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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-N-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2,4-dimethylpiperazine-1-carboxamide —— C18H25N5O
(2S)-N-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2,4-dimethylpiperazine-1-carboxamide
—— 1-[(1R)-2,2-dimethylcyclohexyl]-3-[[1-(2-methoxyethyl)-3,5-dimethylpyrazol-4-yl]methyl]urea —— C18H32N4O2
1-[(1R)-2,2-dimethylcyclohexyl]-3-[[1-(2-methoxyethyl)-3,5-dimethylpyrazol-4-yl]methyl]urea
—— 3-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-5-thiophen-2-yl-1,2-oxazole —— C15H17N3O2S
3-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-5-thiophen-2-yl-1,2-oxazole
—— (4R)-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-N-methyl-2-oxoimidazolidine-4-carboxamide —— C17H21N5O2
(4R)-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-N-methyl-2-oxoimidazolidine-4-carboxamide
—— (2R)-N-[(2-methylpyrazol-3-yl)methyl]-2-(2-phenylimidazol-1-yl)propanamide —— C17H19N5O
(2R)-N-[(2-methylpyrazol-3-yl)methyl]-2-(2-phenylimidazol-1-yl)propanamide
—— 3-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-5-methyl-1,2-oxazole —— C12H17N3O2
3-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-5-methyl-1,2-oxazole
—— 3-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-5-propan-2-yl-1,2,4-oxadiazole —— C13H20N4O2
3-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-5-propan-2-yl-1,2,4-oxadiazole
—— [1-(4-bromophenyl)-3,5-dimethylpyrazol-4-yl]-[(3R)-3-[(1S)-1-hydroxyethyl]piperidin-1-yl]methanone —— C19H24BrN3O2
[1-(4-bromophenyl)-3,5-dimethylpyrazol-4-yl]-[(3R)-3-[(1S)-1-hydroxyethyl]piperidin-1-yl]methanone
—— (3S,8aS)-N-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine-2-carboxamide —— C20H27N5O
(3S,8aS)-N-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine-2-carboxamide
—— methyl (2R)-2-[3,5-dimethyl-1-[(1-phenyltetrazol-5-yl)methyl]pyrazol-4-yl]propanoate —— C17H20N6O2
methyl (2R)-2-[3,5-dimethyl-1-[(1-phenyltetrazol-5-yl)methyl]pyrazol-4-yl]propanoate
—— (7R)-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-7-carboxamide —— C20H23N5O
(7R)-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-7-carboxamide
—— 1-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-2-[(3S)-3-(hydroxymethyl)piperidin-1-yl]ethane-1,2-dione —— C20H22F3N3O3
1-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-2-[(3S)-3-(hydroxymethyl)piperidin-1-yl]ethane-1,2-dione
—— 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]-2-oxo-N-prop-2-ynylacetamide —— C20H21N3O4S
2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]-2-oxo-N-prop-2-ynylacetamide
—— 1-benzyl-2-[(1S)-1-ethoxyethyl]imidazole —— C14H18N2O
1-benzyl-2-[(1S)-1-ethoxyethyl]imidazole
—— N-[[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]ethanamine —— C21H30F2N4
N-[[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]ethanamine
—— 2-methyl-5-[[(4R)-4-methyl-4,5-dihydro-1,3-thiazol-2-yl]sulfanylmethyl]-1,3,4-oxadiazole —— C8H11N3OS2
2-methyl-5-[[(4R)-4-methyl-4,5-dihydro-1,3-thiazol-2-yl]sulfanylmethyl]-1,3,4-oxadiazole
—— 2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-1-hydroxypropan-2-yl]acetamide —— C16H19Cl2N3O2
2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-1-hydroxypropan-2-yl]acetamide
—— (3R)-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide —— C18H22N4O2
(3R)-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
—— (2R)-2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl-methylamino]propanoic acid —— C16H21N3O2
(2R)-2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl-methylamino]propanoic acid
—— N-[[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]ethanamine —— C21H30F2N4
N-[[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]ethanamine
—— 2-methyl-5-[[(4S)-4-methyl-4,5-dihydro-1,3-thiazol-2-yl]sulfanylmethyl]-1,3,4-oxadiazole —— C8H11N3OS2
2-methyl-5-[[(4S)-4-methyl-4,5-dihydro-1,3-thiazol-2-yl]sulfanylmethyl]-1,3,4-oxadiazole
—— 4-[[2-[(1S)-1-ethoxyethyl]imidazol-1-yl]methyl]-2-propan-2-yl-1,3-thiazole —— C14H21N3OS
4-[[2-[(1S)-1-ethoxyethyl]imidazol-1-yl]methyl]-2-propan-2-yl-1,3-thiazole
—— (5-chloro-1,3-dimethylpyrazol-4-yl)-[(2R)-2,4-dimethylpiperazin-1-yl]methanone —— C12H19ClN4O
(5-chloro-1,3-dimethylpyrazol-4-yl)-[(2R)-2,4-dimethylpiperazin-1-yl]methanone
—— 4-[[2-[(1S)-1-ethoxyethyl]imidazol-1-yl]methyl]-3,5-dimethyl-1,2-oxazole —— C13H19N3O2
4-[[2-[(1S)-1-ethoxyethyl]imidazol-1-yl]methyl]-3,5-dimethyl-1,2-oxazole
—— (1R)-N-[2-(1,1-dioxo-1,2-thiazolidin-2-yl)ethyl]-1-[4-(2-methylimidazol-1-yl)phenyl]ethanamine —— C17H24N4O2S
(1R)-N-[2-(1,1-dioxo-1,2-thiazolidin-2-yl)ethyl]-1-[4-(2-methylimidazol-1-yl)phenyl]ethanamine
—— 5-chloro-1,3-dimethyl-N-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]pyrazole-4-carboxamide —— C17H18ClN5O2
5-chloro-1,3-dimethyl-N-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]pyrazole-4-carboxamide
