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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[2-[(1S)-1-ethoxyethyl]-1,3-thiazol-4-yl]-N-[(3R)-3-methyloxolan-3-yl]acetamide —— C14H22N2O3S
2-[2-[(1S)-1-ethoxyethyl]-1,3-thiazol-4-yl]-N-[(3R)-3-methyloxolan-3-yl]acetamide
—— ethyl 2-[(1S)-1-cyano-2-(furan-2-ylmethylamino)-2-oxoethyl]-1,3-thiazole-4-carboxylate —— C14H13N3O4S
ethyl 2-[(1S)-1-cyano-2-(furan-2-ylmethylamino)-2-oxoethyl]-1,3-thiazole-4-carboxylate
—— ethyl 4-methyl-2-[(1R)-1-(3-phenylprop-2-ynoylamino)ethyl]-1,3-thiazole-5-carboxylate —— C18H18N2O3S
ethyl 4-methyl-2-[(1R)-1-(3-phenylprop-2-ynoylamino)ethyl]-1,3-thiazole-5-carboxylate
—— ethyl 2-[[(4R)-6,7-dihydro-4H-thieno[3,2-c]thiopyran-4-carbonyl]amino]-4-propan-2-yl-1,3-thiazole-5-carboxylate —— C17H20N2O3S3
ethyl 2-[[(4R)-6,7-dihydro-4H-thieno[3,2-c]thiopyran-4-carbonyl]amino]-4-propan-2-yl-1,3-thiazole-5-carboxylate
—— ethyl 2-[(1R)-1-[[(1S,5R)-bicyclo[3.1.0]hexane-6-carbonyl]amino]ethyl]-4-methyl-1,3-thiazole-5-carboxylate —— C16H22N2O3S
ethyl 2-[(1R)-1-[[(1S,5R)-bicyclo[3.1.0]hexane-6-carbonyl]amino]ethyl]-4-methyl-1,3-thiazole-5-carboxylate
—— 2-[2-[(1R)-1-ethoxyethyl]-1,3-thiazol-4-yl]-N-[(3S)-3-methyloxolan-3-yl]acetamide —— C14H22N2O3S
2-[2-[(1R)-1-ethoxyethyl]-1,3-thiazol-4-yl]-N-[(3S)-3-methyloxolan-3-yl]acetamide
—— ethyl 3,5-dimethyl-4-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]sulfonyl-1H-pyrrole-2-carboxylate —— C21H25N5O4S
ethyl 3,5-dimethyl-4-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]sulfonyl-1H-pyrrole-2-carboxylate
—— ethyl (4R)-4-(furan-2-yl)-2-oxo-6-[[4-(1,2,4-triazol-1-yl)benzoyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H19N5O6
ethyl (4R)-4-(furan-2-yl)-2-oxo-6-[[4-(1,2,4-triazol-1-yl)benzoyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-[(1S)-1-[[(1S,5R)-bicyclo[3.1.0]hexane-6-carbonyl]amino]ethyl]-4-methyl-1,3-thiazole-5-carboxylate —— C16H22N2O3S
ethyl 2-[(1S)-1-[[(1S,5R)-bicyclo[3.1.0]hexane-6-carbonyl]amino]ethyl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[[(4S)-6,7-dihydro-4H-thieno[3,2-c]thiopyran-4-carbonyl]amino]-4-propan-2-yl-1,3-thiazole-5-carboxylate —— C17H20N2O3S3
ethyl 2-[[(4S)-6,7-dihydro-4H-thieno[3,2-c]thiopyran-4-carbonyl]amino]-4-propan-2-yl-1,3-thiazole-5-carboxylate
—— ethyl 4-methyl-2-[(1S)-1-[(3-methylfuran-2-carbonyl)amino]ethyl]-1,3-thiazole-5-carboxylate —— C15H18N2O4S
ethyl 4-methyl-2-[(1S)-1-[(3-methylfuran-2-carbonyl)amino]ethyl]-1,3-thiazole-5-carboxylate
—— ethyl 4-methyl-2-[(1S)-1-(3-phenylprop-2-ynoylamino)ethyl]-1,3-thiazole-5-carboxylate —— C18H18N2O3S
ethyl 4-methyl-2-[(1S)-1-(3-phenylprop-2-ynoylamino)ethyl]-1,3-thiazole-5-carboxylate
—— ethyl 2-[(1R)-1-cyano-2-(furan-2-ylmethylamino)-2-oxoethyl]-1,3-thiazole-4-carboxylate —— C14H13N3O4S
ethyl 2-[(1R)-1-cyano-2-(furan-2-ylmethylamino)-2-oxoethyl]-1,3-thiazole-4-carboxylate
—— (2R)-N-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-2-ethoxypropanamide —— C11H18N4O2
(2R)-N-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-2-ethoxypropanamide
—— ethyl 2-[[(2R)-2-but-3-enoxypropanoyl]amino]-4-propan-2-yl-1,3-thiazole-5-carboxylate —— C16H24N2O4S
ethyl 2-[[(2R)-2-but-3-enoxypropanoyl]amino]-4-propan-2-yl-1,3-thiazole-5-carboxylate
—— ethyl 2-[(1S)-1-cyano-2-oxo-2-(propan-2-ylamino)ethyl]-1,3-thiazole-4-carboxylate —— C12H15N3O3S
