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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-2-cycloheptyloxy-N-[(2-oxo-3H-1,3-thiazol-4-yl)methyl]propanamide —— C14H22N2O3S
(2R)-2-cycloheptyloxy-N-[(2-oxo-3H-1,3-thiazol-4-yl)methyl]propanamide
—— 2-(4-methyl-2-sulfanylidene-3H-1,3-thiazol-5-yl)-N-[(2-oxo-3H-1,3-thiazol-4-yl)methyl]acetamide —— C10H11N3O2S3
2-(4-methyl-2-sulfanylidene-3H-1,3-thiazol-5-yl)-N-[(2-oxo-3H-1,3-thiazol-4-yl)methyl]acetamide
—— (1S)-1-(2-ethyl-4-methyl-1,3-thiazol-5-yl)-N-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]ethanamine —— C13H20N4OS
(1S)-1-(2-ethyl-4-methyl-1,3-thiazol-5-yl)-N-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]ethanamine
—— (2S)-N-[(1R,2S)-2-(3-methylbutoxy)cyclohexyl]-2-(1,3,5-trimethylpyrazol-4-yl)propanamide —— C20H35N3O2
(2S)-N-[(1R,2S)-2-(3-methylbutoxy)cyclohexyl]-2-(1,3,5-trimethylpyrazol-4-yl)propanamide
—— (2R)-N-[(1R,2S)-2-(3-methylbutoxy)cyclohexyl]-2-(1,3,5-trimethylpyrazol-4-yl)propanamide —— C20H35N3O2
(2R)-N-[(1R,2S)-2-(3-methylbutoxy)cyclohexyl]-2-(1,3,5-trimethylpyrazol-4-yl)propanamide
—— (2R)-N-[(1S,2S)-2-(3-methylbutoxy)cyclohexyl]-2-(1,3,5-trimethylpyrazol-4-yl)propanamide —— C20H35N3O2
(2R)-N-[(1S,2S)-2-(3-methylbutoxy)cyclohexyl]-2-(1,3,5-trimethylpyrazol-4-yl)propanamide
—— benzyl N-[1-[[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]-2,5-dioxopyrrolidin-3-yl]carbamate —— C47H43N3O8S
benzyl N-[1-[[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]-2,5-dioxopyrrolidin-3-yl]carbamate
—— 2-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]isoindole-1,3-dione —— C35H31N5O6S
2-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]isoindole-1,3-dione
—— 4-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(1R)-1-(1-phenyltriazol-4-yl)ethyl]piperidine —— C18H23N7
4-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(1R)-1-(1-phenyltriazol-4-yl)ethyl]piperidine
—— 2-[(7R)-5,7-dihydro-4H-thieno[2,3-c]pyran-7-yl]-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)acetamide —— C20H21N3O3S
2-[(7R)-5,7-dihydro-4H-thieno[2,3-c]pyran-7-yl]-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)acetamide
—— (2S)-N-[(1S,2S)-2-(3-methylbutoxy)cyclohexyl]-2-(1,3,5-trimethylpyrazol-4-yl)propanamide —— C20H35N3O2
(2S)-N-[(1S,2S)-2-(3-methylbutoxy)cyclohexyl]-2-(1,3,5-trimethylpyrazol-4-yl)propanamide
—— 2-[(7S)-5,7-dihydro-4H-thieno[2,3-c]pyran-7-yl]-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)acetamide —— C20H21N3O3S
2-[(7S)-5,7-dihydro-4H-thieno[2,3-c]pyran-7-yl]-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)acetamide
—— 1-[[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]-3-ethylurea —— C38H39N3O5S
1-[[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]-3-ethylurea
—— 4-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(1S)-1-(1-phenyltriazol-4-yl)ethyl]piperidine —— C18H23N7
4-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(1S)-1-(1-phenyltriazol-4-yl)ethyl]piperidine
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C36H33N7O4S
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— 1-(1-adamantyl)-3-[[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]urea —— C46H49N3O5S
