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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-3-oxopiperazine-1-carboxamide —— C17H21N5O2
N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-3-oxopiperazine-1-carboxamide
—— (3R)-N-(2,2-dicyclopropylethyl)-N'-methyl-3-[(1-methylpyrazol-4-yl)methyl]pyrrolidine-1-carboximidamide —— C19H31N5
(3R)-N-(2,2-dicyclopropylethyl)-N'-methyl-3-[(1-methylpyrazol-4-yl)methyl]pyrrolidine-1-carboximidamide
—— 5-[(1S)-1-chloroethyl]-3-[(1S)-1-methoxyethyl]-1,2,4-oxadiazole —— C7H11ClN2O2
5-[(1S)-1-chloroethyl]-3-[(1S)-1-methoxyethyl]-1,2,4-oxadiazole
—— 1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,2R)-2,4,4-trimethylcyclohexyl]urea —— C17H29N5O
1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,2R)-2,4,4-trimethylcyclohexyl]urea
—— 1-[(2R)-2-cyclopropyl-2-hydroxyethyl]-3-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]urea —— C18H24N4O2
1-[(2R)-2-cyclopropyl-2-hydroxyethyl]-3-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]urea
—— 1-cyclopropyl-3-[(1S)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(1S)-1-pyridin-2-ylethyl]urea —— C18H24N4OS
1-cyclopropyl-3-[(1S)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(1S)-1-pyridin-2-ylethyl]urea
—— 1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1R,3S)-3-ethylsulfanylcyclopentyl]urea —— C15H25N5OS
1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1R,3S)-3-ethylsulfanylcyclopentyl]urea
—— 1-[(2S)-2-cyclopropyl-2-hydroxyethyl]-3-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]urea —— C18H24N4O2
1-[(2S)-2-cyclopropyl-2-hydroxyethyl]-3-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]urea
—— 1-cyclopropyl-3-[(R)-cyclopropyl(1,3-thiazol-2-yl)methyl]-1-[(2R)-3-methylbutan-2-yl]urea —— C16H25N3OS
1-cyclopropyl-3-[(R)-cyclopropyl(1,3-thiazol-2-yl)methyl]-1-[(2R)-3-methylbutan-2-yl]urea
—— 4-(hydroxymethyl)-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]piperidine-1-carboxamide —— C19H26N4O2
4-(hydroxymethyl)-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]piperidine-1-carboxamide
—— N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-3-oxopiperazine-1-carboxamide —— C17H21N5O2
N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-3-oxopiperazine-1-carboxamide
—— 1-cyclopropyl-3-[(1R)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(2R)-3-methylbutan-2-yl]urea —— C16H27N3OS
1-cyclopropyl-3-[(1R)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(2R)-3-methylbutan-2-yl]urea
—— 1-cyclopentyl-3-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-1-[[(2R)-oxolan-2-yl]methyl]urea —— C18H29N5O2
1-cyclopentyl-3-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-1-[[(2R)-oxolan-2-yl]methyl]urea
—— 1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1R,3S)-3-ethoxy-2,2-diethylcyclobutyl]urea —— C18H31N5O2
1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1R,3S)-3-ethoxy-2,2-diethylcyclobutyl]urea
—— (3R)-3-(hydroxymethyl)-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]piperidine-1-carboxamide —— C19H26N4O2
(3R)-3-(hydroxymethyl)-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]piperidine-1-carboxamide
—— (2S)-2-(hydroxymethyl)-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]pyrrolidine-1-carboxamide —— C18H24N4O2
(2S)-2-(hydroxymethyl)-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]pyrrolidine-1-carboxamide
—— 1-cyclopropyl-3-[(1R)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(2S)-3-methylbutan-2-yl]urea —— C16H27N3OS
1-cyclopropyl-3-[(1R)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(2S)-3-methylbutan-2-yl]urea
—— 1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1R,2R)-2,4,4-trimethylcyclohexyl]urea —— C17H29N5O
1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1R,2R)-2,4,4-trimethylcyclohexyl]urea
—— 1-cyclopropyl-1-[(1R)-1-(furan-2-yl)ethyl]-3-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)propyl]urea —— C19H28N4O2
1-cyclopropyl-1-[(1R)-1-(furan-2-yl)ethyl]-3-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)propyl]urea
—— 4-(hydroxymethyl)-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]piperidine-1-carboxamide —— C19H26N4O2
4-(hydroxymethyl)-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]piperidine-1-carboxamide
—— 1-cyclopropyl-3-[[2-(dimethylamino)-3-methylimidazol-4-yl]methyl]-1-[(1R)-1-(furan-2-yl)ethyl]urea —— C17H25N5O2
1-cyclopropyl-3-[[2-(dimethylamino)-3-methylimidazol-4-yl]methyl]-1-[(1R)-1-(furan-2-yl)ethyl]urea
—— (3S)-3-(hydroxymethyl)-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]piperidine-1-carboxamide —— C19H26N4O2
(3S)-3-(hydroxymethyl)-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]piperidine-1-carboxamide
—— 1-cyclopropyl-3-[[2-(dimethylamino)-3-methylimidazol-4-yl]methyl]-1-[(1S)-1-(furan-2-yl)ethyl]urea —— C17H25N5O2
1-cyclopropyl-3-[[2-(dimethylamino)-3-methylimidazol-4-yl]methyl]-1-[(1S)-1-(furan-2-yl)ethyl]urea
—— 1-ethyl-1-(2-hydroxyethyl)-3-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]urea —— C17H24N4O2
1-ethyl-1-(2-hydroxyethyl)-3-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]urea
—— 1-cyclopropyl-1-[(1S)-1-(furan-2-yl)ethyl]-3-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)propyl]urea —— C19H28N4O2
1-cyclopropyl-1-[(1S)-1-(furan-2-yl)ethyl]-3-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)propyl]urea
