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中文名称 英文名称 CAS号 化学式 结构式图片
—— [(1S)-2,2,2-trifluoro-1-(1,3,5-trimethylpyrazol-4-yl)ethyl] 2,5-dimethylpyrazole-3-carboxylate —— C14H17F3N4O2
[(1S)-2,2,2-trifluoro-1-(1,3,5-trimethylpyrazol-4-yl)ethyl] 2,5-dimethylpyrazole-3-carboxylate
—— (2S,3S)-2-methyl-N-[(2R)-1-(5-methyl-2-phenylpyrazol-3-yl)propan-2-yl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide —— C23H25N3O3
(2S,3S)-2-methyl-N-[(2R)-1-(5-methyl-2-phenylpyrazol-3-yl)propan-2-yl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide
—— N-[(1R)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]pyridine-2-sulfonamide —— C18H20N4O2S
N-[(1R)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]pyridine-2-sulfonamide
—— N-[(2S)-1-(1H-imidazol-5-yl)-3-phenylpropan-2-yl]-3-methyl-4-(1,2,4-triazol-1-yl)benzamide —— C22H22N6O
N-[(2S)-1-(1H-imidazol-5-yl)-3-phenylpropan-2-yl]-3-methyl-4-(1,2,4-triazol-1-yl)benzamide
—— 3-[(2R)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]-1-methyl-1-[(1S,3S)-3-methylsulfanylcyclopentyl]urea —— C17H30N4OS
3-[(2R)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]-1-methyl-1-[(1S,3S)-3-methylsulfanylcyclopentyl]urea
—— N-[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]pyridine-2-sulfonamide —— C18H20N4O2S
N-[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]pyridine-2-sulfonamide
—— (2E,4E)-N-[(1R)-1-(4-pyridin-4-yl-1,3-thiazol-2-yl)ethyl]hexa-2,4-dienamide —— C16H17N3OS
(2E,4E)-N-[(1R)-1-(4-pyridin-4-yl-1,3-thiazol-2-yl)ethyl]hexa-2,4-dienamide
—— (1S,2S)-N-[[2-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-2-(furan-2-yl)cyclopropane-1-carboxamide —— C20H21N3O2
(1S,2S)-N-[[2-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-2-(furan-2-yl)cyclopropane-1-carboxamide
—— (2S)-N-[[5-(3-cyanophenyl)-1H-imidazol-2-yl]methyl]-2-(3,5-dimethylpyrazol-1-yl)propanamide —— C19H20N6O
(2S)-N-[[5-(3-cyanophenyl)-1H-imidazol-2-yl]methyl]-2-(3,5-dimethylpyrazol-1-yl)propanamide
—— 1-[[2-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-3-[(3S)-2-oxopiperidin-3-yl]urea —— C18H23N5O2
1-[[2-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-3-[(3S)-2-oxopiperidin-3-yl]urea
—— 1-(2,5-dimethylpyrazol-3-yl)-3-[(2R)-2-hydroxy-4-methoxy-2-methylbutyl]urea —— C12H22N4O3
1-(2,5-dimethylpyrazol-3-yl)-3-[(2R)-2-hydroxy-4-methoxy-2-methylbutyl]urea
—— N-[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-2-(1,2-oxazol-3-yl)acetamide —— C18H20N4O2
N-[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-2-(1,2-oxazol-3-yl)acetamide
—— (2S)-2-(4-chloro-2-methylphenoxy)-N-(5-phenyl-1H-pyrazol-4-yl)propanamide —— C19H18ClN3O2
(2S)-2-(4-chloro-2-methylphenoxy)-N-(5-phenyl-1H-pyrazol-4-yl)propanamide
—— 3-[(2R)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]-1-methyl-1-[(1R,3S)-3-methylsulfanylcyclopentyl]urea —— C17H30N4OS
3-[(2R)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]-1-methyl-1-[(1R,3S)-3-methylsulfanylcyclopentyl]urea
—— methyl 2-[(2S)-4-[[4-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]morpholin-2-yl]acetate —— C19H25N3O3
methyl 2-[(2S)-4-[[4-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]morpholin-2-yl]acetate
—— (3S)-N-[[4-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-N-methyl-1,1-dioxothiolan-3-amine —— C17H23N3O2S
(3S)-N-[[4-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-N-methyl-1,1-dioxothiolan-3-amine
—— (2S,3S)-2-methyl-N-[(2S)-1-(5-methyl-2-phenylpyrazol-3-yl)propan-2-yl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide —— C23H25N3O3
