中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
N-[(1R)-7-fluoro-1,2,3,4-tetrahydronaphthalen-1-yl]-4-(1,2,4-triazol-4-yl)benzamide |
—— |
C19H17FN4O |
|
—— |
6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid |
—— |
C32H35N5O6S |
|
—— |
N'-(2-aminophenyl)-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]pentanediamide |
—— |
C37H39N7O6S |
|
—— |
N'-(2-aminophenyl)-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]heptanediamide |
—— |
C38H41N7O6S |
|
—— |
(3R)-3-(3-chlorophenyl)-N-methyl-5-phenyl-3,4-dihydropyrazole-2-carbothioamide |
—— |
C17H16ClN3S |
|
—— |
N'-(2-aminophenyl)-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]hexanediamide |
—— |
C37H39N7O5S |
|
—— |
N'-hydroxy-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]heptanediamide |
—— |
C32H36N6O6S |
|
—— |
[2-(cyclopropylamino)-1,3-thiazol-4-yl]-[(3S)-3-(1-methylpiperidin-4-yl)pyrrolidin-1-yl]methanone |
—— |
C17H26N4OS |
|
—— |
8-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-8-oxooctanoic acid |
—— |
C33H37N5O6S |
|
—— |
2-chloro-5-[[(2S)-2-[(2R)-1-methylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-1,3-thiazole |
—— |
C13H20ClN3S |
|
—— |
[(3S)-3-(1-methylpiperidin-4-yl)pyrrolidin-1-yl]-(1-phenyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)methanone |
—— |
C23H27N5OS |
|
—— |
7-[[4-[(2R,4R,6S)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-7-oxoheptanoic acid |
—— |
C29H33Cl2N3O6 |
|
—— |
(3S)-N-methyl-1-(1-methylpiperidin-4-yl)-N-[[1-[4-(trifluoromethyl)phenyl]tetrazol-5-yl]methyl]pyrrolidin-3-amine |
—— |
C20H28F3N7 |
|
—— |
N'-(2-aminophenyl)-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]heptanediamide |
—— |
C39H43N7O5S |
|
—— |
N'-(2-aminophenyl)-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]octanediamide |
—— |
C40H45N7O5S |
|
—— |
5-[[(2S)-2-[(2S)-1-methylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-2-phenyl-1,3-thiazole |
—— |
C19H25N3S |
|
—— |
5-[[(2S)-2-[(2R)-1-methylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-2-phenyl-1,3-thiazole |
—— |
C19H25N3S |
|
—— |
[2-(4-methoxyphenyl)-1,3-thiazol-4-yl]-[(3S)-3-(4-methylpiperazin-1-yl)azepan-1-yl]methanone |
—— |
C22H30N4O2S |
|
—— |
5-[[4-[(2R,4R,6S)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-5-oxopentanoic acid |
—— |
C27H29Cl2N3O6 |
|
—— |
[2-(cyclopropylamino)-1,3-thiazol-4-yl]-[(3R)-3-(1-methylpiperidin-4-yl)pyrrolidin-1-yl]methanone |
—— |
C17H26N4OS |
|
—— |
2-chloro-5-[[(2S)-2-[(2S)-1-methylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-1,3-thiazole |
—— |
C13H20ClN3S |
|
—— |
(3R)-N-methyl-1-(1-methylpiperidin-4-yl)-N-[[1-[4-(trifluoromethyl)phenyl]tetrazol-5-yl]methyl]pyrrolidin-3-amine |
—— |
C20H28F3N7 |
|
—— |
[(3R)-3-(1-methylpiperidin-4-yl)pyrrolidin-1-yl]-(1-phenyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)methanone |
—— |
C23H27N5OS |
|
—— |
(2R,3S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-(2-methoxyethyl)-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C28H41N3O8 |
|
—— |
4-[(2R,3S,4S)-6-[4-(1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one |
—— |
C34H42N4O7 |
|
—— |
4-[(2S,4S)-2-[2-(2-hydroxyethoxy)ethoxy]-6-(piperidine-1-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one |
—— |
C26H35N3O6 |
|
—— |
(2S,3S,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C39H44N4O7S |
|
—— |
prop-2-enyl (2R,3S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxylate |
—— |
C28H38N2O8 |
|
—— |
(2S,4S)-N-(1H-benzimidazol-2-ylmethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(3-hydroxypropoxy)-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C28H31N5O5 |
|
—— |
N-[(1R,5S)-9-methyl-9-azabicyclo[3.3.1]nonan-3-yl]-2-(tetrazol-1-yl)benzamide |
—— |
C17H22N6O |
|
—— |
(2R,3S,4S)-N-(cyclopropylmethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C29H41N3O7 |
|
—— |
(2R)-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]propanamide |
—— |
C13H15N3OS |
|
—— |
(2R,3S,4S)-N-(cyclopropylmethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C26H35N3O5 |
|
—— |
(2R,4R)-N-(1H-benzimidazol-2-ylmethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(3-hydroxypropoxy)-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C28H31N5O5 |
|
—— |
(2S)-N-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-N-methyl-2-methylsulfonylpropanamide |
—— |
C11H18N4O3S |
|
—— |
(2S,3S,4R)-N-(2,2-dimethoxyethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-N-methyl-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C27H39N3O7 |
|
—— |
(2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-N-(4-hydroxyphenyl)-2-(3-hydroxypropoxy)-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C26H29N3O6 |
|
—— |
(2S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-N-[(4-fluorophenyl)methyl]-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C35H39FN4O8S |
|
—— |
8-[(2S,3S,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carbonyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one |
—— |
C35H43N5O6 |
|
—— |
(2R,4R)-2-[2-(2-hydroxyethoxy)ethoxy]-N-(1H-imidazol-2-ylmethyl)-4-thiophen-3-yl-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C18H23N3O5S |
|
—— |
(2S,3R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C33H40N4O6 |
|
—— |
(2S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(4-hydroxybutoxy)-N-[2-[(5-nitropyridin-2-yl)amino]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C28H34N6O7 |
|
—— |
4-[(2S,3S,4R)-6-(azocane-1-carbonyl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one |
—— |
C32H47N3O7 |
|
—— |
(2S,3S,4R)-N-(1H-benzimidazol-2-ylmethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C33H41N5O7 |
|
—— |
(2S,3R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C39H44N4O7S |
|
—— |
(2S,4S)-2-[2-(2-hydroxyethoxy)ethoxy]-N-[2-(1H-imidazol-5-yl)ethyl]-4-thiophen-2-yl-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C19H25N3O5S |
|
—— |
(2R)-N-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-N-methyl-2-methylsulfonylpropanamide |
—— |
C11H18N4O3S |
|
—— |
(2S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carboxylic acid |
—— |
C25H26N2O6 |
|
—— |
prop-2-enyl (2S,3R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxylate |
—— |
C25H32N2O6 |
|
—— |
(2S,3S,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamide |
—— |
C33H40N4O6 |
|