—— (2S)-2-(hydroxymethyl)-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]pyrrolidine-1-carboxamide —— C18H24N4O2
(2S)-2-(hydroxymethyl)-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]pyrrolidine-1-carboxamide
—— (3S)-3-ethyl-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]morpholine-4-carboxamide —— C19H26N4O2
(3S)-3-ethyl-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]morpholine-4-carboxamide
—— 1-[(2S,6R)-2,6-dimethylcyclohexyl]-3-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]urea —— C16H28N4O2
1-[(2S,6R)-2,6-dimethylcyclohexyl]-3-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]urea
—— 1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,2S)-2,4,4-trimethylcyclohexyl]urea —— C17H29N5O
1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,2S)-2,4,4-trimethylcyclohexyl]urea
—— 1-cyclopentyl-3-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-1-[[(2S)-oxolan-2-yl]methyl]urea —— C18H29N5O2
1-cyclopentyl-3-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-1-[[(2S)-oxolan-2-yl]methyl]urea
—— 1-cyclopropyl-1-[(1S)-1-(furan-2-yl)ethyl]-3-[(1R,2S)-2-imidazol-1-ylcyclopentyl]urea —— C18H24N4O2
1-cyclopropyl-1-[(1S)-1-(furan-2-yl)ethyl]-3-[(1R,2S)-2-imidazol-1-ylcyclopentyl]urea
—— 1-cyclopropyl-1-[(1S)-1-(2-fluorophenyl)ethyl]-3-[(5-methyl-1,3-thiazol-2-yl)methyl]urea —— C17H20FN3OS
1-cyclopropyl-1-[(1S)-1-(2-fluorophenyl)ethyl]-3-[(5-methyl-1,3-thiazol-2-yl)methyl]urea
—— (3R)-3-ethyl-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]morpholine-4-carboxamide —— C19H26N4O2
(3R)-3-ethyl-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]morpholine-4-carboxamide
—— 1-cyclopropyl-3-[(1S)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(1R)-1-pyridin-2-ylethyl]urea —— C18H24N4OS
1-cyclopropyl-3-[(1S)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(1R)-1-pyridin-2-ylethyl]urea
—— 1-cyclopropyl-3-[(1S)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(2R)-3-methylbutan-2-yl]urea —— C16H27N3OS
1-cyclopropyl-3-[(1S)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(2R)-3-methylbutan-2-yl]urea
—— 1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,3S)-3-ethylsulfanylcyclopentyl]urea —— C15H25N5OS
1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,3S)-3-ethylsulfanylcyclopentyl]urea
—— 1-cyclopropyl-1-[(1R)-1-(furan-2-yl)ethyl]-3-[(1R,2S)-2-imidazol-1-ylcyclopentyl]urea —— C18H24N4O2
1-cyclopropyl-1-[(1R)-1-(furan-2-yl)ethyl]-3-[(1R,2S)-2-imidazol-1-ylcyclopentyl]urea
—— 1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,3R)-3-ethoxy-2,2-diethylcyclobutyl]urea —— C18H31N5O2
1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,3R)-3-ethoxy-2,2-diethylcyclobutyl]urea
—— 1-[(2R)-2-cyclopropyl-2-hydroxyethyl]-3-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]urea —— C18H24N4O2
1-[(2R)-2-cyclopropyl-2-hydroxyethyl]-3-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]urea
—— 1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,3S)-3-ethoxy-2,2-diethylcyclobutyl]urea —— C18H31N5O2
1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,3S)-3-ethoxy-2,2-diethylcyclobutyl]urea
—— (3R)-3-ethyl-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]morpholine-4-carboxamide —— C19H26N4O2
(3R)-3-ethyl-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]morpholine-4-carboxamide
—— 1-[(2R,6R)-2,6-dimethylcyclohexyl]-3-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]urea —— C16H28N4O2
1-[(2R,6R)-2,6-dimethylcyclohexyl]-3-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]urea
—— 1-cyclopropyl-1-[(2R)-3-methylbutan-2-yl]-3-[(1R)-1-[3-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C19H27N5O
1-cyclopropyl-1-[(2R)-3-methylbutan-2-yl]-3-[(1R)-1-[3-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— 1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1R,3R)-3-ethoxy-2,2-diethylcyclobutyl]urea —— C18H31N5O2
1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1R,3R)-3-ethoxy-2,2-diethylcyclobutyl]urea
—— 1-cyclopropyl-1-[(2S)-3-methylbutan-2-yl]-3-[(1R)-1-[3-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C19H27N5O
1-cyclopropyl-1-[(2S)-3-methylbutan-2-yl]-3-[(1R)-1-[3-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— (3S)-3-ethyl-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]morpholine-4-carboxamide —— C19H26N4O2
(3S)-3-ethyl-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]morpholine-4-carboxamide
—— 1-[(2S)-2-cyclopropyl-2-hydroxyethyl]-3-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]urea —— C18H24N4O2
1-[(2S)-2-cyclopropyl-2-hydroxyethyl]-3-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]urea
—— 1-cyclopropyl-3-[(1R)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(1S)-1-pyridin-2-ylethyl]urea —— C18H24N4OS
1-cyclopropyl-3-[(1R)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(1S)-1-pyridin-2-ylethyl]urea
—— 1-cyclopropyl-3-[(1S)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(2S)-3-methylbutan-2-yl]urea —— C16H27N3OS
1-cyclopropyl-3-[(1S)-1-(5-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(2S)-3-methylbutan-2-yl]urea
—— 1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,3R)-3-ethylsulfanylcyclopentyl]urea —— C15H25N5OS
1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-3-[(1S,3R)-3-ethylsulfanylcyclopentyl]urea