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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5E)-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-[[2-(3,5-dimethylpiperidin-1-yl)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C30H30N6O3S2
(5E)-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-[[2-(3,5-dimethylpiperidin-1-yl)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-(2,5-dimethylpyrrol-1-yl)-1-methyl-N-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]pyrazole-4-carboxamide —— C20H30N4O2
5-(2,5-dimethylpyrrol-1-yl)-1-methyl-N-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]pyrazole-4-carboxamide
—— (5E)-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-[(4-oxo-2-piperidin-1-ylpyrido[1,2-a]pyrimidin-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C28H26N6O3S2
(5E)-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-[(4-oxo-2-piperidin-1-ylpyrido[1,2-a]pyrimidin-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-(2,5-dimethylpyrrol-1-yl)-1-methyl-N-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]pyrazole-4-carboxamide —— C20H30N4O2
5-(2,5-dimethylpyrrol-1-yl)-1-methyl-N-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]pyrazole-4-carboxamide
—— (2R)-4-[[3-(3-methoxy-4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-methylmorpholine —— C16H21N3O3
(2R)-4-[[3-(3-methoxy-4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-methylmorpholine
—— [(2R)-2-(3,4-dimethylphenyl)pyrrolidin-1-yl]-[1-(2-fluorophenyl)pyrazol-3-yl]methanone —— C22H22FN3O
[(2R)-2-(3,4-dimethylphenyl)pyrrolidin-1-yl]-[1-(2-fluorophenyl)pyrazol-3-yl]methanone
—— 3-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-4-hydroxy-1-methoxybutan-2-yl]propanamide —— C17H22FN3O4
3-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-4-hydroxy-1-methoxybutan-2-yl]propanamide
—— 1-[(1R)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]-3-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C15H21N3O3S
1-[(1R)-2-methoxy-1-(5-methylfuran-2-yl)ethyl]-3-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— 3-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-4-hydroxy-1-methoxybutan-2-yl]propanamide —— C17H22FN3O4
3-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-4-hydroxy-1-methoxybutan-2-yl]propanamide
—— 5-(2,5-dimethylpyrrol-1-yl)-1-methyl-N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]pyrazole-4-carboxamide —— C20H30N4O2
5-(2,5-dimethylpyrrol-1-yl)-1-methyl-N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]pyrazole-4-carboxamide
—— 5-(4-chlorophenyl)-3-[[(S)-(3,4-dimethylphenyl)sulfinyl]methyl]-1,2,4-oxadiazole —— C17H15ClN2O2S
5-(4-chlorophenyl)-3-[[(S)-(3,4-dimethylphenyl)sulfinyl]methyl]-1,2,4-oxadiazole
—— (2S)-4-[[3-(3-methoxy-4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-methylmorpholine —— C16H21N3O3
(2S)-4-[[3-(3-methoxy-4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-methylmorpholine
—— 3-tert-butyl-5-[[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]sulfanylmethyl]-1,2,4-oxadiazole —— C18H21FN4O2S
3-tert-butyl-5-[[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]sulfanylmethyl]-1,2,4-oxadiazole
—— 3-(3-fluoro-4-methylphenyl)-5-[(1S)-1-pyridin-2-ylsulfanylethyl]-1,2,4-oxadiazole —— C16H14FN3OS
3-(3-fluoro-4-methylphenyl)-5-[(1S)-1-pyridin-2-ylsulfanylethyl]-1,2,4-oxadiazole
—— 3-tert-butyl-5-[[(1R)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]sulfanylmethyl]-1,2,4-oxadiazole —— C18H21FN4O2S
3-tert-butyl-5-[[(1R)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]sulfanylmethyl]-1,2,4-oxadiazole
—— (4R)-N-tert-butyl-3-(1-phenylpyrazole-3-carbonyl)-1,3-thiazolidine-4-carboxamide —— C18H22N4O2S
(4R)-N-tert-butyl-3-(1-phenylpyrazole-3-carbonyl)-1,3-thiazolidine-4-carboxamide
—— (3S)-1-[(1R)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-phenylpyrrolidin-3-amine —— C21H23FN4O
(3S)-1-[(1R)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-phenylpyrrolidin-3-amine
—— [(1R,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-[5-(4-methylphenyl)-1,3-oxazol-4-yl]methanone —— C17H18N2O2
[(1R,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-[5-(4-methylphenyl)-1,3-oxazol-4-yl]methanone
—— (3S)-1-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-phenylpyrrolidin-3-amine —— C21H23FN4O
(3S)-1-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-phenylpyrrolidin-3-amine
—— 5-(4-chlorophenyl)-3-[[(R)-(3,4-dimethylphenyl)sulfinyl]methyl]-1,2,4-oxadiazole —— C17H15ClN2O2S
5-(4-chlorophenyl)-3-[[(R)-(3,4-dimethylphenyl)sulfinyl]methyl]-1,2,4-oxadiazole
—— 3-tert-butyl-N-[(2S)-2-[4-(difluoromethoxy)phenyl]-2-hydroxyethyl]-1-(4-methylphenyl)pyrazole-4-carboxamide —— C24H27F2N3O3
3-tert-butyl-N-[(2S)-2-[4-(difluoromethoxy)phenyl]-2-hydroxyethyl]-1-(4-methylphenyl)pyrazole-4-carboxamide
—— [3-tert-butyl-1-(4-methylphenyl)pyrazol-4-yl]-[4-[[(2S)-1,4-dioxan-2-yl]methyl]piperazin-1-yl]methanone —— C24H34N4O3
[3-tert-butyl-1-(4-methylphenyl)pyrazol-4-yl]-[4-[[(2S)-1,4-dioxan-2-yl]methyl]piperazin-1-yl]methanone
—— (5E)-2-(4-Bromophenyl)-5-({3-[4-(isopentyloxy)phenyl]-1-phenyl-1H-pyrazol-4-YL}methylene)[1,3]thiazolo[3,2-B][1,2,4]triazol-6(5H)-one —— C31H26BrN5O2S
(5E)-2-(4-Bromophenyl)-5-({3-[4-(isopentyloxy)phenyl]-1-phenyl-1H-pyrazol-4-YL}methylene)[1,3]thiazolo[3,2-B][1,2,4]triazol-6(5H)-one
—— (2R)-N-cyclohexyl-N,3-dimethyl-2-[1-(4-methylphenyl)tetrazol-5-yl]sulfanylbutanamide —— C20H29N5OS
(2R)-N-cyclohexyl-N,3-dimethyl-2-[1-(4-methylphenyl)tetrazol-5-yl]sulfanylbutanamide
—— N-[[(2R)-1,4-dioxan-2-yl]methyl]-2-[5-(4-methylphenyl)-1,3-oxazol-2-yl]benzamide —— C22H22N2O4
N-[[(2R)-1,4-dioxan-2-yl]methyl]-2-[5-(4-methylphenyl)-1,3-oxazol-2-yl]benzamide
—— (1E)-1-[[4-chloro-3-([1,3]oxazolo[4,5-b]pyridin-2-yl)anilino]methylidene]naphthalen-2-one —— C23H14ClN3O2
(1E)-1-[[4-chloro-3-([1,3]oxazolo[4,5-b]pyridin-2-yl)anilino]methylidene]naphthalen-2-one
—— 5-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methylsulfanyl]-1-(4-methylphenyl)tetrazole —— C17H16N4OS
5-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methylsulfanyl]-1-(4-methylphenyl)tetrazole
—— (4S)-N-tert-butyl-3-(1-phenylpyrazole-3-carbonyl)-1,3-thiazolidine-4-carboxamide —— C18H22N4O2S
(4S)-N-tert-butyl-3-(1-phenylpyrazole-3-carbonyl)-1,3-thiazolidine-4-carboxamide
—— [(2S)-2-(3,4-dimethylphenyl)pyrrolidin-1-yl]-[1-(2-fluorophenyl)pyrazol-3-yl]methanone —— C22H22FN3O
[(2S)-2-(3,4-dimethylphenyl)pyrrolidin-1-yl]-[1-(2-fluorophenyl)pyrazol-3-yl]methanone
—— (2S)-2-methyl-1-[[1-(4-methylphenyl)tetrazol-5-yl]amino]-3-methylsulfanylpropan-2-ol —— C13H19N5OS
(2S)-2-methyl-1-[[1-(4-methylphenyl)tetrazol-5-yl]amino]-3-methylsulfanylpropan-2-ol
—— 2-[2-[(R)-(2,5-dichlorophenyl)sulfinyl]ethyl]-5-(4-methylphenyl)tetrazole —— C16H14Cl2N4OS
2-[2-[(R)-(2,5-dichlorophenyl)sulfinyl]ethyl]-5-(4-methylphenyl)tetrazole
—— (2R)-3,3-dimethyl-2-[(3-phenyltriazolo[4,5-d]pyrimidin-7-yl)amino]butan-1-ol —— C16H20N6O
(2R)-3,3-dimethyl-2-[(3-phenyltriazolo[4,5-d]pyrimidin-7-yl)amino]butan-1-ol
—— [3-tert-butyl-1-(4-methylphenyl)pyrazol-4-yl]-[4-[[(2R)-1,4-dioxan-2-yl]methyl]piperazin-1-yl]methanone —— C24H34N4O3
[3-tert-butyl-1-(4-methylphenyl)pyrazol-4-yl]-[4-[[(2R)-1,4-dioxan-2-yl]methyl]piperazin-1-yl]methanone
