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中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S)-3-(hydroxymethyl)-N-[(1S)-1-(3-pyrazol-1-ylphenyl)ethyl]piperidine-1-carboxamide —— C18H24N4O2
(3S)-3-(hydroxymethyl)-N-[(1S)-1-(3-pyrazol-1-ylphenyl)ethyl]piperidine-1-carboxamide
—— (1S)-N-(2-phenylethyl)-1-(2-pyrazol-1-ylphenyl)ethanamine —— C19H21N3
(1S)-N-(2-phenylethyl)-1-(2-pyrazol-1-ylphenyl)ethanamine
—— N-methyl-3-phenyl-N-[(1R)-1-phenylethyl]-1,2-thiazole-5-carboxamide —— C19H18N2OS
N-methyl-3-phenyl-N-[(1R)-1-phenylethyl]-1,2-thiazole-5-carboxamide
—— N-methyl-3-phenyl-N-[(1S)-1-phenylethyl]-1,2-thiazole-5-carboxamide —— C19H18N2OS
N-methyl-3-phenyl-N-[(1S)-1-phenylethyl]-1,2-thiazole-5-carboxamide
—— (2S,3R)-3-phenyl-2-[(2-pyridin-2-yl-1,3-thiazol-5-yl)methylamino]butan-1-ol —— C19H21N3OS
(2S,3R)-3-phenyl-2-[(2-pyridin-2-yl-1,3-thiazol-5-yl)methylamino]butan-1-ol
—— N-[(1S)-1-(furan-2-yl)ethyl]-2-(5-oxo-3-phenyl-1,2,4-oxadiazol-4-yl)acetamide —— C16H15N3O4
N-[(1S)-1-(furan-2-yl)ethyl]-2-(5-oxo-3-phenyl-1,2,4-oxadiazol-4-yl)acetamide
—— 1-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-3-[(1R)-1-phenylethyl]thiourea —— C15H16N4S2
1-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-3-[(1R)-1-phenylethyl]thiourea
—— (3-tert-butyl-1-phenylpyrazol-4-yl)-[4-[(1S)-1-pyridin-3-ylethyl]piperazin-1-yl]methanone —— C25H31N5O
(3-tert-butyl-1-phenylpyrazol-4-yl)-[4-[(1S)-1-pyridin-3-ylethyl]piperazin-1-yl]methanone
—— (1S)-1-(2-chlorophenyl)-N-[[2-(1-methylpyrazol-4-yl)-1,3-thiazol-4-yl]methyl]ethanamine —— C16H17ClN4S
(1S)-1-(2-chlorophenyl)-N-[[2-(1-methylpyrazol-4-yl)-1,3-thiazol-4-yl]methyl]ethanamine
—— (3S)-3-(hydroxymethyl)-N-[(1R)-1-(3-pyrazol-1-ylphenyl)ethyl]piperidine-1-carboxamide —— C18H24N4O2
(3S)-3-(hydroxymethyl)-N-[(1R)-1-(3-pyrazol-1-ylphenyl)ethyl]piperidine-1-carboxamide
—— 4-[5-[(1R)-1-naphthalen-1-ylethyl]sulfanyltetrazol-1-yl]phenol —— C19H16N4OS
4-[5-[(1R)-1-naphthalen-1-ylethyl]sulfanyltetrazol-1-yl]phenol
—— 5-[[(R)-[(1R)-1-(2-fluorophenyl)ethyl]sulfinyl]methyl]-1-phenyltetrazole —— C16H15FN4OS
5-[[(R)-[(1R)-1-(2-fluorophenyl)ethyl]sulfinyl]methyl]-1-phenyltetrazole
—— 3-(2-fluorophenyl)-4-methyl-5-[(1R)-1-phenylethyl]sulfonyl-1,2,4-triazole —— C17H16FN3O2S
3-(2-fluorophenyl)-4-methyl-5-[(1R)-1-phenylethyl]sulfonyl-1,2,4-triazole
—— (3Z)-3-[[2-(2-amino-1,3-thiazol-4-yl)acetyl]hydrazinylidene]-N-cyclohexylbutanamide —— C15H23N5O2S
(3Z)-3-[[2-(2-amino-1,3-thiazol-4-yl)acetyl]hydrazinylidene]-N-cyclohexylbutanamide
—— (1R)-N-(2-phenylethyl)-1-(2-pyrazol-1-ylphenyl)ethanamine —— C19H21N3
