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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[2-(3,4-dihydro-2H-pyrrol-5-ylamino)-5-methyl-1,3-thiazol-4-yl]ethanone —— C10H13N3OS
1-[2-(3,4-dihydro-2H-pyrrol-5-ylamino)-5-methyl-1,3-thiazol-4-yl]ethanone
—— N-benzyl-5-methyl-N-[[(2S)-oxolan-2-yl]methyl]-1-propylpyrazole-4-carboxamide —— C20H27N3O2
N-benzyl-5-methyl-N-[[(2S)-oxolan-2-yl]methyl]-1-propylpyrazole-4-carboxamide
—— [3-[(2S)-2-methylpiperidin-1-yl]azetidin-1-yl]-(3-methyl-1-propylpyrazol-4-yl)methanone —— C17H28N4O
[3-[(2S)-2-methylpiperidin-1-yl]azetidin-1-yl]-(3-methyl-1-propylpyrazol-4-yl)methanone
—— N-benzyl-5-methyl-N-[[(2R)-oxolan-2-yl]methyl]-1-propylpyrazole-4-carboxamide —— C20H27N3O2
N-benzyl-5-methyl-N-[[(2R)-oxolan-2-yl]methyl]-1-propylpyrazole-4-carboxamide
—— (1-methylpyrazol-4-yl)-[(2S)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C14H19N5O2
(1-methylpyrazol-4-yl)-[(2S)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— 1-(3-chloro-4-fluorophenyl)-5-[(2R)-oxan-2-yl]-1,2,4-triazole —— C13H13ClFN3O
1-(3-chloro-4-fluorophenyl)-5-[(2R)-oxan-2-yl]-1,2,4-triazole
—— (3S)-1-cyclopentyl-N-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-N-methyl-6-oxopiperidine-3-carboxamide —— C22H27FN4O2
(3S)-1-cyclopentyl-N-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-N-methyl-6-oxopiperidine-3-carboxamide
—— (1-methylpyrazol-4-yl)-[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C14H19N5O2
(1-methylpyrazol-4-yl)-[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— [(3S)-3-ethyl-4-propan-2-ylpiperazin-1-yl]-(5-methyl-1-propylpyrazol-4-yl)methanone —— C17H30N4O
[(3S)-3-ethyl-4-propan-2-ylpiperazin-1-yl]-(5-methyl-1-propylpyrazol-4-yl)methanone
—— N-[(2R)-2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl]-3-(1,2,4-triazol-4-yl)benzamide —— C18H15F3N4O2
N-[(2R)-2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl]-3-(1,2,4-triazol-4-yl)benzamide
—— (3R)-1-cyclopentyl-N-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-N-methyl-6-oxopiperidine-3-carboxamide —— C22H27FN4O2
(3R)-1-cyclopentyl-N-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-N-methyl-6-oxopiperidine-3-carboxamide
—— 2-[(5-ethyl-1H-1,2,4-triazol-3-yl)sulfanyl]-N-[(1R)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide —— C18H21FN6OS
2-[(5-ethyl-1H-1,2,4-triazol-3-yl)sulfanyl]-N-[(1R)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide
—— N-[(2S)-2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl]-3-(1,2,4-triazol-4-yl)benzamide —— C18H15F3N4O2
N-[(2S)-2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl]-3-(1,2,4-triazol-4-yl)benzamide
—— 3-(2-fluorophenyl)-N-[1-[[(2S)-oxolan-2-yl]methyl]piperidin-4-yl]-1H-pyrazole-5-carboxamide —— C20H25FN4O2
3-(2-fluorophenyl)-N-[1-[[(2S)-oxolan-2-yl]methyl]piperidin-4-yl]-1H-pyrazole-5-carboxamide
—— 3-(2-fluorophenyl)-N-[1-[[(2R)-oxolan-2-yl]methyl]piperidin-4-yl]-1H-pyrazole-5-carboxamide —— C20H25FN4O2
3-(2-fluorophenyl)-N-[1-[[(2R)-oxolan-2-yl]methyl]piperidin-4-yl]-1H-pyrazole-5-carboxamide
—— 1-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-propylurea —— C19H26N4O
1-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-propylurea
—— 1-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-propylurea —— C19H26N4O
1-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-propylurea
—— N-[(4R)-1-(3-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-5-propan-2-yl-1H-pyrazole-3-carboxamide —— C22H26FN5O
