyrrolidin-1-yl]-(2-phenyltriazol-4-yl)methanone
—— [(2S)-2-[(S)-hydroxy-(4-methoxyphenyl)methyl]pyrrolidin-1-yl]-(2-phenyltriazol-4-yl)methanone —— C21H22N4O3
[(2S)-2-[(S)-hydroxy-(4-methoxyphenyl)methyl]pyrrolidin-1-yl]-(2-phenyltriazol-4-yl)methanone
—— [(2R)-2-[(R)-hydroxy-(4-methoxyphenyl)methyl]pyrrolidin-1-yl]-(2-phenyltriazol-4-yl)methanone —— C21H22N4O3
[(2R)-2-[(R)-hydroxy-(4-methoxyphenyl)methyl]pyrrolidin-1-yl]-(2-phenyltriazol-4-yl)methanone
—— N'-[(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-1-phenyl-3-thiophen-2-ylpyrazole-4-carbohydrazide —— C22H18N4O3S
N'-[(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-1-phenyl-3-thiophen-2-ylpyrazole-4-carbohydrazide
—— 3-(methoxymethyl)-5-[(4S)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,2,4-oxadiazole —— C11H14N4O2
3-(methoxymethyl)-5-[(4S)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,2,4-oxadiazole
—— 3-(methoxymethyl)-5-[(4R)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,2,4-oxadiazole —— C11H14N4O2
3-(methoxymethyl)-5-[(4R)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,2,4-oxadiazole
—— (1R,3S)-1-[4-(hydroxymethyl)phenyl]-4-[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylbutane-1,3-diol —— C18H20N4O4S
(1R,3S)-1-[4-(hydroxymethyl)phenyl]-4-[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylbutane-1,3-diol
—— (8S)-2-(methoxymethyl)-N-[(1-phenylpyrazol-4-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-amine —— C18H22N6O
(8S)-2-(methoxymethyl)-N-[(1-phenylpyrazol-4-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-amine
—— (8R)-2-(methoxymethyl)-N-[(1-phenylpyrazol-4-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-amine —— C18H22N6O
(8R)-2-(methoxymethyl)-N-[(1-phenylpyrazol-4-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-amine
—— 3-[(1S)-cyclohex-2-en-1-yl]-5-(methoxymethyl)-1,3,4-oxadiazol-2-one —— C10H14N2O3
3-[(1S)-cyclohex-2-en-1-yl]-5-(methoxymethyl)-1,3,4-oxadiazol-2-one
—— 3-[(1R)-cyclohex-2-en-1-yl]-5-(methoxymethyl)-1,3,4-oxadiazol-2-one —— C10H14N2O3
3-[(1R)-cyclohex-2-en-1-yl]-5-(methoxymethyl)-1,3,4-oxadiazol-2-one
—— (2-methoxypyridin-3-yl)-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone —— C19H19N5O2
(2-methoxypyridin-3-yl)-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone
—— 4-[5-[[(4S,5R,6R)-2-(3-aminophenyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-4-yl]methylsulfanyl]tetrazol-1-yl]phenol —— C26H27N5O4S
4-[5-[[(4S,5R,6R)-2-(3-aminophenyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-4-yl]methylsulfanyl]tetrazol-1-yl]phenol
—— (2-methoxypyridin-3-yl)-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone —— C19H19N5O2
(2-methoxypyridin-3-yl)-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone
—— N-[3-[(4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]quinoline-8-sulfonamide —— C42H35N3O6S2
N-[3-[(4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]quinoline-8-sulfonamide
—— 8-[[4-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-8-oxooctanoic acid —— C42H44N2O7S
8-[[4-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-8-oxooctanoic acid
—— 5-[(1R,6S)-7-bicyclo[4.1.0]heptanyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C12H18N2O2
5-[(1R,6S)-7-bicyclo[4.1.0]heptanyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— 8-[3-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-8-oxooctanoic acid —— C41H42N2O7S
8-[3-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-8-oxooctanoic acid
—— N'-(2-aminophenyl)-N-[4-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]heptanediamide —— C46H46N4O6S
N'-(2-aminophenyl)-N-[4-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]heptanediamide
—— (2R)-2-(4-bromophenoxy)-1-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]propan-1-one —— C21H21BrN4O2
(2R)-2-(4-bromophenoxy)-1-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]propan-1-one
—— 1-ethyl-3-[[4-[(4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]urea —— C29H32N6O5S
1-ethyl-3-[[4-[(4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]urea