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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[(4R)-1-(3,5-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-propan-2-ylurea —— C17H20F2N4O
1-[(4R)-1-(3,5-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-propan-2-ylurea
—— [(3S)-3-(1-ethylimidazol-2-yl)piperidin-1-yl]-[5-(3-methylphenyl)-1H-pyrazol-4-yl]methanone —— C21H25N5O
[(3S)-3-(1-ethylimidazol-2-yl)piperidin-1-yl]-[5-(3-methylphenyl)-1H-pyrazol-4-yl]methanone
—— (2R)-1-[3-(3,5-dimethylpyrazol-1-yl)azetidin-1-yl]-2-pyrazol-1-ylbutan-1-one —— C15H21N5O
(2R)-1-[3-(3,5-dimethylpyrazol-1-yl)azetidin-1-yl]-2-pyrazol-1-ylbutan-1-one
—— (2S)-1-[3-(3,5-dimethylpyrazol-1-yl)azetidin-1-yl]-2-pyrazol-1-ylbutan-1-one —— C15H21N5O
(2S)-1-[3-(3,5-dimethylpyrazol-1-yl)azetidin-1-yl]-2-pyrazol-1-ylbutan-1-one
—— methyl 4-chloro-2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-1,3-thiazole-5-carboxylate —— C13H18ClN3O2S
methyl 4-chloro-2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-1,3-thiazole-5-carboxylate
—— N-[(1S)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]-4-(1H-1,2,4-triazol-5-yl)benzamide —— C21H20N6O
N-[(1S)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]-4-(1H-1,2,4-triazol-5-yl)benzamide
—— 5-(3-fluorophenyl)-N-[(1S)-1-(1,3-thiazol-2-yl)propyl]-1H-pyrazole-4-carboxamide —— C16H15FN4OS
5-(3-fluorophenyl)-N-[(1S)-1-(1,3-thiazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
—— 5-[(1S)-1-[4-(6-chloro-1,3-benzodioxol-5-yl)triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine —— C13H11ClN6O2S
5-[(1S)-1-[4-(6-chloro-1,3-benzodioxol-5-yl)triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine
—— 4-methyl-2-propan-2-yl-N-[(3S)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-1,3-thiazole-5-carboxamide —— C18H25N3OS2
4-methyl-2-propan-2-yl-N-[(3S)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-1,3-thiazole-5-carboxamide
—— 4-(5-tert-butyl-1H-pyrazol-3-yl)-1-[(2S)-1-imidazol-1-ylbutan-2-yl]triazole —— C16H23N7
4-(5-tert-butyl-1H-pyrazol-3-yl)-1-[(2S)-1-imidazol-1-ylbutan-2-yl]triazole
—— 2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]-1-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethanone —— C17H18N6O2S
2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]-1-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethanone
—— 4-[2-[(2R)-butan-2-yl]oxy-3-methoxyphenyl]-1-(oxan-4-yl)triazole —— C18H25N3O3
4-[2-[(2R)-butan-2-yl]oxy-3-methoxyphenyl]-1-(oxan-4-yl)triazole
—— [(3R)-3-(1-ethylimidazol-2-yl)piperidin-1-yl]-[5-(3-methylphenyl)-1H-pyrazol-4-yl]methanone —— C21H25N5O
[(3R)-3-(1-ethylimidazol-2-yl)piperidin-1-yl]-[5-(3-methylphenyl)-1H-pyrazol-4-yl]methanone
—— (2S)-N-methyl-N-[(1-phenylpyrazol-4-yl)methyl]-3,4-dihydro-2H-chromene-2-carboxamide —— C21H21N3O2
(2S)-N-methyl-N-[(1-phenylpyrazol-4-yl)methyl]-3,4-dihydro-2H-chromene-2-carboxamide
—— 4-(5-tert-butyl-1H-pyrazol-3-yl)-1-[(2R)-1-imidazol-1-ylbutan-2-yl]triazole —— C16H23N7
4-(5-tert-butyl-1H-pyrazol-3-yl)-1-[(2R)-1-imidazol-1-ylbutan-2-yl]triazole
—— 5-[(1R)-1-[4-(6-chloro-1,3-benzodioxol-5-yl)triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine —— C13H11ClN6O2S
5-[(1R)-1-[4-(6-chloro-1,3-benzodioxol-5-yl)triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine
—— (2R)-N-methyl-N-[(1-phenylpyrazol-4-yl)methyl]-3,4-dihydro-2H-chromene-2-carboxamide —— C21H21N3O2
(2R)-N-methyl-N-[(1-phenylpyrazol-4-yl)methyl]-3,4-dihydro-2H-chromene-2-carboxamide
—— 2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]-1-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethanone —— C17H18N6O2S
2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]-1-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethanone
—— 1-ethyl-3-[(4S)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]urea —— C19H26N4O2
1-ethyl-3-[(4S)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]urea
—— 4-[2-[(2S)-butan-2-yl]oxy-3-methoxyphenyl]-1-(oxan-4-yl)triazole —— C18H25N3O3
4-[2-[(2S)-butan-2-yl]oxy-3-methoxyphenyl]-1-(oxan-4-yl)triazole
—— N-[(4S)-1-(3-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-5-methyl-1H-pyrazole-3-carboxamide —— C20H22FN5O
N-[(4S)-1-(3-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-5-methyl-1H-pyrazole-3-carboxamide
—— N-[(1R)-1-[1-(2,4-difluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-hydroxypropanamide —— C15H17F2N3O2
N-[(1R)-1-[1-(2,4-difluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-hydroxypropanamide
—— 1-[(4S)-1-(3,5-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-propan-2-ylurea —— C17H20F2N4O
1-[(4S)-1-(3,5-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-propan-2-ylurea
—— (4R)-4-[[ethyl(methyl)sulfamoyl]amino]-6,6-dimethyl-1-phenyl-5,7-dihydro-4H-indazole —— C18H26N4O2S
(4R)-4-[[ethyl(methyl)sulfamoyl]amino]-6,6-dimethyl-1-phenyl-5,7-dihydro-4H-indazole
—— (4S)-4-[[ethyl(methyl)sulfamoyl]amino]-6,6-dimethyl-1-phenyl-5,7-dihydro-4H-indazole —— C18H26N4O2S
(4S)-4-[[ethyl(methyl)sulfamoyl]amino]-6,6-dimethyl-1-phenyl-5,7-dihydro-4H-indazole
—— [4-(1H-pyrazol-5-yl)phenyl]-[(4R)-4-pyridin-3-yl-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methanone —— C21H18N6O
[4-(1H-pyrazol-5-yl)phenyl]-[(4R)-4-pyridin-3-yl-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methanone
—— N-[(1S)-1-[1-(2,4-difluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-hydroxypropanamide —— C15H17F2N3O2
N-[(1S)-1-[1-(2,4-difluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-hydroxypropanamide
—— 4-N-[(4R)-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]pyrimidine-4,6-diamine —— C19H22N6
4-N-[(4R)-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]pyrimidine-4,6-diamine
—— 2-methyl-4-[(1S)-1-[4-(3-pyrazol-1-ylphenyl)triazol-1-yl]ethyl]-1,3-thiazole —— C17H16N6S
2-methyl-4-[(1S)-1-[4-(3-pyrazol-1-ylphenyl)triazol-1-yl]ethyl]-1,3-thiazole
—— 4-N-[(4S)-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]pyrimidine-4,6-diamine —— C19H22N6
4-N-[(4S)-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]pyrimidine-4,6-diamine
—— 1-[(4S)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-phenylurea —— C20H18F2N4O
1-[(4S)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-phenylurea
—— 2-methyl-4-[(1R)-1-[4-(3-pyrazol-1-ylphenyl)triazol-1-yl]ethyl]-1,3-thiazole —— C17H16N6S
2-methyl-4-[(1R)-1-[4-(3-pyrazol-1-ylphenyl)triazol-1-yl]ethyl]-1,3-thiazole
—— N-[2-[(2R)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-4-methyl-2-propan-2-yl-1,3-thiazole-5-carboxamide —— C16H27N3O2S
N-[2-[(2R)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-4-methyl-2-propan-2-yl-1,3-thiazole-5-carboxamide