1-(1-adamantyl)-3-[[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]urea
—— 2-[3-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]isoindole-1,3-dione —— C34H29N5O5S
2-[3-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]isoindole-1,3-dione
—— methyl (2R,6R)-4-[(4-imidazol-1-ylphenyl)methyl]-6-methylmorpholine-2-carboxylate —— C17H21N3O3
methyl (2R,6R)-4-[(4-imidazol-1-ylphenyl)methyl]-6-methylmorpholine-2-carboxylate
—— N-[[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]pyridine-3-carboxamide —— C41H37N3O5S
N-[[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]pyridine-3-carboxamide
—— 2,2,2-trichloro-N-[3-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-5-methyl-1,3-dioxan-2-yl]phenyl]acetamide —— C28H26Cl3N5O5S
2,2,2-trichloro-N-[3-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-5-methyl-1,3-dioxan-2-yl]phenyl]acetamide
—— methyl (2S,6R)-4-[[1-(4-fluorophenyl)pyrazol-3-yl]methyl]-6-methylmorpholine-2-carboxylate —— C17H20FN3O3
methyl (2S,6R)-4-[[1-(4-fluorophenyl)pyrazol-3-yl]methyl]-6-methylmorpholine-2-carboxylate
—— methyl (2R,6R)-4-[[1-(4-fluorophenyl)pyrazol-3-yl]methyl]-6-methylmorpholine-2-carboxylate —— C17H20FN3O3
methyl (2R,6R)-4-[[1-(4-fluorophenyl)pyrazol-3-yl]methyl]-6-methylmorpholine-2-carboxylate
—— methyl (2S,6R)-4-[(4-imidazol-1-ylphenyl)methyl]-6-methylmorpholine-2-carboxylate —— C17H21N3O3
methyl (2S,6R)-4-[(4-imidazol-1-ylphenyl)methyl]-6-methylmorpholine-2-carboxylate
—— N-[3-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]acetamide —— C36H34N2O5S
N-[3-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]acetamide
—— 1-(1-adamantyl)-3-[3-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea —— C37H42N6O4S
1-(1-adamantyl)-3-[3-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea
—— benzyl N-[1-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]-2,5-dioxopyrrolidin-3-yl]carbamate —— C39H38N6O7S
benzyl N-[1-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]-2,5-dioxopyrrolidin-3-yl]carbamate
—— (2-methylsulfanyl-3-phenylimidazol-4-yl)-[(3S)-spiro[1,2-dihydroindene-3,2'-morpholine]-4'-yl]methanone —— C23H23N3O2S
(2-methylsulfanyl-3-phenylimidazol-4-yl)-[(3S)-spiro[1,2-dihydroindene-3,2'-morpholine]-4'-yl]methanone
—— (2-methylsulfanyl-3-phenylimidazol-4-yl)-[(3R)-spiro[1,2-dihydroindene-3,2'-morpholine]-4'-yl]methanone —— C23H23N3O2S
(2-methylsulfanyl-3-phenylimidazol-4-yl)-[(3R)-spiro[1,2-dihydroindene-3,2'-morpholine]-4'-yl]methanone
—— 3-[[(S)-methylsulfinyl]methyl]-N-[(2-phenyltriazol-4-yl)methyl]aniline —— C17H18N4OS
3-[[(S)-methylsulfinyl]methyl]-N-[(2-phenyltriazol-4-yl)methyl]aniline
—— (E,2R)-5-(6-chloropyridin-3-yl)-3-oxo-2-(4-propan-2-yl-1,3-thiazol-2-yl)pent-4-enenitrile —— C16H14ClN3OS
(E,2R)-5-(6-chloropyridin-3-yl)-3-oxo-2-(4-propan-2-yl-1,3-thiazol-2-yl)pent-4-enenitrile
—— [(1S)-1-cyclopropylprop-2-ynyl] 4-(3,5-dimethylpyrazol-1-yl)benzoate —— C18H18N2O2
[(1S)-1-cyclopropylprop-2-ynyl] 4-(3,5-dimethylpyrazol-1-yl)benzoate
—— (E,2R)-5-(6-chloropyridin-3-yl)-2-(4-methyl-1,3-thiazol-2-yl)-3-oxopent-4-enenitrile —— C14H10ClN3OS
(E,2R)-5-(6-chloropyridin-3-yl)-2-(4-methyl-1,3-thiazol-2-yl)-3-oxopent-4-enenitrile
