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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4S)-6-amino-4-(3-methoxy-4-propoxyphenyl)-3-methyl-1-(4-methylphenyl)-4H-pyrano[2,3-c]pyrazole-5-carbonitrile —— C25H26N4O3
(4S)-6-amino-4-(3-methoxy-4-propoxyphenyl)-3-methyl-1-(4-methylphenyl)-4H-pyrano[2,3-c]pyrazole-5-carbonitrile
—— N-[(4S)-2,2-dimethyloxan-4-yl]-3-(5-phenyl-1,3-oxazol-2-yl)propanamide —— C19H24N2O3
N-[(4S)-2,2-dimethyloxan-4-yl]-3-(5-phenyl-1,3-oxazol-2-yl)propanamide
—— N-[(4R)-2,2-dimethyloxan-4-yl]-3-(5-phenyl-1,3-oxazol-2-yl)propanamide —— C19H24N2O3
N-[(4R)-2,2-dimethyloxan-4-yl]-3-(5-phenyl-1,3-oxazol-2-yl)propanamide
—— 2-bromo-N-[(4R)-2,2-dimethyloxan-4-yl]-5-propan-2-yl-1,3-thiazole-4-carboxamide —— C14H21BrN2O2S
2-bromo-N-[(4R)-2,2-dimethyloxan-4-yl]-5-propan-2-yl-1,3-thiazole-4-carboxamide
—— [(2R)-1-[[(2R)-1-[(5-methyl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]methyl]pyrrolidin-2-yl]methanol —— C15H25N3O2
[(2R)-1-[[(2R)-1-[(5-methyl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]methyl]pyrrolidin-2-yl]methanol
—— (3S,5S,8S)-3,8-dimethyl-3-[2-(prop-2-enylamino)-1,3-thiazol-4-yl]-2,7-dioxaspiro[4.4]nonane-1,6-dione —— C15H18N2O4S
(3S,5S,8S)-3,8-dimethyl-3-[2-(prop-2-enylamino)-1,3-thiazol-4-yl]-2,7-dioxaspiro[4.4]nonane-1,6-dione
—— [(2R)-1-[[(2S)-1-[(5-methyl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]methyl]pyrrolidin-2-yl]methanol —— C15H25N3O2
[(2R)-1-[[(2S)-1-[(5-methyl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]methyl]pyrrolidin-2-yl]methanol
—— 2-ethyl-1-[(4S)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one —— C22H29N3O3
2-ethyl-1-[(4S)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one
—— (1S,2R,5R)-2-[4-ethyl-3-[(5-phenyltetrazol-2-yl)methyl]-5-sulfanylidene-1,2,4-triazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one —— C18H19N7O3S
(1S,2R,5R)-2-[4-ethyl-3-[(5-phenyltetrazol-2-yl)methyl]-5-sulfanylidene-1,2,4-triazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one
—— (3R)-1-[1-(2,4-dimethylphenyl)pyrazolo[3,4-d]pyrimidin-4-yl]-N,N-diethylpiperidine-3-carboxamide —— C23H30N6O
(3R)-1-[1-(2,4-dimethylphenyl)pyrazolo[3,4-d]pyrimidin-4-yl]-N,N-diethylpiperidine-3-carboxamide
—— 2-(1H-indol-3-yl)-1-[(2R)-2-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethanone —— C23H22N4O3
2-(1H-indol-3-yl)-1-[(2R)-2-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethanone
—— (2R,8R)-1,6,7,12-tetrazatricyclo[7.3.0.03,7]dodeca-3,5,9,11-tetraene-2,8-diol —— C8H8N4O2
(2R,8R)-1,6,7,12-tetrazatricyclo[7.3.0.03,7]dodeca-3,5,9,11-tetraene-2,8-diol
—— 2-(1H-indol-3-yl)-1-[(2S)-2-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethanone —— C23H22N4O3
2-(1H-indol-3-yl)-1-[(2S)-2-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethanone
—— 2-ethyl-1-[(4R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one —— C22H29N3O3
2-ethyl-1-[(4R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-8-oxa-2-azaspiro[4.5]decan-2-yl]butan-1-one
—— 1-(2-methoxy-5-methylphenyl)-N-(4-methyl-3-oxopyrazin-2-yl)pyrazole-3-carboxamide —— C17H17N5O3
1-(2-methoxy-5-methylphenyl)-N-(4-methyl-3-oxopyrazin-2-yl)pyrazole-3-carboxamide
—— (2R,4R)-1-[2-ethoxy-5-(tetrazol-1-yl)phenyl]sulfonyl-2,4-dimethylpiperidine —— C16H23N5O3S
(2R,4R)-1-[2-ethoxy-5-(tetrazol-1-yl)phenyl]sulfonyl-2,4-dimethylpiperidine
—— N-[(1R,2R)-2-methylcyclohexyl]-2-[5-[2-(tetrazol-1-yl)phenyl]tetrazol-2-yl]acetamide —— C17H21N9O
N-[(1R,2R)-2-methylcyclohexyl]-2-[5-[2-(tetrazol-1-yl)phenyl]tetrazol-2-yl]acetamide
—— 2-[2-[4-(4-Hydroxybenzoyl)piperazin-1-yl]ethyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C19H21N5O3
