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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[[(1R)-cyclohex-3-en-1-yl]methyl]-1-(3-imidazol-1-ylpropyl)-1-methylurea —— C15H24N4O
3-[[(1R)-cyclohex-3-en-1-yl]methyl]-1-(3-imidazol-1-ylpropyl)-1-methylurea
—— 2-[[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl-methylamino]methyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C17H18N4O3
2-[[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl-methylamino]methyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— (3R)-3-(diethylamino)-N-[2-methyl-5-(1,3-oxazol-2-yl)phenyl]pyrrolidine-1-carboxamide —— C19H26N4O2
(3R)-3-(diethylamino)-N-[2-methyl-5-(1,3-oxazol-2-yl)phenyl]pyrrolidine-1-carboxamide
—— (2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[2-(2-hydroxyethoxy)ethoxy]-N-[2-[(5-nitropyridin-2-yl)amino]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide —— C28H34N6O8
(2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[2-(2-hydroxyethoxy)ethoxy]-N-[2-[(5-nitropyridin-2-yl)amino]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide
—— 3-fluoro-N-[(2S)-2-hydroxy-3-methoxypropyl]-N-methyl-4-pyrazol-1-ylbenzenesulfonamide —— C14H18FN3O4S
3-fluoro-N-[(2S)-2-hydroxy-3-methoxypropyl]-N-methyl-4-pyrazol-1-ylbenzenesulfonamide
—— (2S,4S)-N-[5-(2-aminoanilino)-5-oxopentyl]-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carboxamide —— C32H41N5O6
(2S,4S)-N-[5-(2-aminoanilino)-5-oxopentyl]-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carboxamide
—— 1-[(2R)-2-hydroxy-3-methoxypropyl]-1-methyl-3-[2-(4-pyrazol-1-ylphenyl)ethyl]urea —— C17H24N4O3
1-[(2R)-2-hydroxy-3-methoxypropyl]-1-methyl-3-[2-(4-pyrazol-1-ylphenyl)ethyl]urea
—— 1-[(2S)-2-hydroxy-3-methoxypropyl]-1-methyl-3-[2-(4-pyrazol-1-ylphenyl)ethyl]urea —— C17H24N4O3
1-[(2S)-2-hydroxy-3-methoxypropyl]-1-methyl-3-[2-(4-pyrazol-1-ylphenyl)ethyl]urea
—— (2R,3S,4S)-N-cyclohexyl-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-methyl-3,4-dihydro-2H-pyran-6-carboxamide —— C32H47N3O7
(2R,3S,4S)-N-cyclohexyl-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-methyl-3,4-dihydro-2H-pyran-6-carboxamide
—— 3-fluoro-N-[(2R)-2-hydroxy-3-methoxypropyl]-N-methyl-4-pyrazol-1-ylbenzenesulfonamide —— C14H18FN3O4S
3-fluoro-N-[(2R)-2-hydroxy-3-methoxypropyl]-N-methyl-4-pyrazol-1-ylbenzenesulfonamide
—— 3-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-1-[(3R)-1,1-dioxothiolan-3-yl]-1-methylurea —— C12H19N5O3S
