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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-2-(4-nitrophenyl)sulfanyl-N-[3-(1H-pyrazol-4-yl)phenyl]propanamide —— C18H16N4O3S
(2S)-2-(4-nitrophenyl)sulfanyl-N-[3-(1H-pyrazol-4-yl)phenyl]propanamide
—— N-[(1S)-1-[5-(3,4-dichlorophenyl)-1H-imidazol-2-yl]ethyl]-2,5-dimethylfuran-3-carboxamide —— C18H17Cl2N3O2
N-[(1S)-1-[5-(3,4-dichlorophenyl)-1H-imidazol-2-yl]ethyl]-2,5-dimethylfuran-3-carboxamide
—— 1-[1-[(2S)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)oxyethanone —— C23H25N5O3
1-[1-[(2S)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)oxyethanone
—— benzyl N-[1-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]-2,5-dioxopyrrolidin-3-yl]carbamate —— C37H34N6O7S
benzyl N-[1-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]-2,5-dioxopyrrolidin-3-yl]carbamate
—— (2S)-2-(2,3-dichlorophenoxy)-N-[2-(triazol-1-yl)phenyl]propanamide —— C17H14Cl2N4O2
(2S)-2-(2,3-dichlorophenoxy)-N-[2-(triazol-1-yl)phenyl]propanamide
—— N-[(1R)-1-[5-(3,4-dichlorophenyl)-1H-imidazol-2-yl]ethyl]-2,5-dimethylfuran-3-carboxamide —— C18H17Cl2N3O2
N-[(1R)-1-[5-(3,4-dichlorophenyl)-1H-imidazol-2-yl]ethyl]-2,5-dimethylfuran-3-carboxamide
—— 2-[2,5-dimethyl-3-(2-methyl-1,3-thiazol-4-yl)pyrrol-1-yl]-N-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]acetamide —— C20H27N5OS
2-[2,5-dimethyl-3-(2-methyl-1,3-thiazol-4-yl)pyrrol-1-yl]-N-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]acetamide
—— N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]benzenesulfonamide —— C31H29N5O5S2
N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]benzenesulfonamide
—— 6-acetamido-N-[4-[(2R,4R,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C41H43N3O6S
6-acetamido-N-[4-[(2R,4R,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 2-[2,5-dimethyl-3-(2-methyl-1,3-thiazol-4-yl)pyrrol-1-yl]-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]acetamide —— C20H27N5OS
2-[2,5-dimethyl-3-(2-methyl-1,3-thiazol-4-yl)pyrrol-1-yl]-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]acetamide
—— 6-acetamido-N-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C33H38N6O6S
6-acetamido-N-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 1-ethyl-3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea —— C28H30N6O5S
1-ethyl-3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea
—— 2,2,2-trichloro-N-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]acetamide —— C27H24Cl3N5O4S
2,2,2-trichloro-N-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]acetamide
—— N-[4-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]acetamide —— C35H32N2O5S
N-[4-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]acetamide
—— prop-2-enyl N-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]carbamate —— C29H29N5O6S
prop-2-enyl N-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]carbamate
—— 1-ethyl-3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea —— C28H30N6O5S
1-ethyl-3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea
—— 6-acetamido-N-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C33H38N6O5S
6-acetamido-N-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 4-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-4-oxobutanoic acid —— C29H29N5O7S
4-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-4-oxobutanoic acid
—— 1-[4-[(2R,4R,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]-3-ethylurea —— C36H35N3O5S
1-[4-[(2R,4R,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]-3-ethylurea
—— N-[(2R)-2-(2,5-dimethylfuran-3-yl)-2-hydroxypropyl]-1-methylimidazole-4-sulfonamide —— C13H19N3O4S
N-[(2R)-2-(2,5-dimethylfuran-3-yl)-2-hydroxypropyl]-1-methylimidazole-4-sulfonamide
—— 4-[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-4-oxobutanoic acid —— C30H31N5O6S
4-[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-4-oxobutanoic acid
—— 1-benzyl-3-[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]urea —— C42H39N3O5S
1-benzyl-3-[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]urea
—— (2R)-2-(4-nitrophenyl)sulfanyl-N-[3-(1H-pyrazol-4-yl)phenyl]propanamide —— C18H16N4O3S
(2R)-2-(4-nitrophenyl)sulfanyl-N-[3-(1H-pyrazol-4-yl)phenyl]propanamide
—— (2R)-2-(2,3-dichlorophenoxy)-N-[2-(triazol-1-yl)phenyl]propanamide —— C17H14Cl2N4O2
(2R)-2-(2,3-dichlorophenoxy)-N-[2-(triazol-1-yl)phenyl]propanamide
—— 2,2,2-trichloro-N-[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]acetamide —— C36H31Cl3N2O5S
2,2,2-trichloro-N-[4-[(2R,4R,5S,6S)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]acetamide
—— 4-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-4-oxobutanoic acid —— C30H31N5O6S
4-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-4-oxobutanoic acid
—— (1R,2S)-2-(2,3-difluorophenyl)-N-[2-(5-methyl-1H-imidazol-2-yl)phenyl]cyclopropane-1-carboxamide —— C20H17F2N3O
(1R,2S)-2-(2,3-difluorophenyl)-N-[2-(5-methyl-1H-imidazol-2-yl)phenyl]cyclopropane-1-carboxamide