2-[2-[4-(4-Hydroxybenzoyl)piperazin-1-yl]ethyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— 2-(2,4-dimethylphenyl)-N-(4-methyl-3-oxopyrazin-2-yl)-1,3-thiazole-4-carboxamide —— C17H16N4O2S
2-(2,4-dimethylphenyl)-N-(4-methyl-3-oxopyrazin-2-yl)-1,3-thiazole-4-carboxamide
—— 4-amino-3-[(2S)-oxolan-2-yl]-1H-1,2,4-triazole-5-thione —— C6H10N4OS
4-amino-3-[(2S)-oxolan-2-yl]-1H-1,2,4-triazole-5-thione
—— 8-[[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2S)-oxolan-2-yl]methyl]-1H-purin-6-one —— C22H23N5O3S
8-[[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2S)-oxolan-2-yl]methyl]-1H-purin-6-one
—— 8-[[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2S)-oxolan-2-yl]methyl]-1H-purin-6-one —— C21H20ClN5O3S
8-[[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2S)-oxolan-2-yl]methyl]-1H-purin-6-one
—— 8-[[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2R)-oxolan-2-yl]methyl]-1H-purin-6-one —— C22H23N5O3S
8-[[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2R)-oxolan-2-yl]methyl]-1H-purin-6-one
—— 8-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2R)-oxolan-2-yl]methyl]-1H-purin-6-one —— C22H23N5O3S
8-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2R)-oxolan-2-yl]methyl]-1H-purin-6-one
—— 8-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2S)-oxolan-2-yl]methyl]-1H-purin-6-one —— C22H23N5O3S
8-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2S)-oxolan-2-yl]methyl]-1H-purin-6-one
—— 8-[[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2R)-oxolan-2-yl]methyl]-1H-purin-6-one —— C21H20ClN5O3S
8-[[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methylsulfanyl]-9-[[(2R)-oxolan-2-yl]methyl]-1H-purin-6-one
—— ethyl (3S)-3-phenyl-3-[(4-phenyl-7-thia-2,3,5,10-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5-triene-10-carbonyl)amino]propanoate —— C25H25N5O3S
ethyl (3S)-3-phenyl-3-[(4-phenyl-7-thia-2,3,5,10-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5-triene-10-carbonyl)amino]propanoate
—— ethyl (3S)-3-[[4-(4-fluorophenyl)-7-thia-2,3,5,10-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5-triene-10-carbonyl]amino]-3-phenylpropanoate —— C25H24FN5O3S
ethyl (3S)-3-[[4-(4-fluorophenyl)-7-thia-2,3,5,10-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5-triene-10-carbonyl]amino]-3-phenylpropanoate
—— ethyl (3R)-3-[[4-(4-fluorophenyl)-7-thia-2,3,5,10-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5-triene-10-carbonyl]amino]-3-phenylpropanoate —— C25H24FN5O3S
ethyl (3R)-3-[[4-(4-fluorophenyl)-7-thia-2,3,5,10-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5-triene-10-carbonyl]amino]-3-phenylpropanoate
—— methyl 2-[[3-methylbutyl-[(1R,2R)-2-phenylcyclopropanecarbonyl]amino]methyl]-1,3-thiazole-4-carboxylate —— C21H26N2O3S
methyl 2-[[3-methylbutyl-[(1R,2R)-2-phenylcyclopropanecarbonyl]amino]methyl]-1,3-thiazole-4-carboxylate
—— (2R)-N-(2,6-dimethylphenyl)-2-[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide —— C25H29N3O2S
(2R)-N-(2,6-dimethylphenyl)-2-[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide
—— [(3R,3aR,7E)-3-thiophen-2-yl-7-(thiophen-2-ylmethylidene)-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-(4-chloro-1-ethylpyrazol-3-yl)methanone —— C22H21ClN4OS2
[(3R,3aR,7E)-3-thiophen-2-yl-7-(thiophen-2-ylmethylidene)-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-(4-chloro-1-ethylpyrazol-3-yl)methanone
—— ethyl (3R)-3-phenyl-3-[(4-phenyl-7-thia-2,3,5,10-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5-triene-10-carbonyl)amino]propanoate —— C25H25N5O3S
ethyl (3R)-3-phenyl-3-[(4-phenyl-7-thia-2,3,5,10-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5-triene-10-carbonyl)amino]propanoate
