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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4,5-dimethyl-2-[(3S)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]-1,3-thiazole —— C17H25N5S
4,5-dimethyl-2-[(3S)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]-1,3-thiazole
—— (5S)-3-(2,4-dichlorophenyl)-N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H17Cl2N3O2S
(5S)-3-(2,4-dichlorophenyl)-N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-1-[(2S,3R)-2-(1-methylpyrazol-4-yl)oxolan-3-yl]methanamine —— C15H22N4OS
N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-1-[(2S,3R)-2-(1-methylpyrazol-4-yl)oxolan-3-yl]methanamine
—— 1-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[3-(2-oxopyridin-1-yl)propyl]urea —— C16H22N4O2S
1-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[3-(2-oxopyridin-1-yl)propyl]urea
—— N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-2-pyrrol-1-yl-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxamide —— C19H21N3OS3
N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-2-pyrrol-1-yl-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxamide
—— methyl 4-methyl-2-[[(5S)-5-phenyl-4,5-dihydro-1,2-oxazole-3-carbonyl]amino]-1,3-thiazole-5-carboxylate —— C16H15N3O4S
methyl 4-methyl-2-[[(5S)-5-phenyl-4,5-dihydro-1,2-oxazole-3-carbonyl]amino]-1,3-thiazole-5-carboxylate
—— N-[(1R,2R)-2-(2,4-difluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide —— C16H13F2N5OS
N-[(1R,2R)-2-(2,4-difluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide
—— 2-[(1S)-cyclohex-2-en-1-yl]sulfanyl-5-(2,4-dimethyl-1,3-thiazol-5-yl)-1,3,4-oxadiazole —— C13H15N3OS2
2-[(1S)-cyclohex-2-en-1-yl]sulfanyl-5-(2,4-dimethyl-1,3-thiazol-5-yl)-1,3,4-oxadiazole
—— methyl 4-methyl-2-[[(5R)-5-phenyl-4,5-dihydro-1,2-oxazole-3-carbonyl]amino]-1,3-thiazole-5-carboxylate —— C16H15N3O4S
methyl 4-methyl-2-[[(5R)-5-phenyl-4,5-dihydro-1,2-oxazole-3-carbonyl]amino]-1,3-thiazole-5-carboxylate
—— N-[(1R,2R)-2-(2-chlorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide —— C16H14ClN5OS
N-[(1R,2R)-2-(2-chlorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide
—— methyl (2S)-3-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoylamino]-2-phenylpropanoate —— C16H19N3O3S
methyl (2S)-3-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoylamino]-2-phenylpropanoate
—— N-methyl-2-(4-methyl-2-sulfanylidene-3H-1,3-thiazol-5-yl)-N-[(1S)-1-thiophen-2-ylethyl]acetamide —— C13H16N2OS3
N-methyl-2-(4-methyl-2-sulfanylidene-3H-1,3-thiazol-5-yl)-N-[(1S)-1-thiophen-2-ylethyl]acetamide
—— N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-1-[(2R,3R)-2-(1-methylpyrazol-4-yl)oxolan-3-yl]methanamine —— C15H22N4OS
N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-1-[(2R,3R)-2-(1-methylpyrazol-4-yl)oxolan-3-yl]methanamine
—— N-[(1S,2R)-2-(2,4-difluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide —— C16H13F2N5OS
N-[(1S,2R)-2-(2,4-difluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide
—— 2-(4-fluorophenyl)-N-[(1R)-4-hydroxy-1-phenylbutyl]-4-methyl-1,3-thiazole-5-carboxamide —— C21H21FN2O2S
2-(4-fluorophenyl)-N-[(1R)-4-hydroxy-1-phenylbutyl]-4-methyl-1,3-thiazole-5-carboxamide
—— [(1R,2S)-2-methoxycyclohexyl] 2-benzyl-4-methyl-1,3-thiazole-5-carboxylate —— C19H23NO3S
[(1R,2S)-2-methoxycyclohexyl] 2-benzyl-4-methyl-1,3-thiazole-5-carboxylate
—— 1-[[(3R,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-3-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]urea —— C15H24N4O2S