3-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-1-[(3R)-1,1-dioxothiolan-3-yl]-1-methylurea
—— 3-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-1-[(3S)-1,1-dioxothiolan-3-yl]-1-methylurea —— C12H19N5O3S
3-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-1-[(3S)-1,1-dioxothiolan-3-yl]-1-methylurea
—— (3S)-3-(diethylamino)-N-[2-methyl-5-(1,3-oxazol-2-yl)phenyl]pyrrolidine-1-carboxamide —— C19H26N4O2
(3S)-3-(diethylamino)-N-[2-methyl-5-(1,3-oxazol-2-yl)phenyl]pyrrolidine-1-carboxamide
—— (3S)-3-hydroxy-N-[2-methyl-5-(1,3-oxazol-2-yl)phenyl]pyrrolidine-1-carboxamide —— C15H17N3O3
(3S)-3-hydroxy-N-[2-methyl-5-(1,3-oxazol-2-yl)phenyl]pyrrolidine-1-carboxamide
—— N-[2-[(1-phenylpyrazol-4-yl)methyl]pyrazol-3-yl]pyridine-3-carboxamide —— C19H16N6O
N-[2-[(1-phenylpyrazol-4-yl)methyl]pyrazol-3-yl]pyridine-3-carboxamide
—— 5-[(3R)-3-(dimethylamino)-3,4-dihydro-2H-quinoline-1-carbonyl]-2-phenylpyrazole-3-carboxamide —— C22H23N5O2
5-[(3R)-3-(dimethylamino)-3,4-dihydro-2H-quinoline-1-carbonyl]-2-phenylpyrazole-3-carboxamide
—— 1-[(2S)-4-[[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methyl]morpholin-2-yl]-N,N-dimethylmethanamine —— C17H22FN3OS
1-[(2S)-4-[[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methyl]morpholin-2-yl]-N,N-dimethylmethanamine
—— [(2S)-hex-5-en-2-yl] 1-methylpyrazole-4-carboxylate —— C11H16N2O2
[(2S)-hex-5-en-2-yl] 1-methylpyrazole-4-carboxylate
—— (3R)-3-hydroxy-N-[2-methyl-5-(1,3-oxazol-2-yl)phenyl]pyrrolidine-1-carboxamide —— C15H17N3O3
(3R)-3-hydroxy-N-[2-methyl-5-(1,3-oxazol-2-yl)phenyl]pyrrolidine-1-carboxamide
—— (3R)-3-(dimethylamino)-N-[(2-pyrazol-1-ylphenyl)methyl]piperidine-1-carboxamide —— C18H25N5O
(3R)-3-(dimethylamino)-N-[(2-pyrazol-1-ylphenyl)methyl]piperidine-1-carboxamide
—— [(2R)-hex-5-en-2-yl] 1-methylpyrazole-4-carboxylate —— C11H16N2O2
[(2R)-hex-5-en-2-yl] 1-methylpyrazole-4-carboxylate
—— 1-[(2R)-4-[[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methyl]morpholin-2-yl]-N,N-dimethylmethanamine —— C17H22FN3OS
1-[(2R)-4-[[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methyl]morpholin-2-yl]-N,N-dimethylmethanamine
—— 5-[(3S)-3-(dimethylamino)-3,4-dihydro-2H-quinoline-1-carbonyl]-2-phenylpyrazole-3-carboxamide —— C22H23N5O2
5-[(3S)-3-(dimethylamino)-3,4-dihydro-2H-quinoline-1-carbonyl]-2-phenylpyrazole-3-carboxamide
—— 4-(5-amino-4-cyanopyrazol-1-yl)-N-[(1R)-3-hydroxy-1-phenylpropyl]-N-methylbenzamide —— C21H21N5O2