—— benzyl N-[1-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]-2,5-dioxopyrrolidin-3-yl]carbamate —— C38H36N6O7S
benzyl N-[1-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]-2,5-dioxopyrrolidin-3-yl]carbamate
—— benzyl N-[1-[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]-2,5-dioxopyrrolidin-3-yl]carbamate —— C38H36N6O7S
benzyl N-[1-[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]-2,5-dioxopyrrolidin-3-yl]carbamate
—— prop-2-enyl N-[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]carbamate —— C30H31N5O5S
prop-2-enyl N-[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]carbamate
—— 3-[4-[(2S)-2,4-dimethylpiperazine-1-carbonyl]phenyl]-4-methyl-1H-imidazol-2-one —— C17H22N4O2
3-[4-[(2S)-2,4-dimethylpiperazine-1-carbonyl]phenyl]-4-methyl-1H-imidazol-2-one
—— 3-[4-[(2R)-2,4-dimethylpiperazine-1-carbonyl]phenyl]-4-methyl-1H-imidazol-2-one —— C17H22N4O2
3-[4-[(2R)-2,4-dimethylpiperazine-1-carbonyl]phenyl]-4-methyl-1H-imidazol-2-one
—— (4S)-N-[2-(5-methyl-1H-imidazol-2-yl)phenyl]-6,7-dihydro-4H-thieno[3,2-c]thiopyran-4-carboxamide —— C18H17N3OS2
(4S)-N-[2-(5-methyl-1H-imidazol-2-yl)phenyl]-6,7-dihydro-4H-thieno[3,2-c]thiopyran-4-carboxamide
—— (1S,2R)-2-(2,3-difluorophenyl)-N-[2-(5-methyl-1H-imidazol-2-yl)phenyl]cyclopropane-1-carboxamide —— C20H17F2N3O
(1S,2R)-2-(2,3-difluorophenyl)-N-[2-(5-methyl-1H-imidazol-2-yl)phenyl]cyclopropane-1-carboxamide
—— (1R,2R)-2-(2,3-difluorophenyl)-N-[2-(5-methyl-1H-imidazol-2-yl)phenyl]cyclopropane-1-carboxamide —— C20H17F2N3O
(1R,2R)-2-(2,3-difluorophenyl)-N-[2-(5-methyl-1H-imidazol-2-yl)phenyl]cyclopropane-1-carboxamide
—— 5-[2-[(R)-3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfinyl]ethyl]-4-methyl-1,3-thiazole —— C15H17NO3S2
5-[2-[(R)-3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfinyl]ethyl]-4-methyl-1,3-thiazole
—— (4R)-N-[2-(5-methyl-1H-imidazol-2-yl)phenyl]-6,7-dihydro-4H-thieno[3,2-c]thiopyran-4-carboxamide —— C18H17N3OS2
(4R)-N-[2-(5-methyl-1H-imidazol-2-yl)phenyl]-6,7-dihydro-4H-thieno[3,2-c]thiopyran-4-carboxamide
—— 5-[2-[(S)-3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfinyl]ethyl]-4-methyl-1,3-thiazole —— C15H17NO3S2
5-[2-[(S)-3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfinyl]ethyl]-4-methyl-1,3-thiazole
—— N-[(3S)-1-(5-chloro-2-methoxyphenyl)pyrrolidin-3-yl]-3-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide —— C22H23ClN4O3
N-[(3S)-1-(5-chloro-2-methoxyphenyl)pyrrolidin-3-yl]-3-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide
—— (2R)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-phenylpropane-1-sulfonamide —— C14H18N2O2S2
(2R)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-phenylpropane-1-sulfonamide
—— 1-(2-chlorophenyl)-3-methyl-N-[(2S)-2-morpholin-4-yl-2-thiophen-2-ylethyl]thieno[2,3-c]pyrazole-5-carboxamide —— C23H23ClN4O2S2
1-(2-chlorophenyl)-3-methyl-N-[(2S)-2-morpholin-4-yl-2-thiophen-2-ylethyl]thieno[2,3-c]pyrazole-5-carboxamide
—— (2S)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-phenylpropane-1-sulfonamide —— C14H18N2O2S2
(2S)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-phenylpropane-1-sulfonamide
—— (3R)-N-methyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-N-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-amine —— C18H28N4OS
(3R)-N-methyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-N-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-amine
—— N-[(3R)-1-(5-chloro-2-methoxyphenyl)pyrrolidin-3-yl]-3-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide —— C22H23ClN4O3
N-[(3R)-1-(5-chloro-2-methoxyphenyl)pyrrolidin-3-yl]-3-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide
—— prop-2-enyl N-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-5-methyl-1,3-dioxan-2-yl]phenyl]carbamate —— C30H31N5O6S
prop-2-enyl N-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-5-methyl-1,3-dioxan-2-yl]phenyl]carbamate
—— 1-(2-chlorophenyl)-3-methyl-N-[(2R)-2-morpholin-4-yl-2-thiophen-2-ylethyl]thieno[2,3-c]pyrazole-5-carboxamide —— C23H23ClN4O2S2
1-(2-chlorophenyl)-3-methyl-N-[(2R)-2-morpholin-4-yl-2-thiophen-2-ylethyl]thieno[2,3-c]pyrazole-5-carboxamide
—— 5-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C31H33N5O6S
5-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— (3S)-N-methyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-N-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-amine —— C18H28N4OS
(3S)-N-methyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-N-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-amine
—— 1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(2R,4R)-4-hydroxy-4-phenylbutan-2-yl]urea —— C18H25N3O2S
1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(2R,4R)-4-hydroxy-4-phenylbutan-2-yl]urea
—— 2-[(3S,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]-N,4-dimethyl-1,3-thiazole-5-carboxamide —— C13H19N3O2S
2-[(3S,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]-N,4-dimethyl-1,3-thiazole-5-carboxamide