1-[[(3R,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-3-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]urea
—— [(1S,2R)-2-methoxycyclohexyl] 2-benzyl-4-methyl-1,3-thiazole-5-carboxylate —— C19H23NO3S
[(1S,2R)-2-methoxycyclohexyl] 2-benzyl-4-methyl-1,3-thiazole-5-carboxylate
—— N-[2-[(2S)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]piperidin-2-yl]ethyl]methanesulfonamide —— C14H25N3O2S2
N-[2-[(2S)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]piperidin-2-yl]ethyl]methanesulfonamide
—— (3R)-N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]thian-3-amine —— C11H18N2S2
(3R)-N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]thian-3-amine
—— (E)-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methoxy]-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethanimine —— C17H19ClN2O3S
(E)-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methoxy]-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethanimine
—— (1S,2S)-2-[3-(4,5-dimethyl-2-oxo-1,3-thiazol-3-yl)propanoylamino]cyclopentane-1-carboxamide —— C14H21N3O3S
(1S,2S)-2-[3-(4,5-dimethyl-2-oxo-1,3-thiazol-3-yl)propanoylamino]cyclopentane-1-carboxamide
—— (1S,2R)-2-[3-(4,5-dimethyl-2-oxo-1,3-thiazol-3-yl)propanoylamino]cyclopentane-1-carboxamide —— C14H21N3O3S
(1S,2R)-2-[3-(4,5-dimethyl-2-oxo-1,3-thiazol-3-yl)propanoylamino]cyclopentane-1-carboxamide
—— (2R)-2-[(2-chloro-6-fluorophenyl)methyl]-N-(4,5-dimethyl-1,3-oxazol-2-yl)pyrrolidine-1-carboxamide —— C17H19ClFN3O2
(2R)-2-[(2-chloro-6-fluorophenyl)methyl]-N-(4,5-dimethyl-1,3-oxazol-2-yl)pyrrolidine-1-carboxamide
—— (3R)-1-(2-tert-butyl-4-methyl-1,3-thiazole-5-carbonyl)pyrrolidine-3-carboxamide —— C14H21N3O2S
(3R)-1-(2-tert-butyl-4-methyl-1,3-thiazole-5-carbonyl)pyrrolidine-3-carboxamide
—— (1R,2R)-2-[3-(4,5-dimethyl-2-oxo-1,3-thiazol-3-yl)propanoylamino]cyclopentane-1-carboxamide —— C14H21N3O3S
(1R,2R)-2-[3-(4,5-dimethyl-2-oxo-1,3-thiazol-3-yl)propanoylamino]cyclopentane-1-carboxamide
—— 1-cyclopropyl-3-[3-(4,5-dimethyl-1,3-oxazol-2-yl)phenyl]-1-[[(3S)-oxolan-3-yl]methyl]urea —— C20H25N3O3
1-cyclopropyl-3-[3-(4,5-dimethyl-1,3-oxazol-2-yl)phenyl]-1-[[(3S)-oxolan-3-yl]methyl]urea
—— N-[4-thiophen-2-yl-2-[(2Z)-2-(thiophen-2-ylmethylidene)hydrazinyl]-1,3-thiazol-5-yl]furan-2-carboxamide —— C17H12N4O2S3
N-[4-thiophen-2-yl-2-[(2Z)-2-(thiophen-2-ylmethylidene)hydrazinyl]-1,3-thiazol-5-yl]furan-2-carboxamide
—— 1-(4,5-dimethyl-1,3-oxazol-2-yl)-3-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]urea —— C14H19N5O2
1-(4,5-dimethyl-1,3-oxazol-2-yl)-3-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]urea
—— [(2S)-2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-(2,4-dimethyl-1,3-thiazol-5-yl)methanone —— C15H18N4O2S
[(2S)-2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-(2,4-dimethyl-1,3-thiazol-5-yl)methanone
—— (5R)-3-(2,4-dichlorophenyl)-N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H17Cl2N3O2S
(5R)-3-(2,4-dichlorophenyl)-N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (2S)-N-[2-(4-methoxyphenyl)ethyl]-2-[(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)methylsulfanyl]propanamide —— C21H24N2O3S2
(2S)-N-[2-(4-methoxyphenyl)ethyl]-2-[(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)methylsulfanyl]propanamide
—— [(2R)-2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-(2,4-dimethyl-1,3-thiazol-5-yl)methanone —— C15H18N4O2S
[(2R)-2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-(2,4-dimethyl-1,3-thiazol-5-yl)methanone
—— (E)-1-(2,4-dimethyl-1,3-thiazol-5-yl)-N-[(4-pyrazol-1-ylphenyl)methoxy]ethanimine —— C17H18N4OS
