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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl (3R)-3-[[(3S)-3-hydroxybutyl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate —— C17H23N3O4
ethyl (3R)-3-[[(3S)-3-hydroxybutyl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate
—— ethyl N-[(2R)-1-[[5-(2,5-difluorophenyl)-1,2,4-oxadiazole-3-carbonyl]amino]-4-methylpentan-2-yl]carbamate —— C18H22F2N4O4
ethyl N-[(2R)-1-[[5-(2,5-difluorophenyl)-1,2,4-oxadiazole-3-carbonyl]amino]-4-methylpentan-2-yl]carbamate
—— ethyl (3R)-3-[(5-phenyl-1,3-thiazol-2-yl)carbamoylamino]butanoate —— C16H19N3O3S
ethyl (3R)-3-[(5-phenyl-1,3-thiazol-2-yl)carbamoylamino]butanoate
—— (3R)-3-(4-ethylpiperazin-1-yl)-N-[5-[(3-fluorophenyl)methyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide —— C20H27FN6OS
(3R)-3-(4-ethylpiperazin-1-yl)-N-[5-[(3-fluorophenyl)methyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide
—— N-[(3R)-1-(ethylcarbamoyl)pyrrolidin-3-yl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide —— C16H20N4O2S2
N-[(3R)-1-(ethylcarbamoyl)pyrrolidin-3-yl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide
—— 1-(4-chlorophenyl)-N-[(3R)-1-(ethylcarbamoyl)pyrrolidin-3-yl]-5-(furan-2-yl)pyrazole-3-carboxamide —— C21H22ClN5O3
1-(4-chlorophenyl)-N-[(3R)-1-(ethylcarbamoyl)pyrrolidin-3-yl]-5-(furan-2-yl)pyrazole-3-carboxamide
—— 1-(4-chlorophenyl)-N-[(3S)-1-(ethylcarbamoyl)pyrrolidin-3-yl]-5-(furan-2-yl)pyrazole-3-carboxamide —— C21H22ClN5O3
1-(4-chlorophenyl)-N-[(3S)-1-(ethylcarbamoyl)pyrrolidin-3-yl]-5-(furan-2-yl)pyrazole-3-carboxamide
—— 2-(ethylamino)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1,3-thiazole-5-carboxamide —— C18H20FN5OS
2-(ethylamino)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1,3-thiazole-5-carboxamide
—— N-[(3S)-1-(ethylcarbamoyl)pyrrolidin-3-yl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide —— C16H20N4O2S2
N-[(3S)-1-(ethylcarbamoyl)pyrrolidin-3-yl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide
—— 1-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-3-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]urea —— C17H25N7O
1-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-3-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]urea
—— 2-(ethylamino)-4-methyl-N-[(1S)-2-methyl-1-(5-methyl-1H-1,2,4-triazol-3-yl)propyl]-1,3-thiazole-5-carboxamide —— C14H22N6OS
2-(ethylamino)-4-methyl-N-[(1S)-2-methyl-1-(5-methyl-1H-1,2,4-triazol-3-yl)propyl]-1,3-thiazole-5-carboxamide
—— 2-(ethylamino)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1,3-thiazole-5-carboxamide —— C18H20FN5OS
2-(ethylamino)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1,3-thiazole-5-carboxamide
—— methyl (1S,2S)-2-[[2-(1,2-oxazol-3-yl)acetyl]amino]cyclohexane-1-carboxylate —— C13H18N2O4
methyl (1S,2S)-2-[[2-(1,2-oxazol-3-yl)acetyl]amino]cyclohexane-1-carboxylate
—— methyl (1R,2R)-2-[[2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]acetyl]amino]cyclohexane-1-carboxylate —— C16H23F2N3O3
methyl (1R,2R)-2-[[2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]acetyl]amino]cyclohexane-1-carboxylate
—— 1-[(3S)-1-ethylpyrrolidin-3-yl]-N-[(2-thiophen-3-yl-1,3-thiazol-4-yl)methyl]methanamine —— C15H21N3S2
1-[(3S)-1-ethylpyrrolidin-3-yl]-N-[(2-thiophen-3-yl-1,3-thiazol-4-yl)methyl]methanamine
—— N-[[(2R)-4-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]morpholin-2-yl]methyl]-N-ethylpyridazin-3-amine —— C17H25N5O2