ethyl 2-[(1S)-1-cyano-2-oxo-2-(propan-2-ylamino)ethyl]-1,3-thiazole-4-carboxylate
—— ethyl 3-[cyclopropylmethyl-[(7R)-4,5,6,7-tetrahydro-1H-indazole-7-carbonyl]amino]propanoate —— C17H25N3O3
ethyl 3-[cyclopropylmethyl-[(7R)-4,5,6,7-tetrahydro-1H-indazole-7-carbonyl]amino]propanoate
—— 5-(4-Chlorophenyl)-1,2,3-triaza-4-azanidacyclopenta-2,5-diene —— C7H4ClN4-
5-(4-Chlorophenyl)-1,2,3-triaza-4-azanidacyclopenta-2,5-diene
—— [(2R)-1-methylsulfanylpropan-2-yl] 4-(triazol-1-yl)benzoate —— C13H15N3O2S
[(2R)-1-methylsulfanylpropan-2-yl] 4-(triazol-1-yl)benzoate
—— ethyl (4R)-4-(furan-2-yl)-2-oxo-6-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H20N6O5S
ethyl (4R)-4-(furan-2-yl)-2-oxo-6-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-(furan-2-yl)-2-oxo-6-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H20N6O5S
ethyl (4S)-4-(furan-2-yl)-2-oxo-6-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-(3-fluoropropylsulfonyl)-2-[(2R)-oxolan-2-yl]-1,3-thiazole-5-carboxamide —— C11H15FN2O4S2
N-(3-fluoropropylsulfonyl)-2-[(2R)-oxolan-2-yl]-1,3-thiazole-5-carboxamide
—— (Z)-2-cyano-3-ethoxy-N-[(1R)-1-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]prop-2-enamide —— C17H18N4O4
(Z)-2-cyano-3-ethoxy-N-[(1R)-1-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]prop-2-enamide
—— ethyl 3-[cyclopropylmethyl-[(7S)-4,5,6,7-tetrahydro-1H-indazole-7-carbonyl]amino]propanoate —— C17H25N3O3
ethyl 3-[cyclopropylmethyl-[(7S)-4,5,6,7-tetrahydro-1H-indazole-7-carbonyl]amino]propanoate
—— N-ethyl-6-[[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]pyridine-3-carboxamide —— C18H20N6O
N-ethyl-6-[[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]pyridine-3-carboxamide
—— (Z)-2-cyano-3-ethoxy-N-[(1S)-1-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]prop-2-enamide —— C17H18N4O4
(Z)-2-cyano-3-ethoxy-N-[(1S)-1-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]prop-2-enamide
—— [(2S)-1-methylsulfanylpropan-2-yl] 4-(triazol-1-yl)benzoate —— C13H15N3O2S
[(2S)-1-methylsulfanylpropan-2-yl] 4-(triazol-1-yl)benzoate
—— 2-(ethylamino)-N-[[2-[(1R)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-N-methyl-1,3-thiazole-4-carboxamide —— C14H20N4O2S2
2-(ethylamino)-N-[[2-[(1R)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-N-methyl-1,3-thiazole-4-carboxamide
—— ethyl (4S)-4-(furan-2-yl)-2-oxo-6-[[4-(1,2,4-triazol-1-yl)benzoyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H19N5O6
ethyl (4S)-4-(furan-2-yl)-2-oxo-6-[[4-(1,2,4-triazol-1-yl)benzoyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 1-[(1R)-1-[3-(4-bromophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-3-ethylurea —— C13H15BrN4O2
1-[(1R)-1-[3-(4-bromophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-3-ethylurea
—— N-(3-fluoropropylsulfonyl)-2-[(2S)-oxolan-2-yl]-1,3-thiazole-5-carboxamide —— C11H15FN2O4S2
N-(3-fluoropropylsulfonyl)-2-[(2S)-oxolan-2-yl]-1,3-thiazole-5-carboxamide
—— 2-(ethylamino)-N-[(2R)-1-ethylsulfanylpropan-2-yl]-N-methyl-1,3-thiazole-4-carboxamide —— C12H21N3OS2
2-(ethylamino)-N-[(2R)-1-ethylsulfanylpropan-2-yl]-N-methyl-1,3-thiazole-4-carboxamide
—— 5-(2-Fluorophenyl)-1,2,3-triaza-4-azanidacyclopenta-2,5-diene —— C7H4FN4-
5-(2-Fluorophenyl)-1,2,3-triaza-4-azanidacyclopenta-2,5-diene