(1R)-N-(2-phenylethyl)-1-(2-pyrazol-1-ylphenyl)ethanamine
—— (1R,4S)-N-[(1S)-1-(3-pyrazol-1-ylphenyl)ethyl]-2-azabicyclo[2.2.1]heptane-2-carboxamide —— C18H22N4O
(1R,4S)-N-[(1S)-1-(3-pyrazol-1-ylphenyl)ethyl]-2-azabicyclo[2.2.1]heptane-2-carboxamide
—— 3-(4-fluorophenyl)-5-[(3S)-1-[(1R)-1-(3-fluorophenyl)ethyl]piperidin-3-yl]-1,2,4-oxadiazole —— C21H21F2N3O
3-(4-fluorophenyl)-5-[(3S)-1-[(1R)-1-(3-fluorophenyl)ethyl]piperidin-3-yl]-1,2,4-oxadiazole
—— 1-[4-[[(R)-[(1R)-1-(2-fluorophenyl)ethyl]sulfinyl]methyl]phenyl]pyrazole —— C18H17FN2OS
1-[4-[[(R)-[(1R)-1-(2-fluorophenyl)ethyl]sulfinyl]methyl]phenyl]pyrazole
—— (1R)-1-(2-chlorophenyl)-N-[[2-(1-methylpyrazol-4-yl)-1,3-thiazol-4-yl]methyl]ethanamine —— C16H17ClN4S
(1R)-1-(2-chlorophenyl)-N-[[2-(1-methylpyrazol-4-yl)-1,3-thiazol-4-yl]methyl]ethanamine
—— (2E)-2-[[4-(dimethylamino)phenyl]methylidene]-6-(4-nitrophenyl)imidazo[2,1-b][1,3]thiazol-3-one —— C20H16N4O3S
(2E)-2-[[4-(dimethylamino)phenyl]methylidene]-6-(4-nitrophenyl)imidazo[2,1-b][1,3]thiazol-3-one
—— 2-[(2Z,5E)-2-(3,3-dimethyl-2-oxobutylidene)-4-oxo-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-3-yl]-N-pentan-2-ylacetamide —— C21H28N2O3S2
2-[(2Z,5E)-2-(3,3-dimethyl-2-oxobutylidene)-4-oxo-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-3-yl]-N-pentan-2-ylacetamide
—— [(2R)-1-[[(1S)-1-(2,4-dichlorophenyl)ethyl]amino]-1-oxopropan-2-yl] 2-(methylamino)-1,3-thiazole-5-carboxylate —— C16H17Cl2N3O3S
[(2R)-1-[[(1S)-1-(2,4-dichlorophenyl)ethyl]amino]-1-oxopropan-2-yl] 2-(methylamino)-1,3-thiazole-5-carboxylate
—— (1R,4S)-N-[(1R)-1-(3-pyrazol-1-ylphenyl)ethyl]-2-azabicyclo[2.2.1]heptane-2-carboxamide —— C18H22N4O
(1R,4S)-N-[(1R)-1-(3-pyrazol-1-ylphenyl)ethyl]-2-azabicyclo[2.2.1]heptane-2-carboxamide
—— 5-cyclopropyl-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]-1-phenyltriazole-4-carboxamide —— C22H24N4O3
5-cyclopropyl-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]-1-phenyltriazole-4-carboxamide
—— (3R)-3-(hydroxymethyl)-N-[(1S)-1-(3-pyrazol-1-ylphenyl)ethyl]piperidine-1-carboxamide —— C18H24N4O2
(3R)-3-(hydroxymethyl)-N-[(1S)-1-(3-pyrazol-1-ylphenyl)ethyl]piperidine-1-carboxamide
—— 3-(4-fluorophenyl)-5-[(3S)-1-[(1S)-1-(3-fluorophenyl)ethyl]piperidin-3-yl]-1,2,4-oxadiazole —— C21H21F2N3O
3-(4-fluorophenyl)-5-[(3S)-1-[(1S)-1-(3-fluorophenyl)ethyl]piperidin-3-yl]-1,2,4-oxadiazole
—— [(2R)-1-[[(1R)-1-(2,4-dichlorophenyl)ethyl]amino]-1-oxopropan-2-yl] 2-(methylamino)-1,3-thiazole-5-carboxylate —— C16H17Cl2N3O3S
