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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-4-methylsulfonyl-2-[[4-(3-pyrazol-1-ylphenyl)triazol-1-yl]methyl]morpholine —— C17H20N6O3S
(2S)-4-methylsulfonyl-2-[[4-(3-pyrazol-1-ylphenyl)triazol-1-yl]methyl]morpholine
—— (5R)-7-propan-2-yl-2-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5R)-7-propan-2-yl-2-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propan-2-yl-2-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5S)-7-propan-2-yl-2-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (2R)-2-phenoxy-N-(2-phenyl-4,6-dihydrothieno[3,4-c]pyrazol-3-yl)propanamide —— C20H19N3O2S
(2R)-2-phenoxy-N-(2-phenyl-4,6-dihydrothieno[3,4-c]pyrazol-3-yl)propanamide
—— (5S)-2-[[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C21H27FN4O
(5S)-2-[[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 2-[(2R)-2-[4-(3-chloro-5-fluoro-4-methoxyphenyl)triazol-1-yl]propyl]pyrazine —— C16H15ClFN5O
2-[(2R)-2-[4-(3-chloro-5-fluoro-4-methoxyphenyl)triazol-1-yl]propyl]pyrazine
—— (5R)-2-[[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C21H27FN4O
(5R)-2-[[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— [(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C21H28N4O3
[(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— 5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-[(2-methoxyphenoxy)methyl]-1,3-oxazole-4-carbonitrile —— C19H23N3O3
5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-[(2-methoxyphenoxy)methyl]-1,3-oxazole-4-carbonitrile
—— (4R)-4-[4-(2,2-dimethyl-3H-1-benzofuran-5-yl)triazol-1-yl]-1-(2-methoxyethyl)pyrrolidin-2-one —— C19H24N4O3
(4R)-4-[4-(2,2-dimethyl-3H-1-benzofuran-5-yl)triazol-1-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
—— 5-[(1R)-1-[4-[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]triazol-1-yl]ethyl]-2H-tetrazole —— C16H16FN9
5-[(1R)-1-[4-[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]triazol-1-yl]ethyl]-2H-tetrazole
—— N-[5-(1-adamantyl)-1,3,4-thiadiazol-2-yl]-4-chloro-N-methylbutanamide —— C17H24ClN3OS
N-[5-(1-adamantyl)-1,3,4-thiadiazol-2-yl]-4-chloro-N-methylbutanamide
—— (4S)-4-(dimethylsulfamoylamino)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazole —— C18H26N4O3S
(4S)-4-(dimethylsulfamoylamino)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazole
—— 4-(1-methylimidazol-2-yl)-1-[(1S)-1-(2-pyrazol-1-ylphenyl)ethyl]triazole —— C17H17N7
4-(1-methylimidazol-2-yl)-1-[(1S)-1-(2-pyrazol-1-ylphenyl)ethyl]triazole
—— [(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C21H28N4O3
[(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— (4S)-4-[4-(2,2-dimethyl-3H-1-benzofuran-5-yl)triazol-1-yl]-1-(2-methoxyethyl)pyrrolidin-2-one —— C19H24N4O3
(4S)-4-[4-(2,2-dimethyl-3H-1-benzofuran-5-yl)triazol-1-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
—— (5R)-7-(2-hydroxyethyl)-2-[3-(1,2,4-triazol-4-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H23N5O3
(5R)-7-(2-hydroxyethyl)-2-[3-(1,2,4-triazol-4-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
—— [(2R)-2-(furan-2-yl)pyrrolidin-1-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone —— C18H17N3O2
[(2R)-2-(furan-2-yl)pyrrolidin-1-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone
—— (5S)-7-(2-hydroxyethyl)-2-[3-(1,2,4-triazol-4-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H23N5O3
(5S)-7-(2-hydroxyethyl)-2-[3-(1,2,4-triazol-4-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
—— N-[(4S)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]pyrrolidine-1-sulfonamide —— C20H28N4O3S
N-[(4S)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]pyrrolidine-1-sulfonamide
—— 4-(1-methylimidazol-2-yl)-1-[(1R)-1-(2-pyrazol-1-ylphenyl)ethyl]triazole —— C17H17N7
4-(1-methylimidazol-2-yl)-1-[(1R)-1-(2-pyrazol-1-ylphenyl)ethyl]triazole
—— (4R)-4-(dimethylsulfamoylamino)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazole —— C18H26N4O3S
(4R)-4-(dimethylsulfamoylamino)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazole
—— 2-[(2S)-2-[4-(3-chloro-5-fluoro-4-methoxyphenyl)triazol-1-yl]propyl]pyrazine —— C16H15ClFN5O
2-[(2S)-2-[4-(3-chloro-5-fluoro-4-methoxyphenyl)triazol-1-yl]propyl]pyrazine
—— N-[[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-5-[(2S)-oxolan-2-yl]thiophene-2-carboxamide —— C19H19N3O3S
N-[[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-5-[(2S)-oxolan-2-yl]thiophene-2-carboxamide
—— N-[(4R)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]pyrrolidine-1-sulfonamide —— C20H28N4O3S
N-[(4R)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]pyrrolidine-1-sulfonamide