(2S,3S)-2-methyl-N-[(2S)-1-(5-methyl-2-phenylpyrazol-3-yl)propan-2-yl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide
—— (2R)-N-[[5-(3-cyanophenyl)-1H-imidazol-2-yl]methyl]-2-(3,5-dimethylpyrazol-1-yl)propanamide —— C19H20N6O
(2R)-N-[[5-(3-cyanophenyl)-1H-imidazol-2-yl]methyl]-2-(3,5-dimethylpyrazol-1-yl)propanamide
—— (2R)-1-[3-(3,5-dimethylpyrazol-1-yl)azetidin-1-yl]-3-(thiophen-2-ylmethoxy)propan-2-ol —— C16H23N3O2S
(2R)-1-[3-(3,5-dimethylpyrazol-1-yl)azetidin-1-yl]-3-(thiophen-2-ylmethoxy)propan-2-ol
—— 6-(Benzylthio)-3-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazine —— C18H13FN4S
6-(Benzylthio)-3-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazine
—— 3-[(2S)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]-1-methyl-1-[(1R,3S)-3-methylsulfanylcyclopentyl]urea —— C17H30N4OS
3-[(2S)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]-1-methyl-1-[(1R,3S)-3-methylsulfanylcyclopentyl]urea
—— methyl 2-[(2R)-4-[[4-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]morpholin-2-yl]acetate —— C19H25N3O3
methyl 2-[(2R)-4-[[4-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]morpholin-2-yl]acetate
—— 1-[(1S)-1-cyclohexyl-3-hydroxypropyl]-3-(2,5-dimethylpyrazol-3-yl)urea —— C15H26N4O2
1-[(1S)-1-cyclohexyl-3-hydroxypropyl]-3-(2,5-dimethylpyrazol-3-yl)urea
—— 1-[(2R)-2,4-dimethylpiperazin-1-yl]-2-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethanone —— C19H26N4O
1-[(2R)-2,4-dimethylpiperazin-1-yl]-2-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethanone
—— 3-[(5-Ethylsulfanyl-4-phenyl-1,2,4-triazol-3-yl)methyl]-1,3-benzothiazol-2-one —— C18H16N4OS2
3-[(5-Ethylsulfanyl-4-phenyl-1,2,4-triazol-3-yl)methyl]-1,3-benzothiazol-2-one
—— 1-[2-[2-chloro-5-(trifluoromethyl)phenyl]-5-methylpyrazol-3-yl]-3-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea —— C17H17ClF3N7O
1-[2-[2-chloro-5-(trifluoromethyl)phenyl]-5-methylpyrazol-3-yl]-3-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea
—— 3-[(2S)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]-1-methyl-1-[(1S,3S)-3-methylsulfanylcyclopentyl]urea —— C17H30N4OS
3-[(2S)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]-1-methyl-1-[(1S,3S)-3-methylsulfanylcyclopentyl]urea
—— [(2R)-2-(5-methyl-1,3,4-oxadiazol-2-yl)pyrrolidin-1-yl]-[2-methyl-4-(1,2,4-triazol-1-yl)phenyl]methanone —— C17H18N6O2
[(2R)-2-(5-methyl-1,3,4-oxadiazol-2-yl)pyrrolidin-1-yl]-[2-methyl-4-(1,2,4-triazol-1-yl)phenyl]methanone
—— N-[(2R)-1-(1H-imidazol-5-yl)-3-phenylpropan-2-yl]-3-methyl-4-(1,2,4-triazol-1-yl)benzamide —— C22H22N6O
N-[(2R)-1-(1H-imidazol-5-yl)-3-phenylpropan-2-yl]-3-methyl-4-(1,2,4-triazol-1-yl)benzamide
—— (2S)-1-[3-(3,5-dimethylpyrazol-1-yl)azetidin-1-yl]-3-(thiophen-2-ylmethoxy)propan-2-ol —— C16H23N3O2S
(2S)-1-[3-(3,5-dimethylpyrazol-1-yl)azetidin-1-yl]-3-(thiophen-2-ylmethoxy)propan-2-ol
—— 5-(2,5-dimethylpyrazol-3-yl)-3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazole —— C11H14N4O2
5-(2,5-dimethylpyrazol-3-yl)-3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazole
—— (2S)-3-[[4-bromo-2-(3,5-dimethylphenyl)-5-methylpyrazol-3-yl]carbamoyl-methylamino]-N,2-dimethylpropanamide —— C19H26BrN5O2
(2S)-3-[[4-bromo-2-(3,5-dimethylphenyl)-5-methylpyrazol-3-yl]carbamoyl-methylamino]-N,2-dimethylpropanamide
—— [(1R)-2,2,2-trifluoro-1-(1,3,5-trimethylpyrazol-4-yl)ethyl] 2,5-dimethylpyrazole-3-carboxylate —— C14H17F3N4O2
[(1R)-2,2,2-trifluoro-1-(1,3,5-trimethylpyrazol-4-yl)ethyl] 2,5-dimethylpyrazole-3-carboxylate
—— Methyl 5-methyl-2-[2-methyl-1-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]-1,3-oxazole-4-carboxylate —— C15H24N2O5