N-[(4R)-1-(3-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-5-propan-2-yl-1H-pyrazole-3-carboxamide
—— (2S)-N-[(1-phenyltetrazol-5-yl)methyl]-2-pyrazol-1-ylbutanamide —— C15H17N7O
(2S)-N-[(1-phenyltetrazol-5-yl)methyl]-2-pyrazol-1-ylbutanamide
—— (2R)-N-[(1-phenyltetrazol-5-yl)methyl]-2-pyrazol-1-ylbutanamide —— C15H17N7O
(2R)-N-[(1-phenyltetrazol-5-yl)methyl]-2-pyrazol-1-ylbutanamide
—— (3R)-3-(furan-2-yl)-3-(4-phenyl-5-pyridin-3-ylimidazol-1-yl)propanoic acid —— C21H17N3O3
(3R)-3-(furan-2-yl)-3-(4-phenyl-5-pyridin-3-ylimidazol-1-yl)propanoic acid
—— N-[(4S)-1-(3-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-5-propan-2-yl-1H-pyrazole-3-carboxamide —— C22H26FN5O
N-[(4S)-1-(3-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-5-propan-2-yl-1H-pyrazole-3-carboxamide
—— (2-propyl-1,3-thiazol-4-yl)-[(1S)-1-pyridin-2-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone —— C19H20N4OS
(2-propyl-1,3-thiazol-4-yl)-[(1S)-1-pyridin-2-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone
—— (2-propyl-1,3-thiazol-4-yl)-[(1R)-1-pyridin-2-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone —— C19H20N4OS
(2-propyl-1,3-thiazol-4-yl)-[(1R)-1-pyridin-2-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone
—— (1-methylpyrrol-2-yl)-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C18H18N4O2
(1-methylpyrrol-2-yl)-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— (1-methylpyrrol-2-yl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C18H18N4O2
(1-methylpyrrol-2-yl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— N-[[(1S)-3,4-dihydro-1H-isochromen-1-yl]methyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide —— C20H18FN3O2
N-[[(1S)-3,4-dihydro-1H-isochromen-1-yl]methyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
—— (3S)-3-(4-methoxyphenyl)-5-naphthalen-2-yl-2-phenyl-3,4-dihydropyrazole —— C26H22N2O
(3S)-3-(4-methoxyphenyl)-5-naphthalen-2-yl-2-phenyl-3,4-dihydropyrazole
—— 2-cyclopropyl-N-[(1S)-1-[1-(2-methoxyphenyl)pyrazol-4-yl]ethyl]-6-oxo-1H-pyrimidine-5-carboxamide —— C20H21N5O3
2-cyclopropyl-N-[(1S)-1-[1-(2-methoxyphenyl)pyrazol-4-yl]ethyl]-6-oxo-1H-pyrimidine-5-carboxamide
—— 1-methyl-4-phenyl-2-[(1'R,8'S,9'S)-spiro[cyclopropane-1,10'-tricyclo[6.2.1.02,7]undeca-2,4,6-triene]-9'-yl]-1,2,4-triazolidine-3,5-dione —— C22H21N3O2
1-methyl-4-phenyl-2-[(1'R,8'S,9'S)-spiro[cyclopropane-1,10'-tricyclo[6.2.1.02,7]undeca-2,4,6-triene]-9'-yl]-1,2,4-triazolidine-3,5-dione
—— (4-ethyl-2-methyl-1,3-thiazol-5-yl)-[(3R)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methanone —— C16H27N3OS
(4-ethyl-2-methyl-1,3-thiazol-5-yl)-[(3R)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methanone
—— N-[(4S)-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]cyclopropanesulfonamide —— C18H23N3O2S
N-[(4S)-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]cyclopropanesulfonamide
—— 1-methyl-4-phenyl-2-[(1'R,8'S,9'R)-spiro[cyclopropane-1,10'-tricyclo[6.2.1.02,7]undeca-2,4,6-triene]-9'-yl]-1,2,4-triazolidine-3,5-dione —— C22H21N3O2
1-methyl-4-phenyl-2-[(1'R,8'S,9'R)-spiro[cyclopropane-1,10'-tricyclo[6.2.1.02,7]undeca-2,4,6-triene]-9'-yl]-1,2,4-triazolidine-3,5-dione
—— N-[(4R)-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]cyclopropanesulfonamide —— C18H23N3O2S
N-[(4R)-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]cyclopropanesulfonamide