—— N-[2-[(2S)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-4-methyl-2-propan-2-yl-1,3-thiazole-5-carboxamide —— C16H27N3O2S
N-[2-[(2S)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-4-methyl-2-propan-2-yl-1,3-thiazole-5-carboxamide
—— 1-[(4R)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-phenylurea —— C20H18F2N4O
1-[(4R)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-3-phenylurea
—— N-[(4R)-1-(3-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-5-methyl-1H-pyrazole-3-carboxamide —— C20H22FN5O
N-[(4R)-1-(3-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-5-methyl-1H-pyrazole-3-carboxamide
—— [(3S)-3-aminopyrrolidin-1-yl]-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]methanone —— C15H18N4O2
[(3S)-3-aminopyrrolidin-1-yl]-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]methanone
—— N-[(1S)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-pyrrolidin-1-ylbutanamide —— C20H27FN4O
N-[(1S)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-pyrrolidin-1-ylbutanamide
—— (3R)-3-[[4-(1-methylimidazol-2-yl)triazol-1-yl]methyl]thiolane 1,1-dioxide —— C11H15N5O2S
(3R)-3-[[4-(1-methylimidazol-2-yl)triazol-1-yl]methyl]thiolane 1,1-dioxide
—— 2-methyl-N-[(1R)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]-2-pyrrol-1-ylpropanamide —— C20H24N4O
2-methyl-N-[(1R)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]-2-pyrrol-1-ylpropanamide
—— N-[(1S)-2-imidazol-1-yl-1-phenylethyl]-4-methyl-2-propan-2-yl-1,3-thiazole-5-carboxamide —— C19H22N4OS
N-[(1S)-2-imidazol-1-yl-1-phenylethyl]-4-methyl-2-propan-2-yl-1,3-thiazole-5-carboxamide
—— N-[(1R)-2-imidazol-1-yl-1-phenylethyl]-4-methyl-2-propan-2-yl-1,3-thiazole-5-carboxamide —— C19H22N4OS
N-[(1R)-2-imidazol-1-yl-1-phenylethyl]-4-methyl-2-propan-2-yl-1,3-thiazole-5-carboxamide
—— (3S)-3-[[4-(1-methylimidazol-2-yl)triazol-1-yl]methyl]thiolane 1,1-dioxide —— C11H15N5O2S
(3S)-3-[[4-(1-methylimidazol-2-yl)triazol-1-yl]methyl]thiolane 1,1-dioxide
—— [(3R)-3-aminopyrrolidin-1-yl]-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]methanone —— C15H18N4O2
[(3R)-3-aminopyrrolidin-1-yl]-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]methanone
—— [4-(1H-pyrazol-5-yl)phenyl]-[(4S)-4-pyridin-3-yl-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methanone —— C21H18N6O
[4-(1H-pyrazol-5-yl)phenyl]-[(4S)-4-pyridin-3-yl-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methanone
—— N-[(1S)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]-2-(2H-tetrazol-5-yl)benzamide —— C20H19N7O
N-[(1S)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]-2-(2H-tetrazol-5-yl)benzamide
—— 5-(3-methoxyphenyl)-N-[(1S)-1-(3-methylpyridin-2-yl)propyl]-1H-pyrazole-4-carboxamide —— C20H22N4O2
5-(3-methoxyphenyl)-N-[(1S)-1-(3-methylpyridin-2-yl)propyl]-1H-pyrazole-4-carboxamide
—— 4-[(2R)-1-[2-(5-chloro-2-methoxyphenyl)-1,2,4-triazol-3-yl]propan-2-yl]morpholine —— C16H21ClN4O2
4-[(2R)-1-[2-(5-chloro-2-methoxyphenyl)-1,2,4-triazol-3-yl]propan-2-yl]morpholine
—— N-[(1R)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-pyrrolidin-1-ylbutanamide —— C20H27FN4O
N-[(1R)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-pyrrolidin-1-ylbutanamide
—— 4-[(2S)-1-[2-(5-chloro-2-methoxyphenyl)-1,2,4-triazol-3-yl]propan-2-yl]morpholine —— C16H21ClN4O2
4-[(2S)-1-[2-(5-chloro-2-methoxyphenyl)-1,2,4-triazol-3-yl]propan-2-yl]morpholine