Methyl 5-methyl-2-[2-methyl-1-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]-1,3-oxazole-4-carboxylate
—— 1,2-dimethyl-3-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]guanidine —— C14H19N5O
1,2-dimethyl-3-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]guanidine
—— 3-(2-Methyl-4-nitroimidazol-1-yl)-1-[4-(3-phenylprop-2-enyl)piperazin-1-yl]propan-1-one —— C20H25N5O3
3-(2-Methyl-4-nitroimidazol-1-yl)-1-[4-(3-phenylprop-2-enyl)piperazin-1-yl]propan-1-one
—— methyl 1-[(2S)-2-hydroxy-3-(4-methylpiperidin-1-yl)propyl]-4,5,6,7-tetrahydroindazole-3-carboxylate —— C18H29N3O3
methyl 1-[(2S)-2-hydroxy-3-(4-methylpiperidin-1-yl)propyl]-4,5,6,7-tetrahydroindazole-3-carboxylate
—— methyl 1-[(2R)-2-hydroxy-3-(4-methylpiperidin-1-yl)propyl]-4,5,6,7-tetrahydroindazole-3-carboxylate —— C18H29N3O3
methyl 1-[(2R)-2-hydroxy-3-(4-methylpiperidin-1-yl)propyl]-4,5,6,7-tetrahydroindazole-3-carboxylate
—— 1,2-dimethyl-3-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]guanidine —— C14H19N5O
1,2-dimethyl-3-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]guanidine
—— Methyl 5-[2-[4-methoxycarbonyl-2-[2-methyl-1-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]-1,3-oxazol-5-yl]ethyl]-2-[2-methyl-1-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]-1,3-oxazole-4-carboxylate —— C30H46N4O10
Methyl 5-[2-[4-methoxycarbonyl-2-[2-methyl-1-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]-1,3-oxazol-5-yl]ethyl]-2-[2-methyl-1-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]-1,3-oxazole-4-carboxylate
—— (2R)-2-(4-chloro-2-methylphenoxy)-N-(5-phenyl-1H-pyrazol-4-yl)propanamide —— C19H18ClN3O2
(2R)-2-(4-chloro-2-methylphenoxy)-N-(5-phenyl-1H-pyrazol-4-yl)propanamide
—— (2R)-3-[[4-bromo-2-(3,5-dimethylphenyl)-5-methylpyrazol-3-yl]carbamoyl-methylamino]-N,2-dimethylpropanamide —— C19H26BrN5O2
(2R)-3-[[4-bromo-2-(3,5-dimethylphenyl)-5-methylpyrazol-3-yl]carbamoyl-methylamino]-N,2-dimethylpropanamide
—— [(2S)-2-(5-methyl-1,3,4-oxadiazol-2-yl)pyrrolidin-1-yl]-[2-methyl-4-(1,2,4-triazol-1-yl)phenyl]methanone —— C17H18N6O2
[(2S)-2-(5-methyl-1,3,4-oxadiazol-2-yl)pyrrolidin-1-yl]-[2-methyl-4-(1,2,4-triazol-1-yl)phenyl]methanone
—— 5-(Cyclopropylmethyl)-1-(3,5-dimethylphenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C17H18N4O
5-(Cyclopropylmethyl)-1-(3,5-dimethylphenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— (1R)-N-[(1S)-1-(2,5-dimethylfuran-3-yl)ethyl]-1-[4-(1,2,4-triazol-1-yl)phenyl]ethanamine —— C18H22N4O
(1R)-N-[(1S)-1-(2,5-dimethylfuran-3-yl)ethyl]-1-[4-(1,2,4-triazol-1-yl)phenyl]ethanamine
—— (1S)-N-[(1S)-1-(2,5-dimethylfuran-3-yl)ethyl]-1-[4-(1,2,4-triazol-1-yl)phenyl]ethanamine —— C18H22N4O
(1S)-N-[(1S)-1-(2,5-dimethylfuran-3-yl)ethyl]-1-[4-(1,2,4-triazol-1-yl)phenyl]ethanamine
—— (1R)-N-[(1R)-1-(2,5-dimethylfuran-3-yl)ethyl]-1-[4-(1,2,4-triazol-1-yl)phenyl]ethanamine —— C18H22N4O
(1R)-N-[(1R)-1-(2,5-dimethylfuran-3-yl)ethyl]-1-[4-(1,2,4-triazol-1-yl)phenyl]ethanamine
—— (1S)-N-[(1R)-1-(2,5-dimethylfuran-3-yl)ethyl]-1-[4-(1,2,4-triazol-1-yl)phenyl]ethanamine —— C18H22N4O
(1S)-N-[(1R)-1-(2,5-dimethylfuran-3-yl)ethyl]-1-[4-(1,2,4-triazol-1-yl)phenyl]ethanamine
—— 1-[1-[(2R)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)oxyethanone —— C23H25N5O3
1-[1-[(2R)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)oxyethanone
—— N-[(2S)-2-(2,5-dimethylfuran-3-yl)-2-hydroxypropyl]-1-methylimidazole-4-sulfonamide —— C13H19N3O4S
N-[(2S)-2-(2,5-dimethylfuran-3-yl)-2-hydroxypropyl]-1-methylimidazole-4-sulfonamide