4-(5-amino-4-cyanopyrazol-1-yl)-N-[(1R)-3-hydroxy-1-phenylpropyl]-N-methylbenzamide
—— (3S)-3-(dimethylamino)-N-[(2-pyrazol-1-ylphenyl)methyl]piperidine-1-carboxamide —— C18H25N5O
(3S)-3-(dimethylamino)-N-[(2-pyrazol-1-ylphenyl)methyl]piperidine-1-carboxamide
—— [(2S)-hex-5-en-2-yl] 5-methyl-1,3-oxazole-4-carboxylate —— C11H15NO3
[(2S)-hex-5-en-2-yl] 5-methyl-1,3-oxazole-4-carboxylate
—— 4-(5-amino-4-cyanopyrazol-1-yl)-N-[(1S)-3-hydroxy-1-phenylpropyl]-N-methylbenzamide —— C21H21N5O2
4-(5-amino-4-cyanopyrazol-1-yl)-N-[(1S)-3-hydroxy-1-phenylpropyl]-N-methylbenzamide
—— 1-[(4-ethyl-1,2,4-triazol-3-yl)methyl]-3-[[(3S)-oxolan-3-yl]methyl]urea —— C11H19N5O2
1-[(4-ethyl-1,2,4-triazol-3-yl)methyl]-3-[[(3S)-oxolan-3-yl]methyl]urea
—— 4-(4-ethyl-1,2,4-triazol-3-yl)-N-[(1R)-1-[5-methyl-1-(4-methylphenyl)pyrazol-4-yl]ethyl]benzamide —— C24H26N6O
4-(4-ethyl-1,2,4-triazol-3-yl)-N-[(1R)-1-[5-methyl-1-(4-methylphenyl)pyrazol-4-yl]ethyl]benzamide
—— N-[(2R)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-4-(4-ethyl-1,2,4-triazol-3-yl)benzamide —— C23H26ClN5O2
N-[(2R)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-4-(4-ethyl-1,2,4-triazol-3-yl)benzamide
—— [(2S)-1-prop-2-ynylpyrrolidin-2-yl]methyl 1-ethylpyrazole-4-carboxylate —— C14H19N3O2
[(2S)-1-prop-2-ynylpyrrolidin-2-yl]methyl 1-ethylpyrazole-4-carboxylate
—— 1-[(2R)-2-cyclohexyl-2-(dimethylamino)ethyl]-3-[(4-ethyl-1,2,4-triazol-3-yl)methyl]urea —— C16H30N6O
1-[(2R)-2-cyclohexyl-2-(dimethylamino)ethyl]-3-[(4-ethyl-1,2,4-triazol-3-yl)methyl]urea
—— 1-[(4-ethyl-1,2,4-triazol-3-yl)methyl]-3-[(4R)-1-(2-hydroxyethyl)-4,5,6,7-tetrahydroindazol-4-yl]urea —— C15H23N7O2
1-[(4-ethyl-1,2,4-triazol-3-yl)methyl]-3-[(4R)-1-(2-hydroxyethyl)-4,5,6,7-tetrahydroindazol-4-yl]urea
—— 4-(4-ethyl-1,2,4-triazol-3-yl)-N-[(1S)-1-[5-methyl-1-(4-methylphenyl)pyrazol-4-yl]ethyl]benzamide —— C24H26N6O
4-(4-ethyl-1,2,4-triazol-3-yl)-N-[(1S)-1-[5-methyl-1-(4-methylphenyl)pyrazol-4-yl]ethyl]benzamide
—— [(2R)-hex-5-en-2-yl] 5-methyl-1,3-oxazole-4-carboxylate —— C11H15NO3
[(2R)-hex-5-en-2-yl] 5-methyl-1,3-oxazole-4-carboxylate
—— 1-[(4-ethyl-1,2,4-triazol-3-yl)methyl]-3-[(2S)-1-pyrazol-1-ylpropan-2-yl]urea —— C12H19N7O
1-[(4-ethyl-1,2,4-triazol-3-yl)methyl]-3-[(2S)-1-pyrazol-1-ylpropan-2-yl]urea
—— [(1S,6R,7S)-8,8-dimethyl-2-oxabicyclo[4.2.0]octan-7-yl] 1-ethylpyrazole-4-carboxylate —— C15H22N2O3
[(1S,6R,7S)-8,8-dimethyl-2-oxabicyclo[4.2.0]octan-7-yl] 1-ethylpyrazole-4-carboxylate