[(2R)-1-[[(1R)-1-(2,4-dichlorophenyl)ethyl]amino]-1-oxopropan-2-yl] 2-(methylamino)-1,3-thiazole-5-carboxylate
—— 6-nitro-N-[(1S)-1-(4-pyrazol-1-ylphenyl)ethyl]pyridin-3-amine —— C16H15N5O2
6-nitro-N-[(1S)-1-(4-pyrazol-1-ylphenyl)ethyl]pyridin-3-amine
—— N-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-2-(2-phenyltriazol-4-yl)acetamide —— C21H22N4O3
N-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-2-(2-phenyltriazol-4-yl)acetamide
—— [(2S)-1-[[(1S)-1-(2,4-dichlorophenyl)ethyl]amino]-1-oxopropan-2-yl] 2-(methylamino)-1,3-thiazole-5-carboxylate —— C16H17Cl2N3O3S
[(2S)-1-[[(1S)-1-(2,4-dichlorophenyl)ethyl]amino]-1-oxopropan-2-yl] 2-(methylamino)-1,3-thiazole-5-carboxylate
—— [(1S)-1-(6-bromo-1H-imidazo[4,5-b]pyridin-2-yl)ethyl] 1-(2-chlorophenyl)pyrazole-4-carboxylate —— C18H13BrClN5O2
[(1S)-1-(6-bromo-1H-imidazo[4,5-b]pyridin-2-yl)ethyl] 1-(2-chlorophenyl)pyrazole-4-carboxylate
—— (1R)-1-phenyl-1-pyridin-2-yl-N-[(2-pyridin-2-yl-1,3-thiazol-5-yl)methyl]methanamine —— C21H18N4S
(1R)-1-phenyl-1-pyridin-2-yl-N-[(2-pyridin-2-yl-1,3-thiazol-5-yl)methyl]methanamine
—— 1-phenyl-2-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]sulfonylimidazole —— C18H15F3N2O3S
1-phenyl-2-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]sulfonylimidazole
—— 5-cyclopropyl-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]-1-phenyltriazole-4-carboxamide —— C22H24N4O3
5-cyclopropyl-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]-1-phenyltriazole-4-carboxamide
—— N-[(Z)-1-(furan-2-yl)ethylideneamino]-2-(2-methyl-1,3-thiazol-4-yl)acetamide —— C12H13N3O2S
N-[(Z)-1-(furan-2-yl)ethylideneamino]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
—— (1S)-1-phenyl-1-pyridin-2-yl-N-[(2-pyridin-2-yl-1,3-thiazol-5-yl)methyl]methanamine —— C21H18N4S
(1S)-1-phenyl-1-pyridin-2-yl-N-[(2-pyridin-2-yl-1,3-thiazol-5-yl)methyl]methanamine
—— 1-phenyl-2-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]sulfonylimidazole —— C18H15F3N2O3S
1-phenyl-2-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]sulfonylimidazole
—— 2-[[4-(4-methylphenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-1-thiophen-2-ylethylideneamino]acetamide —— C23H21N5OS2
2-[[4-(4-methylphenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-1-thiophen-2-ylethylideneamino]acetamide
—— [(1S)-1-(2-fluoro-6-pyrazol-1-ylphenyl)ethyl] 3-(2-oxopyrrolidin-1-yl)propanoate —— C18H20FN3O3
[(1S)-1-(2-fluoro-6-pyrazol-1-ylphenyl)ethyl] 3-(2-oxopyrrolidin-1-yl)propanoate
—— (5E)-5-[[3-[4-[(4-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-3-[(4-methylphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C34H26ClN3O2S2