—— 2-(ethylamino)-N-[(2S)-1-ethylsulfanylpropan-2-yl]-N-methyl-1,3-thiazole-4-carboxamide —— C12H21N3OS2
2-(ethylamino)-N-[(2S)-1-ethylsulfanylpropan-2-yl]-N-methyl-1,3-thiazole-4-carboxamide
—— (Z)-N-[(1S)-1-(3-tert-butyl-1,2,4-oxadiazol-5-yl)ethyl]-2-cyano-3-ethoxyprop-2-enamide —— C14H20N4O3
(Z)-N-[(1S)-1-(3-tert-butyl-1,2,4-oxadiazol-5-yl)ethyl]-2-cyano-3-ethoxyprop-2-enamide
—— N-ethyl-6-[[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]pyridine-3-carboxamide —— C18H20N6O
N-ethyl-6-[[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]pyridine-3-carboxamide
—— 4-(2-chlorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]-1,3-thiazol-2-amine —— C14H15ClN2OS
4-(2-chlorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]-1,3-thiazol-2-amine
—— 1-[(2R)-2-(4-ethylpiperazin-1-yl)propyl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C16H29N5OS
1-[(2R)-2-(4-ethylpiperazin-1-yl)propyl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— (Z)-N-[(1R)-1-(3-tert-butyl-1,2,4-oxadiazol-5-yl)ethyl]-2-cyano-3-ethoxyprop-2-enamide —— C14H20N4O3
(Z)-N-[(1R)-1-(3-tert-butyl-1,2,4-oxadiazol-5-yl)ethyl]-2-cyano-3-ethoxyprop-2-enamide
—— 5-[2-(3,5-Dimethylpyrazol-1-yl)-5-nitrophenyl]-1,2,3-triaza-4-azanidacyclopenta-2,5-diene —— C12H10N7O2-
5-[2-(3,5-Dimethylpyrazol-1-yl)-5-nitrophenyl]-1,2,3-triaza-4-azanidacyclopenta-2,5-diene
—— 4-ethyl-N-[(1R)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]piperazine-1-carboxamide —— C17H23N5O2
4-ethyl-N-[(1R)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]piperazine-1-carboxamide
—— [2-(ethylamino)-1,3-thiazol-4-yl]-[(2S)-2-[4-(2-methylpropyl)-1,2,4-triazol-3-yl]pyrrolidin-1-yl]methanone —— C16H24N6OS
[2-(ethylamino)-1,3-thiazol-4-yl]-[(2S)-2-[4-(2-methylpropyl)-1,2,4-triazol-3-yl]pyrrolidin-1-yl]methanone
—— 1-(4-Nitrophenyl)-5-(trifluoromethyl)pyrazole-4-carboxylate —— C11H5F3N3O4-
1-(4-Nitrophenyl)-5-(trifluoromethyl)pyrazole-4-carboxylate
—— 1-[[(3R)-1-ethylpyrrolidin-3-yl]methyl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C14H24N4OS
1-[[(3R)-1-ethylpyrrolidin-3-yl]methyl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— N'-[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-N-ethylbutanediamide —— C19H26N4O2
N'-[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-N-ethylbutanediamide
—— [(1S)-1-(2-fluoro-6-pyrazol-1-ylphenyl)ethyl] 5-(ethylamino)-5-oxopentanoate —— C18H22FN3O3
[(1S)-1-(2-fluoro-6-pyrazol-1-ylphenyl)ethyl] 5-(ethylamino)-5-oxopentanoate
—— [2-(ethylamino)-1,3-thiazol-4-yl]-[(2R)-2-[4-(2-methylpropyl)-1,2,4-triazol-3-yl]pyrrolidin-1-yl]methanone —— C16H24N6OS
[2-(ethylamino)-1,3-thiazol-4-yl]-[(2R)-2-[4-(2-methylpropyl)-1,2,4-triazol-3-yl]pyrrolidin-1-yl]methanone
—— (3R)-3-(4-ethylpiperazin-1-yl)-N-[5-[(3-methoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide —— C21H30N6O2S
(3R)-3-(4-ethylpiperazin-1-yl)-N-[5-[(3-methoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide
—— (3S)-3-(4-ethylpiperazin-1-yl)-N-[5-[(3-methoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide —— C21H30N6O2S
(3S)-3-(4-ethylpiperazin-1-yl)-N-[5-[(3-methoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide
—— 1-[(2S)-2-(4-ethylpiperazin-1-yl)propyl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C16H29N5OS
1-[(2S)-2-(4-ethylpiperazin-1-yl)propyl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea