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中文名称 英文名称 CAS号 化学式 结构式图片
—— (3R)-1-cyclopentyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide —— C18H27N3O2S
(3R)-1-cyclopentyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
—— (2S)-N-[2-(2-pyrazin-2-yl-1,3-thiazol-4-yl)ethyl]-2-pyrazol-1-ylbutanamide —— C16H18N6OS
(2S)-N-[2-(2-pyrazin-2-yl-1,3-thiazol-4-yl)ethyl]-2-pyrazol-1-ylbutanamide
—— (4R)-1-(2,4-difluorophenyl)-4-[[ethyl(methyl)sulfamoyl]amino]-4,5,6,7-tetrahydroindazole —— C16H20F2N4O2S
(4R)-1-(2,4-difluorophenyl)-4-[[ethyl(methyl)sulfamoyl]amino]-4,5,6,7-tetrahydroindazole
—— (3S)-2-(2-methoxyphenyl)-3-(3-nitrophenyl)-5-phenyl-3,4-dihydropyrazole —— C22H19N3O3
(3S)-2-(2-methoxyphenyl)-3-(3-nitrophenyl)-5-phenyl-3,4-dihydropyrazole
—— 5-tert-butyl-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3,4-oxadiazol-2-amine —— C11H18N6O
5-tert-butyl-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3,4-oxadiazol-2-amine
—— 4-(3,4-dichlorophenyl)-1-[(1S)-1-(furan-2-yl)ethyl]triazole —— C14H11Cl2N3O
4-(3,4-dichlorophenyl)-1-[(1S)-1-(furan-2-yl)ethyl]triazole
—— 2-[(1R)-1-[4-[2-(furan-2-yl)phenyl]triazol-1-yl]ethyl]-3-methylpyridine —— C20H18N4O
2-[(1R)-1-[4-[2-(furan-2-yl)phenyl]triazol-1-yl]ethyl]-3-methylpyridine
—— 3-(4-methoxyphenyl)-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide —— C16H18N6O2
3-(4-methoxyphenyl)-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
—— [(3R)-4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-[3-(1,2,4-triazol-4-yl)phenyl]methanone —— C20H23N5O3
[(3R)-4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-[3-(1,2,4-triazol-4-yl)phenyl]methanone
—— [(3S)-4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-[3-(1,2,4-triazol-4-yl)phenyl]methanone —— C20H23N5O3
[(3S)-4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-[3-(1,2,4-triazol-4-yl)phenyl]methanone
—— (4S)-1-(2,4-difluorophenyl)-4-[[ethyl(methyl)sulfamoyl]amino]-4,5,6,7-tetrahydroindazole —— C16H20F2N4O2S
(4S)-1-(2,4-difluorophenyl)-4-[[ethyl(methyl)sulfamoyl]amino]-4,5,6,7-tetrahydroindazole
—— N-methyl-N-[[(3S)-1-propan-2-ylpiperidin-3-yl]methyl]-4-(1,2,4-triazol-4-yl)benzamide —— C19H27N5O
N-methyl-N-[[(3S)-1-propan-2-ylpiperidin-3-yl]methyl]-4-(1,2,4-triazol-4-yl)benzamide
—— (5R)-7-ethyl-2-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H27N3O3
(5R)-7-ethyl-2-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (2R)-N-[2-(2-pyrazin-2-yl-1,3-thiazol-4-yl)ethyl]-2-pyrazol-1-ylbutanamide —— C16H18N6OS
(2R)-N-[2-(2-pyrazin-2-yl-1,3-thiazol-4-yl)ethyl]-2-pyrazol-1-ylbutanamide
—— (5S)-7-ethyl-2-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H27N3O3
(5S)-7-ethyl-2-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 4-(3,4-dichlorophenyl)-1-[(1R)-1-(furan-2-yl)ethyl]triazole —— C14H11Cl2N3O
4-(3,4-dichlorophenyl)-1-[(1R)-1-(furan-2-yl)ethyl]triazole
—— [(3S)-3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methanone —— C20H24FN3O2
[(3S)-3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methanone
—— (4S)-3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-(1-phenyltetrazol-5-yl)piperidin-4-ol —— C19H28N6O2
(4S)-3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-(1-phenyltetrazol-5-yl)piperidin-4-ol
—— N-[(4R)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2-propoxyacetamide —— C18H21F2N3O2
N-[(4R)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2-propoxyacetamide
—— (4R)-3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-(1-phenyltetrazol-5-yl)piperidin-4-ol —— C19H28N6O2
(4R)-3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-(1-phenyltetrazol-5-yl)piperidin-4-ol
—— [(3R)-3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methanone —— C20H24FN3O2
[(3R)-3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methanone
—— N-[(4S)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2-propoxyacetamide —— C18H21F2N3O2
N-[(4S)-1-(2,4-difluorophenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2-propoxyacetamide
—— (5R)-1-[2-(4-methoxyphenyl)ethyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C23H25N3O3
(5R)-1-[2-(4-methoxyphenyl)ethyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5S)-1-[2-(4-methoxyphenyl)ethyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C23H25N3O3
(5S)-1-[2-(4-methoxyphenyl)ethyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— N-[(4S)-1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrrole-2-carboxamide —— C20H22N4O
N-[(4S)-1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrrole-2-carboxamide
—— N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide —— C16H14N6OS
N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
—— 2-[3-[1-[(1S)-1-(1-methylpyrazol-4-yl)ethyl]triazol-4-yl]phenoxy]acetamide —— C16H18N6O2
2-[3-[1-[(1S)-1-(1-methylpyrazol-4-yl)ethyl]triazol-4-yl]phenoxy]acetamide
—— 2-(2-phenylimidazol-1-yl)-N-[(2R)-1-thiophen-2-ylpropan-2-yl]acetamide —— C18H19N3OS
2-(2-phenylimidazol-1-yl)-N-[(2R)-1-thiophen-2-ylpropan-2-yl]acetamide
—— N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide —— C16H14N6OS
N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
—— N-[(4R)-1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrrole-2-carboxamide —— C20H22N4O
N-[(4R)-1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrrole-2-carboxamide
—— 2-[3-[1-[(1R)-1-(1-methylpyrazol-4-yl)ethyl]triazol-4-yl]phenoxy]acetamide —— C16H18N6O2
2-[3-[1-[(1R)-1-(1-methylpyrazol-4-yl)ethyl]triazol-4-yl]phenoxy]acetamide
—— (2R)-3-[4-(6-methoxy-1,3-benzodioxol-5-yl)triazol-1-yl]propane-1,2-diol —— C13H15N3O5
(2R)-3-[4-(6-methoxy-1,3-benzodioxol-5-yl)triazol-1-yl]propane-1,2-diol
—— N-[2-[(2R)-1-methylsulfonylpiperidin-2-yl]ethyl]-2-propyl-1,3-thiazole-4-carboxamide —— C15H25N3O3S2
N-[2-[(2R)-1-methylsulfonylpiperidin-2-yl]ethyl]-2-propyl-1,3-thiazole-4-carboxamide
—— 3-chloro-N-[(1R)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]thiophene-2-carboxamide —— C17H16ClN3OS
3-chloro-N-[(1R)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]thiophene-2-carboxamide
—— (2S)-3-[4-(6-methoxy-1,3-benzodioxol-5-yl)triazol-1-yl]propane-1,2-diol —— C13H15N3O5
(2S)-3-[4-(6-methoxy-1,3-benzodioxol-5-yl)triazol-1-yl]propane-1,2-diol
—— N-[2-[(2S)-1-methylsulfonylpiperidin-2-yl]ethyl]-2-propyl-1,3-thiazole-4-carboxamide —— C15H25N3O3S2
N-[2-[(2S)-1-methylsulfonylpiperidin-2-yl]ethyl]-2-propyl-1,3-thiazole-4-carboxamide
—— (5-phenyl-1H-pyrazol-4-yl)-[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone —— C20H23N5O
(5-phenyl-1H-pyrazol-4-yl)-[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone
—— N-[(R)-cyclopropyl-(1-methylimidazol-2-yl)methyl]-5-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide —— C19H21N5O2
N-[(R)-cyclopropyl-(1-methylimidazol-2-yl)methyl]-5-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
—— 2-(2-phenylimidazol-1-yl)-N-[(2S)-1-thiophen-2-ylpropan-2-yl]acetamide —— C18H19N3OS
2-(2-phenylimidazol-1-yl)-N-[(2S)-1-thiophen-2-ylpropan-2-yl]acetamide
—— N-[(S)-cyclopropyl-(1-methylimidazol-2-yl)methyl]-5-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide —— C19H21N5O2
N-[(S)-cyclopropyl-(1-methylimidazol-2-yl)methyl]-5-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
—— (5-phenyl-1H-pyrazol-4-yl)-[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone —— C20H23N5O
(5-phenyl-1H-pyrazol-4-yl)-[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone
—— 3-(4-methoxyphenyl)-N-methyl-N-[(1R)-1-(3-phenyl-1H-pyrazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide —— C23H23N5O2
3-(4-methoxyphenyl)-N-methyl-N-[(1R)-1-(3-phenyl-1H-pyrazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
—— N-[2-[(2S)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C19H26N4O3
N-[2-[(2S)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— [2-[(dimethylamino)methyl]-1,3-thiazol-4-yl]-[(3S)-3-[[3-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methanone —— C19H25N3O2S
[2-[(dimethylamino)methyl]-1,3-thiazol-4-yl]-[(3S)-3-[[3-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methanone
—— N-[(1S)-2-methoxy-1-pyridin-2-ylethyl]-N,4-dimethyl-2-propan-2-yl-1,3-thiazole-5-carboxamide —— C17H23N3O2S
N-[(1S)-2-methoxy-1-pyridin-2-ylethyl]-N,4-dimethyl-2-propan-2-yl-1,3-thiazole-5-carboxamide
—— N-[(1R)-1-[1-(4-methoxyphenyl)-5-methylpyrazol-4-yl]ethyl]-1,1-dioxothiane-4-carboxamide —— C19H25N3O4S
N-[(1R)-1-[1-(4-methoxyphenyl)-5-methylpyrazol-4-yl]ethyl]-1,1-dioxothiane-4-carboxamide
—— N-[2-[(2R)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C19H26N4O3
N-[2-[(2R)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— [2-[(dimethylamino)methyl]-1,3-thiazol-4-yl]-[(3R)-3-[[3-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methanone —— C19H25N3O2S
[2-[(dimethylamino)methyl]-1,3-thiazol-4-yl]-[(3R)-3-[[3-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methanone
—— [(2R)-oxolan-2-yl]-[4-[3-(1,2,4-triazol-4-yl)benzoyl]-1,4-diazepan-1-yl]methanone —— C19H23N5O3
[(2R)-oxolan-2-yl]-[4-[3-(1,2,4-triazol-4-yl)benzoyl]-1,4-diazepan-1-yl]methanone
—— [(2S)-oxolan-2-yl]-[4-[3-(1,2,4-triazol-4-yl)benzoyl]-1,4-diazepan-1-yl]methanone —— C19H23N5O3
[(2S)-oxolan-2-yl]-[4-[3-(1,2,4-triazol-4-yl)benzoyl]-1,4-diazepan-1-yl]methanone