—— 1-[(4-ethyl-1,2,4-triazol-3-yl)methyl]-3-[(4S)-1-(2-hydroxyethyl)-4,5,6,7-tetrahydroindazol-4-yl]urea —— C15H23N7O2
1-[(4-ethyl-1,2,4-triazol-3-yl)methyl]-3-[(4S)-1-(2-hydroxyethyl)-4,5,6,7-tetrahydroindazol-4-yl]urea
—— 1-[3-(1-ethylimidazol-2-yl)phenyl]-3-[(1R)-1-pyridin-4-ylethyl]urea —— C19H21N5O
1-[3-(1-ethylimidazol-2-yl)phenyl]-3-[(1R)-1-pyridin-4-ylethyl]urea
—— N-[(2S)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-4-(4-ethyl-1,2,4-triazol-3-yl)benzamide —— C23H26ClN5O2
N-[(2S)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-4-(4-ethyl-1,2,4-triazol-3-yl)benzamide
—— [(2R)-1-methoxy-3-(1,2,4-triazol-1-yl)propan-2-yl] 1-ethylpyrazole-4-carboxylate —— C12H17N5O3
[(2R)-1-methoxy-3-(1,2,4-triazol-1-yl)propan-2-yl] 1-ethylpyrazole-4-carboxylate
—— [(2S)-5-(diethylamino)pent-3-yn-2-yl] 1-ethylpyrazole-4-carboxylate —— C15H23N3O2
[(2S)-5-(diethylamino)pent-3-yn-2-yl] 1-ethylpyrazole-4-carboxylate
—— 1-[(2S,3S)-2-(1-ethylpyrazol-4-yl)oxolan-3-yl]-N-[(4-methyl-1,3-thiazol-5-yl)methyl]methanamine —— C15H22N4OS
1-[(2S,3S)-2-(1-ethylpyrazol-4-yl)oxolan-3-yl]-N-[(4-methyl-1,3-thiazol-5-yl)methyl]methanamine
—— 1-[3-(1-ethylimidazol-2-yl)phenyl]-3-[(1S)-1-pyridin-4-ylethyl]urea —— C19H21N5O
1-[3-(1-ethylimidazol-2-yl)phenyl]-3-[(1S)-1-pyridin-4-ylethyl]urea
—— 1-ethyl-N-methyl-N-[(1S)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]pyrazole-4-carboxamide —— C16H24N4OS
1-ethyl-N-methyl-N-[(1S)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]pyrazole-4-carboxamide
—— 1-[(4-ethyl-1,2,4-triazol-3-yl)methyl]-3-[(2R)-1-pyrazol-1-ylpropan-2-yl]urea —— C12H19N7O
1-[(4-ethyl-1,2,4-triazol-3-yl)methyl]-3-[(2R)-1-pyrazol-1-ylpropan-2-yl]urea
—— 1-[(2S,3R)-2-(1-ethylpyrazol-4-yl)oxolan-3-yl]-N-[(4-methyl-1,3-thiazol-5-yl)methyl]methanamine —— C15H22N4OS
1-[(2S,3R)-2-(1-ethylpyrazol-4-yl)oxolan-3-yl]-N-[(4-methyl-1,3-thiazol-5-yl)methyl]methanamine
—— 1-[(2S)-2-cyclohexyl-2-(dimethylamino)ethyl]-3-[(4-ethyl-1,2,4-triazol-3-yl)methyl]urea —— C16H30N6O
1-[(2S)-2-cyclohexyl-2-(dimethylamino)ethyl]-3-[(4-ethyl-1,2,4-triazol-3-yl)methyl]urea
—— [(2S)-1-methoxy-3-(1,2,4-triazol-1-yl)propan-2-yl] 1-ethylpyrazole-4-carboxylate —— C12H17N5O3
[(2S)-1-methoxy-3-(1,2,4-triazol-1-yl)propan-2-yl] 1-ethylpyrazole-4-carboxylate
—— 1-ethyl-N-[(1S)-1-[4-(triazol-1-yl)phenyl]ethyl]pyrazole-4-carboxamide —— C16H18N6O
1-ethyl-N-[(1S)-1-[4-(triazol-1-yl)phenyl]ethyl]pyrazole-4-carboxamide