(5E)-5-[[3-[4-[(4-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-3-[(4-methylphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— [(2S)-1-[[(1R)-1-(2,4-dichlorophenyl)ethyl]amino]-1-oxopropan-2-yl] 2-(methylamino)-1,3-thiazole-5-carboxylate —— C16H17Cl2N3O3S
[(2S)-1-[[(1R)-1-(2,4-dichlorophenyl)ethyl]amino]-1-oxopropan-2-yl] 2-(methylamino)-1,3-thiazole-5-carboxylate
—— (5E)-3-ethyl-5-{[3-(4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methylene}-2-thioxo-1,3-thiazolidin-4-one —— C22H19N3O2S2
(5E)-3-ethyl-5-{[3-(4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methylene}-2-thioxo-1,3-thiazolidin-4-one
—— [(1R)-1-(6-bromo-1H-imidazo[4,5-b]pyridin-2-yl)ethyl] 1-(2-chlorophenyl)pyrazole-4-carboxylate —— C18H13BrClN5O2
[(1R)-1-(6-bromo-1H-imidazo[4,5-b]pyridin-2-yl)ethyl] 1-(2-chlorophenyl)pyrazole-4-carboxylate
—— 2-[[4-cyclohexyl-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-(2,4,6-trimethoxyphenyl)methylideneamino]acetamide —— C27H33N5O4S
2-[[4-cyclohexyl-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-(2,4,6-trimethoxyphenyl)methylideneamino]acetamide
—— 6-nitro-N-[(1R)-1-(4-pyrazol-1-ylphenyl)ethyl]pyridin-3-amine —— C16H15N5O2
6-nitro-N-[(1R)-1-(4-pyrazol-1-ylphenyl)ethyl]pyridin-3-amine
—— (4Z)-2-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-5-methyl-4-(1,3-thiazol-2-ylhydrazinylidene)pyrazol-3-one —— C16H11BrN6OS2
(4Z)-2-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-5-methyl-4-(1,3-thiazol-2-ylhydrazinylidene)pyrazol-3-one
—— 4-[4-[(E)-(3-butyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1-phenylpyrazol-3-yl]-N,N-dimethylbenzenesulfonamide —— C25H26N4O3S3
4-[4-[(E)-(3-butyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1-phenylpyrazol-3-yl]-N,N-dimethylbenzenesulfonamide
—— [(1R)-1-(2-fluoro-6-pyrazol-1-ylphenyl)ethyl] 3-(2-oxopyrrolidin-1-yl)propanoate —— C18H20FN3O3
[(1R)-1-(2-fluoro-6-pyrazol-1-ylphenyl)ethyl] 3-(2-oxopyrrolidin-1-yl)propanoate
—— ethyl (2Z)-2-cyano-2-[(5Z)-5-[(2-methyl-6-phenylimidazo[2,1-b][1,3,4]thiadiazol-5-yl)methylidene]-4-oxo-3-phenyl-1,3-thiazolidin-2-ylidene]acetate —— C26H19N5O3S2
ethyl (2Z)-2-cyano-2-[(5Z)-5-[(2-methyl-6-phenylimidazo[2,1-b][1,3,4]thiadiazol-5-yl)methylidene]-4-oxo-3-phenyl-1,3-thiazolidin-2-ylidene]acetate
—— ethyl 4-(5-{(Z)-[2-(4-ethoxyphenyl)-6-oxo[1,3]thiazolo[3,2-b][1,2,4]triazol-5(6H)-ylidene]methyl}furan-2-yl)benzoate —— C26H21N3O5S
ethyl 4-(5-{(Z)-[2-(4-ethoxyphenyl)-6-oxo[1,3]thiazolo[3,2-b][1,2,4]triazol-5(6H)-ylidene]methyl}furan-2-yl)benzoate