—— (Z)-[[amino-[(4-bromo-2-methyl-5-oxo-1-phenylpyrazol-3-yl)methylsulfanyl]methylidene]amino]-[(4-methoxyphenyl)methylidene]azanium —— C20H21BrN5O2S+
(Z)-[[amino-[(4-bromo-2-methyl-5-oxo-1-phenylpyrazol-3-yl)methylsulfanyl]methylidene]amino]-[(4-methoxyphenyl)methylidene]azanium
—— N-[(2R)-2-hydroxy-3-methylbutyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide —— C16H20N2O3
N-[(2R)-2-hydroxy-3-methylbutyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide
—— 3-(3-fluoro-4-methylphenyl)-5-[(1R)-1-pyridin-2-ylsulfanylethyl]-1,2,4-oxadiazole —— C16H14FN3OS
3-(3-fluoro-4-methylphenyl)-5-[(1R)-1-pyridin-2-ylsulfanylethyl]-1,2,4-oxadiazole
—— N-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]cyclopentanesulfonamide —— C17H23N3O2S
N-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]cyclopentanesulfonamide
—— 1-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]-3-[[(2R)-oxolan-2-yl]methyl]thiourea —— C18H24N4OS
1-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]-3-[[(2R)-oxolan-2-yl]methyl]thiourea
—— N-[(2S)-2-hydroxy-3-methylbutyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide —— C16H20N2O3
N-[(2S)-2-hydroxy-3-methylbutyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide
—— 2-[5-(4-methylphenyl)tetrazol-2-yl]-N-[(1R,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C20H27N5O
2-[5-(4-methylphenyl)tetrazol-2-yl]-N-[(1R,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— 2-chloro-N-[(Z)-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)methylideneamino]-5-(trifluoromethyl)aniline —— C21H14ClF3N4S
2-chloro-N-[(Z)-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)methylideneamino]-5-(trifluoromethyl)aniline
—— [(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-[5-(4-methylphenyl)-1,3-oxazol-4-yl]methanone —— C17H18N2O2
[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-[5-(4-methylphenyl)-1,3-oxazol-4-yl]methanone
—— (5E)-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-[[2-(3-methylpiperidin-1-yl)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H28N6O3S2
(5E)-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-[[2-(3-methylpiperidin-1-yl)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— N-[(1R)-2,2-dimethyl-1-thiophen-2-ylpropyl]-1-phenylpyrazole-3-carboxamide —— C19H21N3OS
N-[(1R)-2,2-dimethyl-1-thiophen-2-ylpropyl]-1-phenylpyrazole-3-carboxamide
—— (2S)-3,3-dimethyl-2-[(3-phenyltriazolo[4,5-d]pyrimidin-7-yl)amino]butan-1-ol —— C16H20N6O
(2S)-3,3-dimethyl-2-[(3-phenyltriazolo[4,5-d]pyrimidin-7-yl)amino]butan-1-ol
—— 3-tert-butyl-N-[(2R)-2-[4-(difluoromethoxy)phenyl]-2-hydroxyethyl]-1-(4-methylphenyl)pyrazole-4-carboxamide —— C24H27F2N3O3
3-tert-butyl-N-[(2R)-2-[4-(difluoromethoxy)phenyl]-2-hydroxyethyl]-1-(4-methylphenyl)pyrazole-4-carboxamide
—— (2S)-N-cyclohexyl-N,3-dimethyl-2-[1-(4-methylphenyl)tetrazol-5-yl]sulfanylbutanamide —— C20H29N5OS
(2S)-N-cyclohexyl-N,3-dimethyl-2-[1-(4-methylphenyl)tetrazol-5-yl]sulfanylbutanamide
—— 3-(2-bromophenyl)-4-[(Z)-(2-bromophenyl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C15H10Br2N4S
3-(2-bromophenyl)-4-[(Z)-(2-bromophenyl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— 1-(4-amino-1,2,5-oxadiazol-3-yl)-N'-[(1Z)-1-(2-chlorophenyl)ethylidene]-5-phenyl-1H-1,2,3-triazole-4-carbohydrazide —— C19H15ClN8O2
1-(4-amino-1,2,5-oxadiazol-3-yl)-N'-[(1Z)-1-(2-chlorophenyl)ethylidene]-5-phenyl-1H-1,2,3-triazole-4-carbohydrazide
—— N-[(2S)-2-hydroxy-3-(2-methylpropoxy)propyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide —— C18H24N2O4
N-[(2S)-2-hydroxy-3-(2-methylpropoxy)propyl]-5-(4-methylphenyl)-1,3-oxazole-4-carboxamide