(E)-1-(2,4-dimethyl-1,3-thiazol-5-yl)-N-[(4-pyrazol-1-ylphenyl)methoxy]ethanimine
—— (5S)-3-(2,4-dichlorophenyl)-N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H17Cl2N3O2S
(5S)-3-(2,4-dichlorophenyl)-N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (1R,2S)-2-[3-(4,5-dimethyl-2-oxo-1,3-thiazol-3-yl)propanoylamino]cyclopentane-1-carboxamide —— C14H21N3O3S
(1R,2S)-2-[3-(4,5-dimethyl-2-oxo-1,3-thiazol-3-yl)propanoylamino]cyclopentane-1-carboxamide
—— (3S)-3-[(2-methyl-3-phenylimidazol-4-yl)methylamino]-N-propan-2-ylbutanamide —— C18H26N4O
(3S)-3-[(2-methyl-3-phenylimidazol-4-yl)methylamino]-N-propan-2-ylbutanamide
—— [(2R)-2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)methanone —— C17H22N4O2S
[(2R)-2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)methanone
—— N-[3-(4,5-dimethyl-1,3-oxazol-2-yl)phenyl]-2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetamide —— C21H19N3O3S
N-[3-(4,5-dimethyl-1,3-oxazol-2-yl)phenyl]-2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetamide
—— (3R)-N-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-N-[(2-fluorophenyl)methyl]-1-methylpyrrolidin-3-amine —— C18H24FN3O
(3R)-N-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-N-[(2-fluorophenyl)methyl]-1-methylpyrrolidin-3-amine
—— N-cyclopropyl-2-[(R)-(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)methylsulfinyl]acetamide —— C14H16N2O3S2
N-cyclopropyl-2-[(R)-(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)methylsulfinyl]acetamide
—— (5S)-3-(5-chlorothiophen-2-yl)-N-[3-(4,5-dimethyl-1,3-oxazol-2-yl)phenyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H16ClN3O3S
(5S)-3-(5-chlorothiophen-2-yl)-N-[3-(4,5-dimethyl-1,3-oxazol-2-yl)phenyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 1-(4,5-dimethyl-1,3-oxazol-2-yl)-3-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]urea —— C15H25N3O3
1-(4,5-dimethyl-1,3-oxazol-2-yl)-3-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]urea
—— (2,4-dimethyl-1,3-oxazol-5-yl)-[(1R,6S)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methanone —— C16H25N3O2
(2,4-dimethyl-1,3-oxazol-5-yl)-[(1R,6S)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methanone
—— 2-hydroxy-N'-{(Z)-1-[5-methyl-1-(3-nitrophenyl)-1H-1,2,3-triazol-4-yl]ethylidene}benzohydrazide 624725-44-6 C18H16N6O4
2-hydroxy-N'-{(Z)-1-[5-methyl-1-(3-nitrophenyl)-1H-1,2,3-triazol-4-yl]ethylidene}benzohydrazide
—— [(1S)-1-(1,3-benzodioxol-5-yl)ethyl] 1-(3-methoxyphenyl)-5-methyltriazole-4-carboxylate —— C20H19N3O5
[(1S)-1-(1,3-benzodioxol-5-yl)ethyl] 1-(3-methoxyphenyl)-5-methyltriazole-4-carboxylate
—— (2,4-dimethyl-1,3-oxazol-5-yl)-[(1S,6R)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methanone —— C16H25N3O2
(2,4-dimethyl-1,3-oxazol-5-yl)-[(1S,6R)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methanone
—— 1-cyclopropyl-3-[3-(4,5-dimethyl-1,3-oxazol-2-yl)phenyl]-1-[[(3R)-oxolan-3-yl]methyl]urea —— C20H25N3O3
1-cyclopropyl-3-[3-(4,5-dimethyl-1,3-oxazol-2-yl)phenyl]-1-[[(3R)-oxolan-3-yl]methyl]urea
—— (3S)-1-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-N-methyl-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-3-amine —— C17H27N5O2
(3S)-1-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-N-methyl-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-3-amine
—— 1-(3-methoxyphenyl)-5-methyl-N-[(1R,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]triazole-4-carboxamide —— C21H28N4O2
1-(3-methoxyphenyl)-5-methyl-N-[(1R,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]triazole-4-carboxamide