—— N-[[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-5-[(2R)-oxolan-2-yl]thiophene-2-carboxamide —— C19H19N3O3S
N-[[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-5-[(2R)-oxolan-2-yl]thiophene-2-carboxamide
—— (3S)-3-butyl-4-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1-methylpiperazin-2-one —— C20H26N4O3
(3S)-3-butyl-4-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1-methylpiperazin-2-one
—— 5-[(1S)-1-[4-[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]triazol-1-yl]ethyl]-2H-tetrazole —— C16H16FN9
5-[(1S)-1-[4-[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]triazol-1-yl]ethyl]-2H-tetrazole
—— 5-[4-[(3S)-oxolan-3-yl]triazol-1-yl]pentan-1-ol —— C11H19N3O2
5-[4-[(3S)-oxolan-3-yl]triazol-1-yl]pentan-1-ol
—— 5-cyclopropyl-N-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrazole-3-carboxamide —— C22H25N5O
5-cyclopropyl-N-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrazole-3-carboxamide
—— 5-[(2R)-oxolan-2-yl]-N-[(1-phenyltetrazol-5-yl)methyl]thiophene-2-carboxamide —— C17H17N5O2S
5-[(2R)-oxolan-2-yl]-N-[(1-phenyltetrazol-5-yl)methyl]thiophene-2-carboxamide
—— [(3R)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl]methanol —— C15H26N2O2S
[(3R)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl]methanol
—— 5-[4-[(3R)-oxolan-3-yl]triazol-1-yl]pentan-1-ol —— C11H19N3O2
5-[4-[(3R)-oxolan-3-yl]triazol-1-yl]pentan-1-ol
—— N-[(3R)-1-(4-chlorophenyl)-5-oxopyrrolidin-3-yl]-5-phenyl-1H-pyrazole-4-carboxamide —— C20H17ClN4O2
N-[(3R)-1-(4-chlorophenyl)-5-oxopyrrolidin-3-yl]-5-phenyl-1H-pyrazole-4-carboxamide
—— N-[(3S)-1-(4-chlorophenyl)-5-oxopyrrolidin-3-yl]-5-phenyl-1H-pyrazole-4-carboxamide —— C20H17ClN4O2
N-[(3S)-1-(4-chlorophenyl)-5-oxopyrrolidin-3-yl]-5-phenyl-1H-pyrazole-4-carboxamide
—— 1-[(1S,3R)-3-(dimethylamino)cyclopentyl]-3-[[2-(3-methylpyrazol-1-yl)phenyl]methyl]urea —— C19H27N5O
1-[(1S,3R)-3-(dimethylamino)cyclopentyl]-3-[[2-(3-methylpyrazol-1-yl)phenyl]methyl]urea
—— [(3S)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl]methanol —— C15H26N2O2S
[(3S)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl]methanol
—— (3R)-3-butyl-4-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1-methylpiperazin-2-one —— C20H26N4O3
(3R)-3-butyl-4-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1-methylpiperazin-2-one
—— 1-[(1R,3S)-3-(dimethylamino)cyclopentyl]-3-[[2-(3-methylpyrazol-1-yl)phenyl]methyl]urea —— C19H27N5O
1-[(1R,3S)-3-(dimethylamino)cyclopentyl]-3-[[2-(3-methylpyrazol-1-yl)phenyl]methyl]urea
—— 1-[(1S,3S)-3-(dimethylamino)cyclopentyl]-3-[[2-(3-methylpyrazol-1-yl)phenyl]methyl]urea —— C19H27N5O
1-[(1S,3S)-3-(dimethylamino)cyclopentyl]-3-[[2-(3-methylpyrazol-1-yl)phenyl]methyl]urea
—— 5-cyclopropyl-N-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrazole-3-carboxamide —— C22H25N5O
5-cyclopropyl-N-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrazole-3-carboxamide
—— [(2S)-2-(furan-2-yl)pyrrolidin-1-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone —— C18H17N3O2
[(2S)-2-(furan-2-yl)pyrrolidin-1-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone
—— 5-[(2S)-oxolan-2-yl]-N-[(1-phenyltetrazol-5-yl)methyl]thiophene-2-carboxamide —— C17H17N5O2S
5-[(2S)-oxolan-2-yl]-N-[(1-phenyltetrazol-5-yl)methyl]thiophene-2-carboxamide
—— 1-[(1R,3R)-3-(dimethylamino)cyclopentyl]-3-[[2-(3-methylpyrazol-1-yl)phenyl]methyl]urea —— C19H27N5O
1-[(1R,3R)-3-(dimethylamino)cyclopentyl]-3-[[2-(3-methylpyrazol-1-yl)phenyl]methyl]urea
—— [(3S)-3-(imidazol-1-ylmethyl)piperidin-1-yl]-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]methanone —— C20H23N5O2
[(3S)-3-(imidazol-1-ylmethyl)piperidin-1-yl]-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]methanone
—— N-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]methanesulfonamide —— C16H21N3O2S
N-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]methanesulfonamide
—— 1-[(1R,3R)-3-(dimethylamino)cyclopentyl]-3-[(4-propan-2-yl-1,3-thiazol-2-yl)methyl]urea —— C15H26N4OS
1-[(1R,3R)-3-(dimethylamino)cyclopentyl]-3-[(4-propan-2-yl-1,3-thiazol-2-yl)methyl]urea
—— N-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]methanesulfonamide —— C16H21N3O2S
N-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]methanesulfonamide
—— [(3R)-3-(imidazol-1-ylmethyl)piperidin-1-yl]-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]methanone —— C20H23N5O2
[(3R)-3-(imidazol-1-ylmethyl)piperidin-1-yl]-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]methanone
—— 4-(1H-imidazol-2-yl)-1-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]triazole —— C14H19N7
4-(1H-imidazol-2-yl)-1-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]triazole