N-[[(2R)-4-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]morpholin-2-yl]methyl]-N-ethylpyridazin-3-amine
—— (3S)-3-(4-ethylpiperazin-1-yl)-N-[5-[(3-fluorophenyl)methyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide —— C20H27FN6OS
(3S)-3-(4-ethylpiperazin-1-yl)-N-[5-[(3-fluorophenyl)methyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide
—— N-[[(2S)-4-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]morpholin-2-yl]methyl]-N-ethylpyridazin-3-amine —— C17H25N5O2
N-[[(2S)-4-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]morpholin-2-yl]methyl]-N-ethylpyridazin-3-amine
—— N-[(3R)-1-ethylpiperidin-3-yl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide —— C18H25N5O2
N-[(3R)-1-ethylpiperidin-3-yl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide
—— N-[[(2R)-4-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]morpholin-2-yl]methyl]-N-ethylpyridazin-3-amine —— C17H25N5OS
N-[[(2R)-4-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]morpholin-2-yl]methyl]-N-ethylpyridazin-3-amine
—— N-ethyl-N-[4-[[(3S)-3-(5-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl]-1,3-thiazol-2-yl]acetamide —— C17H25N5OS
N-ethyl-N-[4-[[(3S)-3-(5-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl]-1,3-thiazol-2-yl]acetamide
—— 1-[(3R)-1-ethylpyrrolidin-3-yl]-N-[(2-thiophen-3-yl-1,3-thiazol-4-yl)methyl]methanamine —— C15H21N3S2
1-[(3R)-1-ethylpyrrolidin-3-yl]-N-[(2-thiophen-3-yl-1,3-thiazol-4-yl)methyl]methanamine
—— methyl (1R,2S)-2-[[2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]acetyl]amino]cyclohexane-1-carboxylate —— C16H23F2N3O3
methyl (1R,2S)-2-[[2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]acetyl]amino]cyclohexane-1-carboxylate
—— methyl (1S,2S)-2-[[2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]acetyl]amino]cyclohexane-1-carboxylate —— C16H23F2N3O3
methyl (1S,2S)-2-[[2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]acetyl]amino]cyclohexane-1-carboxylate
—— methyl (1R,2R)-2-[[2-(1,2-oxazol-3-yl)acetyl]amino]cyclohexane-1-carboxylate —— C13H18N2O4
methyl (1R,2R)-2-[[2-(1,2-oxazol-3-yl)acetyl]amino]cyclohexane-1-carboxylate
—— 3-[3-(3,5-dimethylpyrazol-1-yl)phenyl]-1-[(3R,4R)-1-ethyl-3-methylpiperidin-4-yl]-1-methylurea —— C21H31N5O
3-[3-(3,5-dimethylpyrazol-1-yl)phenyl]-1-[(3R,4R)-1-ethyl-3-methylpiperidin-4-yl]-1-methylurea
—— methyl (1S,2R)-2-[[2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]acetyl]amino]cyclohexane-1-carboxylate —— C16H23F2N3O3
methyl (1S,2R)-2-[[2-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]acetyl]amino]cyclohexane-1-carboxylate
—— 1-ethyl-3-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-1-[[(2S)-oxolan-2-yl]methyl]urea —— C17H22N4O3
1-ethyl-3-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-1-[[(2S)-oxolan-2-yl]methyl]urea
—— N-[(3S)-1-ethylpiperidin-3-yl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide —— C18H25N5O2
N-[(3S)-1-ethylpiperidin-3-yl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide
—— N-[[(2S)-4-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]morpholin-2-yl]methyl]-N-ethylpyridazin-3-amine —— C17H25N5OS
N-[[(2S)-4-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]morpholin-2-yl]methyl]-N-ethylpyridazin-3-amine
—— 1-[(1S,6R)-3-ethyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)ethanone —— C19H25N3O2S
1-[(1S,6R)-3-ethyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)ethanone
—— N-ethyl-N-[4-[[(3R)-3-(5-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl]-1,3-thiazol-2-yl]acetamide —— C17H25N5OS