—— 1-[(4aS,9bR)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-2-[1-(4-chlorophenyl)tetrazol-5-yl]sulfanylethanone —— C22H23ClN6OS
1-[(4aS,9bR)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-2-[1-(4-chlorophenyl)tetrazol-5-yl]sulfanylethanone
—— methyl 2-[[[(1R,2R)-2-phenylcyclopropanecarbonyl]-propylamino]methyl]-1,3-thiazole-4-carboxylate —— C19H22N2O3S
methyl 2-[[[(1R,2R)-2-phenylcyclopropanecarbonyl]-propylamino]methyl]-1,3-thiazole-4-carboxylate
—— (2S)-N-cyclohexyl-2-(4-methyl-N-[2-(5-phenyltetrazol-2-yl)acetyl]anilino)-2-pyridin-2-ylacetamide —— C29H31N7O2
(2S)-N-cyclohexyl-2-(4-methyl-N-[2-(5-phenyltetrazol-2-yl)acetyl]anilino)-2-pyridin-2-ylacetamide
—— (2S)-2-[[4-(4-methylphenyl)-5-(phenoxymethyl)-1,2,4-triazol-3-yl]sulfanyl]propanoic acid —— C19H19N3O3S
(2S)-2-[[4-(4-methylphenyl)-5-(phenoxymethyl)-1,2,4-triazol-3-yl]sulfanyl]propanoic acid
—— (2S)-1-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonyl-2-methyl-2,3-dihydroindole —— C20H20ClN3O2S
(2S)-1-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]sulfonyl-2-methyl-2,3-dihydroindole
—— 1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]piperidine-4-carboxamide —— C22H30N4O4S
1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]piperidine-4-carboxamide
—— 1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]piperidine-4-carboxamide —— C22H30N4O4S
1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonyl-N-[[(2S)-oxolan-2-yl]methyl]piperidine-4-carboxamide
—— 1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]piperidine-4-carboxamide —— C27H32N4O3S
1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]piperidine-4-carboxamide
—— 1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]piperidine-4-carboxamide —— C27H32N4O3S
1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]piperidine-4-carboxamide
—— methyl 2-[[cyclohexyl-[(1R,2R)-2-phenylcyclopropanecarbonyl]amino]methyl]-1,3-thiazole-4-carboxylate —— C22H26N2O3S
methyl 2-[[cyclohexyl-[(1R,2R)-2-phenylcyclopropanecarbonyl]amino]methyl]-1,3-thiazole-4-carboxylate
—— [1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonylpiperidin-4-yl]-[(2R)-2-methyl-2,3-dihydroindol-1-yl]methanone —— C26H30N4O3S
[1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonylpiperidin-4-yl]-[(2R)-2-methyl-2,3-dihydroindol-1-yl]methanone
—— (2S)-N-cyclopentyl-2-(furan-2-yl)-2-[furan-2-ylmethyl-[2-[5-(4-methoxyphenyl)tetrazol-2-yl]acetyl]amino]acetamide —— C26H28N6O5
(2S)-N-cyclopentyl-2-(furan-2-yl)-2-[furan-2-ylmethyl-[2-[5-(4-methoxyphenyl)tetrazol-2-yl]acetyl]amino]acetamide
—— 3,5-dimethyl-1-(4-methylphenyl)-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazole-4-sulfonamide —— C22H25N3O2S
3,5-dimethyl-1-(4-methylphenyl)-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazole-4-sulfonamide
—— (2R)-2-[[5-(4-chlorophenyl)-1H-imidazol-2-yl]sulfanyl]-N-(4-methyl-3-nitrophenyl)propanamide —— C19H17ClN4O3S
(2R)-2-[[5-(4-chlorophenyl)-1H-imidazol-2-yl]sulfanyl]-N-(4-methyl-3-nitrophenyl)propanamide
—— 3,5-dimethyl-1-(4-methylphenyl)-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazole-4-sulfonamide —— C22H25N3O2S
3,5-dimethyl-1-(4-methylphenyl)-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazole-4-sulfonamide
—— N-[(2S)-butan-2-yl]-1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonylpiperidine-4-carboxamide —— C21H30N4O3S
N-[(2S)-butan-2-yl]-1-(3,5-dimethyl-1-phenylpyrazol-4-yl)sulfonylpiperidine-4-carboxamide
—— (3R,5S)-5-(2-methylpropoxymethyl)-3-[(2Z)-2-[(4-phenyl-1,3-thiazol-2-yl)hydrazinylidene]propyl]oxolan-2-one —— C21H27N3O3S
(3R,5S)-5-(2-methylpropoxymethyl)-3-[(2Z)-2-[(4-phenyl-1,3-thiazol-2-yl)hydrazinylidene]propyl]oxolan-2-one