—— (E,2S)-5-(6-chloropyridin-3-yl)-3-oxo-2-(4-propan-2-yl-1,3-thiazol-2-yl)pent-4-enenitrile —— C16H14ClN3OS
(E,2S)-5-(6-chloropyridin-3-yl)-3-oxo-2-(4-propan-2-yl-1,3-thiazol-2-yl)pent-4-enenitrile
—— [(1R)-1-cyclopropylprop-2-ynyl] 4-(3,5-dimethylpyrazol-1-yl)benzoate —— C18H18N2O2
[(1R)-1-cyclopropylprop-2-ynyl] 4-(3,5-dimethylpyrazol-1-yl)benzoate
—— 3-[[(R)-methylsulfinyl]methyl]-N-[(2-phenyltriazol-4-yl)methyl]aniline —— C17H18N4OS
3-[[(R)-methylsulfinyl]methyl]-N-[(2-phenyltriazol-4-yl)methyl]aniline
—— (E,2S)-5-(6-chloropyridin-3-yl)-2-(4-methyl-1,3-thiazol-2-yl)-3-oxopent-4-enenitrile —— C14H10ClN3OS
(E,2S)-5-(6-chloropyridin-3-yl)-2-(4-methyl-1,3-thiazol-2-yl)-3-oxopent-4-enenitrile
—— N-[(3R)-3-cyanothiolan-3-yl]-2-(2-methoxyphenyl)-1,3-thiazole-4-carboxamide —— C16H15N3O2S2
N-[(3R)-3-cyanothiolan-3-yl]-2-(2-methoxyphenyl)-1,3-thiazole-4-carboxamide
—— 3-(2-methoxyphenyl)-4-[(3S)-2-methylsulfonyl-5-phenyl-3,4-dihydropyrazol-3-yl]-1-phenylpyrazole —— C26H24N4O3S
3-(2-methoxyphenyl)-4-[(3S)-2-methylsulfonyl-5-phenyl-3,4-dihydropyrazol-3-yl]-1-phenylpyrazole
—— 5-tert-butyl-2-[(1R)-1-(5-methylpyrimidin-2-yl)sulfonylethyl]-1,3-oxazole —— C14H19N3O3S
5-tert-butyl-2-[(1R)-1-(5-methylpyrimidin-2-yl)sulfonylethyl]-1,3-oxazole
—— (3R)-2-methylsulfonyl-3-(4-nitrophenyl)-5-phenyl-3,4-dihydropyrazole —— C16H15N3O4S
(3R)-2-methylsulfonyl-3-(4-nitrophenyl)-5-phenyl-3,4-dihydropyrazole
—— 1-(1-ethyl-3,5-dimethylpyrazol-4-yl)-3-[(1S,3S)-3-(trifluoromethyl)cyclohexyl]urea —— C15H23F3N4O
1-(1-ethyl-3,5-dimethylpyrazol-4-yl)-3-[(1S,3S)-3-(trifluoromethyl)cyclohexyl]urea
—— 1-(1-ethyl-3,5-dimethylpyrazol-4-yl)-3-[(1R,3R)-3-(trifluoromethyl)cyclohexyl]urea —— C15H23F3N4O
1-(1-ethyl-3,5-dimethylpyrazol-4-yl)-3-[(1R,3R)-3-(trifluoromethyl)cyclohexyl]urea
—— 1-[(1S,2S)-2-cyclohexylcyclopropyl]-3-(1-ethyl-3,5-dimethylpyrazol-4-yl)urea —— C17H28N4O
1-[(1S,2S)-2-cyclohexylcyclopropyl]-3-(1-ethyl-3,5-dimethylpyrazol-4-yl)urea
—— 1-(3-imidazol-1-ylpropyl)-3-[(1S)-2-methylsulfonyl-1-phenylethyl]urea —— C16H22N4O3S
1-(3-imidazol-1-ylpropyl)-3-[(1S)-2-methylsulfonyl-1-phenylethyl]urea
—— 5-tert-butyl-2-[(1S)-1-(5-methylpyrimidin-2-yl)sulfonylethyl]-1,3-oxazole —— C14H19N3O3S
5-tert-butyl-2-[(1S)-1-(5-methylpyrimidin-2-yl)sulfonylethyl]-1,3-oxazole
—— (3S)-2-methylsulfonyl-3-(4-nitrophenyl)-5-phenyl-3,4-dihydropyrazole —— C16H15N3O4S
(3S)-2-methylsulfonyl-3-(4-nitrophenyl)-5-phenyl-3,4-dihydropyrazole
—— N-[(3S)-3-cyanothiolan-3-yl]-2-(2-methoxyphenyl)-1,3-thiazole-4-carboxamide —— C16H15N3O2S2
N-[(3S)-3-cyanothiolan-3-yl]-2-(2-methoxyphenyl)-1,3-thiazole-4-carboxamide
—— (2S)-2-(2-phenylimidazol-1-yl)-N-[(3-sulfamoylphenyl)methyl]propanamide —— C19H20N4O3S
(2S)-2-(2-phenylimidazol-1-yl)-N-[(3-sulfamoylphenyl)methyl]propanamide
—— (2R)-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]-N-prop-2-enylpropanamide —— C16H19N3OS
(2R)-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]-N-prop-2-enylpropanamide
—— 1-[(1R,2S)-2-cyclohexylcyclopropyl]-3-(1-ethyl-3,5-dimethylpyrazol-4-yl)urea —— C17H28N4O
1-[(1R,2S)-2-cyclohexylcyclopropyl]-3-(1-ethyl-3,5-dimethylpyrazol-4-yl)urea