N-ethyl-N-[4-[[(3R)-3-(5-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl]-1,3-thiazol-2-yl]acetamide
—— 3-[3-(3,5-dimethylpyrazol-1-yl)phenyl]-1-[(3R,4S)-1-ethyl-3-methylpiperidin-4-yl]-1-methylurea —— C21H31N5O
3-[3-(3,5-dimethylpyrazol-1-yl)phenyl]-1-[(3R,4S)-1-ethyl-3-methylpiperidin-4-yl]-1-methylurea
—— 1-ethyl-3-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-1-[[(2R)-oxolan-2-yl]methyl]urea —— C17H22N4O3
1-ethyl-3-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-1-[[(2R)-oxolan-2-yl]methyl]urea
—— methyl (1S,2R)-2-[[2-(1,2-oxazol-3-yl)acetyl]amino]cyclohexane-1-carboxylate —— C13H18N2O4
methyl (1S,2R)-2-[[2-(1,2-oxazol-3-yl)acetyl]amino]cyclohexane-1-carboxylate
—— 1-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-3-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]urea —— C17H25N7O
1-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-3-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]urea
—— methyl (1R,2S)-2-[[2-(1,2-oxazol-3-yl)acetyl]amino]cyclohexane-1-carboxylate —— C13H18N2O4
methyl (1R,2S)-2-[[2-(1,2-oxazol-3-yl)acetyl]amino]cyclohexane-1-carboxylate
—— 3-[(1R)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-1,1-diethylurea —— C18H26N4O
3-[(1R)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-1,1-diethylurea
—— [(2S)-2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-(4-methyl-2-propyl-1,3-thiazol-5-yl)methanone —— C17H22N4O2S
[(2S)-2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-(4-methyl-2-propyl-1,3-thiazol-5-yl)methanone
—— (3S)-3-[[ethyl(methyl)amino]methyl]-N-[3-(5-methyl-1,3-oxazol-2-yl)phenyl]pyrrolidine-1-carboxamide —— C19H26N4O2
(3S)-3-[[ethyl(methyl)amino]methyl]-N-[3-(5-methyl-1,3-oxazol-2-yl)phenyl]pyrrolidine-1-carboxamide
—— [(2R)-5-(diethylamino)pent-3-yn-2-yl] 1-benzylpyrazole-4-carboxylate —— C20H25N3O2
[(2R)-5-(diethylamino)pent-3-yn-2-yl] 1-benzylpyrazole-4-carboxylate
—— [(2S)-5-(diethylamino)pent-3-yn-2-yl] 1-benzylpyrazole-4-carboxylate —— C20H25N3O2
[(2S)-5-(diethylamino)pent-3-yn-2-yl] 1-benzylpyrazole-4-carboxylate
—— N-ethyl-1-methyl-N-[(1R)-1-pyridin-4-ylethyl]pyrazole-4-carboxamide —— C14H18N4O
N-ethyl-1-methyl-N-[(1R)-1-pyridin-4-ylethyl]pyrazole-4-carboxamide
—— 3-[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-1,1-diethylurea —— C18H26N4O
3-[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-1,1-diethylurea
—— (3S)-3-[[ethyl(methyl)amino]methyl]-N-[(3-imidazol-1-ylphenyl)methyl]pyrrolidine-1-carboxamide —— C19H27N5O
(3S)-3-[[ethyl(methyl)amino]methyl]-N-[(3-imidazol-1-ylphenyl)methyl]pyrrolidine-1-carboxamide
—— 3-[[(2R)-oxolan-2-yl]methyl]-5-propyl-1,3,4-oxadiazol-2-one —— C10H16N2O3
3-[[(2R)-oxolan-2-yl]methyl]-5-propyl-1,3,4-oxadiazol-2-one
—— 1-[(2S,4S)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-(5-propyl-1,3,4-thiadiazol-2-yl)urea —— C14H20N4O3S
1-[(2S,4S)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-(5-propyl-1,3,4-thiadiazol-2-yl)urea
—— 1-[(2R,4R)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-(5-propyl-1,3,4-thiadiazol-2-yl)urea —— C14H20N4O3S
1-[(2R,4R)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-(5-propyl-1,3,4-thiadiazol-2-yl)urea
—— N-[2-(2-hydroxyethyl)-5-(4-propylphenyl)pyrazol-3-yl]acetamide —— C16H21N3O2
N-[2-(2-hydroxyethyl)-5-(4-propylphenyl)pyrazol-3-yl]acetamide
—— [(3R,4S)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-(2-propyl-1,3-thiazol-5-yl)methanone —— C17H27N3O2S
[(3R,4S)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-(2-propyl-1,3-thiazol-5-yl)methanone