—— 4-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-5-methyl-2-phenyl-1,3-oxazole —— C18H21N3O2
4-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-5-methyl-2-phenyl-1,3-oxazole
—— (4S)-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-N-methyl-2-oxoimidazolidine-4-carboxamide —— C17H21N5O2
(4S)-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-N-methyl-2-oxoimidazolidine-4-carboxamide
—— 3-[[2-[(1S)-1-ethoxyethyl]imidazol-1-yl]methyl]-5-ethyl-1,2,4-oxadiazole —— C12H18N4O2
3-[[2-[(1S)-1-ethoxyethyl]imidazol-1-yl]methyl]-5-ethyl-1,2,4-oxadiazole
—— 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]-2-oxo-N-prop-2-ynylacetamide —— C20H21N3O4S
2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]-2-oxo-N-prop-2-ynylacetamide
—— (1R)-N-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[4-(tetrazol-1-yl)phenyl]ethanamine —— C14H17N7O
(1R)-N-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[4-(tetrazol-1-yl)phenyl]ethanamine
—— methyl (2S)-2-[3,5-dimethyl-1-[(1-phenyltetrazol-5-yl)methyl]pyrazol-4-yl]propanoate —— C17H20N6O2
methyl (2S)-2-[3,5-dimethyl-1-[(1-phenyltetrazol-5-yl)methyl]pyrazol-4-yl]propanoate
—— 1-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-2-[(3R)-3-(hydroxymethyl)piperidin-1-yl]ethane-1,2-dione —— C20H22F3N3O3
1-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-2-[(3R)-3-(hydroxymethyl)piperidin-1-yl]ethane-1,2-dione
—— 2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-1-hydroxypropan-2-yl]acetamide —— C16H19Cl2N3O2
2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-1-hydroxypropan-2-yl]acetamide
—— 1-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3-[[(2S)-2-methylthiolan-2-yl]methyl]urea —— C18H24N4OS
1-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3-[[(2S)-2-methylthiolan-2-yl]methyl]urea
—— 4-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-3,5-dimethyl-1,2-oxazole —— C13H19N3O2
4-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-3,5-dimethyl-1,2-oxazole
—— (1R)-1-(2-ethyl-4-methyl-1,3-thiazol-5-yl)-N-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]ethanamine —— C13H20N4OS
(1R)-1-(2-ethyl-4-methyl-1,3-thiazol-5-yl)-N-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]ethanamine
—— (1R)-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-1-(2-methyl-1,3-thiazol-5-yl)ethanamine —— C16H19ClN2O2S
(1R)-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-1-(2-methyl-1,3-thiazol-5-yl)ethanamine
—— (2S)-N-[(2-methylpyrazol-3-yl)methyl]-2-(2-phenylimidazol-1-yl)propanamide —— C17H19N5O
(2S)-N-[(2-methylpyrazol-3-yl)methyl]-2-(2-phenylimidazol-1-yl)propanamide
—— (1S)-N-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[4-(tetrazol-1-yl)phenyl]ethanamine —— C14H17N7O
(1S)-N-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[4-(tetrazol-1-yl)phenyl]ethanamine
—— (5-chloro-1,3-dimethylpyrazol-4-yl)-[(2S)-2,4-dimethylpiperazin-1-yl]methanone —— C12H19ClN4O
(5-chloro-1,3-dimethylpyrazol-4-yl)-[(2S)-2,4-dimethylpiperazin-1-yl]methanone
—— (2S)-2-(2-cyanophenoxy)-N-[(4-phenyl-1,2,4-triazol-3-yl)methyl]propanamide —— C19H17N5O2
(2S)-2-(2-cyanophenoxy)-N-[(4-phenyl-1,2,4-triazol-3-yl)methyl]propanamide
—— 5-chloro-1,3-dimethyl-N-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]pyrazole-4-carboxamide —— C17H18ClN5O2
5-chloro-1,3-dimethyl-N-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]pyrazole-4-carboxamide
—— 4-hydroxy-N,3-dimethyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1H-pyrazole-5-carboxamide —— C16H18N6O2
4-hydroxy-N,3-dimethyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1H-pyrazole-5-carboxamide
—— 2,2,2-trifluoro-N'-[(1R)-1-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)ethoxy]ethanimidamide —— C10H9F3N4O2S
2,2,2-trifluoro-N'-[(1R)-1-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)ethoxy]ethanimidamide
—— 4-hydroxy-N,3-dimethyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1H-pyrazole-5-carboxamide —— C16H18N6O2
4-hydroxy-N,3-dimethyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1H-pyrazole-5-carboxamide
—— [1-(4-bromophenyl)-3,5-dimethylpyrazol-4-yl]-[(3S)-3-[(1S)-1-hydroxyethyl]piperidin-1-yl]methanone —— C19H24BrN3O2
[1-(4-bromophenyl)-3,5-dimethylpyrazol-4-yl]-[(3S)-3-[(1S)-1-hydroxyethyl]piperidin-1-yl]methanone
—— 5-(2-fluorophenyl)-N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1H-pyrazole-4-carboxamide —— C19H16FN3O2
5-(2-fluorophenyl)-N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1H-pyrazole-4-carboxamide
—— (1S)-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-1-(2-methyl-1,3-thiazol-5-yl)ethanamine —— C16H19ClN2O2S
(1S)-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-1-(2-methyl-1,3-thiazol-5-yl)ethanamine
—— 2,2,2-trifluoro-N'-[(1S)-1-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)ethoxy]ethanimidamide —— C10H9F3N4O2S
2,2,2-trifluoro-N'-[(1S)-1-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)ethoxy]ethanimidamide