—— 2-cyclopropyl-N-[(1R)-1-[1-(2-methoxyphenyl)pyrazol-4-yl]ethyl]-6-oxo-1H-pyrimidine-5-carboxamide —— C20H21N5O3
2-cyclopropyl-N-[(1R)-1-[1-(2-methoxyphenyl)pyrazol-4-yl]ethyl]-6-oxo-1H-pyrimidine-5-carboxamide
—— [(3R)-3-[[4-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]-[4-(1H-1,2,4-triazol-5-yl)phenyl]methanone —— C21H22N4O2
[(3R)-3-[[4-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]-[4-(1H-1,2,4-triazol-5-yl)phenyl]methanone
—— (4-ethyl-2-methyl-1,3-thiazol-5-yl)-[(3S)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methanone —— C16H27N3OS
(4-ethyl-2-methyl-1,3-thiazol-5-yl)-[(3S)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methanone
—— N-[[(1R)-3,4-dihydro-1H-isochromen-1-yl]methyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide —— C20H18FN3O2
N-[[(1R)-3,4-dihydro-1H-isochromen-1-yl]methyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
—— N-[(4R)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]pyridine-3-sulfonamide —— C21H24N4O2S
N-[(4R)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]pyridine-3-sulfonamide
—— 5-ethyl-N-[(4R)-1-(4-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-1H-pyrazole-3-carboxamide —— C21H24FN5O
5-ethyl-N-[(4R)-1-(4-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-1H-pyrazole-3-carboxamide
—— 1-(2-methoxyphenyl)-N-[(2R)-2-(N-methylanilino)propyl]pyrazole-4-carboxamide —— C21H24N4O2
1-(2-methoxyphenyl)-N-[(2R)-2-(N-methylanilino)propyl]pyrazole-4-carboxamide
—— N,4-dimethyl-N-[3-[(2S)-oxolan-2-yl]propyl]-2-propan-2-yl-1,3-thiazole-5-carboxamide —— C16H26N2O2S
N,4-dimethyl-N-[3-[(2S)-oxolan-2-yl]propyl]-2-propan-2-yl-1,3-thiazole-5-carboxamide
—— N,4-dimethyl-N-[3-[(2R)-oxolan-2-yl]propyl]-2-propan-2-yl-1,3-thiazole-5-carboxamide —— C16H26N2O2S
N,4-dimethyl-N-[3-[(2R)-oxolan-2-yl]propyl]-2-propan-2-yl-1,3-thiazole-5-carboxamide
—— 1-(4-chlorophenyl)-4-oxo-2H-pyrazolo[3,4-b]pyridine-5-carboxylate —— C13H7ClN3O3-
1-(4-chlorophenyl)-4-oxo-2H-pyrazolo[3,4-b]pyridine-5-carboxylate
—— 2-[[4-Ethyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetate —— C13H14N3O2S-
2-[[4-Ethyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 4-[(3aR,6aS)-5-(4-fluorophenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-d][1,2]oxazole-3-carbonyl]-5-methyl-1-(4-methylphenyl)pyrazole-3-carboxylate —— C26H21FN4O6
ethyl 4-[(3aR,6aS)-5-(4-fluorophenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-d][1,2]oxazole-3-carbonyl]-5-methyl-1-(4-methylphenyl)pyrazole-3-carboxylate
—— ethyl 4-[(3aR,6aR)-5-(4-fluorophenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-d][1,2]oxazole-3-carbonyl]-5-methyl-1-(4-methylphenyl)pyrazole-3-carboxylate —— C26H21FN4O6
ethyl 4-[(3aR,6aR)-5-(4-fluorophenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-d][1,2]oxazole-3-carbonyl]-5-methyl-1-(4-methylphenyl)pyrazole-3-carboxylate
—— [(3S)-3-[[4-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]-[4-(1H-1,2,4-triazol-5-yl)phenyl]methanone —— C21H22N4O2
[(3S)-3-[[4-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]-[4-(1H-1,2,4-triazol-5-yl)phenyl]methanone
—— [5-[1-[(1R)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]triazol-4-yl]furan-2-yl]methanol —— C16H18N4O2S
[5-[1-[(1R)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]triazol-4-yl]furan-2-yl]methanol
—— 1-(2-methoxyphenyl)-N-[(2S)-2-(N-methylanilino)propyl]pyrazole-4-carboxamide —— C21H24N4O2
1-(2-methoxyphenyl)-N-[(2S)-2-(N-methylanilino)propyl]pyrazole-4-carboxamide